ATE533775T1 - Verfahren zur herstellung von 17-vinyl-triflaten als intermediate - Google Patents

Verfahren zur herstellung von 17-vinyl-triflaten als intermediate

Info

Publication number: ATE533775T1
Authority: AT; Austria
Prior art keywords: producing; formula; vinyl triflates; triflates; vinyl
Prior art date: 2004-08-24

Application number

AT05781067T

Other languages

English (en)

Inventor

Paul Stanley Bury

Original Assignee

Btg Int Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2004-08-24

Filing date

2005-08-23

Publication date

2011-12-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35311370&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE533775(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2004-08-24 Priority claimed from GB0418901A external-priority patent/GB0418901D0/en

2004-08-24 Priority claimed from GBGB0418900.7A external-priority patent/GB0418900D0/en

2005-08-23 Application filed by Btg Int Ltd filed Critical Btg Int Ltd

2011-12-15 Application granted granted Critical

2011-12-15 Publication of ATE533775T1 publication Critical patent/ATE533775T1/de

Links

238000004519 manufacturing process Methods 0.000 title 1
229920002554 vinyl polymer Polymers 0.000 title 1
239000002253 acid Substances 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
-1 heterocyclic amine Chemical class 0.000 abstract 1
150000002576 ketones Chemical class 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
ITMCEJHCFYSIIV-UHFFFAOYSA-M triflate Chemical compound [O-]S(=O)(=O)C(F)(F)F ITMCEJHCFYSIIV-UHFFFAOYSA-M 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Pyridine Compounds (AREA)

AT05781067T 2004-08-24 2005-08-23 Verfahren zur herstellung von 17-vinyl-triflaten als intermediate ATE533775T1 (de)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US60355804P	2004-08-24	2004-08-24
GB0418901A GB0418901D0 (en)	2004-08-24	2004-08-24	Synthetic method
GBGB0418900.7A GB0418900D0 (en)	2004-08-24	2004-08-24	Novel salt forms
PCT/GB2005/003283 WO2006021777A1 (en)	2004-08-24	2005-08-23	Process fot the preparation of 17-0-vinyl- triflates as intermediates

Publications (1)

Publication Number	Publication Date
ATE533775T1 true ATE533775T1 (de)	2011-12-15

Family

ID=35311370

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT05781067T ATE533775T1 (de)	2004-08-24	2005-08-23	Verfahren zur herstellung von 17-vinyl-triflaten als intermediate

Country Status (11)

Country	Link
US (2)	US8236946B2 (de)
EP (2)	EP1781683B1 (de)
JP (1)	JP5199667B2 (de)
AT (1)	ATE533775T1 (de)
CY (1)	CY1112283T1 (de)
DK (2)	DK1781683T3 (de)
ES (2)	ES2377074T3 (de)
PL (2)	PL2428519T3 (de)
PT (2)	PT2428519E (de)
SI (2)	SI1781683T1 (de)
WO (1)	WO2006021777A1 (de)

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CN102816200B (zh) *	2012-09-05	2015-04-15	中山大学	一种醋酸阿比特龙的制备方法
ITMI20121788A1 (it)	2012-10-22	2014-04-23	Olon Spa	Procedimento per la purificazione di abiraterone acetato
EP2917226A1 (de)	2012-11-09	2015-09-16	Synthon BV	Verfahren zur herstellung des 17-triflat-zwischenprodukts von abirateron-3-acetat
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WO2014075978A1 (en)	2012-11-16	2014-05-22	Synthon B.V.	Process for the production of abiraterone-3-acetate involving an enol trliflation reaction in the presence of an alkoxy-pyridine compound
CA2895356A1 (en)	2012-12-19	2014-06-26	Bayer Pharma Aktiengesellschaft	Combination comprising radium-223 for the treatment of cancer
EP2938625B1 (de) *	2012-12-31	2018-02-21	Hetero Research Foundation	Verfahren zur herstellung von abirateronacetat
EP2792682B1 (de)	2013-04-19	2016-11-09	Zach System	Verfahren zur Herstellung einer festen Form von Abirateron-Azetat
CN103242410B (zh) *	2013-05-09	2015-08-26	苏州明锐医药科技有限公司	醋酸阿比特龙的制备方法
IN2013MU02133A (de) *	2013-06-24	2015-06-05	Sun Pharmaceutical Ind Ltd
JP6474799B2 (ja) *	2013-06-28	2019-02-27	サイノファームタイワン，リミティド	アビラテロン及びその中間体の調製方法
ES2581317T3 (es)	2013-07-29	2016-09-05	Industriale Chimica S.R.L.	Proceso de preparación de abiraterona o acetato de abiraterona
ES2663469T3 (es)	2013-07-29	2018-04-12	Industriale Chimica S.R.L.	Proceso para la preparación de abiraterona y acetato de abiraterona
ITMI20131861A1 (it) *	2013-11-08	2015-05-09	Ind Chimica Srl	Processo per la preparazione di abiraterone e abiraterone acetato
CN104418930B (zh) *	2013-08-23	2018-01-12	四川海思科制药有限公司	一种高纯度醋酸乌利司他
ES2741505T3 (es)	2014-01-28	2020-02-11	Olon Spa	Procedimiento para la preparación de acetato de abiraterona y sus productos intermedios
CN103965282B (zh)	2014-04-21	2016-01-20	武汉百科药物开发有限公司	一种醋酸阿比特龙的制备方法
US9315541B2 (en)	2014-05-20	2016-04-19	Olon S.P.A.	Process for the preparation of unsaturated trifluoromethanesulfonate steroid derivatives
WO2016001208A1 (en)	2014-06-30	2016-01-07	Galenicum Health S.L.	Stable pharmaceutical compositions in the form of immediate release tablets
CZ2014475A3 (cs)	2014-07-09	2016-01-20	Zentiva, K.S.	Způsob přípravy Abirateron acetátu o vysoké čistotě aplikovatelný v průmyslovém měřítku
CN105622703B (zh) *	2014-11-05	2019-09-27	兰州大学	一种制备醋酸阿比特龙的方法
CN104447934B (zh) *	2014-12-08	2017-03-15	深圳科兴生物工程有限公司	一种醋酸阿比特龙的纯化方法
HU231297B1 (hu)	2018-07-31	2022-09-28	Richter Gedeon Nyrt	Stabil gyógyszerkészítmények és eljárás az előállításukra
CN112812147A (zh) *	2019-11-15	2021-05-18	江苏佳尔科药业集团股份有限公司	一种醋酸阿比特龙的合成方法及其中间体
EP3944860A1 (de)	2020-07-30	2022-02-02	Galenicum Health S.L.U.	Abirateron zur verwendung in einem verfahren zur behandlung von krebs
KR102583796B1 (ko)	2021-07-28	2023-09-27	오스템임플란트 주식회사	골 이식량 결정 방법 및 장치, 컴퓨터 판독 가능한 기록 매체 및 컴퓨터 프로그램
WO2023213151A1 (zh)	2022-05-06	2023-11-09	奥锐特药业股份有限公司	一种醋酸阿比特龙及其中间体的制备方法

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2005
- 2005-08-23 US US11/660,792 patent/US8236946B2/en active Active
- 2005-08-23 PT PT111780052T patent/PT2428519E/pt unknown
- 2005-08-23 EP EP05781067A patent/EP1781683B1/de not_active Expired - Lifetime
- 2005-08-23 JP JP2007528971A patent/JP5199667B2/ja not_active Expired - Lifetime
- 2005-08-23 DK DK05781067.3T patent/DK1781683T3/da active
- 2005-08-23 PT PT05781067T patent/PT1781683E/pt unknown
- 2005-08-23 AT AT05781067T patent/ATE533775T1/de active
- 2005-08-23 PL PL11178005T patent/PL2428519T3/pl unknown
- 2005-08-23 WO PCT/GB2005/003283 patent/WO2006021777A1/en not_active Ceased
- 2005-08-23 SI SI200531462T patent/SI1781683T1/sl unknown
- 2005-08-23 DK DK11178005T patent/DK2428519T3/en active
- 2005-08-23 ES ES05781067T patent/ES2377074T3/es not_active Expired - Lifetime
- 2005-08-23 ES ES11178005.2T patent/ES2534587T3/es not_active Expired - Lifetime
- 2005-08-23 SI SI200531956T patent/SI2428519T1/sl unknown
- 2005-08-23 EP EP11178005.2A patent/EP2428519B1/de not_active Revoked
- 2005-08-23 PL PL05781067T patent/PL1781683T3/pl unknown
2011
- 2011-07-27 US US13/137,193 patent/US8389714B2/en not_active Expired - Lifetime
2012
- 2012-01-27 CY CY20121100095T patent/CY1112283T1/el unknown

Also Published As

Publication number	Publication date
PT1781683E (pt)	2012-02-13
JP2008510781A (ja)	2008-04-10
ES2377074T3 (es)	2012-03-22
CY1112283T1 (el)	2015-12-09
US20110288288A1 (en)	2011-11-24
EP1781683A1 (de)	2007-05-09
US20070282109A1 (en)	2007-12-06
PL1781683T3 (pl)	2012-04-30
DK1781683T3 (da)	2012-02-06
EP2428519A3 (de)	2014-01-15
EP2428519A2 (de)	2012-03-14
EP2428519B1 (de)	2015-01-21
ES2534587T3 (es)	2015-04-24
PL2428519T3 (pl)	2015-09-30
WO2006021777A1 (en)	2006-03-02
HK1167658A1 (en)	2012-12-07
JP5199667B2 (ja)	2013-05-15
SI2428519T1 (sl)	2015-07-31
SI1781683T1 (sl)	2012-06-29
EP1781683B1 (de)	2011-11-16
PT2428519E (pt)	2015-04-29
DK2428519T3 (en)	2015-04-13
US8236946B2 (en)	2012-08-07
US8389714B2 (en)	2013-03-05

Publication	Publication Date	Title
ATE533775T1 (de)	2011-12-15	Verfahren zur herstellung von 17-vinyl-triflaten als intermediate
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ATE422200T1 (de)	2009-02-15	Verfahren zur herstellung substituierter nikotinsäureester
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DE602006021411D1 (de)	2011-06-01	Verfahren zur herstellung von optional 2-substituierten 1,6-dihydro-6-oxo-4-pyrimidincarboxylsäuren
EA200701470A1 (ru)	2008-02-28	Способы получения производных 4-(фенокси-5-метилпиримидин-4-илокси)пиперидин-1-карбоновой кислоты и родственных соединений
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ATE255103T1 (de)	2003-12-15	Verfahren zur herstellung von pyridinmethanol- verbindungen
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