ATE315573T1 - 13-substituierte milbemycinderivate, ihre herstellung und ihre verwendung gegen insekten und andere schadorganismen - Google Patents

13-substituierte milbemycinderivate, ihre herstellung und ihre verwendung gegen insekten und andere schadorganismen

Info

Publication number: ATE315573T1
Authority: AT; Austria
Prior art keywords: production; against insects; use against; harmful organisms; milbemycin derivatives
Prior art date: 2000-04-27

Application number

AT01925985T

Other languages

English (en)

Inventor

Akio Saito

Yoko Sugiyama

Toshimitsu Toyama

Toshihiko Nanba

Original Assignee

Sankyo Lifetech Company Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-04-27

Filing date

2001-04-26

Publication date

2006-02-15

2001-04-26 Application filed by Sankyo Lifetech Company Ltd filed Critical Sankyo Lifetech Company Ltd

2006-02-15 Application granted granted Critical

2006-02-15 Publication of ATE315573T1 publication Critical patent/ATE315573T1/de

Links

241000238631 Hexapoda Species 0.000 title 1
FXWHFKOXMBTCMP-WMEDONTMSA-N milbemycin Natural products COC1C2OCC3=C/C=C/C(C)CC(=CCC4CC(CC5(O4)OC(C)C(C)C(OC(=O)C(C)CC(C)C)C5O)OC(=O)C(C=C1C)C23O)C FXWHFKOXMBTCMP-WMEDONTMSA-N 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

Life Sciences & Earth Sciences (AREA)
Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Agronomy & Crop Science (AREA)
Zoology (AREA)
Environmental Sciences (AREA)
Tropical Medicine & Parasitology (AREA)
Dentistry (AREA)
Plant Pathology (AREA)
Pest Control & Pesticides (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Wood Science & Technology (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AT01925985T 2000-04-27 2001-04-26 13-substituierte milbemycinderivate, ihre herstellung und ihre verwendung gegen insekten und andere schadorganismen ATE315573T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP2000127209		2000-04-27

Publications (1)

Publication Number	Publication Date
ATE315573T1 true ATE315573T1 (de)	2006-02-15

Family

ID=18636847

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT01925985T ATE315573T1 (de)	2000-04-27	2001-04-26	13-substituierte milbemycinderivate, ihre herstellung und ihre verwendung gegen insekten und andere schadorganismen

Country Status (23)

Country	Link
US (1)	US6653342B2 (de)
EP (1)	EP1276748B1 (de)
KR (1)	KR100711931B1 (de)
CN (1)	CN1247607C (de)
AR (1)	AR029250A1 (de)
AT (1)	ATE315573T1 (de)
AU (2)	AU5261301A (de)
BR (1)	BR0110385A (de)
CA (1)	CA2407611A1 (de)
CZ (1)	CZ20023565A3 (de)
DE (1)	DE60116615T2 (de)
DK (1)	DK1276748T3 (de)
ES (1)	ES2254400T3 (de)
HU (1)	HUP0301040A3 (de)
IL (1)	IL152449A0 (de)
MX (1)	MXPA02010587A (de)
NO (1)	NO323751B1 (de)
NZ (1)	NZ522247A (de)
PL (1)	PL357598A1 (de)
RU (1)	RU2226531C1 (de)
TW (1)	TWI285206B (de)
WO (1)	WO2001083500A1 (de)
ZA (1)	ZA200208630B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
KR20040047962A (ko) *	2001-10-25	2004-06-05	상꾜 라이프테크 가부시키가이샤	기생충 구제 조성물
AR045142A1 (es)	2003-07-30	2005-10-19	Novartis Ag	Composicion veterinaria masticable ductil de buen sabor
US20090281175A1 (en) *	2006-09-28	2009-11-12	Galderma S.A.	Avermectin compounds and treatment of dermatological disorders in humans therewith
TWI457347B (zh)	2008-12-04	2014-10-21	Merial Ltd	二聚合的阿佛菌素（ａｖｅｒｍｅｃｔｉｎ）及密倍脈心（ｍｉｌｂｅｍｙｃｉｎ）衍生物
RU2413513C2 (ru) *	2009-04-06	2011-03-10	Государственное образовательное учреждение высшего профессионального образования "Казанский государственный университет им. В.И. Ульянова-Ленина"	Антигельминтная композиция на основе соли четвертичного фосфония и замещенного динитробензофуроксана
US8980896B2 (en)	2009-12-17	2015-03-17	Merial, Inc.	Compositions comprising macrocyclic lactone compounds and spirodioxepinoindoles
MX379693B (es)	2011-12-02	2025-03-11	Merial Ltd	Formulaciones de moxidectina inyectables de larga acción y formas de cristal de moxidectina novedosas.
PL2983712T3 (pl)	2013-04-12	2021-05-31	Zoetis Services Llc	Kompozycja makrocyklicznych laktonów, lewamizolu, aminocukru i dodatkowego środka przeciwpasożytniczego
CA3123852A1 (en) *	2018-12-21	2020-06-25	Bayer Healthcare Llc	Parasiticidal formulations and use thereof

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4201861A (en)	1977-10-03	1980-05-06	Merck & Co., Inc.	Acyl derivatives of C-076 compounds
US4206205A (en)	1977-10-03	1980-06-03	Merck & Co., Inc.	Monosaccharide and aglycone derivatives of C-076
NZ188459A (en)	1977-10-03	1982-09-07	Merck & Co Inc	Derivatives of c-076 compounds and pesticidal compositions
US4171314A (en)	1977-12-19	1979-10-16	Merck & Co., Inc.	13-Halo and 13-deoxy C-076 compounds
US4173571A (en)	1977-12-19	1979-11-06	Merck & Co., Inc.	13-Halo and 13-deoxy derivatives of C-076 compounds
US4203976A (en)	1978-08-02	1980-05-20	Merck & Co., Inc.	Sugar derivatives of C-076 compounds
US4200581A (en)	1978-08-04	1980-04-29	Merck & Co., Inc.	Alkyl derivatives of C-076 compounds
US4289760A (en)	1980-05-02	1981-09-15	Merck & Co., Inc.	23-Keto derivatives of C-076 compounds
JPS57120589A (en)	1981-01-20	1982-07-27	Sankyo Co Ltd	5-methoxy and 5-lower alkanoyloxy derivative, its preparation and acaricide and parasiticide
IT1144368B (it)	1981-05-20	1986-10-29	Gaudino Di P Gaudino & C Sas O	Perfezionamenti nei laminatoi con almeno un campo di stiro per la filatura diretta di pettinato e semipettinato
US4457920A (en)	1981-09-03	1984-07-03	Merck & Co., Inc.	4a-Substituted avermectin compounds
US4423209A (en)	1982-02-26	1983-12-27	Merck & Co., Inc.	Processes for the interconversion of avermectin compounds
JPS5916894A (ja)	1982-07-21	1984-01-28	Sankyo Co Ltd	ミルベマイシンｄの５−アシルオキシ誘導体
JPS5920285A (ja)	1982-07-23	1984-02-01	Sankyo Co Ltd	ミルベマイシンｄの５−二塩基酸エステル誘導体及びその塩
JPS59108785A (ja)	1982-11-25	1984-06-23	Sankyo Co Ltd	ミルベマイシン類の５−オキシム誘導体
US4469682A (en)	1983-01-28	1984-09-04	Merck & Co., Inc.	Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
US4579864A (en)	1984-06-11	1986-04-01	Merck & Co., Inc.	Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives
US4547491A (en)	1984-07-18	1985-10-15	Merck & Co., Inc.	C-8A-Oxo-avermectin and milbemycin derivatives, pharmaceutical compositions and method of use
EP0180539A1 (de)	1984-09-18	1986-05-07	Ciba-Geigy Ag	13-Halo- und 13-Hydroximilbemycine
US4696922A (en)	1984-11-26	1987-09-29	Ciba-Geigy Corporation	5-azolylacetoxymilbemycins as ecto- and endoparasites
JPS6289685A (ja)	1985-05-31	1987-04-24	Sankyo Co Ltd	１３−ハロゲンミルベマイシン誘導体
RU2024527C1 (ru)	1986-03-25	1994-12-15	Санкио Компани Лимитед	Способ получения макролидных соединений
US5614470A (en) *	1994-04-01	1997-03-25	Sankyo Company, Limited	13-substituted milbemycin derivatives, their preparation and their use
PT765879E (pt)	1995-09-29	2001-05-31	Sankyo Co	Derivados 13-substituidos de milbemicina-5-oxima sua preparacao e utilizacao contra insectos e outras pragas

2001
- 2001-04-26 NZ NZ522247A patent/NZ522247A/en unknown
- 2001-04-26 TW TW090109990A patent/TWI285206B/zh not_active IP Right Cessation
- 2001-04-26 AT AT01925985T patent/ATE315573T1/de not_active IP Right Cessation
- 2001-04-26 CA CA002407611A patent/CA2407611A1/en not_active Abandoned
- 2001-04-26 EP EP01925985A patent/EP1276748B1/de not_active Expired - Lifetime
- 2001-04-26 RU RU2002131794/04A patent/RU2226531C1/ru not_active IP Right Cessation
- 2001-04-26 MX MXPA02010587A patent/MXPA02010587A/es active IP Right Grant
- 2001-04-26 BR BR0110385-7A patent/BR0110385A/pt not_active IP Right Cessation
- 2001-04-26 CZ CZ20023565A patent/CZ20023565A3/cs unknown
- 2001-04-26 DE DE60116615T patent/DE60116615T2/de not_active Expired - Fee Related
- 2001-04-26 IL IL15244901A patent/IL152449A0/xx unknown
- 2001-04-26 WO PCT/JP2001/003656 patent/WO2001083500A1/en not_active Ceased
- 2001-04-26 AU AU5261301A patent/AU5261301A/xx active Pending
- 2001-04-26 PL PL01357598A patent/PL357598A1/xx unknown
- 2001-04-26 CN CNB018119832A patent/CN1247607C/zh not_active Expired - Fee Related
- 2001-04-26 ES ES01925985T patent/ES2254400T3/es not_active Expired - Lifetime
- 2001-04-26 HU HU0301040A patent/HUP0301040A3/hu unknown
- 2001-04-26 DK DK01925985T patent/DK1276748T3/da active
- 2001-04-26 KR KR1020027013834A patent/KR100711931B1/ko not_active Expired - Fee Related
- 2001-04-26 AU AU2001252613A patent/AU2001252613B2/en not_active Ceased
- 2001-04-27 AR ARP010102004A patent/AR029250A1/es not_active Application Discontinuation
2002
- 2002-10-22 US US10/277,993 patent/US6653342B2/en not_active Expired - Fee Related
- 2002-10-24 ZA ZA200208630A patent/ZA200208630B/en unknown
- 2002-10-25 NO NO20025141A patent/NO323751B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
DE60116615D1 (de)	2006-04-06
US6653342B2 (en)	2003-11-25
RU2226531C1 (ru)	2004-04-10
PL357598A1 (en)	2004-07-26
NZ522247A (en)	2004-07-30
DE60116615T2 (de)	2006-09-07
ES2254400T3 (es)	2006-06-16
CA2407611A1 (en)	2001-11-08
KR20020087987A (ko)	2002-11-23
MXPA02010587A (es)	2003-03-10
IL152449A0 (en)	2003-05-29
CN1439016A (zh)	2003-08-27
NO323751B1 (no)	2007-07-02
EP1276748A1 (de)	2003-01-22
US20030139601A1 (en)	2003-07-24
RU2002131794A (ru)	2004-02-27
KR100711931B1 (ko)	2007-05-02
CN1247607C (zh)	2006-03-29
NO20025141D0 (no)	2002-10-25
TWI285206B (en)	2007-08-11
WO2001083500A1 (en)	2001-11-08
BR0110385A (pt)	2003-02-04
EP1276748B1 (de)	2006-01-11
HUP0301040A2 (hu)	2003-08-28
ZA200208630B (en)	2004-02-12
HUP0301040A3 (en)	2005-11-28
NO20025141L (no)	2002-12-16
HK1057757A1 (en)	2004-04-16
DK1276748T3 (da)	2006-03-20
CZ20023565A3 (cs)	2003-04-16
WO2001083500A8 (en)	2003-05-08
AR029250A1 (es)	2003-06-18
AU5261301A (en)	2001-11-12
AU2001252613B2 (en)	2004-05-13

Legal Events

Date

Code

Title

Description

2006-10-15

UEP

Publication of translation of european patent specification

Ref document number: 1276748

Country of ref document: EP

2011-01-15

REN

Ceased due to non-payment of the annual fee

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