AU2935300A - New pharmaceutical combinations for nos inhibitors - Google Patents

New pharmaceutical combinations for nos inhibitors Download PDF

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Publication number
AU2935300A
AU2935300A AU29353/00A AU2935300A AU2935300A AU 2935300 A AU2935300 A AU 2935300A AU 29353/00 A AU29353/00 A AU 29353/00A AU 2935300 A AU2935300 A AU 2935300A AU 2935300 A AU2935300 A AU 2935300A
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AU
Australia
Prior art keywords
pyridin
phenyl
ylamine
amino
ethoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
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AU29353/00A
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English (en)
Inventor
John Adams Lowe Iii
Mario David Saltarelli
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Pfizer Products Inc
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Pfizer Products Inc
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Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of AU2935300A publication Critical patent/AU2935300A/en
Abandoned legal-status Critical Current

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
AU29353/00A 1999-05-21 2000-03-16 New pharmaceutical combinations for nos inhibitors Abandoned AU2935300A (en)

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US13552099P 1999-05-21 1999-05-21
US60135520 1999-05-21
PCT/IB2000/000295 WO2000071107A2 (fr) 1999-05-21 2000-03-16 Nouvelles combinaisons pharmaceutiques pour les inhibiteurs de nos

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KR (1) KR20020010916A (fr)
CN (1) CN1617743A (fr)
AP (1) AP2001002326A0 (fr)
AR (1) AR022640A1 (fr)
AU (1) AU2935300A (fr)
BG (1) BG106208A (fr)
BR (1) BR0010820A (fr)
CA (1) CA2374668A1 (fr)
CO (1) CO5160295A1 (fr)
DZ (1) DZ3041A1 (fr)
EA (1) EA200101110A1 (fr)
EE (1) EE200100611A (fr)
GT (1) GT200000071A (fr)
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HR (1) HRP20010862A2 (fr)
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PL (1) PL358538A1 (fr)
SK (1) SK16602001A3 (fr)
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TR (1) TR200103351T2 (fr)
UY (1) UY26148A1 (fr)
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DE10001785A1 (de) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma NK¶1¶-Rezeptor-Antagonisten zur Behandlung des Restless Legs Syndroms
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
DOP2002000467A (es) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-amino-6 (fenilo sustituido en las posiciones 2,4,5)-piridinas
BRPI0411608A (pt) * 2003-06-24 2006-08-08 Neurosearch As derivado de 8-aza-biciclo [3.2.1] octano, composição farmacêutica, uso do composto, e, método de tratamento, prevenção ou alìvio de uma doença, um distúrbio ou uma condição de um organismo animal vivo
EP1634598A1 (fr) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Utilisation de dérivés de piperazine et ses analogues pour prevenir et traiter des désordres liés à l'ingestion de nourriture
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
EP2152271B1 (fr) 2007-06-08 2015-10-21 Janssen Pharmaceutica, N.V. Dérivés de piperidine/piperazine
ES2536406T3 (es) 2007-06-08 2015-05-25 Janssen Pharmaceutica, N.V. Derivados de piperidina/piperazina
JP5464709B2 (ja) 2007-06-08 2014-04-09 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ピペリジン／ピペラジン誘導体
PE20100083A1 (es) 2008-06-05 2010-02-17 Janssen Pharmaceutica Nv Combinaciones de drogas que comprenden un inhibidor de dgat y un agonista de ppar
JP5642661B2 (ja) * 2009-03-05 2014-12-17 塩野義製薬株式会社 Ｎｐｙｙ５受容体拮抗作用を有するピペリジンおよびピロリジン誘導体
US20140206667A1 (en) 2012-11-14 2014-07-24 Michela Gallagher Methods and compositions for treating schizophrenia
AU2020291468A1 (en) * 2019-06-14 2022-01-06 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)
US12115154B2 (en) 2020-12-16 2024-10-15 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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Publication number Publication date
IL145955A0 (en) 2002-07-25
NO20015651L (no) 2002-01-18
PE20010157A1 (es) 2001-02-16
TR200103351T2 (tr) 2002-06-21
AP2001002326A0 (en) 2001-12-31
EP1178784A1 (fr) 2002-02-13
CA2374668A1 (fr) 2000-11-30
SK16602001A3 (sk) 2003-03-04
CO5160295A1 (es) 2002-05-30
EE200100611A (et) 2003-02-17
TNSN00106A1 (fr) 2005-11-10
IS6126A (is) 2001-10-26
PA8494601A1 (es) 2002-08-29
BR0010820A (pt) 2002-03-05
MXPA01011978A (es) 2002-05-06
CN1617743A (zh) 2005-05-18
KR20020010916A (ko) 2002-02-06
AR022640A1 (es) 2002-09-04
HN2000000045A (es) 2001-03-02
HRP20010862A2 (en) 2003-06-30
HUP0301287A3 (en) 2005-03-29
BG106208A (en) 2002-09-30
UY26148A1 (es) 2000-12-29
JP2003523941A (ja) 2003-08-12
DZ3041A1 (fr) 2004-03-27
MA26732A1 (fr) 2004-12-20
GT200000071A (es) 2001-11-08
OA11943A (en) 2006-04-12
WO2000071107A2 (fr) 2000-11-30
WO2000071107A8 (fr) 2002-01-24
EA200101110A1 (ru) 2002-08-29
PL358538A1 (en) 2004-08-09
HUP0301287A2 (hu) 2003-08-28
NO20015651D0 (no) 2001-11-20
ZA200109555B (en) 2004-04-07

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