NO322496B1 - 1-trifluormetyl-4-hydroksy-7-piperidinyl-aminometylkromanderivater, anvendelse derav og farmasoytisk blanding. - Google Patents

1-trifluormetyl-4-hydroksy-7-piperidinyl-aminometylkromanderivater, anvendelse derav og farmasoytisk blanding. Download PDF

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Publication number
NO322496B1
NO322496B1 NO20015652A NO20015652A NO322496B1 NO 322496 B1 NO322496 B1 NO 322496B1 NO 20015652 A NO20015652 A NO 20015652A NO 20015652 A NO20015652 A NO 20015652A NO 322496 B1 NO322496 B1 NO 322496B1
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Prior art keywords
compound
reaction
methyl
compounds
disorders
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NO20015652A
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English (en)
Norwegian (no)
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NO20015652D0 (no
NO20015652L (no
Inventor
Ronald Scott Obach
Douglas Alan Scully
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Pfizer Prod Inc
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Publication of NO20015652D0 publication Critical patent/NO20015652D0/no
Publication of NO20015652L publication Critical patent/NO20015652L/no
Publication of NO322496B1 publication Critical patent/NO322496B1/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Gynecology & Obstetrics (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
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NO20015652A 1999-05-21 2001-11-20 1-trifluormetyl-4-hydroksy-7-piperidinyl-aminometylkromanderivater, anvendelse derav og farmasoytisk blanding. NO322496B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13539999P 1999-05-21 1999-05-21
PCT/IB2000/000493 WO2000071538A2 (en) 1999-05-21 2000-04-20 1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives

Publications (3)

Publication Number Publication Date
NO20015652D0 NO20015652D0 (no) 2001-11-20
NO20015652L NO20015652L (no) 2002-01-14
NO322496B1 true NO322496B1 (no) 2006-10-16

Family

ID=22467939

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Application Number Title Priority Date Filing Date
NO20015652A NO322496B1 (no) 1999-05-21 2001-11-20 1-trifluormetyl-4-hydroksy-7-piperidinyl-aminometylkromanderivater, anvendelse derav og farmasoytisk blanding.

Country Status (49)

Country Link
US (1) US6239147B1 (de)
EP (1) EP1178984B1 (de)
JP (1) JP3802762B2 (de)
KR (1) KR100453301B1 (de)
CN (1) CN1140525C (de)
AP (1) AP1396A (de)
AR (1) AR020294A1 (de)
AT (1) ATE234832T1 (de)
AU (1) AU775861B2 (de)
BG (1) BG106152A (de)
BR (1) BR0011284A (de)
CA (1) CA2374643C (de)
CO (1) CO5170464A1 (de)
CR (1) CR6503A (de)
CZ (1) CZ20014164A3 (de)
DE (1) DE60001736T2 (de)
DK (1) DK1178984T3 (de)
DZ (1) DZ3044A1 (de)
EA (1) EA004233B1 (de)
EE (1) EE04719B1 (de)
ES (1) ES2190781T3 (de)
GC (1) GC0000254A (de)
GE (1) GEP20043225B (de)
GT (1) GT200000073A (de)
HK (1) HK1046280B (de)
HN (1) HN2000000057A (de)
HR (1) HRP20010861A2 (de)
HU (1) HUP0201443A3 (de)
IL (1) IL145949A0 (de)
IS (1) IS6123A (de)
MA (1) MA26734A1 (de)
MX (1) MXPA01011977A (de)
MY (1) MY123373A (de)
NO (1) NO322496B1 (de)
NZ (1) NZ514698A (de)
OA (1) OA11944A (de)
PA (1) PA8495201A1 (de)
PE (1) PE20010165A1 (de)
PL (1) PL198658B1 (de)
PT (1) PT1178984E (de)
SK (1) SK285819B6 (de)
SV (1) SV2002000077A (de)
TN (1) TNSN00105A1 (de)
TR (1) TR200103332T2 (de)
TW (1) TWI275588B (de)
UA (1) UA71004C2 (de)
UY (1) UY26147A1 (de)
WO (1) WO2000071538A2 (de)
ZA (1) ZA200109554B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists
EP1095939B1 (de) * 1999-10-18 2004-01-07 Pfizer Products Inc. Verfahren zur Herstellung von zyklischen Piperidinylaminomethyl-trifluoromethyl-etherderivaten
DE10311984A1 (de) * 2003-03-12 2004-09-23 Freie Universität Berlin Verwendung von NEP-assoziierten Molekülen zur Behandlung von nichtimmunogenen-nichthypertensiven Zivilisationskrankheiten
US7122700B2 (en) * 2004-07-30 2006-10-17 Xerox Corporation Arylamine processes
US7868016B2 (en) * 2005-07-13 2011-01-11 Baxter International Inc. Pharmaceutical formulations of endo-N-(9-methyl-9-azabicyclo[3,3.1]non-3-yl)-1-methyl-1H-indazole-3-carboxamide hydrochloride
WO2009109001A1 (en) * 2008-03-04 2009-09-11 Adelaide Research & Innovation Pty Ltd Method for preventing and/or treating a disease, condition or state associated with reduced dopaminergic neuron function
JP5753780B2 (ja) 2008-06-25 2015-07-22 アレイ バイオファーマ、インコーポレイテッド 6−置換フェノキシクロマンカルボン酸誘導体
CN117343036A (zh) * 2023-03-20 2024-01-05 江苏联环药业股份有限公司 异苯并二氢吡喃类化合物及其药物组合物和应用

Family Cites Families (7)

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Publication number Priority date Publication date Assignee Title
MY110227A (en) * 1991-08-12 1998-03-31 Ciba Geigy Ag 1-acylpiperindine compounds.
GB9317987D0 (en) * 1993-08-26 1993-10-13 Glaxo Group Ltd Chemical compounds
KR19980703354A (ko) * 1995-03-27 1998-10-15 나카토미히로타카 피페리딘 유도체
TW475930B (en) * 1995-04-24 2002-02-11 Novartis Ag Novel compound, its use and pharmaceutical composition comprising it
JP3042894B2 (ja) * 1995-07-07 2000-05-22 ファイザー製薬株式会社 サブスタンスpアンタゴニストとしての置換ベンゾラクタム化合物
TW340842B (en) * 1995-08-24 1998-09-21 Pfizer Substituted benzylaminopiperidine compounds
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists

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TWI275588B (en) 2007-03-11
JP3802762B2 (ja) 2006-07-26
WO2000071538A2 (en) 2000-11-30
EP1178984B1 (de) 2003-03-19
ZA200109554B (en) 2002-11-20
ATE234832T1 (de) 2003-04-15
CN1140525C (zh) 2004-03-03
HN2000000057A (es) 2001-03-02
CR6503A (es) 2004-02-03
DZ3044A1 (fr) 2004-03-27
MY123373A (en) 2006-05-31
PE20010165A1 (es) 2001-02-20
GC0000254A (en) 2006-11-01
BG106152A (en) 2002-06-28
WO2000071538A3 (en) 2001-02-22
KR100453301B1 (ko) 2004-10-20
CA2374643A1 (en) 2000-11-30
SK285819B6 (sk) 2007-09-06
NO20015652D0 (no) 2001-11-20
EE04719B1 (et) 2006-10-16
ES2190781T3 (es) 2003-08-16
JP2003500405A (ja) 2003-01-07
PA8495201A1 (es) 2002-08-26
AP1396A (en) 2005-04-19
HK1046280B (zh) 2004-10-21
PT1178984E (pt) 2003-06-30
BR0011284A (pt) 2002-03-05
AU775861B2 (en) 2004-08-19
CZ20014164A3 (cs) 2003-01-15
EP1178984A2 (de) 2002-02-13
EA004233B1 (ru) 2004-02-26
EA200101109A1 (ru) 2002-04-25
AR020294A1 (es) 2002-05-02
TR200103332T2 (tr) 2002-04-22
NO20015652L (no) 2002-01-14
SV2002000077A (es) 2002-07-03
DE60001736T2 (de) 2003-09-18
US6239147B1 (en) 2001-05-29
CA2374643C (en) 2006-02-14
DK1178984T3 (da) 2003-06-10
MA26734A1 (fr) 2004-12-20
IL145949A0 (en) 2002-07-25
CO5170464A1 (es) 2002-06-27
DE60001736D1 (de) 2003-04-24
GT200000073A (es) 2001-11-09
EE200100612A (et) 2003-02-17
KR20020016793A (ko) 2002-03-06
IS6123A (is) 2001-10-23
MXPA01011977A (es) 2002-05-06
SK16592001A3 (sk) 2003-03-04
AU3667300A (en) 2000-12-12
UA71004C2 (uk) 2004-11-15
PL198658B1 (pl) 2008-07-31
HUP0201443A3 (en) 2005-09-28
AP2001002327A0 (en) 2001-12-31
HUP0201443A2 (en) 2002-08-28
PL352409A1 (en) 2003-08-25
CN1355799A (zh) 2002-06-26
UY26147A1 (es) 2000-12-29
HRP20010861A2 (en) 2003-04-30
NZ514698A (en) 2005-01-28
OA11944A (en) 2006-04-12
GEP20043225B (en) 2004-04-26
HK1046280A1 (en) 2003-01-03
TNSN00105A1 (fr) 2005-11-10

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