CZ206599A3 - Benzothiofenkarboxamidové deriváty a antagonisty PGD2, které je obsahují - Google Patents

Benzothiofenkarboxamidové deriváty a antagonisty PGD2, které je obsahují Download PDF

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Publication number
CZ206599A3
CZ206599A3 CZ992065A CZ206599A CZ206599A3 CZ 206599 A3 CZ206599 A3 CZ 206599A3 CZ 992065 A CZ992065 A CZ 992065A CZ 206599 A CZ206599 A CZ 206599A CZ 206599 A3 CZ206599 A3 CZ 206599A3
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CZ
Czechia
Prior art keywords
pgd
cables
antagonists containing
cable
benzothiophenecarboxamide
Prior art date
Application number
CZ992065A
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English (en)
Other versions
CZ297324B6 (cs
Inventor
Tsunetoshi Honma
Yoshiharu Hiramatsu
Akinori Arimura
Original Assignee
Shionogi & Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co., Ltd. filed Critical Shionogi & Co., Ltd.
Publication of CZ206599A3 publication Critical patent/CZ206599A3/cs
Publication of CZ297324B6 publication Critical patent/CZ297324B6/cs

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Description

Zařízení pro ochranu přebytečných délek připojovacích a spojovacích kabelů.
Oblast techniky
Vynález se týká oboru spotřebního průmyslu.
Dosavadní stav techniky
V současné době přebytečné délky připojovacích a spojovacích kabelů volně leží na stolech či podlaze domácností a kanceláří. Zřízení pro jejich ochranu není nikde v obchodní síti ani v katalogách zahraničních sítí obchodní či zásilkových společností.
Podstata vynálezu
Nevýhodu volně ležících kabelů odstraní zařízení jehož podstata spočívá v tom, že přebytečná délka připojovacího nebo propojovacího kabelu se navine do schránky.
V této schránce je kabel chráněn proti poškození, jetím umožněn úklid míst kde původně ležel přebytečný kabel a zlepší se vzhled prostoru. Zařízení umožňuje navinout kabely i bez rozpojení kabelů. Zařízení je možné vyrobit v různých velikostech dle síly kabelů a je možné je sestavovat v bloky o různém počtu jednotlivých zařízení.
Přehled obrázků na výkresu
Příklad provedení vynálezu je blíže znázorněn na schematickém výkresu znázorňujícím nárys a bokorys zařízení v řezech.
Příklad provedení vynálezu
Zařízení se skládá z pláště L, který má na obvodě otvor pro vsunutí smyčky kabelu 5^
Při otáčení vnitřního bubínku 2 pomocí tyčky 3 zachytí kolíček 4 ,který je spojen s bubínkem 2 , za vsunutou smyčku kabelu a začne vtahovat a navíjet kabel do schránky L Otáčení se provádí tak dlouho až žádná přebytečná délka kabelu neleží zbytečně mimo zařízení. Jednotlivá zařízení, která mohou být vybavena držáky 6 , lze zasunout do lišt 7 a sestavovat vedle sebe v neomezeném počtu.

Claims (1)

  1. PATENTOVÉ NÁROKY
    Zařízení pro ochranu přebytečných délek připojovacích a spojovacích kabelů skládající se ze schránky a navíjecího mechanismu je význačné tím, že umožňuje navinout kabely i bez rozpojení a je dále význačné tím, že umožňuje použití, jak samostatně, tak sestaveno v blocích.
CZ0206599A 1996-12-13 1997-12-10 Benzothiofenkarboxamidové deriváty a antagonisty PGD2, které je obsahují CZ297324B6 (cs)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP33349596 1996-12-13
JP25400197 1997-09-19

Publications (2)

Publication Number Publication Date
CZ206599A3 true CZ206599A3 (cs) 1999-11-17
CZ297324B6 CZ297324B6 (cs) 2006-11-15

Family

ID=26541496

Family Applications (1)

Application Number Title Priority Date Filing Date
CZ0206599A CZ297324B6 (cs) 1996-12-13 1997-12-10 Benzothiofenkarboxamidové deriváty a antagonisty PGD2, které je obsahují

Country Status (25)

Country Link
US (1) US6083974A (cs)
EP (1) EP0944614B1 (cs)
JP (1) JP3215441B2 (cs)
KR (1) KR100433568B1 (cs)
CN (2) CN1105112C (cs)
AR (1) AR008939A1 (cs)
AT (1) ATE223911T1 (cs)
AU (1) AU718958B2 (cs)
BR (1) BR9714016A (cs)
CA (1) CA2274591C (cs)
CZ (1) CZ297324B6 (cs)
DE (1) DE69715448T2 (cs)
DK (1) DK0944614T3 (cs)
ES (1) ES2181039T3 (cs)
HU (1) HU226458B1 (cs)
ID (1) ID22753A (cs)
IL (1) IL130660A (cs)
NO (1) NO992838L (cs)
NZ (1) NZ336143A (cs)
PL (1) PL191760B1 (cs)
PT (1) PT944614E (cs)
RU (1) RU2161617C1 (cs)
TR (1) TR199901280T2 (cs)
TW (1) TW438790B (cs)
WO (1) WO1998025919A1 (cs)

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AR038136A1 (es) 2002-01-24 2004-12-29 Merck Frosst Canada Inc Cicloalcanindoles con sustitucion con fluor composiciones que contienen estos compuestos y metodos de tratamiento
CN100378083C (zh) 2002-03-19 2008-04-02 小野药品工业株式会社 羧酸化合物和含有所述化合物作为活性成分的药物制剂
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TWI532737B (zh) 2010-06-30 2016-05-11 艾諾屋製藥公司 可溶性鳥苷酸環化酶(sGC)刺激物
US20130259830A1 (en) 2010-07-12 2013-10-03 Ironwood Pharmaceuticals, Inc. Crth2 modulators
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CA2861804C (en) 2011-12-27 2021-10-26 Ironwood Pharmaceuticals, Inc. 2-benzyl,3(pyrimidin-2-yl)substituted pyrazoles useful as sgc stimulators
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Also Published As

Publication number Publication date
US6083974A (en) 2000-07-04
PL191760B1 (pl) 2006-06-30
HUP0002869A3 (en) 2003-01-28
AU5409798A (en) 1998-07-03
HK1020045A1 (en) 2000-03-10
CN1240438A (zh) 2000-01-05
ATE223911T1 (de) 2002-09-15
KR100433568B1 (ko) 2004-05-31
ID22753A (id) 1999-12-09
CA2274591A1 (en) 1998-06-18
AU718958B2 (en) 2000-05-04
KR20000069402A (ko) 2000-11-25
TR199901280T2 (xx) 1999-10-21
DK0944614T3 (da) 2003-01-13
IL130660A0 (en) 2000-06-01
EP0944614A1 (en) 1999-09-29
HUP0002869A2 (hu) 2001-06-28
CZ297324B6 (cs) 2006-11-15
AR008939A1 (es) 2000-02-23
TW438790B (en) 2001-06-07
CN1445225A (zh) 2003-10-01
RU2161617C1 (ru) 2001-01-10
EP0944614B1 (en) 2002-09-11
CN1105112C (zh) 2003-04-09
JP2000514824A (ja) 2000-11-07
DE69715448T2 (de) 2003-08-07
CA2274591C (en) 2005-06-14
NO992838D0 (no) 1999-06-10
HU226458B1 (en) 2008-12-29
PT944614E (pt) 2003-01-31
NZ336143A (en) 2002-05-31
WO1998025919A1 (en) 1998-06-18
JP3215441B2 (ja) 2001-10-09
IL130660A (en) 2002-03-10
PL334072A1 (en) 2000-01-31
NO992838L (no) 1999-07-20
BR9714016A (pt) 2000-02-29
CN1185226C (zh) 2005-01-19
ES2181039T3 (es) 2003-02-16
DE69715448D1 (de) 2002-10-17

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MM4A Patent lapsed due to non-payment of fee

Effective date: 20091210