UA77329C2 - Combination of alpha-2-delta ligand and a pdev inhibitor for use in therapy of pain - Google Patents

Combination of alpha-2-delta ligand and a pdev inhibitor for use in therapy of pain Download PDF

Info

Publication number: UA77329C2
Authority: UA; Ukraine
Prior art keywords: acid; pain; methyl; alpha; alkyl
Prior art date: 2002-08-15

Application number

UAA200501347A

Other languages

English (en)

Ukrainian (uk)

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-08-15

Filing date

2003-04-08

Publication date

2006-11-15

2003-04-08 Application filed by Pfizer filed Critical Pfizer

2006-11-15 Publication of UA77329C2 publication Critical patent/UA77329C2/uk

Links

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Health & Medical Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Epidemiology (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Orthopedic Medicine & Surgery (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Cardiology (AREA)
Physical Education & Sports Medicine (AREA)
Rheumatology (AREA)
Psychiatry (AREA)
Immunology (AREA)
Vascular Medicine (AREA)
Gynecology & Obstetrics (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Hospice & Palliative Care (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

UAA200501347A 2002-08-15 2003-04-08 Combination of alpha-2-delta ligand and a pdev inhibitor for use in therapy of pain UA77329C2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB0219024.7A GB0219024D0 (en)	2002-08-15	2002-08-15	Synergistic combinations
PCT/IB2003/003476 WO2004016259A1 (en)	2002-08-15	2003-08-04	Synergistic combination of an alpha-2-delta ligand and a pdev inhibitor for use in the treatment of pain

Publications (1)

Publication Number	Publication Date
UA77329C2 true UA77329C2 (en)	2006-11-15

Family

ID=9942388

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UAA200501347A UA77329C2 (en)	2002-08-15	2003-04-08	Combination of alpha-2-delta ligand and a pdev inhibitor for use in therapy of pain

Country Status (40)

Country	Link
EP (1)	EP1536782B1 (de)
JP (1)	JP2006502139A (de)
KR (2)	KR20070009746A (de)
CN (1)	CN1674884A (de)
AP (1)	AP2005003227A0 (de)
AR (1)	AR040871A1 (de)
AT (1)	ATE359775T1 (de)
AU (1)	AU2003249476B2 (de)
BR (1)	BR0313484A (de)
CA (1)	CA2495433A1 (de)
CR (1)	CR7687A (de)
DE (1)	DE60313330T2 (de)
DK (1)	DK1536782T3 (de)
EA (1)	EA007504B1 (de)
EC (1)	ECSP055593A (de)
ES (1)	ES2285230T3 (de)
GB (1)	GB0219024D0 (de)
GE (1)	GEP20084366B (de)
GT (1)	GT200300173A (de)
HN (1)	HN2003000247A (de)
HR (1)	HRP20050136A2 (de)
IL (1)	IL166415A0 (de)
IS (1)	IS7643A (de)
MA (1)	MA27381A1 (de)
MX (1)	MXPA05001835A (de)
NO (1)	NO20050782L (de)
NZ (1)	NZ537818A (de)
OA (1)	OA12899A (de)
PA (1)	PA8577301A1 (de)
PE (1)	PE20040992A1 (de)
PL (1)	PL375553A1 (de)
PT (1)	PT1536782E (de)
RS (1)	RS20050078A (de)
SI (1)	SI1536782T1 (de)
TN (1)	TNSN05042A1 (de)
TW (1)	TW200404531A (de)
UA (1)	UA77329C2 (de)
UY (1)	UY27936A1 (de)
WO (1)	WO2004016259A1 (de)
ZA (1)	ZA200500369B (de)

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NI200300043A (es)	2002-03-28	2003-11-05	Warner Lambert Co	AMINOACIDOS CON AFINIDAD POR LA PROTEINA a2DELTA.
JP2007505095A (ja) *	2003-09-12	2007-03-08	ワーナー−ランバートカンパニーリミティドライアビリティーカンパニー	うつ病及び不安障害の治療のためのアルファ−２−デルタリガンド及びｓｓｒｉ及び／又はｓｎｒｉを含む組み合わせ
CA2539976A1 (en)	2003-09-25	2005-04-07	Warner-Lambert Company Llc	Therapeutic beta aminoacids
OA13258A (en) *	2003-09-25	2007-01-31	Warner Lambert Co	Amino acids with affinity for the alpha2delta-protein.
GB0405200D0 (en) *	2004-03-08	2004-04-21	Pfizer Ltd	Combinations comprising alpha-2-delta ligands
MXPA06014662A (es) *	2004-07-09	2007-02-12	Warner Lambert Co	Preparacion de beta-amino acidos que tienen afinidad por la proteina alfa-2-delta.
ITMI20041447A1 (it) *	2004-07-20	2004-10-20	Zambon Spa	Composizione farmaceutica comprendente gabapentina
US20090227562A1 (en) *	2004-08-10	2009-09-10	Pfizer Inc.	Combination of a Selective Noradrenaline Reuptake Unhibitor and a PDEV Inhibitor
EP1791599A1 (de) *	2004-09-07	2007-06-06	Pfizer Limited	Kombination aus einem 5-ht(1) rezeptor-agonisten und einem alpha-2-delta-liganden zur behandlung von migräne
WO2006092692A1 (en) *	2005-03-01	2006-09-08	Pfizer Limited	Use of combinations of pde7 inhibitors and alpha-2-delty ligands for the treatment of neuropathic pain
CA2685395A1 (en) *	2007-04-30	2008-11-06	Adolor Corporation	Compositions of (-)-e-10-oh-nt and methods for their synthesis and use
WO2008132589A1 (en) *	2007-05-01	2008-11-06	Pfizer Limited	Combinations comprising pregabalin
US20090148532A1 (en) *	2007-12-06	2009-06-11	Venkatesh Gopi M	Preparation of controlled release skeletal muscle relaxant dosage forms
TWI531362B (zh)	2008-07-21	2016-05-01	艾爾康股份有限公司	具有治療劑遞送能力之眼科裝置
CA2805371C (en) *	2010-07-30	2017-10-31	Toray Industries, Inc.	Therapeutic agent or prophylactic agent for neuropathic pain
PL2710005T3 (pl)	2011-05-17	2017-07-31	Principia Biopharma Inc.	Inhibitory kinazy tyrozynowej
ES2770550T3 (es)	2011-05-17	2020-07-02	Univ California	Inhibidores de quinasa
WO2012158795A1 (en)	2011-05-17	2012-11-22	Principia Biopharma Inc.	Pyrazolopyrimidine derivatives as tyrosine kinase inhibitors
WO2013084182A1 (en) *	2011-12-08	2013-06-13	Glenmark Pharmaceuticals S.A.	Pharmaceutical composition that includes a pde4 enzyme inhibitor and an analgesic agent
SI2892900T1 (en)	2012-09-10	2018-01-31	Principia Biopharma Inc.	Pyrazolopyrimidine compounds as kinase inhibitors
US8957080B2 (en)	2013-04-09	2015-02-17	Principia Biopharma Inc.	Tyrosine kinase inhibitors
CN112353806A (zh)	2014-02-21	2021-02-12	普林斯匹亚生物制药公司	Btk抑制剂的盐和固体形式
SG11201704808VA (en)	2014-12-18	2017-07-28	Principia Biopharma Inc	Treatment of pemphigus
WO2016210165A1 (en)	2015-06-24	2016-12-29	Principia Biopharma Inc.	Tyrosine kinase inhibitors
CN115054586B (zh)	2016-06-29	2024-08-02	普林斯匹亚生物制药公司	改性的释放制剂
US20210106584A1 (en)	2019-10-14	2021-04-15	Principia Biopharma Inc.	Methods for treating immune thrombocytopenia by administering (r)-2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile
US11814390B2 (en)	2020-01-22	2023-11-14	Principia Biopharma Inc.	Crystalline forms of 2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)-1H-pyrazolo[3,4-D]pyrimidin-1-yl]piperidine-1-carbonyl]-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile
CN114195661B (zh) *	2021-12-21	2023-12-22	苏州楚凯药业有限公司	一种苯磺酸米洛巴林的制备方法

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2002
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2003
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2005
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- 2005-02-14 NO NO20050782A patent/NO20050782L/no not_active Application Discontinuation
- 2005-02-15 MA MA28104A patent/MA27381A1/fr unknown
- 2005-02-15 TN TNP2005000042A patent/TNSN05042A1/fr unknown

Also Published As

Publication number	Publication date
CA2495433A1 (en)	2004-02-26
NZ537818A (en)	2007-07-27
UY27936A1 (es)	2004-03-31
NO20050782L (no)	2005-04-08
IS7643A (is)	2005-01-12
EA007504B1 (ru)	2006-10-27
PA8577301A1 (es)	2004-03-10
MA27381A1 (fr)	2005-06-01
RS20050078A (sr)	2007-09-21
AR040871A1 (es)	2005-04-20
AU2003249476B2 (en)	2008-06-26
MXPA05001835A (es)	2005-09-30
SI1536782T1 (sl)	2007-08-31
GEP20084366B (en)	2008-05-13
EA200500207A1 (ru)	2005-08-25
HRP20050136A2 (en)	2005-06-30
JP2006502139A (ja)	2006-01-19
CN1674884A (zh)	2005-09-28
AP2005003227A0 (en)	2005-03-31
EP1536782B1 (de)	2007-04-18
GB0219024D0 (en)	2002-09-25
HN2003000247A (es)	2007-12-14
OA12899A (en)	2006-10-13
BR0313484A (pt)	2005-06-21
ZA200500369B (en)	2006-10-25
DE60313330T2 (de)	2008-01-03
TNSN05042A1 (fr)	2007-05-14
GT200300173A (es)	2007-03-29
ECSP055593A (es)	2005-04-18
PE20040992A1 (es)	2004-12-29
KR20050042154A (ko)	2005-05-04
IL166415A0 (en)	2006-01-15
TW200404531A (en)	2004-04-01
WO2004016259A1 (en)	2004-02-26
EP1536782A1 (de)	2005-06-08
DE60313330D1 (de)	2007-05-31
KR20070009746A (ko)	2007-01-18
PT1536782E (pt)	2007-06-27
ATE359775T1 (de)	2007-05-15
PL375553A1 (en)	2005-11-28
AU2003249476A1 (en)	2004-03-03
DK1536782T3 (da)	2007-07-30
CR7687A (es)	2005-07-08
ES2285230T3 (es)	2007-11-16

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