DK1781683T3 - Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata - Google Patents

Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata

Info

Publication number
DK1781683T3
DK1781683T3 DK05781067.3T DK05781067T DK1781683T3 DK 1781683 T3 DK1781683 T3 DK 1781683T3 DK 05781067 T DK05781067 T DK 05781067T DK 1781683 T3 DK1781683 T3 DK 1781683T3
Authority
DK
Denmark
Prior art keywords
semi
preparation
finished products
vinyl triflates
formula
Prior art date
Application number
DK05781067.3T
Other languages
English (en)
Inventor
Paul Stanley Bury
Original Assignee
Btg Int Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35311370&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1781683(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0418901A external-priority patent/GB0418901D0/en
Priority claimed from GBGB0418900.7A external-priority patent/GB0418900D0/en
Application filed by Btg Int Ltd filed Critical Btg Int Ltd
Application granted granted Critical
Publication of DK1781683T3 publication Critical patent/DK1781683T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pyridine Compounds (AREA)
DK05781067.3T 2004-08-24 2005-08-23 Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata DK1781683T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US60355804P 2004-08-24 2004-08-24
GB0418901A GB0418901D0 (en) 2004-08-24 2004-08-24 Synthetic method
GBGB0418900.7A GB0418900D0 (en) 2004-08-24 2004-08-24 Novel salt forms
PCT/GB2005/003283 WO2006021777A1 (en) 2004-08-24 2005-08-23 Process fot the preparation of 17-0-vinyl- triflates as intermediates

Publications (1)

Publication Number Publication Date
DK1781683T3 true DK1781683T3 (da) 2012-02-06

Family

ID=35311370

Family Applications (2)

Application Number Title Priority Date Filing Date
DK11178005T DK2428519T3 (da) 2004-08-24 2005-08-23 Sammensætning til præparation af 17-vinyl-triflater som intermediater
DK05781067.3T DK1781683T3 (da) 2004-08-24 2005-08-23 Fremgangsmåde til fremstilling af 17-vinyl-triflater som halvfabrikata

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK11178005T DK2428519T3 (da) 2004-08-24 2005-08-23 Sammensætning til præparation af 17-vinyl-triflater som intermediater

Country Status (11)

Country Link
US (2) US8236946B2 (da)
EP (2) EP1781683B1 (da)
JP (1) JP5199667B2 (da)
AT (1) ATE533775T1 (da)
CY (1) CY1112283T1 (da)
DK (2) DK2428519T3 (da)
ES (2) ES2534587T3 (da)
PL (2) PL2428519T3 (da)
PT (2) PT1781683E (da)
SI (2) SI2428519T1 (da)
WO (1) WO2006021777A1 (da)

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102030798B (zh) * 2010-12-17 2012-10-17 深圳万乐药业有限公司 一种醋酸阿比特龙的纯化方法
CN104066744B (zh) 2011-10-10 2017-03-22 扎克系统公司 用于制备17‑取代的甾体的方法
CN103172690B (zh) * 2011-12-23 2016-08-24 重庆医药工业研究院有限责任公司 醋酸阿比特龙及其中间体的制备方法
EP2607371A1 (en) 2011-12-23 2013-06-26 Crystal Pharma, S.A.U. Processes for the preparation of abiraterone and related compouds
CN103193849B (zh) * 2012-01-04 2016-05-04 连云港润众制药有限公司 一种高纯度醋酸阿比特龙的制备方法
CN103254265B (zh) 2012-02-21 2016-07-13 上海希迈医药科技有限公司 醋酸阿比特龙三氟乙酸盐及其制备方法和应用
US9511152B2 (en) * 2012-04-05 2016-12-06 The Board Of Regents Of The University Of Texas System Multicolored pH-activatable fluorescence nanoplatform
WO2014009436A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Nanosuspension of abiraterone acetate
WO2014009437A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Oxidation stability of abiraterone acetate
WO2014009434A1 (en) 2012-07-11 2014-01-16 Sandoz Ag Self-microemulsifying drug delivery system of abiraterone or abiraterone acetate
WO2014016830A1 (en) * 2012-07-25 2014-01-30 Mapi Pharma Ltd. Process and intermediates for the preparation of abiraterone acetate
CN102816200B (zh) * 2012-09-05 2015-04-15 中山大学 一种醋酸阿比特龙的制备方法
ITMI20121788A1 (it) 2012-10-22 2014-04-23 Olon Spa Procedimento per la purificazione di abiraterone acetato
EP2917226A1 (en) 2012-11-09 2015-09-16 Synthon BV Process for making the 17-triflate intermediate of abiraterone-3-acetate
WO2014071984A1 (en) 2012-11-09 2014-05-15 Synthon Bv Process for making abiraterone-3-acetate
WO2014075978A1 (en) 2012-11-16 2014-05-22 Synthon B.V. Process for the production of abiraterone-3-acetate involving an enol trliflation reaction in the presence of an alkoxy-pyridine compound
US20150343099A1 (en) 2012-12-19 2015-12-03 Bayer Pharma Aktiengesellschaft Combination comprising radium-223 for the treatment of cancer
WO2014102833A2 (en) * 2012-12-31 2014-07-03 Hetero Research Foundation Process for abiraterone acetate
PL2792682T3 (pl) 2013-04-19 2017-04-28 Zach System Sposób wytwarzania stałej postaci octanu abirateronu
CN103242410B (zh) * 2013-05-09 2015-08-26 苏州明锐医药科技有限公司 醋酸阿比特龙的制备方法
US20160176915A1 (en) * 2013-06-24 2016-06-23 Sun Pharmaceutical Industries Limited Process for preparation of abiraterone acetate
CN105377871B (zh) * 2013-06-28 2017-06-06 台湾神隆股份有限公司 阿比特龙及其中间体的制备方法
ITMI20131861A1 (it) * 2013-11-08 2015-05-09 Ind Chimica Srl Processo per la preparazione di abiraterone e abiraterone acetato
US9650410B2 (en) 2013-07-29 2017-05-16 Industriale Chimica S.R.L. Process for the preparation of abiraterone and abiraterone acetate
CA2919484C (en) 2013-07-29 2021-05-11 Industriale Chimica S.R.L. Process for the preparation of abiraterone or abiraterone acetate
CN104418930B (zh) * 2013-08-23 2018-01-12 四川海思科制药有限公司 一种高纯度醋酸乌利司他
US9556219B2 (en) 2014-01-28 2017-01-31 Olon S.P.A. Procedure for the preparation of abiraterone acetate and intermediates thereof
CN103965282B (zh) * 2014-04-21 2016-01-20 武汉百科药物开发有限公司 一种醋酸阿比特龙的制备方法
US9315541B2 (en) * 2014-05-20 2016-04-19 Olon S.P.A. Process for the preparation of unsaturated trifluoromethanesulfonate steroid derivatives
EP3160450A1 (en) 2014-06-30 2017-05-03 Galenicum Health S.L. Stable pharmaceutical compositions in the form of immediate release tablets
CZ2014475A3 (cs) 2014-07-09 2016-01-20 Zentiva, K.S. Způsob přípravy Abirateron acetátu o vysoké čistotě aplikovatelný v průmyslovém měřítku
CN105622703B (zh) * 2014-11-05 2019-09-27 兰州大学 一种制备醋酸阿比特龙的方法
CN104447934B (zh) * 2014-12-08 2017-03-15 深圳科兴生物工程有限公司 一种醋酸阿比特龙的纯化方法
HU231297B1 (hu) 2018-07-31 2022-09-28 Richter Gedeon Nyrt Stabil gyógyszerkészítmények és eljárás az előállításukra
CN112812147A (zh) * 2019-11-15 2021-05-18 江苏佳尔科药业集团股份有限公司 一种醋酸阿比特龙的合成方法及其中间体
EP3944860A1 (en) 2020-07-30 2022-02-02 Galenicum Health S.L.U. Abiraterone for use in a method of treating cancer
KR102583796B1 (ko) 2021-07-28 2023-09-27 오스템임플란트 주식회사 골 이식량 결정 방법 및 장치, 컴퓨터 판독 가능한 기록 매체 및 컴퓨터 프로그램
WO2023213151A1 (zh) 2022-05-06 2023-11-09 奥锐特药业股份有限公司 一种醋酸阿比特龙及其中间体的制备方法

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4207851A1 (de) * 1992-03-12 1993-09-16 Bayer Ag Mittel und verfahren zur ausruestung von textilien
ES2138618T3 (es) * 1992-03-31 2000-01-16 Btg Int Ltd Esteroides 17-sustituidos utiles en el tratamiento del cancer.
US5338875A (en) * 1992-11-19 1994-08-16 Merck & Co., Inc. Boron containing intermediates useful in the preparation of carbapenems
ES2127413T3 (es) 1993-09-30 1999-04-16 Btg Int Ltd Sintesis de esteroides 17-(3-piridilo).
US5466770A (en) * 1994-05-26 1995-11-14 Minnesota Mining And Manufacturing Company Fluorine-efficient oil- and water-repellent compositions
JP3982012B2 (ja) * 1997-01-30 2007-09-26 ダイキン工業株式会社 新規組成物および処理剤
US5994334A (en) 1997-02-05 1999-11-30 University Of Maryland Androgen synthesis inhibitors
JP3399286B2 (ja) * 1997-04-11 2003-04-21 ダイキン工業株式会社 防汚加工剤組成物
JPH10316719A (ja) * 1997-05-20 1998-12-02 Daikin Ind Ltd 新規重合体およびそれを含む防汚加工剤組成物
US6059868A (en) * 1998-10-29 2000-05-09 Hewlett-Packard Company Ink-jet inks with improved performance
US6753376B1 (en) * 1998-12-22 2004-06-22 Daikin Industries Ltd. Aqueous water-and oil-repellent dispersion
JP2000212549A (ja) * 1999-01-25 2000-08-02 Asahi Glass Co Ltd 撥水撥油剤組成物およびその製造方法
US6274060B1 (en) * 1999-02-04 2001-08-14 Daikin Industries, Ltd. Water- and oil-repellent
JP5298399B2 (ja) * 2000-09-21 2013-09-25 ダイキン工業株式会社 撥水撥油剤水性分散液組成物およびその製造方法
WO2002064696A1 (en) * 2001-01-30 2002-08-22 Daikin Industries, Ltd. Water- and oil-repellent composition, process for producing the same and use thereof
EP1380628A4 (en) * 2001-03-09 2006-09-13 Daikin Ind Ltd HYDROPHOBIC AND OLEOPHOBIC COMPOSITION WITH IMPROVED COLD CURING BEHAVIOR
DE60233192D1 (de) * 2001-04-13 2009-09-17 Asahi Glass Co Ltd Hydrophobe und lipophobe zusammensetzung
EP1477543A4 (en) * 2002-01-21 2007-10-31 Daikin Ind Ltd AQUEOUS HYDRO AND OLEOPHOBY DISPERSION
US20050209477A1 (en) * 2002-06-20 2005-09-22 Sachiko Kato Process for producing vinyl perfluoroalkanesulfonate derivative
TW200416277A (en) * 2002-10-15 2004-09-01 Asahi Glass Co Ltd Water-and-oil repellant composition
GB0418900D0 (en) * 2004-08-24 2004-09-29 Btg Int Ltd Novel salt forms

Also Published As

Publication number Publication date
PT1781683E (pt) 2012-02-13
SI1781683T1 (sl) 2012-06-29
EP1781683A1 (en) 2007-05-09
US20110288288A1 (en) 2011-11-24
EP2428519A2 (en) 2012-03-14
US8236946B2 (en) 2012-08-07
EP1781683B1 (en) 2011-11-16
WO2006021777A1 (en) 2006-03-02
EP2428519B1 (en) 2015-01-21
ATE533775T1 (de) 2011-12-15
PT2428519E (pt) 2015-04-29
DK2428519T3 (da) 2015-04-13
PL1781683T3 (pl) 2012-04-30
CY1112283T1 (el) 2015-12-09
ES2377074T3 (es) 2012-03-22
US8389714B2 (en) 2013-03-05
PL2428519T3 (pl) 2015-09-30
HK1167658A1 (en) 2012-12-07
JP2008510781A (ja) 2008-04-10
SI2428519T1 (sl) 2015-07-31
EP2428519A3 (en) 2014-01-15
JP5199667B2 (ja) 2013-05-15
ES2534587T3 (es) 2015-04-24
US20070282109A1 (en) 2007-12-06

Similar Documents

Publication Publication Date Title
PL1781683T3 (pl) Sposób wytwarzania 17-winylo-trifluorometanosulfonianów jako związków pośrednich
ATE497957T1 (de) Pyridinderivate als fungizide verbindungen
BRPI0516911A (pt) método para a preparação de um composto e composto de anilina
BRPI0411268C8 (pt) Processo para a preparação de compostos 3-aril butil-amina substituído
GB0418900D0 (en) Novel salt forms
PL1954264T3 (pl) Sposób wytwarzania epoksybutanolowych związków pośrednich
DK1740544T3 (da) 2 pyridinylcycloalkylcarboxamidderivater, der er egnede som fungicider
EA200701470A1 (ru) Способы получения производных 4-(фенокси-5-метилпиримидин-4-илокси)пиперидин-1-карбоновой кислоты и родственных соединений
NO20040388L (no) Fremgangsmåte for fremstilling av beraprost og salter derav, samt forbindelser som er mellomprodukter i fremgangsmåten
BR0308345A (pt) Processo para derivados de ácido trans-4-amino-1-cicloexanocarboxìlico
IS7978A (is) Aðferð til að framleiða súr viðbótarsölt af fjölsýrðum basískum samböndum
EA200701738A1 (ru) Способ получения транс-1-((1r,3s)-6-хлор-3-фенилиндан-1-ил)-3,3-диметилпиперазина
BR0315112A (pt) Sal de adição ácido, e, processo para a preparação de um composto
EA200500688A1 (ru) Новый способ получения синтетических промежуточных соединений для пестицидов
DK1272480T3 (da) Fremgangsmåde til fremstilling af spirocycliske tetronsyrederivater
DK1907396T3 (da) Fremgangsmåde til fremstilling af 4-beta-amino-4'-demethyl-4-deoxypodophyllotoxin
WO2007143014A3 (en) Methods for preparing glutamic acid derivatives and intermediates thereof
EA200700767A1 (ru) Способ получения пиразолов
BRPI0400141A (pt) Composição de incenso inseticida, e emulsão e processo para produção da mesma
DE602006014001D1 (de) Herstellung von 2-aminothiazol-5-carbonsäurederivaten
DK1581504T3 (da) Fremgangsmåde til fremstilling af subsituterede imidazolderivater og intermediater anvendt i fremgangsmåden
DE502006005865D1 (de) Herstellung von 1,7` -dimethyl-2` -propyl-2,5` -bi-1h-benzimidazol
DE602006015458D1 (de) Verfahren zur herstellung eines carbonsäureamidderivats
DE602007012989D1 (de) Verfahren zur Herstellung von Entacapon
DK1807401T3 (da) Fremgangsmåde til fremstilling af phenyl-2-pyrimidinylketoner samt deres nye mellemprodukter