BR0110385A - Composto, composição anti-helmìntica, acaricida ou inseticida, método de proteção de plantas ou animais de danos causados por parasitas, e, uso de um composto - Google Patents
Composto, composição anti-helmìntica, acaricida ou inseticida, método de proteção de plantas ou animais de danos causados por parasitas, e, uso de um compostoInfo
- Publication number
- BR0110385A BR0110385A BR0110385-7A BR0110385A BR0110385A BR 0110385 A BR0110385 A BR 0110385A BR 0110385 A BR0110385 A BR 0110385A BR 0110385 A BR0110385 A BR 0110385A
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- optionally substituted
- anthelmintic
- acaricidal
- parasites
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 5
- 241001465754 Metazoa Species 0.000 title abstract 2
- 230000000895 acaricidal effect Effects 0.000 title abstract 2
- 230000000507 anthelmentic effect Effects 0.000 title abstract 2
- 230000000749 insecticidal effect Effects 0.000 title abstract 2
- 244000045947 parasite Species 0.000 title abstract 2
- 239000002361 compost Substances 0.000 title 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
- 125000001589 carboacyl group Chemical group 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 239000002917 insecticide Substances 0.000 abstract 1
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- 125000002914 sec-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
- 125000005017 substituted alkenyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Agronomy & Crop Science (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Dentistry (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Wood Science & Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
"COMPOSTO, COMPOSIçãO ANTI-HELMìNTICA, ACARICIDA OU INSETICIDA, MéTODO DE PROTEçãO DE PLANTAS OU ANIMAIS DE DANOS CAUSADOS POR PARASITAS, E, USO DE UM COMPOSTO". Compostos de fórmula (I) e seus sais, em que: R^ 1^ representa metila, etila, isopropila ou s-butila; R^ 2^ representa hidrogênio ou alquila; R^ 3^ representa hidrogênio, alcanoíla opcionalmente substituído, alquenoíla opcionalmente substituído, alquinoíla opcionalmente substituído, alquilsulfonila, ou alcoxicarbonila, ou R^ 2^ e R^ 3^ juntamente com o átomo de nitrogênio ao qual estão ligados formam um grupo de anel heterocíclico saturado com de 4 a 6 membros opcionalmente substituído; e a porção -a- juntamente com o átomo de carbono ao qual está ligada forma um grupo cicloalquila com de 3 a 6 membros. Estes compostos têm atividade anti-helmíntica, acaricida e inseticida.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000127209 | 2000-04-27 | ||
| PCT/JP2001/003656 WO2001083500A1 (en) | 2000-04-27 | 2001-04-26 | 13-substituted milbemycin derivatives, their preparation and their use against insects and other pests |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0110385A true BR0110385A (pt) | 2003-02-04 |
Family
ID=18636847
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0110385-7A BR0110385A (pt) | 2000-04-27 | 2001-04-26 | Composto, composição anti-helmìntica, acaricida ou inseticida, método de proteção de plantas ou animais de danos causados por parasitas, e, uso de um composto |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US6653342B2 (pt) |
| EP (1) | EP1276748B1 (pt) |
| KR (1) | KR100711931B1 (pt) |
| CN (1) | CN1247607C (pt) |
| AR (1) | AR029250A1 (pt) |
| AT (1) | ATE315573T1 (pt) |
| AU (2) | AU5261301A (pt) |
| BR (1) | BR0110385A (pt) |
| CA (1) | CA2407611A1 (pt) |
| CZ (1) | CZ20023565A3 (pt) |
| DE (1) | DE60116615T2 (pt) |
| DK (1) | DK1276748T3 (pt) |
| ES (1) | ES2254400T3 (pt) |
| HU (1) | HUP0301040A3 (pt) |
| IL (1) | IL152449A0 (pt) |
| MX (1) | MXPA02010587A (pt) |
| NO (1) | NO323751B1 (pt) |
| NZ (1) | NZ522247A (pt) |
| PL (1) | PL357598A1 (pt) |
| RU (1) | RU2226531C1 (pt) |
| TW (1) | TWI285206B (pt) |
| WO (1) | WO2001083500A1 (pt) |
| ZA (1) | ZA200208630B (pt) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20040047962A (ko) * | 2001-10-25 | 2004-06-05 | 상꾜 라이프테크 가부시키가이샤 | 기생충 구제 조성물 |
| AR045142A1 (es) | 2003-07-30 | 2005-10-19 | Novartis Ag | Composicion veterinaria masticable ductil de buen sabor |
| US20090281175A1 (en) * | 2006-09-28 | 2009-11-12 | Galderma S.A. | Avermectin compounds and treatment of dermatological disorders in humans therewith |
| TWI457347B (zh) | 2008-12-04 | 2014-10-21 | Merial Ltd | 二聚合的阿佛菌素（ａｖｅｒｍｅｃｔｉｎ）及密倍脈心（ｍｉｌｂｅｍｙｃｉｎ）衍生物 |
| RU2413513C2 (ru) * | 2009-04-06 | 2011-03-10 | Государственное образовательное учреждение высшего профессионального образования "Казанский государственный университет им. В.И. Ульянова-Ленина" | Антигельминтная композиция на основе соли четвертичного фосфония и замещенного динитробензофуроксана |
| US8980896B2 (en) | 2009-12-17 | 2015-03-17 | Merial, Inc. | Compositions comprising macrocyclic lactone compounds and spirodioxepinoindoles |
| MX379693B (es) | 2011-12-02 | 2025-03-11 | Merial Ltd | Formulaciones de moxidectina inyectables de larga acción y formas de cristal de moxidectina novedosas. |
| PL2983712T3 (pl) | 2013-04-12 | 2021-05-31 | Zoetis Services Llc | Kompozycja makrocyklicznych laktonów, lewamizolu, aminocukru i dodatkowego środka przeciwpasożytniczego |
| CA3123852A1 (en) * | 2018-12-21 | 2020-06-25 | Bayer Healthcare Llc | Parasiticidal formulations and use thereof |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4201861A (en) | 1977-10-03 | 1980-05-06 | Merck & Co., Inc. | Acyl derivatives of C-076 compounds |
| US4206205A (en) | 1977-10-03 | 1980-06-03 | Merck & Co., Inc. | Monosaccharide and aglycone derivatives of C-076 |
| NZ188459A (en) | 1977-10-03 | 1982-09-07 | Merck & Co Inc | Derivatives of c-076 compounds and pesticidal compositions |
| US4171314A (en) | 1977-12-19 | 1979-10-16 | Merck & Co., Inc. | 13-Halo and 13-deoxy C-076 compounds |
| US4173571A (en) | 1977-12-19 | 1979-11-06 | Merck & Co., Inc. | 13-Halo and 13-deoxy derivatives of C-076 compounds |
| US4203976A (en) | 1978-08-02 | 1980-05-20 | Merck & Co., Inc. | Sugar derivatives of C-076 compounds |
| US4200581A (en) | 1978-08-04 | 1980-04-29 | Merck & Co., Inc. | Alkyl derivatives of C-076 compounds |
| US4289760A (en) | 1980-05-02 | 1981-09-15 | Merck & Co., Inc. | 23-Keto derivatives of C-076 compounds |
| JPS57120589A (en) | 1981-01-20 | 1982-07-27 | Sankyo Co Ltd | 5-methoxy and 5-lower alkanoyloxy derivative, its preparation and acaricide and parasiticide |
| IT1144368B (it) | 1981-05-20 | 1986-10-29 | Gaudino Di P Gaudino & C Sas O | Perfezionamenti nei laminatoi con almeno un campo di stiro per la filatura diretta di pettinato e semipettinato |
| US4457920A (en) | 1981-09-03 | 1984-07-03 | Merck & Co., Inc. | 4a-Substituted avermectin compounds |
| US4423209A (en) | 1982-02-26 | 1983-12-27 | Merck & Co., Inc. | Processes for the interconversion of avermectin compounds |
| JPS5916894A (ja) | 1982-07-21 | 1984-01-28 | Sankyo Co Ltd | ミルベマイシンｄの５−アシルオキシ誘導体 |
| JPS5920285A (ja) | 1982-07-23 | 1984-02-01 | Sankyo Co Ltd | ミルベマイシンｄの５−二塩基酸エステル誘導体及びその塩 |
| JPS59108785A (ja) | 1982-11-25 | 1984-06-23 | Sankyo Co Ltd | ミルベマイシン類の５−オキシム誘導体 |
| US4469682A (en) | 1983-01-28 | 1984-09-04 | Merck & Co., Inc. | Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use |
| US4579864A (en) | 1984-06-11 | 1986-04-01 | Merck & Co., Inc. | Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives |
| US4547491A (en) | 1984-07-18 | 1985-10-15 | Merck & Co., Inc. | C-8A-Oxo-avermectin and milbemycin derivatives, pharmaceutical compositions and method of use |
| EP0180539A1 (de) | 1984-09-18 | 1986-05-07 | Ciba-Geigy Ag | 13-Halo- und 13-Hydroximilbemycine |
| US4696922A (en) | 1984-11-26 | 1987-09-29 | Ciba-Geigy Corporation | 5-azolylacetoxymilbemycins as ecto- and endoparasites |
| JPS6289685A (ja) | 1985-05-31 | 1987-04-24 | Sankyo Co Ltd | １３−ハロゲンミルベマイシン誘導体 |
| RU2024527C1 (ru) | 1986-03-25 | 1994-12-15 | Санкио Компани Лимитед | Способ получения макролидных соединений |
| US5614470A (en) * | 1994-04-01 | 1997-03-25 | Sankyo Company, Limited | 13-substituted milbemycin derivatives, their preparation and their use |
| PT765879E (pt) | 1995-09-29 | 2001-05-31 | Sankyo Co | Derivados 13-substituidos de milbemicina-5-oxima sua preparacao e utilizacao contra insectos e outras pragas |
-
2001
- 2001-04-26 NZ NZ522247A patent/NZ522247A/en unknown
- 2001-04-26 TW TW090109990A patent/TWI285206B/zh not_active IP Right Cessation
- 2001-04-26 AT AT01925985T patent/ATE315573T1/de not_active IP Right Cessation
- 2001-04-26 CA CA002407611A patent/CA2407611A1/en not_active Abandoned
- 2001-04-26 EP EP01925985A patent/EP1276748B1/en not_active Expired - Lifetime
- 2001-04-26 RU RU2002131794/04A patent/RU2226531C1/ru not_active IP Right Cessation
- 2001-04-26 MX MXPA02010587A patent/MXPA02010587A/es active IP Right Grant
- 2001-04-26 BR BR0110385-7A patent/BR0110385A/pt not_active IP Right Cessation
- 2001-04-26 CZ CZ20023565A patent/CZ20023565A3/cs unknown
- 2001-04-26 DE DE60116615T patent/DE60116615T2/de not_active Expired - Fee Related
- 2001-04-26 IL IL15244901A patent/IL152449A0/xx unknown
- 2001-04-26 WO PCT/JP2001/003656 patent/WO2001083500A1/en not_active Ceased
- 2001-04-26 AU AU5261301A patent/AU5261301A/xx active Pending
- 2001-04-26 PL PL01357598A patent/PL357598A1/xx unknown
- 2001-04-26 CN CNB018119832A patent/CN1247607C/zh not_active Expired - Fee Related
- 2001-04-26 ES ES01925985T patent/ES2254400T3/es not_active Expired - Lifetime
- 2001-04-26 HU HU0301040A patent/HUP0301040A3/hu unknown
- 2001-04-26 DK DK01925985T patent/DK1276748T3/da active
- 2001-04-26 KR KR1020027013834A patent/KR100711931B1/ko not_active Expired - Fee Related
- 2001-04-26 AU AU2001252613A patent/AU2001252613B2/en not_active Ceased
- 2001-04-27 AR ARP010102004A patent/AR029250A1/es not_active Application Discontinuation
-
2002
- 2002-10-22 US US10/277,993 patent/US6653342B2/en not_active Expired - Fee Related
- 2002-10-24 ZA ZA200208630A patent/ZA200208630B/en unknown
- 2002-10-25 NO NO20025141A patent/NO323751B1/no not_active IP Right Cessation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B25A | Requested transfer of rights approved |
Owner name: SANKYO COMPANY, LIMITED (JP) , SANKYO LIFETECH COM Free format text: TRANSFERIDO DE: SANKYO COMPANY, LIMITED |
|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6A, 7A E 8A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO PUBLICADO NA RPI 2008 DE 30/06/2009. |