HUP0301577A3 - Spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors, pharmaceutical compositions containing them and their use - Google Patents

Spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors, pharmaceutical compositions containing them and their use

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Publication number
HUP0301577A3
HUP0301577A3 HU0301577A HUP0301577A HUP0301577A3 HU P0301577 A3 HUP0301577 A3 HU P0301577A3 HU 0301577 A HU0301577 A HU 0301577A HU P0301577 A HUP0301577 A HU P0301577A HU P0301577 A3 HUP0301577 A3 HU P0301577A3
Authority
HU
Hungary
Prior art keywords
spiro
pyrimidine
pharmaceutical compositions
compositions containing
metalloproteinase inhibitors
Prior art date
Application number
HU0301577A
Other languages
English (en)
Hungarian (hu)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HUP0301577A2 publication Critical patent/HUP0301577A2/hu
Publication of HUP0301577A3 publication Critical patent/HUP0301577A3/hu

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10Spiro-condensed systems
    • AHUMAN NECESSITIES
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  • Health & Medical Sciences (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
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  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Communicable Diseases (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Cardiology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Virology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
HU0301577A 2000-10-26 2001-10-23 Spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors, pharmaceutical compositions containing them and their use HUP0301577A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24338900P 2000-10-26 2000-10-26
PCT/IB2001/001986 WO2002034753A2 (fr) 2000-10-26 2001-10-23 Inhibiteurs de metalloproteinase spiro-pyrimidine-2,4,6-trione

Publications (2)

Publication Number Publication Date
HUP0301577A2 HUP0301577A2 (hu) 2003-11-28
HUP0301577A3 true HUP0301577A3 (en) 2006-02-28

Family

ID=22918584

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0301577A HUP0301577A3 (en) 2000-10-26 2001-10-23 Spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors, pharmaceutical compositions containing them and their use

Country Status (32)

Country Link
EP (1) EP1332146A2 (fr)
JP (1) JP2004518635A (fr)
KR (1) KR20040004412A (fr)
CN (1) CN1501937A (fr)
AP (1) AP2001002318A0 (fr)
AR (1) AR035069A1 (fr)
AU (1) AU2002210813A1 (fr)
BG (1) BG107653A (fr)
BR (1) BR0114913A (fr)
CA (1) CA2425283A1 (fr)
CZ (1) CZ20031083A3 (fr)
EA (1) EA005762B1 (fr)
EC (1) ECSP034567A (fr)
EE (1) EE200300196A (fr)
GT (1) GT200100213A (fr)
HN (1) HN2001000244A (fr)
HR (1) HRP20030332A2 (fr)
HU (1) HUP0301577A3 (fr)
IL (1) IL154948A0 (fr)
IS (1) IS6762A (fr)
MA (1) MA26957A1 (fr)
MX (1) MXPA03003735A (fr)
NO (1) NO20031853L (fr)
OA (1) OA12529A (fr)
PA (1) PA8531401A1 (fr)
PE (1) PE20020589A1 (fr)
PL (1) PL366201A1 (fr)
SK (1) SK4972003A3 (fr)
SV (1) SV2003000705A (fr)
TN (1) TNSN01149A1 (fr)
WO (1) WO2002034753A2 (fr)
ZA (1) ZA200302190B (fr)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DOP2002000332A (es) 2001-02-14 2002-08-30 Warner Lambert Co Inhibidores de piridina de metaloproteinasas de la matriz
WO2002064571A1 (fr) 2001-02-14 2002-08-22 Warner-Lambert Company Llc Pyrimidine comme inhibiteurs de la métalloprotéinase de matrice
BR0207865A (pt) 2001-02-14 2004-03-23 Warner Lambert Co Benzotiadiazinas inibidores de metaloproteinases de matriz
DOP2002000333A (es) 2001-02-14 2002-09-30 Warner Lambert Co Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
PA8539501A1 (es) 2001-02-14 2002-09-30 Warner Lambert Co Compuestos triazolo como inhibidores de mmp
US6924276B2 (en) 2001-09-10 2005-08-02 Warner-Lambert Company Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
BR0213233A (pt) 2001-10-12 2005-01-04 Warner Lambert Co Alcinos inibidores de metaloproteinase de matriz
US6962922B2 (en) 2001-10-12 2005-11-08 Warner-Lambert Company Llc Alkynylated quinazoline compounds
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