PL358538A1 - New pharmaceutical combinations for nos inhibitors - Google Patents

New pharmaceutical combinations for nos inhibitors

Info

Publication number
PL358538A1
PL358538A1 PL00358538A PL35853800A PL358538A1 PL 358538 A1 PL358538 A1 PL 358538A1 PL 00358538 A PL00358538 A PL 00358538A PL 35853800 A PL35853800 A PL 35853800A PL 358538 A1 PL358538 A1 PL 358538A1
Authority
PL
Poland
Prior art keywords
pharmaceutical combinations
new pharmaceutical
nos inhibitors
inhibitors
nos
Prior art date
Application number
PL00358538A
Other languages
English (en)
Polish (pl)
Inventor
Mario David Saltarelli
John Adams Lowe Iii
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of PL358538A1 publication Critical patent/PL358538A1/xx

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/13—Amines
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    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Anesthesiology (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PL00358538A 1999-05-21 2000-03-16 New pharmaceutical combinations for nos inhibitors PL358538A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13552099P 1999-05-21 1999-05-21
PCT/IB2000/000295 WO2000071107A2 (fr) 1999-05-21 2000-03-16 Nouvelles combinaisons pharmaceutiques pour les inhibiteurs de nos

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EP (1) EP1178784A1 (fr)
JP (1) JP2003523941A (fr)
KR (1) KR20020010916A (fr)
CN (1) CN1617743A (fr)
AP (1) AP2001002326A0 (fr)
AR (1) AR022640A1 (fr)
AU (1) AU2935300A (fr)
BG (1) BG106208A (fr)
BR (1) BR0010820A (fr)
CA (1) CA2374668A1 (fr)
CO (1) CO5160295A1 (fr)
DZ (1) DZ3041A1 (fr)
EA (1) EA200101110A1 (fr)
EE (1) EE200100611A (fr)
GT (1) GT200000071A (fr)
HN (1) HN2000000045A (fr)
HR (1) HRP20010862A2 (fr)
HU (1) HUP0301287A3 (fr)
IL (1) IL145955A0 (fr)
IS (1) IS6126A (fr)
MA (1) MA26732A1 (fr)
MX (1) MXPA01011978A (fr)
NO (1) NO20015651L (fr)
OA (1) OA11943A (fr)
PA (1) PA8494601A1 (fr)
PE (1) PE20010157A1 (fr)
PL (1) PL358538A1 (fr)
SK (1) SK16602001A3 (fr)
TN (1) TNSN00106A1 (fr)
TR (1) TR200103351T2 (fr)
UY (1) UY26148A1 (fr)
WO (1) WO2000071107A2 (fr)
ZA (1) ZA200109555B (fr)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10001785A1 (de) * 2000-01-18 2001-07-19 Boehringer Ingelheim Pharma NK¶1¶-Rezeptor-Antagonisten zur Behandlung des Restless Legs Syndroms
GB0019006D0 (en) * 2000-08-04 2000-09-20 Astrazeneca Ab Novel compounds
US20030045449A1 (en) * 2001-08-15 2003-03-06 Pfizer, Inc. Pharmaceutical combinations for the treatment of neurodegenerative diseases
DOP2002000467A (es) * 2001-10-10 2003-04-15 Pfizer Prod Inc 2-amino-6 (fenilo sustituido en las posiciones 2,4,5)-piridinas
US6803470B2 (en) * 2001-10-10 2004-10-12 Pfizer Inc 2-amino-6-(2,4,5-substituted-phenyl)-pyridines
AU2004249441B2 (en) * 2003-06-24 2009-11-12 Neurosearch A/S Novel 8-aza-bicyclo(3.2.1)octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
EP1634598A1 (fr) * 2004-09-07 2006-03-15 Laboratorios Del Dr. Esteve, S.A. Utilisation de dérivés de piperazine et ses analogues pour prevenir et traiter des désordres liés à l'ingestion de nourriture
EP2152271B1 (fr) 2007-06-08 2015-10-21 Janssen Pharmaceutica, N.V. Dérivés de piperidine/piperazine
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
CA2687918C (fr) 2007-06-08 2016-11-08 Janssen Pharmaceutica N.V. Derives de piperidine/piperazine
AU2008258487B2 (en) 2007-06-08 2012-11-15 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
JP5579170B2 (ja) 2008-06-05 2014-08-27 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Ｄｇａｔ阻害剤とｐｐａｒ作動薬を含有する薬剤組み合わせ物
US8889674B2 (en) 2009-03-05 2014-11-18 Shionogi & Co., Ltd. Piperidine and pyrrolidine derivatives having NPY Y5 receptor antagonism
JP6440625B2 (ja) 2012-11-14 2018-12-19 ザ・ジョンズ・ホプキンス・ユニバーシティー 精神分裂病を処置するための方法および組成物
US20220267269A1 (en) * 2019-06-14 2022-08-25 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (pcsk9)
US12115154B2 (en) 2020-12-16 2024-10-15 Srx Cardio, Llc Compounds for the modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9)

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Publication number Publication date
HN2000000045A (es) 2001-03-02
EP1178784A1 (fr) 2002-02-13
EA200101110A1 (ru) 2002-08-29
CN1617743A (zh) 2005-05-18
IS6126A (is) 2001-10-26
AP2001002326A0 (en) 2001-12-31
KR20020010916A (ko) 2002-02-06
NO20015651L (no) 2002-01-18
EE200100611A (et) 2003-02-17
HRP20010862A2 (en) 2003-06-30
BR0010820A (pt) 2002-03-05
NO20015651D0 (no) 2001-11-20
JP2003523941A (ja) 2003-08-12
CA2374668A1 (fr) 2000-11-30
DZ3041A1 (fr) 2004-03-27
HUP0301287A3 (en) 2005-03-29
MA26732A1 (fr) 2004-12-20
GT200000071A (es) 2001-11-08
IL145955A0 (en) 2002-07-25
TR200103351T2 (tr) 2002-06-21
OA11943A (en) 2006-04-12
SK16602001A3 (sk) 2003-03-04
TNSN00106A1 (fr) 2005-11-10
WO2000071107A2 (fr) 2000-11-30
BG106208A (en) 2002-09-30
CO5160295A1 (es) 2002-05-30
UY26148A1 (es) 2000-12-29
HUP0301287A2 (hu) 2003-08-28
AR022640A1 (es) 2002-09-04
PA8494601A1 (es) 2002-08-29
AU2935300A (en) 2000-12-12
MXPA01011978A (es) 2002-05-06
PE20010157A1 (es) 2001-02-16
ZA200109555B (en) 2004-04-07
WO2000071107A8 (fr) 2002-01-24

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