ATE234832T1 - 1-trifluorotmethyl-4-hydroxy-7-piperidinyl- aminomethylchroman-derivate - Google Patents

1-trifluorotmethyl-4-hydroxy-7-piperidinyl- aminomethylchroman-derivate

Info

Publication number
ATE234832T1
ATE234832T1 AT00915314T AT00915314T ATE234832T1 AT E234832 T1 ATE234832 T1 AT E234832T1 AT 00915314 T AT00915314 T AT 00915314T AT 00915314 T AT00915314 T AT 00915314T AT E234832 T1 ATE234832 T1 AT E234832T1
Authority
AT
Austria
Prior art keywords
trifluorotmethyl
aminomethyl
piperidinyl
hydroxy
chromene derivatives
Prior art date
Application number
AT00915314T
Other languages
English (en)
Inventor
Ronald Scott Obach
Douglas Alan Scully
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of ATE234832T1 publication Critical patent/ATE234832T1/de

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Endocrinology (AREA)
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AT00915314T 1999-05-21 2000-04-20 1-trifluorotmethyl-4-hydroxy-7-piperidinyl- aminomethylchroman-derivate ATE234832T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13539999P 1999-05-21 1999-05-21
PCT/IB2000/000493 WO2000071538A2 (en) 1999-05-21 2000-04-20 1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives

Publications (1)

Publication Number Publication Date
ATE234832T1 true ATE234832T1 (de) 2003-04-15

Family

ID=22467939

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00915314T ATE234832T1 (de) 1999-05-21 2000-04-20 1-trifluorotmethyl-4-hydroxy-7-piperidinyl- aminomethylchroman-derivate

Country Status (49)

Country Link
US (1) US6239147B1 (de)
EP (1) EP1178984B1 (de)
JP (1) JP3802762B2 (de)
KR (1) KR100453301B1 (de)
CN (1) CN1140525C (de)
AP (1) AP1396A (de)
AR (1) AR020294A1 (de)
AT (1) ATE234832T1 (de)
AU (1) AU775861B2 (de)
BG (1) BG106152A (de)
BR (1) BR0011284A (de)
CA (1) CA2374643C (de)
CO (1) CO5170464A1 (de)
CR (1) CR6503A (de)
CZ (1) CZ20014164A3 (de)
DE (1) DE60001736T2 (de)
DK (1) DK1178984T3 (de)
DZ (1) DZ3044A1 (de)
EA (1) EA004233B1 (de)
EE (1) EE04719B1 (de)
ES (1) ES2190781T3 (de)
GC (1) GC0000254A (de)
GE (1) GEP20043225B (de)
GT (1) GT200000073A (de)
HK (1) HK1046280B (de)
HN (1) HN2000000057A (de)
HR (1) HRP20010861A2 (de)
HU (1) HUP0201443A3 (de)
IL (1) IL145949A0 (de)
IS (1) IS6123A (de)
MA (1) MA26734A1 (de)
MX (1) MXPA01011977A (de)
MY (1) MY123373A (de)
NO (1) NO322496B1 (de)
NZ (1) NZ514698A (de)
OA (1) OA11944A (de)
PA (1) PA8495201A1 (de)
PE (1) PE20010165A1 (de)
PL (1) PL198658B1 (de)
PT (1) PT1178984E (de)
SK (1) SK285819B6 (de)
SV (1) SV2002000077A (de)
TN (1) TNSN00105A1 (de)
TR (1) TR200103332T2 (de)
TW (1) TWI275588B (de)
UA (1) UA71004C2 (de)
UY (1) UY26147A1 (de)
WO (1) WO2000071538A2 (de)
ZA (1) ZA200109554B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists
EP1095939B1 (de) * 1999-10-18 2004-01-07 Pfizer Products Inc. Verfahren zur Herstellung von zyklischen Piperidinylaminomethyl-trifluoromethyl-etherderivaten
DE10311984A1 (de) * 2003-03-12 2004-09-23 Freie Universität Berlin Verwendung von NEP-assoziierten Molekülen zur Behandlung von nichtimmunogenen-nichthypertensiven Zivilisationskrankheiten
US7122700B2 (en) * 2004-07-30 2006-10-17 Xerox Corporation Arylamine processes
US7868016B2 (en) * 2005-07-13 2011-01-11 Baxter International Inc. Pharmaceutical formulations of endo-N-(9-methyl-9-azabicyclo[3,3.1]non-3-yl)-1-methyl-1H-indazole-3-carboxamide hydrochloride
WO2009109001A1 (en) * 2008-03-04 2009-09-11 Adelaide Research & Innovation Pty Ltd Method for preventing and/or treating a disease, condition or state associated with reduced dopaminergic neuron function
JP5753780B2 (ja) 2008-06-25 2015-07-22 アレイ バイオファーマ、インコーポレイテッド ６−置換フェノキシクロマンカルボン酸誘導体
CN117343036A (zh) * 2023-03-20 2024-01-05 江苏联环药业股份有限公司 异苯并二氢吡喃类化合物及其药物组合物和应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY110227A (en) * 1991-08-12 1998-03-31 Ciba Geigy Ag 1-acylpiperindine compounds.
GB9317987D0 (en) * 1993-08-26 1993-10-13 Glaxo Group Ltd Chemical compounds
KR19980703354A (ko) * 1995-03-27 1998-10-15 나카토미히로타카 피페리딘 유도체
TW475930B (en) * 1995-04-24 2002-02-11 Novartis Ag Novel compound, its use and pharmaceutical composition comprising it
JP3042894B2 (ja) * 1995-07-07 2000-05-22 ファイザー製薬株式会社 サブスタンスｐアンタゴニストとしての置換ベンゾラクタム化合物
TW340842B (en) * 1995-08-24 1998-09-21 Pfizer Substituted benzylaminopiperidine compounds
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists

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TWI275588B (en) 2007-03-11
JP3802762B2 (ja) 2006-07-26
WO2000071538A2 (en) 2000-11-30
EP1178984B1 (de) 2003-03-19
ZA200109554B (en) 2002-11-20
CN1140525C (zh) 2004-03-03
HN2000000057A (es) 2001-03-02
CR6503A (es) 2004-02-03
DZ3044A1 (fr) 2004-03-27
MY123373A (en) 2006-05-31
PE20010165A1 (es) 2001-02-20
GC0000254A (en) 2006-11-01
BG106152A (en) 2002-06-28
WO2000071538A3 (en) 2001-02-22
KR100453301B1 (ko) 2004-10-20
CA2374643A1 (en) 2000-11-30
SK285819B6 (sk) 2007-09-06
NO20015652D0 (no) 2001-11-20
EE04719B1 (et) 2006-10-16
ES2190781T3 (es) 2003-08-16
JP2003500405A (ja) 2003-01-07
PA8495201A1 (es) 2002-08-26
AP1396A (en) 2005-04-19
HK1046280B (zh) 2004-10-21
PT1178984E (pt) 2003-06-30
NO322496B1 (no) 2006-10-16
BR0011284A (pt) 2002-03-05
AU775861B2 (en) 2004-08-19
CZ20014164A3 (cs) 2003-01-15
EP1178984A2 (de) 2002-02-13
EA004233B1 (ru) 2004-02-26
EA200101109A1 (ru) 2002-04-25
AR020294A1 (es) 2002-05-02
TR200103332T2 (tr) 2002-04-22
NO20015652L (no) 2002-01-14
SV2002000077A (es) 2002-07-03
DE60001736T2 (de) 2003-09-18
US6239147B1 (en) 2001-05-29
CA2374643C (en) 2006-02-14
DK1178984T3 (da) 2003-06-10
MA26734A1 (fr) 2004-12-20
IL145949A0 (en) 2002-07-25
CO5170464A1 (es) 2002-06-27
DE60001736D1 (de) 2003-04-24
GT200000073A (es) 2001-11-09
EE200100612A (et) 2003-02-17
KR20020016793A (ko) 2002-03-06
IS6123A (is) 2001-10-23
MXPA01011977A (es) 2002-05-06
SK16592001A3 (sk) 2003-03-04
AU3667300A (en) 2000-12-12
UA71004C2 (uk) 2004-11-15
PL198658B1 (pl) 2008-07-31
HUP0201443A3 (en) 2005-09-28
AP2001002327A0 (en) 2001-12-31
HUP0201443A2 (en) 2002-08-28
PL352409A1 (en) 2003-08-25
CN1355799A (zh) 2002-06-26
UY26147A1 (es) 2000-12-29
HRP20010861A2 (en) 2003-04-30
NZ514698A (en) 2005-01-28
OA11944A (en) 2006-04-12
GEP20043225B (en) 2004-04-26
HK1046280A1 (en) 2003-01-03
TNSN00105A1 (fr) 2005-11-10

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