TR200103351T2 - Nos inhibitörleri için yeni farmasötik kombinasyonlar. - Google Patents

Nos inhibitörleri için yeni farmasötik kombinasyonlar.

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Publication number
TR200103351T2
TR200103351T2 TR2001/03351T TR200103351T TR200103351T2 TR 200103351 T2 TR200103351 T2 TR 200103351T2 TR 2001/03351 T TR2001/03351 T TR 2001/03351T TR 200103351 T TR200103351 T TR 200103351T TR 200103351 T2 TR200103351 T2 TR 200103351T2
Authority
TR
Turkey
Prior art keywords
nos
inhibitors
new pharmaceutical
pharmaceutical combinations
nos inhibitors
Prior art date
Application number
TR2001/03351T
Other languages
English (en)
Turkish (tr)
Inventor
David Saltarelli Mario
Adams Iii Lowe John
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of TR200103351T2 publication Critical patent/TR200103351T2/xx

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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    • A61K31/13Amines
    • A61K31/15Oximes (>C=N—O—); Hydrazines (>N—N<); Hydrazones (>N—N=) ; Imines (C—N=C)
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    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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TR2001/03351T 1999-05-21 2000-03-16 Nos inhibitörleri için yeni farmasötik kombinasyonlar. TR200103351T2 (tr)

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DE10001785A1 (de) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma NK¶1¶-Rezeptor-Antagonisten zur Behandlung des Restless Legs Syndroms
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
DOP2002000467A (es) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-amino-6 (fenilo sustituido en las posiciones 2,4,5)-piridinas
BRPI0411608A (pt) * 2003-06-24 2006-08-08 Neurosearch As derivado de 8-aza-biciclo [3.2.1] octano, composição farmacêutica, uso do composto, e, método de tratamento, prevenção ou alìvio de uma doença, um distúrbio ou uma condição de um organismo animal vivo
EP1634598A1 (fr) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Utilisation de dérivés de piperazine et ses analogues pour prevenir et traiter des désordres liés à l'ingestion de nourriture
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
EP2152271B1 (fr) 2007-06-08 2015-10-21 Janssen Pharmaceutica, N.V. Dérivés de piperidine/piperazine
ES2536406T3 (es) 2007-06-08 2015-05-25 Janssen Pharmaceutica, N.V. Derivados de piperidina/piperazina
JP5464709B2 (ja) 2007-06-08 2014-04-09 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ピペリジン/ピペラジン誘導体
PE20100083A1 (es) 2008-06-05 2010-02-17 Janssen Pharmaceutica Nv Combinaciones de drogas que comprenden un inhibidor de dgat y un agonista de ppar
JP5642661B2 (ja) * 2009-03-05 2014-12-17 塩野義製薬株式会社 Npyy5受容体拮抗作用を有するピペリジンおよびピロリジン誘導体
US20140206667A1 (en) 2012-11-14 2014-07-24 Michela Gallagher Methods and compositions for treating schizophrenia
AU2020291468A1 (en) * 2019-06-14 2022-01-06 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)
US12115154B2 (en) 2020-12-16 2024-10-15 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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IL145955A0 (en) 2002-07-25
NO20015651L (no) 2002-01-18
PE20010157A1 (es) 2001-02-16
AP2001002326A0 (en) 2001-12-31
EP1178784A1 (fr) 2002-02-13
CA2374668A1 (fr) 2000-11-30
SK16602001A3 (sk) 2003-03-04
CO5160295A1 (es) 2002-05-30
EE200100611A (et) 2003-02-17
TNSN00106A1 (fr) 2005-11-10
IS6126A (is) 2001-10-26
PA8494601A1 (es) 2002-08-29
BR0010820A (pt) 2002-03-05
MXPA01011978A (es) 2002-05-06
CN1617743A (zh) 2005-05-18
KR20020010916A (ko) 2002-02-06
AR022640A1 (es) 2002-09-04
HN2000000045A (es) 2001-03-02
HRP20010862A2 (en) 2003-06-30
HUP0301287A3 (en) 2005-03-29
BG106208A (en) 2002-09-30
UY26148A1 (es) 2000-12-29
JP2003523941A (ja) 2003-08-12
DZ3041A1 (fr) 2004-03-27
MA26732A1 (fr) 2004-12-20
GT200000071A (es) 2001-11-08
OA11943A (en) 2006-04-12
WO2000071107A2 (fr) 2000-11-30
AU2935300A (en) 2000-12-12
WO2000071107A8 (fr) 2002-01-24
EA200101110A1 (ru) 2002-08-29
PL358538A1 (en) 2004-08-09
HUP0301287A2 (hu) 2003-08-28
NO20015651D0 (no) 2001-11-20
ZA200109555B (en) 2004-04-07

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