CZ206599A3 - Benzothiofenkarboxamidové deriváty a antagonisty PGD2, které je obsahují - Google Patents
Benzothiofenkarboxamidové deriváty a antagonisty PGD2, které je obsahují Download PDFInfo
- Publication number
- CZ206599A3 CZ206599A3 CZ992065A CZ206599A CZ206599A3 CZ 206599 A3 CZ206599 A3 CZ 206599A3 CZ 992065 A CZ992065 A CZ 992065A CZ 206599 A CZ206599 A CZ 206599A CZ 206599 A3 CZ206599 A3 CZ 206599A3
- Authority
- CZ
- Czechia
- Prior art keywords
- pgd
- cables
- antagonists containing
- cable
- benzothiophenecarboxamide
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Ophthalmology & Optometry (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Indole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Description
Zařízení pro ochranu přebytečných délek připojovacích a spojovacích kabelů.
Oblast techniky
Vynález se týká oboru spotřebního průmyslu.
Dosavadní stav techniky
V současné době přebytečné délky připojovacích a spojovacích kabelů volně leží na stolech či podlaze domácností a kanceláří. Zřízení pro jejich ochranu není nikde v obchodní síti ani v katalogách zahraničních sítí obchodní či zásilkových společností.
Podstata vynálezu
Nevýhodu volně ležících kabelů odstraní zařízení jehož podstata spočívá v tom, že přebytečná délka připojovacího nebo propojovacího kabelu se navine do schránky.
V této schránce je kabel chráněn proti poškození, jetím umožněn úklid míst kde původně ležel přebytečný kabel a zlepší se vzhled prostoru. Zařízení umožňuje navinout kabely i bez rozpojení kabelů. Zařízení je možné vyrobit v různých velikostech dle síly kabelů a je možné je sestavovat v bloky o různém počtu jednotlivých zařízení.
Přehled obrázků na výkresu
Příklad provedení vynálezu je blíže znázorněn na schematickém výkresu znázorňujícím nárys a bokorys zařízení v řezech.
Příklad provedení vynálezu
Zařízení se skládá z pláště L, který má na obvodě otvor pro vsunutí smyčky kabelu 5^
Při otáčení vnitřního bubínku 2 pomocí tyčky 3 zachytí kolíček 4 ,který je spojen s bubínkem 2 , za vsunutou smyčku kabelu a začne vtahovat a navíjet kabel do schránky L Otáčení se provádí tak dlouho až žádná přebytečná délka kabelu neleží zbytečně mimo zařízení. Jednotlivá zařízení, která mohou být vybavena držáky 6 , lze zasunout do lišt 7 a sestavovat vedle sebe v neomezeném počtu.
Claims (1)
- PATENTOVÉ NÁROKYZařízení pro ochranu přebytečných délek připojovacích a spojovacích kabelů skládající se ze schránky a navíjecího mechanismu je význačné tím, že umožňuje navinout kabely i bez rozpojení a je dále význačné tím, že umožňuje použití, jak samostatně, tak sestaveno v blocích.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP33349596 | 1996-12-13 | ||
| JP25400197 | 1997-09-19 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CZ206599A3 true CZ206599A3 (cs) | 1999-11-17 |
| CZ297324B6 CZ297324B6 (cs) | 2006-11-15 |
Family
ID=26541496
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CZ0206599A CZ297324B6 (cs) | 1996-12-13 | 1997-12-10 | Benzothiofenkarboxamidové deriváty a antagonisty PGD2, které je obsahují |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US6083974A (cs) |
| EP (1) | EP0944614B1 (cs) |
| JP (1) | JP3215441B2 (cs) |
| KR (1) | KR100433568B1 (cs) |
| CN (2) | CN1105112C (cs) |
| AR (1) | AR008939A1 (cs) |
| AT (1) | ATE223911T1 (cs) |
| AU (1) | AU718958B2 (cs) |
| BR (1) | BR9714016A (cs) |
| CA (1) | CA2274591C (cs) |
| CZ (1) | CZ297324B6 (cs) |
| DE (1) | DE69715448T2 (cs) |
| DK (1) | DK0944614T3 (cs) |
| ES (1) | ES2181039T3 (cs) |
| HU (1) | HU226458B1 (cs) |
| ID (1) | ID22753A (cs) |
| IL (1) | IL130660A (cs) |
| NO (1) | NO992838L (cs) |
| NZ (1) | NZ336143A (cs) |
| PL (1) | PL191760B1 (cs) |
| PT (1) | PT944614E (cs) |
| RU (1) | RU2161617C1 (cs) |
| TR (1) | TR199901280T2 (cs) |
| TW (1) | TW438790B (cs) |
| WO (1) | WO1998025919A1 (cs) |
Families Citing this family (38)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2185380C1 (ru) | 1998-03-31 | 2002-07-20 | Сионоги Энд Ко., Лтд. | Способ получения производных бензотиофенкарбоксамида и аминоспиртов (варианты) |
| ID26346A (id) | 1998-03-31 | 2000-12-14 | Shionogi & Co | PROSES PEMBUATAN TURUNAN ASAM 5-HIDROKSIBENZO (b)TIOFEN-3-KARBOKSILAT |
| ES2241283T3 (es) * | 1998-06-03 | 2005-10-16 | SHIONOGI & CO., LTD. | Remedios para el tratamiento del prurito que contienen antagonistas de pgd2. |
| EP1808427A3 (en) * | 1999-07-02 | 2008-06-25 | Shionogi & Co., Ltd. | Novel processes for the preparation of bicyclic aminoalcohols |
| KR20030010589A (ko) | 2000-03-09 | 2003-02-05 | 오노 야꾸힝 고교 가부시키가이샤 | 인돌 유도체, 그 제조 방법 및 용도 |
| ATE311200T1 (de) * | 2000-04-12 | 2005-12-15 | Merck Frosst Canada Inc | Verfahren und zusammensetzungen zur behandlung von allergischen zuständen mit pgd2 rezeptor antagonisten |
| US6410583B1 (en) * | 2000-07-25 | 2002-06-25 | Merck Frosst Canada & Co. | Cyclopentanoindoles, compositions containing such compounds and methods of treatment |
| US7273883B2 (en) | 2000-09-14 | 2007-09-25 | Allergan, Inc. | Prostaglandin EP4 antagonist |
| US7217725B2 (en) | 2000-09-14 | 2007-05-15 | Allergan, Inc. | Prostaglandin D2 antagonist |
| WO2002032892A1 (en) * | 2000-10-17 | 2002-04-25 | Shionogi & Co., Ltd | Process for the preparation of pgd2 antagonist |
| JPWO2002036583A1 (ja) * | 2000-11-01 | 2004-03-11 | 塩野義製薬株式会社 | Pgd2受容体拮抗性医薬組成物 |
| AR038136A1 (es) | 2002-01-24 | 2004-12-29 | Merck Frosst Canada Inc | Cicloalcanindoles con sustitucion con fluor composiciones que contienen estos compuestos y metodos de tratamiento |
| CN100378083C (zh) | 2002-03-19 | 2008-04-02 | 小野药品工业株式会社 | 羧酸化合物和含有所述化合物作为活性成分的药物制剂 |
| JPWO2004006956A1 (ja) * | 2002-07-12 | 2005-11-10 | 独立行政法人科学技術振興機構 | 脳損傷の予後改善薬とそのスクリーニング方法 |
| AU2003242485A1 (en) * | 2002-09-30 | 2004-04-23 | Shionogi And Co., Ltd. | Novel uses of prostaglandin d2, prostaglandin d2 agonist and prostaglandin d2 antagonist |
| EP1558614B1 (en) | 2002-10-30 | 2010-09-01 | Merck Frosst Canada Ltd. | Pyridopyrrolizine and pyridoindolizine derivatives |
| JP4051398B2 (ja) | 2004-03-11 | 2008-02-20 | アクテリオン ファマシューティカルズ リミテッド | テトラヒドロピリドインドール誘導体 |
| JPWO2006068162A1 (ja) * | 2004-12-24 | 2008-06-12 | 塩野義製薬株式会社 | 慢性閉塞性肺疾患の治療剤 |
| TW200716093A (en) * | 2005-04-28 | 2007-05-01 | Shionogi & Co | An antiasthmatic agent containing PGD2 receptor antagonist and leukotriene receptor antagonist |
| TWI410410B (zh) | 2007-08-10 | 2013-10-01 | Ono Pharmaceutical Co | Phenylacetic acid compounds |
| CN102822163B (zh) | 2009-12-23 | 2016-01-20 | 艾恩伍德医药品股份有限公司 | Crth2调节剂 |
| US20130178475A1 (en) | 2010-03-17 | 2013-07-11 | Ironwood Pharmaceuticals, Inc. | sGC STIMULATORS |
| TWI532737B (zh) | 2010-06-30 | 2016-05-11 | 艾諾屋製藥公司 | 可溶性鳥苷酸環化酶(sGC)刺激物 |
| US20130259830A1 (en) | 2010-07-12 | 2013-10-03 | Ironwood Pharmaceuticals, Inc. | Crth2 modulators |
| WO2012009137A1 (en) | 2010-07-12 | 2012-01-19 | Ironwood Pharmaceuticals, Inc. | Crth2 modulators |
| JP5878546B2 (ja) | 2010-11-09 | 2016-03-08 | アイアンウッド ファーマシューティカルズ インコーポレイテッド | sGC刺激剤 |
| CA2861804C (en) | 2011-12-27 | 2021-10-26 | Ironwood Pharmaceuticals, Inc. | 2-benzyl,3(pyrimidin-2-yl)substituted pyrazoles useful as sgc stimulators |
| WO2014047111A1 (en) | 2012-09-18 | 2014-03-27 | Ironwood Pharmaceuticals, Inc. | Sgc stimulators |
| EP2897953B8 (en) | 2012-09-19 | 2019-06-26 | Cyclerion Therapeutics, Inc. | Sgc stimulators |
| ES2911276T3 (es) | 2013-03-15 | 2022-05-18 | Cyclerion Therapeutics Inc | Estimuladores de sGC |
| JP2016540017A (ja) | 2013-12-11 | 2016-12-22 | アイアンウッド ファーマシューティカルズ インコーポレイテッド | sGC刺激物質 |
| WO2015106268A1 (en) | 2014-01-13 | 2015-07-16 | Ironwood Pharmaceuticals, Inc. | USE OF sGC STIMULATORS FOR THE TREATMENT OF NEUROMUSCULAR DISORDERS |
| EP3194382B1 (en) | 2014-09-17 | 2021-09-08 | Cyclerion Therapeutics, Inc. | Pyrazole derivatives as sgc stimulators |
| WO2016044445A2 (en) | 2014-09-17 | 2016-03-24 | Ironwood Pharmaceuticals, Inc. | sGC STIMULATORS |
| US10844064B2 (en) | 2014-09-17 | 2020-11-24 | Cyclerion Therapeutics, Inc. | sGC stimulators |
| JP6770522B2 (ja) | 2015-02-13 | 2020-10-14 | アンスティチュ ナショナル ドゥ ラ サンテ エ ドゥ ラ ルシェルシュ メディカル | 全身性エリテマトーデスを予防し、及び/又は、治療するためのptgdr−1及び/又はptgdr−2アンタゴニスト |
| KR102513343B1 (ko) | 2016-07-07 | 2023-03-22 | 사이클리온 테라퓨틱스, 인크. | sGC 자극제의 인 전구약물 |
| EA039753B1 (ru) | 2016-07-07 | 2022-03-10 | Сайклерион Терапьютикс, Инк. | ТВЕРДЫЕ ФОРМЫ СТИМУЛЯТОРА sGC |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8406906D0 (en) * | 1984-03-16 | 1984-04-18 | Akzo Nv | Benzo-thiazole and benzothiophene derivatives |
| US4560343A (en) * | 1984-06-11 | 1985-12-24 | Honeywell Inc. | Functional check for a hot surface ignitor element |
| JPS6149A (ja) * | 1984-06-12 | 1986-01-06 | Ono Pharmaceut Co Ltd | 新規な13―アザ―14―オキソ―TxA2類似化合物およびそれらを有効成分として含有するトロンボキサン起因疾患治療剤 |
| NZ218115A (en) * | 1985-11-18 | 1990-02-26 | Shionogi & Co | Bicyclic sulphonamides and pharmaceutical compositions |
| CA1294974C (en) * | 1987-05-08 | 1992-01-28 | Sanji Hagishita | Bicyclic sulfonamide derivatives and process therefor |
| US5356926A (en) * | 1992-02-24 | 1994-10-18 | Warner-Lambert Company | 3-alkyloxy-, aryloxy-, or arylalkyloxy-benzo [β]thiophene-2-carboxamides as inhibitors of cell adhesion |
| CA2113787A1 (en) * | 1993-01-29 | 1994-07-30 | Nobuyuki Hamanaka | Carbocyclic sulfonamides |
| DE4317076A1 (de) * | 1993-05-21 | 1994-11-24 | Bayer Ag | Benzthiophencarbonsäureamid-S-oxide |
| US5863936A (en) * | 1995-04-18 | 1999-01-26 | Geron Corporation | Telomerase inhibitors |
| PL185107B1 (pl) * | 1995-06-21 | 2003-02-28 | Shionogi & Co | Bicykliczne związki aminowe, kompozycja farmaceutyczna i jej stosowanie |
| JP2001501946A (ja) * | 1996-10-08 | 2001-02-13 | イーライ・リリー・アンド・カンパニー | 新規セロトニン5―ht▲下1f▼アゴニスト |
-
1997
- 1997-12-10 BR BR9714016-3A patent/BR9714016A/pt active Search and Examination
- 1997-12-10 AU AU54097/98A patent/AU718958B2/en not_active Ceased
- 1997-12-10 KR KR10-1999-7005154A patent/KR100433568B1/ko not_active Expired - Fee Related
- 1997-12-10 PL PL334072A patent/PL191760B1/pl not_active IP Right Cessation
- 1997-12-10 EP EP97947866A patent/EP0944614B1/en not_active Expired - Lifetime
- 1997-12-10 DK DK97947866T patent/DK0944614T3/da active
- 1997-12-10 NZ NZ336143A patent/NZ336143A/en unknown
- 1997-12-10 HU HU0002869A patent/HU226458B1/hu not_active IP Right Cessation
- 1997-12-10 DE DE69715448T patent/DE69715448T2/de not_active Expired - Lifetime
- 1997-12-10 PT PT97947866T patent/PT944614E/pt unknown
- 1997-12-10 JP JP52649298A patent/JP3215441B2/ja not_active Expired - Fee Related
- 1997-12-10 US US09/308,176 patent/US6083974A/en not_active Expired - Lifetime
- 1997-12-10 ES ES97947866T patent/ES2181039T3/es not_active Expired - Lifetime
- 1997-12-10 CA CA002274591A patent/CA2274591C/en not_active Expired - Fee Related
- 1997-12-10 WO PCT/JP1997/004527 patent/WO1998025919A1/en not_active Ceased
- 1997-12-10 AT AT97947866T patent/ATE223911T1/de not_active IP Right Cessation
- 1997-12-10 IL IL13066097A patent/IL130660A/en not_active IP Right Cessation
- 1997-12-10 CZ CZ0206599A patent/CZ297324B6/cs not_active IP Right Cessation
- 1997-12-10 RU RU99115766/04A patent/RU2161617C1/ru not_active IP Right Cessation
- 1997-12-10 TR TR1999/01280T patent/TR199901280T2/xx unknown
- 1997-12-10 ID IDW990472A patent/ID22753A/id unknown
- 1997-12-10 CN CN97180628A patent/CN1105112C/zh not_active Expired - Fee Related
- 1997-12-11 TW TW086118667A patent/TW438790B/zh not_active IP Right Cessation
- 1997-12-12 AR ARP970105862A patent/AR008939A1/es active IP Right Grant
-
1999
- 1999-06-10 NO NO992838A patent/NO992838L/no unknown
-
2002
- 2002-06-11 CN CNB021227608A patent/CN1185226C/zh not_active Expired - Fee Related
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PD00 | Pending as of 2000-06-30 in czech republic | ||
| MM4A | Patent lapsed due to non-payment of fee |
Effective date: 20091210 |