EE04719B1 - 1-trifluorometüül-4-hüdroksü-7-piperidinüül-aminometüülkromaani derivaadid - Google Patents

1-trifluorometüül-4-hüdroksü-7-piperidinüül-aminometüülkromaani derivaadid

Info

Publication number
EE04719B1
EE04719B1 EEP200100612A EEP200100612A EE04719B1 EE 04719 B1 EE04719 B1 EE 04719B1 EE P200100612 A EEP200100612 A EE P200100612A EE P200100612 A EEP200100612 A EE P200100612A EE 04719 B1 EE04719 B1 EE 04719B1
Authority
EE
Estonia
Prior art keywords
aminomethyl
piperidinyl
trifluoromethyl
hydroxy
chroman derivatives
Prior art date
Application number
EEP200100612A
Other languages
English (en)
Estonian (et)
Inventor
Scott Obach Ronald
Alan Scully Douglas
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of EE200100612A publication Critical patent/EE200100612A/xx
Publication of EE04719B1 publication Critical patent/EE04719B1/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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EEP200100612A 1999-05-21 2000-04-20 1-trifluorometüül-4-hüdroksü-7-piperidinüül-aminometüülkromaani derivaadid EE04719B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13539999P 1999-05-21 1999-05-21
PCT/IB2000/000493 WO2000071538A2 (en) 1999-05-21 2000-04-20 1-trifluoromethyl-4-hydroxy-7-piperidinyl-aminomethylchroman derivatives

Publications (2)

Publication Number Publication Date
EE200100612A EE200100612A (et) 2003-02-17
EE04719B1 true EE04719B1 (et) 2006-10-16

Family

ID=22467939

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100612A EE04719B1 (et) 1999-05-21 2000-04-20 1-trifluorometüül-4-hüdroksü-7-piperidinüül-aminometüülkromaani derivaadid

Country Status (49)

Country Link
US (1) US6239147B1 (de)
EP (1) EP1178984B1 (de)
JP (1) JP3802762B2 (de)
KR (1) KR100453301B1 (de)
CN (1) CN1140525C (de)
AP (1) AP1396A (de)
AR (1) AR020294A1 (de)
AT (1) ATE234832T1 (de)
AU (1) AU775861B2 (de)
BG (1) BG106152A (de)
BR (1) BR0011284A (de)
CA (1) CA2374643C (de)
CO (1) CO5170464A1 (de)
CR (1) CR6503A (de)
CZ (1) CZ20014164A3 (de)
DE (1) DE60001736T2 (de)
DK (1) DK1178984T3 (de)
DZ (1) DZ3044A1 (de)
EA (1) EA004233B1 (de)
EE (1) EE04719B1 (de)
ES (1) ES2190781T3 (de)
GC (1) GC0000254A (de)
GE (1) GEP20043225B (de)
GT (1) GT200000073A (de)
HK (1) HK1046280B (de)
HN (1) HN2000000057A (de)
HR (1) HRP20010861A2 (de)
HU (1) HUP0201443A3 (de)
IL (1) IL145949A0 (de)
IS (1) IS6123A (de)
MA (1) MA26734A1 (de)
MX (1) MXPA01011977A (de)
MY (1) MY123373A (de)
NO (1) NO322496B1 (de)
NZ (1) NZ514698A (de)
OA (1) OA11944A (de)
PA (1) PA8495201A1 (de)
PE (1) PE20010165A1 (de)
PL (1) PL198658B1 (de)
PT (1) PT1178984E (de)
SK (1) SK285819B6 (de)
SV (1) SV2002000077A (de)
TN (1) TNSN00105A1 (de)
TR (1) TR200103332T2 (de)
TW (1) TWI275588B (de)
UA (1) UA71004C2 (de)
UY (1) UY26147A1 (de)
WO (1) WO2000071538A2 (de)
ZA (1) ZA200109554B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists
EP1095939B1 (de) * 1999-10-18 2004-01-07 Pfizer Products Inc. Verfahren zur Herstellung von zyklischen Piperidinylaminomethyl-trifluoromethyl-etherderivaten
DE10311984A1 (de) * 2003-03-12 2004-09-23 Freie Universität Berlin Verwendung von NEP-assoziierten Molekülen zur Behandlung von nichtimmunogenen-nichthypertensiven Zivilisationskrankheiten
US7122700B2 (en) * 2004-07-30 2006-10-17 Xerox Corporation Arylamine processes
US7868016B2 (en) * 2005-07-13 2011-01-11 Baxter International Inc. Pharmaceutical formulations of endo-N-(9-methyl-9-azabicyclo[3,3.1]non-3-yl)-1-methyl-1H-indazole-3-carboxamide hydrochloride
WO2009109001A1 (en) * 2008-03-04 2009-09-11 Adelaide Research & Innovation Pty Ltd Method for preventing and/or treating a disease, condition or state associated with reduced dopaminergic neuron function
JP5753780B2 (ja) 2008-06-25 2015-07-22 アレイ バイオファーマ、インコーポレイテッド ６−置換フェノキシクロマンカルボン酸誘導体
CN117343036A (zh) * 2023-03-20 2024-01-05 江苏联环药业股份有限公司 异苯并二氢吡喃类化合物及其药物组合物和应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY110227A (en) * 1991-08-12 1998-03-31 Ciba Geigy Ag 1-acylpiperindine compounds.
GB9317987D0 (en) * 1993-08-26 1993-10-13 Glaxo Group Ltd Chemical compounds
KR19980703354A (ko) * 1995-03-27 1998-10-15 나카토미히로타카 피페리딘 유도체
TW475930B (en) * 1995-04-24 2002-02-11 Novartis Ag Novel compound, its use and pharmaceutical composition comprising it
JP3042894B2 (ja) * 1995-07-07 2000-05-22 ファイザー製薬株式会社 サブスタンスｐアンタゴニストとしての置換ベンゾラクタム化合物
TW340842B (en) * 1995-08-24 1998-09-21 Pfizer Substituted benzylaminopiperidine compounds
TW426667B (en) * 1997-11-19 2001-03-21 Pfizer Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists

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TWI275588B (en) 2007-03-11
JP3802762B2 (ja) 2006-07-26
WO2000071538A2 (en) 2000-11-30
EP1178984B1 (de) 2003-03-19
ZA200109554B (en) 2002-11-20
ATE234832T1 (de) 2003-04-15
CN1140525C (zh) 2004-03-03
HN2000000057A (es) 2001-03-02
CR6503A (es) 2004-02-03
DZ3044A1 (fr) 2004-03-27
MY123373A (en) 2006-05-31
PE20010165A1 (es) 2001-02-20
GC0000254A (en) 2006-11-01
BG106152A (en) 2002-06-28
WO2000071538A3 (en) 2001-02-22
KR100453301B1 (ko) 2004-10-20
CA2374643A1 (en) 2000-11-30
SK285819B6 (sk) 2007-09-06
NO20015652D0 (no) 2001-11-20
ES2190781T3 (es) 2003-08-16
JP2003500405A (ja) 2003-01-07
PA8495201A1 (es) 2002-08-26
AP1396A (en) 2005-04-19
HK1046280B (zh) 2004-10-21
PT1178984E (pt) 2003-06-30
NO322496B1 (no) 2006-10-16
BR0011284A (pt) 2002-03-05
AU775861B2 (en) 2004-08-19
CZ20014164A3 (cs) 2003-01-15
EP1178984A2 (de) 2002-02-13
EA004233B1 (ru) 2004-02-26
EA200101109A1 (ru) 2002-04-25
AR020294A1 (es) 2002-05-02
TR200103332T2 (tr) 2002-04-22
NO20015652L (no) 2002-01-14
SV2002000077A (es) 2002-07-03
DE60001736T2 (de) 2003-09-18
US6239147B1 (en) 2001-05-29
CA2374643C (en) 2006-02-14
DK1178984T3 (da) 2003-06-10
MA26734A1 (fr) 2004-12-20
IL145949A0 (en) 2002-07-25
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AU3667300A (en) 2000-12-12
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HUP0201443A3 (en) 2005-09-28
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CN1355799A (zh) 2002-06-26
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