UY32904A - Compuestos de aminoquinazolina para combatir plagas de invertebrados - Google Patents

Compuestos de aminoquinazolina para combatir plagas de invertebrados

Info

Publication number
UY32904A
UY32904A UY0001032904A UY32904A UY32904A UY 32904 A UY32904 A UY 32904A UY 0001032904 A UY0001032904 A UY 0001032904A UY 32904 A UY32904 A UY 32904A UY 32904 A UY32904 A UY 32904A
Authority
UY
Uruguay
Prior art keywords
compounds
invertebrate pests
aminoquinazoline
pests
aminoquinazoline compounds
Prior art date
Application number
UY0001032904A
Other languages
English (en)
Inventor
Deborah L Culberston
Dr Narine Arun
Cecille Ebuenga
Dr Langewald Juergen
Dr Pohlman Matthias
Dr Grob Steffen
Dr Rer Nat Rosenbaum Claudia
Dr Phil Deshmukh Prashant
Dr Dickhaut Joachim
Dr Bandur Nina Gertrud
Dr Koerber Karsten
Dr Kaiser Florian
Dr Von Deyn Wolfgang
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of UY32904A publication Critical patent/UY32904A/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/04Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D407/00Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/12Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

La invención se refiere a compuestos de aminoquinazolina o sus enantiómeros o sales veterinariamente aceptables, que son útiles para combatir o controlar plagas de invertebrados, sobre todo, plagas de artrópodos y nematodos. La invención también se refiere a métodos para controlar plagas de invertebrados usando estos compuestos y a material de propagación de planta y a composiciones agrícolas y veterinarias que comprenden dichos compuestos. Donde A1 , A2 , A3 , A4, R 1 , R2, R3, R4, R5d, R5b , R5b, R5d y p tienen las definiciones indicadas en la descripción.
UY0001032904A 2009-09-24 2010-09-24 Compuestos de aminoquinazolina para combatir plagas de invertebrados UY32904A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24532209P 2009-09-24 2009-09-24

Publications (1)

Publication Number Publication Date
UY32904A true UY32904A (es) 2011-03-31

Family

ID=43216941

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032904A UY32904A (es) 2009-09-24 2010-09-24 Compuestos de aminoquinazolina para combatir plagas de invertebrados

Country Status (9)

Country Link
US (1) US8796180B2 (es)
EP (1) EP2480537A1 (es)
JP (1) JP2013505909A (es)
CN (1) CN102574817A (es)
AR (1) AR078441A1 (es)
BR (1) BR112012006615A2 (es)
TW (1) TW201119579A (es)
UY (1) UY32904A (es)
WO (1) WO2011036074A1 (es)

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AU2011354895B2 (en) 2011-01-14 2016-05-05 Sds Biotech K. K. Agri-horticultural pest control compositions comprising 4- (3-butynyl)aminopyrimidine derivatives
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TW201609713A (zh) * 2013-12-19 2016-03-16 H 朗德貝克公司 作爲pde1抑制劑之喹唑啉-thf-胺
CN103819414B (zh) * 2014-02-27 2016-06-01 福建医科大学 一种在水相中催化制备喹唑酮化合物的方法
KR20160138084A (ko) * 2014-04-04 2016-12-02 하. 룬드벡 아크티에셀스카브 Pde1 저해제인 할로겐화된 퀴나졸린-thf-아민
US10626094B2 (en) * 2014-10-14 2020-04-21 Sanford Burnham Prebys Medical Discovery Institute Inhibitors of low molecular weight protein tyrosine phosphatase and uses thereof
EP3226868A4 (en) * 2014-12-05 2018-08-15 Subramaniam Ananthan Novel quinazolines as biogenic amine transport modulators
SI3538512T1 (sl) * 2016-11-11 2021-09-30 Bayer Animal Health Gmbh Novi antihelmintični kinolin-3-karboksamidni derivati
WO2018204176A1 (en) 2017-05-01 2018-11-08 Sanford Burnham Prebys Medical Discovery Institute Inhibitors of low molecular weight protein tyrosine phosphatase (lmptp) and uses thereof
US11548867B2 (en) * 2017-07-19 2023-01-10 Idea Ya Biosciences, Inc. Amido compounds as AhR modulators
CN111039878B (zh) * 2019-12-28 2022-06-17 青岛科技大学 一种4-氨基喹唑啉苯醚类化合物及其应用
CN114436976B (zh) * 2021-01-29 2023-07-11 石药集团中奇制药技术(石家庄)有限公司 一种新型喹唑啉类衍生物及其制备和应用
CN116589414A (zh) * 2023-05-26 2023-08-15 青岛科技大学 一种含氟苯基喹唑啉类化合物及其用途

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Also Published As

Publication number Publication date
AR078441A1 (es) 2011-11-09
WO2011036074A1 (en) 2011-03-31
EP2480537A1 (en) 2012-08-01
CN102574817A (zh) 2012-07-11
US20120178622A1 (en) 2012-07-12
JP2013505909A (ja) 2013-02-21
BR112012006615A2 (pt) 2019-09-24
US8796180B2 (en) 2014-08-05
TW201119579A (en) 2011-06-16

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