UA73804C2 - Anticholinergic agents being used as medicaments, a method for the preparation thereof and a pharmaceutical composition - Google Patents

Anticholinergic agents being used as medicaments, a method for the preparation thereof and a pharmaceutical composition Download PDF

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Publication number
UA73804C2
UA73804C2 UA2003054186A UA2003054186A UA73804C2 UA 73804 C2 UA73804 C2 UA 73804C2 UA 2003054186 A UA2003054186 A UA 2003054186A UA 2003054186 A UA2003054186 A UA 2003054186A UA 73804 C2 UA73804 C2 UA 73804C2
Authority
UA
Ukraine
Prior art keywords
group
methyl
compounds
general formula
residue
Prior art date
Application number
UA2003054186A
Other languages
English (en)
Ukrainian (uk)
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of UA73804C2 publication Critical patent/UA73804C2/uk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Reproductive Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
UA2003054186A 2000-10-14 2001-09-28 Anticholinergic agents being used as medicaments, a method for the preparation thereof and a pharmaceutical composition UA73804C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10050994A DE10050994A1 (de) 2000-10-14 2000-10-14 Neue als Arneimittel einsetzbare Anticholinergika sowie Verfahren zu deren Herstellung
PCT/EP2001/011226 WO2002032899A1 (de) 2000-10-14 2001-09-28 Neue als arzneimittel einsetzbare anticholinergika sowie verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
UA73804C2 true UA73804C2 (en) 2005-09-15

Family

ID=7659808

Family Applications (1)

Application Number Title Priority Date Filing Date
UA2003054186A UA73804C2 (en) 2000-10-14 2001-09-28 Anticholinergic agents being used as medicaments, a method for the preparation thereof and a pharmaceutical composition

Country Status (37)

Country Link
EP (2) EP1382606A3 (sr)
JP (2) JP4109106B2 (sr)
KR (1) KR100830359B1 (sr)
CN (1) CN1275962C (sr)
AR (1) AR035589A1 (sr)
AT (1) ATE259805T1 (sr)
AU (2) AU1397502A (sr)
BG (1) BG66225B1 (sr)
BR (1) BR0114635A (sr)
CA (1) CA2425557C (sr)
DE (2) DE10050994A1 (sr)
DK (1) DK1325001T3 (sr)
EA (1) EA005816B1 (sr)
EC (1) ECSP034542A (sr)
EE (1) EE05179B1 (sr)
ES (1) ES2215147T3 (sr)
HR (1) HRP20030278B1 (sr)
HU (1) HUP0301203A3 (sr)
IL (2) IL155334A0 (sr)
ME (1) MEP39908A (sr)
MX (1) MXPA03003160A (sr)
MY (1) MY127144A (sr)
NO (1) NO328207B1 (sr)
NZ (1) NZ525836A (sr)
PE (1) PE20020433A1 (sr)
PL (1) PL207311B1 (sr)
PT (1) PT1325001E (sr)
RS (1) RS50464B (sr)
SA (1) SA01220414B1 (sr)
SI (1) SI1325001T1 (sr)
SK (1) SK287138B6 (sr)
TR (1) TR200400376T4 (sr)
TW (1) TWI306098B (sr)
UA (1) UA73804C2 (sr)
UY (1) UY26958A1 (sr)
WO (1) WO2002032899A1 (sr)
ZA (1) ZA200302914B (sr)

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DE10216429A1 (de) * 2002-04-12 2003-10-23 Boehringer Ingelheim Pharma Arzneimittel enthaltend Steroide und ein neues Anticholinergikum
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Also Published As

Publication number Publication date
AR035589A1 (es) 2004-06-16
CA2425557A1 (en) 2003-04-11
AU1397502A (en) 2002-04-29
IL155334A (en) 2009-02-11
TWI306098B (en) 2009-02-11
MY127144A (en) 2006-11-30
CN1275962C (zh) 2006-09-20
CN1468236A (zh) 2004-01-14
MEP39908A (en) 2011-02-10
AU2002213975B2 (en) 2006-11-09
EE200300151A (et) 2003-06-16
RS50464B (sr) 2010-03-02
BR0114635A (pt) 2004-02-10
ECSP034542A (es) 2003-06-25
ZA200302914B (en) 2003-11-14
IL155334A0 (en) 2003-11-23
PL207311B1 (pl) 2010-11-30
HUP0301203A3 (en) 2006-05-29
HRP20030278B1 (en) 2006-02-28
HUP0301203A2 (hu) 2003-10-28
YU29503A (sh) 2006-03-03
EP1325001B1 (de) 2004-02-18
JP2004511557A (ja) 2004-04-15
EP1382606A3 (de) 2004-10-13
EP1382606A2 (de) 2004-01-21
WO2002032899A1 (de) 2002-04-25
PT1325001E (pt) 2004-07-30
NO20031693L (no) 2003-05-28
PL360673A1 (en) 2004-09-20
SA01220414B1 (ar) 2007-01-20
EA200300459A1 (ru) 2003-10-30
EP1325001A1 (de) 2003-07-09
KR20030041165A (ko) 2003-05-23
JP2008120834A (ja) 2008-05-29
MXPA03003160A (es) 2005-09-09
UY26958A1 (es) 2002-06-20
NO328207B1 (no) 2010-01-11
PE20020433A1 (es) 2002-06-28
ATE259805T1 (de) 2004-03-15
EE05179B1 (et) 2009-06-15
SK287138B6 (sk) 2010-01-07
TR200400376T4 (tr) 2004-03-22
CA2425557C (en) 2007-11-13
SK4352003A3 (en) 2003-08-05
EA005816B1 (ru) 2005-06-30
BG107688A (bg) 2003-09-30
ES2215147T3 (es) 2004-10-01
JP4109106B2 (ja) 2008-07-02
NZ525836A (en) 2004-09-24
KR100830359B1 (ko) 2008-05-20
DK1325001T3 (da) 2004-06-21
DE10050994A1 (de) 2002-04-18
HK1060566A1 (en) 2004-08-13
BG66225B1 (bg) 2012-06-29
NO20031693D0 (no) 2003-04-11
HRP20030278A2 (en) 2005-02-28
SI1325001T1 (sl) 2004-08-31
DE50101524D1 (de) 2004-03-25

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