ATE422202T1 - Substituierte 4-(indazol-3-yl)phenole als liganden des oestrogenrezeptors und deren verwendung bei der behandlung von entzündlichen erkrankungen - Google Patents

Substituierte 4-(indazol-3-yl)phenole als liganden des oestrogenrezeptors und deren verwendung bei der behandlung von entzündlichen erkrankungen

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Publication number
ATE422202T1
ATE422202T1 AT03799289T AT03799289T ATE422202T1 AT E422202 T1 ATE422202 T1 AT E422202T1 AT 03799289 T AT03799289 T AT 03799289T AT 03799289 T AT03799289 T AT 03799289T AT E422202 T1 ATE422202 T1 AT E422202T1
Authority
AT
Austria
Prior art keywords
indazol
phenols
ligands
substituted
treatment
Prior art date
Application number
AT03799289T
Other languages
English (en)
Inventor
Robert Steffan
Edward Matelan
Mark Ashwell
William Solvibile
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Application granted granted Critical
Publication of ATE422202T1 publication Critical patent/ATE422202T1/de

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    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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AT03799289T 2002-09-25 2003-09-24 Substituierte 4-(indazol-3-yl)phenole als liganden des oestrogenrezeptors und deren verwendung bei der behandlung von entzündlichen erkrankungen ATE422202T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41393102P 2002-09-25 2002-09-25

Publications (1)

Publication Number Publication Date
ATE422202T1 true ATE422202T1 (de) 2009-02-15

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AT03799289T ATE422202T1 (de) 2002-09-25 2003-09-24 Substituierte 4-(indazol-3-yl)phenole als liganden des oestrogenrezeptors und deren verwendung bei der behandlung von entzündlichen erkrankungen

Country Status (21)

Country Link
US (2) US7241791B2 (de)
EP (1) EP1542976B1 (de)
JP (1) JP4459813B2 (de)
KR (1) KR20050053702A (de)
CN (2) CN1321984C (de)
AR (1) AR041378A1 (de)
AT (1) ATE422202T1 (de)
AU (1) AU2003276940A1 (de)
BR (1) BR0314475A (de)
CA (1) CA2499736A1 (de)
CR (1) CR7769A (de)
DE (1) DE60326077D1 (de)
DK (1) DK1542976T3 (de)
EC (1) ECSP055704A (de)
ES (1) ES2319519T3 (de)
MX (1) MXPA05003275A (de)
NO (1) NO20051942L (de)
RU (1) RU2005109387A (de)
TW (1) TW200409759A (de)
WO (1) WO2004031159A1 (de)
ZA (1) ZA200502462B (de)

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RU2005109387A (ru) 2006-01-20
JP4459813B2 (ja) 2010-04-28
US20040167127A1 (en) 2004-08-26
JP2006505544A (ja) 2006-02-16
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BR0314475A (pt) 2005-08-09
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KR20050053702A (ko) 2005-06-08
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CA2499736A1 (en) 2004-04-15
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CN1321984C (zh) 2007-06-20
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TW200409759A (en) 2004-06-16
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AR041378A1 (es) 2005-05-11

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