CZ20031083A3 - 5-Spiropyrimidin-2, 4, 6-trionové inhibitory metaloproteinasy - Google Patents

5-Spiropyrimidin-2, 4, 6-trionové inhibitory metaloproteinasy Download PDF

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Publication number: CZ20031083A3
Authority: CZ; Czechia
Prior art keywords: group; alkyl; pyridin; triazaspiro; ring
Prior art date: 2000-10-26

Application number

CZ20031083A

Other languages

Czech (cs)

English (en)

Inventor

Brian Scott Bronk

Mark Carl Noe

Martin James Wythes

Original Assignee

Pfizer Products Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-10-26

Filing date

2001-10-23

Publication date

2004-03-17

2001-10-23 Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.

2004-03-17 Publication of CZ20031083A3 publication Critical patent/CZ20031083A3/cs

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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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- C07D487/10—Spiro-condensed systems

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Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Physical Education & Sports Medicine (AREA)
Immunology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Rheumatology (AREA)
Oncology (AREA)
Dermatology (AREA)
Communicable Diseases (AREA)
Orthopedic Medicine & Surgery (AREA)
Pain & Pain Management (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Gynecology & Obstetrics (AREA)
Cardiology (AREA)
Pregnancy & Childbirth (AREA)
Virology (AREA)
Ophthalmology & Optometry (AREA)
Heart & Thoracic Surgery (AREA)
Tropical Medicine & Parasitology (AREA)
Hematology (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)

CZ20031083A 2000-10-26 2001-10-23 5-Spiropyrimidin-2, 4, 6-trionové inhibitory metaloproteinasy CZ20031083A3 (cs)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US24338900P	2000-10-26	2000-10-26

Publications (1)

Publication Number	Publication Date
CZ20031083A3 true CZ20031083A3 (cs)	2004-03-17

Family

ID=22918584

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CZ20031083A CZ20031083A3 (cs)	2000-10-26	2001-10-23	5-Spiropyrimidin-2, 4, 6-trionové inhibitory metaloproteinasy

Country Status (32)

Country	Link
EP (1)	EP1332146A2 (fr)
JP (1)	JP2004518635A (fr)
KR (1)	KR20040004412A (fr)
CN (1)	CN1501937A (fr)
AP (1)	AP2001002318A0 (fr)
AR (1)	AR035069A1 (fr)
AU (1)	AU2002210813A1 (fr)
BG (1)	BG107653A (fr)
BR (1)	BR0114913A (fr)
CA (1)	CA2425283A1 (fr)
CZ (1)	CZ20031083A3 (fr)
EA (1)	EA005762B1 (fr)
EC (1)	ECSP034567A (fr)
EE (1)	EE200300196A (fr)
GT (1)	GT200100213A (fr)
HN (1)	HN2001000244A (fr)
HR (1)	HRP20030332A2 (fr)
HU (1)	HUP0301577A3 (fr)
IL (1)	IL154948A0 (fr)
IS (1)	IS6762A (fr)
MA (1)	MA26957A1 (fr)
MX (1)	MXPA03003735A (fr)
NO (1)	NO20031853L (fr)
OA (1)	OA12529A (fr)
PA (1)	PA8531401A1 (fr)
PE (1)	PE20020589A1 (fr)
PL (1)	PL366201A1 (fr)
SK (1)	SK4972003A3 (fr)
SV (1)	SV2003000705A (fr)
TN (1)	TNSN01149A1 (fr)
WO (1)	WO2002034753A2 (fr)
ZA (1)	ZA200302190B (fr)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DOP2002000332A (es)	2001-02-14	2002-08-30	Warner Lambert Co	Inhibidores de piridina de metaloproteinasas de la matriz
WO2002064571A1 (fr)	2001-02-14	2002-08-22	Warner-Lambert Company Llc	Pyrimidine comme inhibiteurs de la métalloprotéinase de matrice
BR0207865A (pt)	2001-02-14	2004-03-23	Warner Lambert Co	Benzotiadiazinas inibidores de metaloproteinases de matriz
DOP2002000333A (es)	2001-02-14	2002-09-30	Warner Lambert Co	Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
PA8539501A1 (es)	2001-02-14	2002-09-30	Warner Lambert Co	Compuestos triazolo como inhibidores de mmp
US6924276B2 (en)	2001-09-10	2005-08-02	Warner-Lambert Company	Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
BR0213233A (pt)	2001-10-12	2005-01-04	Warner Lambert Co	Alcinos inibidores de metaloproteinase de matriz
US6962922B2 (en)	2001-10-12	2005-11-08	Warner-Lambert Company Llc	Alkynylated quinazoline compounds
US6894057B2 (en)	2002-03-08	2005-05-17	Warner-Lambert Company	Oxo-azabicyclic compounds
AU2003228701A1 (en) *	2002-04-25	2003-11-10	Bristol-Myers Squibb Company	Spirobarbituric acid derivatives useful as inhibitors of matrix metalloproteases
WO2003091258A1 (fr) *	2002-04-26	2003-11-06	Pfizer Products Inc.	Inhibiteurs de la metalloproteinase n-substitues-heteroaryloxy-aryl-spiro-pyrimidine-2,4,6-trione
EP1501834B1 (fr) *	2002-04-26	2005-09-07	Pfizer Products Inc.	Inhibiteurs de la triaryl-oxy-aryl-spiro-pyrimidine-2, 4, 6-trione metalloproteinase
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2001
- 2001-10-23 CN CNA018179231A patent/CN1501937A/zh active Pending
- 2001-10-23 AU AU2002210813A patent/AU2002210813A1/en not_active Abandoned
- 2001-10-23 HR HR20030332A patent/HRP20030332A2/hr not_active Application Discontinuation
- 2001-10-23 CZ CZ20031083A patent/CZ20031083A3/cs unknown
- 2001-10-23 EE EEP200300196A patent/EE200300196A/xx unknown
- 2001-10-23 SK SK497-2003A patent/SK4972003A3/sk unknown
- 2001-10-23 OA OA1200300123A patent/OA12529A/en unknown
- 2001-10-23 AP APAP/P/2001/002318A patent/AP2001002318A0/en unknown
- 2001-10-23 MX MXPA03003735A patent/MXPA03003735A/es unknown
- 2001-10-23 IL IL15494801A patent/IL154948A0/xx unknown
- 2001-10-23 WO PCT/IB2001/001986 patent/WO2002034753A2/fr not_active Ceased
- 2001-10-23 EP EP01978721A patent/EP1332146A2/fr not_active Withdrawn
- 2001-10-23 KR KR10-2003-7005753A patent/KR20040004412A/ko not_active Ceased
- 2001-10-23 PL PL01366201A patent/PL366201A1/xx not_active Application Discontinuation
- 2001-10-23 JP JP2002537743A patent/JP2004518635A/ja not_active Withdrawn
- 2001-10-23 BR BR0114913-0A patent/BR0114913A/pt not_active IP Right Cessation
- 2001-10-23 HU HU0301577A patent/HUP0301577A3/hu unknown
- 2001-10-23 EA EA200300306A patent/EA005762B1/ru not_active IP Right Cessation
- 2001-10-23 CA CA002425283A patent/CA2425283A1/fr not_active Abandoned
- 2001-10-24 HN HN2001000244A patent/HN2001000244A/es unknown
- 2001-10-24 AR ARP010104977A patent/AR035069A1/es unknown
- 2001-10-25 TN TNTNSN01149A patent/TNSN01149A1/fr unknown
- 2001-10-25 SV SV2001000705A patent/SV2003000705A/es unknown
- 2001-10-25 PE PE2001001060A patent/PE20020589A1/es not_active Application Discontinuation
- 2001-10-25 GT GT200100213A patent/GT200100213A/es unknown
- 2001-10-26 PA PA20018531401A patent/PA8531401A1/es unknown
2003
- 2003-03-19 ZA ZA200302190A patent/ZA200302190B/en unknown
- 2003-03-20 BG BG107653A patent/BG107653A/bg unknown
- 2003-03-27 IS IS6762A patent/IS6762A/is unknown
- 2003-04-22 MA MA27117A patent/MA26957A1/fr unknown
- 2003-04-24 NO NO20031853A patent/NO20031853L/no not_active Application Discontinuation
- 2003-04-25 EC EC2003004567A patent/ECSP034567A/es unknown

Also Published As

Publication number	Publication date
CN1501937A (zh)	2004-06-02
WO2002034753A2 (fr)	2002-05-02
NO20031853D0 (no)	2003-04-24
KR20040004412A (ko)	2004-01-13
EA005762B1 (ru)	2005-06-30
ECSP034567A (es)	2003-06-25
MA26957A1 (fr)	2004-12-20
EE200300196A (et)	2003-10-15
BR0114913A (pt)	2003-07-01
PE20020589A1 (es)	2002-07-06
WO2002034753A3 (fr)	2002-08-15
ZA200302190B (en)	2004-04-28
IL154948A0 (en)	2003-10-31
MXPA03003735A (es)	2003-07-28
NO20031853L (no)	2003-06-23
PL366201A1 (en)	2005-01-24
EA200300306A1 (ru)	2003-08-28
HUP0301577A3 (en)	2006-02-28
PA8531401A1 (es)	2003-06-30
GT200100213A (es)	2002-07-03
AU2002210813A1 (en)	2002-05-06
TNSN01149A1 (fr)	2005-11-10
HUP0301577A2 (hu)	2003-11-28
CA2425283A1 (fr)	2002-05-02
IS6762A (is)	2003-03-27
SK4972003A3 (en)	2004-05-04
SV2003000705A (es)	2003-01-13
OA12529A (en)	2006-06-02
AR035069A1 (es)	2004-04-14
EP1332146A2 (fr)	2003-08-06
AP2001002318A0 (en)	2001-12-31
BG107653A (bg)	2003-12-31
HRP20030332A2 (en)	2003-06-30
HN2001000244A (es)	2003-11-07
JP2004518635A (ja)	2004-06-24

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