DK1212321T3 - Mellemprodukter til fremstilling af quinolone carboxylsyrederivater - Google Patents

Mellemprodukter til fremstilling af quinolone carboxylsyrederivater

Info

Publication number: DK1212321T3
Authority: DK; Denmark
Prior art keywords: intermediates; preparation; carboxylic acid; acid derivatives; quinolone carboxylic
Prior art date: 1999-09-03

Application number

DK00956706T

Other languages

English (en)

Inventor

Trevor John Grinter

Simon Howie

Original Assignee

Lg Life Sciences Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-09-03

Filing date

2000-09-01

Publication date

2004-10-25

2000-09-01 Application filed by Lg Life Sciences Ltd filed Critical Lg Life Sciences Ltd

2004-10-25 Application granted granted Critical

2004-10-25 Publication of DK1212321T3 publication Critical patent/DK1212321T3/da

Links

XOQQVKDBGLYPGH-UHFFFAOYSA-N 2-oxo-1h-quinoline-3-carboxylic acid Chemical class C1=CC=C2NC(=O)C(C(=O)O)=CC2=C1 XOQQVKDBGLYPGH-UHFFFAOYSA-N 0.000 title 1
239000000543 intermediate Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pyrrole Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

DK00956706T 1999-09-03 2000-09-01 Mellemprodukter til fremstilling af quinolone carboxylsyrederivater DK1212321T3 (da)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GBGB9920919.9A GB9920919D0 (en)	1999-09-03	1999-09-03	Novel compound
EP00956706A EP1212321B1 (en)	1999-09-03	2000-09-01	Intermediates for the production of naphthyridine-3-carboxylic acid derivatives
PCT/GB2000/003358 WO2001017961A2 (en)	1999-09-03	2000-09-01	Intermediates for the production of naphthyridine-3-carboxylic acid derivatives

Publications (1)

Publication Number	Publication Date
DK1212321T3 true DK1212321T3 (da)	2004-10-25

Family

ID=10860355

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK00956706T DK1212321T3 (da)	1999-09-03	2000-09-01	Mellemprodukter til fremstilling af quinolone carboxylsyrederivater

Country Status (30)

Country	Link
US (3)	US6703512B1 (da)
EP (1)	EP1212321B1 (da)
JP (1)	JP4208463B2 (da)
KR (1)	KR100705363B1 (da)
CN (1)	CN1255402C (da)
AR (1)	AR029452A1 (da)
AT (1)	ATE270671T1 (da)
AU (1)	AU773698B2 (da)
BR (1)	BRPI0013750B8 (da)
CA (1)	CA2383751C (da)
CO (1)	CO5180620A1 (da)
CZ (1)	CZ2002759A3 (da)
DE (1)	DE60012028T2 (da)
DK (1)	DK1212321T3 (da)
ES (1)	ES2223570T3 (da)
GB (1)	GB9920919D0 (da)
HK (1)	HK1046908B (da)
HU (1)	HU229391B1 (da)
IL (2)	IL148441A0 (da)
MX (1)	MXPA02002356A (da)
MY (1)	MY126789A (da)
NO (1)	NO322501B1 (da)
NZ (1)	NZ517601A (da)
PL (1)	PL206491B1 (da)
PT (1)	PT1212321E (da)
SI (1)	SI1212321T1 (da)
TR (1)	TR200200548T2 (da)
TW (1)	TWI264435B (da)
WO (1)	WO2001017961A2 (da)
ZA (1)	ZA200201779B (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
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CA2281817C (en) *	1999-06-29	2008-07-29	Smithkline Beecham Corporation	Methods of use of fluoroquinolone compounds against maxillary sinus pathogenic bacteria
GB9920917D0 (en)	1999-09-03	1999-11-10	Sb Pharmco Inc	Novel process
GB9920919D0 (en)	1999-09-03	1999-11-10	Sb Pharmco Inc	Novel compound
PT1412078E (pt)	2001-08-02	2009-01-08	Lg Life Sciences Ltd	Processos para a produção de derivados amino-protegidos da 4- aminometileno-pirrolidin-3-ona, gemifloxacina ou um seu sal
KR100517638B1 (ko)	2002-04-08	2005-09-28	주식회사 엘지생명과학	게미플록사신 산염의 새로운 제조방법
ATE310773T1 (de) *	2002-07-17	2005-12-15	Ciba Sc Holding Ag	Oxidationsverfahren zur herstellung von chinacridonpigmenten
KR100653334B1 (ko)	2003-03-07	2006-12-04	주식회사 엘지생명과학	4-아미노메틸-3-알콕시이미노피롤리딘 메탄설폰산염의 신규한 제조 방법
US8822934B2 (en) *	2006-11-03	2014-09-02	Accuray Incorporated	Collimator changer
CN104693088B (zh) *	2013-12-06	2018-01-05	常州市勇毅生物药业有限公司	一种吉米沙星侧链的制备方法

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JPH0356479A (ja)	1989-07-24	1991-03-12	Takeshi Yokota	水溶性キノロン誘導体のｐ‐トルエンスルホン酸塩
RU2049777C1 (ru)	1989-08-16	1995-12-10	Пфайзер Инк.	Азабицикло-хинолон-карбоновые кислоты или их фармацевтически приемлемые кислотно-аддитивные соли и промежуточные продукты для их получения
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JPH0673056A (ja)	1992-08-26	1994-03-15	Kaken Pharmaceut Co Ltd	キノリンカルボン酸誘導体およびその塩
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JP3449658B2 (ja)	1994-12-21	2003-09-22	杏林製薬株式会社	安定性に優れた８−アルコキシキノロンカルボン酸水和物並びにその製造方法
JP3145715B2 (ja)	1995-06-06	2001-03-12	ファイザー・インコーポレーテッド	無水７−（［１α，５α，６α］−６−アミノ−３−アザビシクロ［３．１．０］ヘキサ−３−イル）−６−フルオロ−１−（２，４−ジフルオロフェニル）−１，４−ジヒドロ−４−オキソ−１，８−ナフチリディン−３−カルボン酸メタンスルホン酸塩の新規な結晶形態
ATE215072T1 (de)	1995-08-11	2002-04-15	Pfizer	(1s,2s)-1-(4-hydroxyphenyl)-2-(4-hydroxy-4- phenylpiperidin-1-yl)-1-propanol-methansulfonat trihydrat
AR006439A1 (es)	1996-03-29	1999-08-25	Smithkline Beecham Corp	Dihidrato de eprosartano y un procedimiento para su produccion y formulacion
MA24500A1 (fr) *	1997-03-21	1998-10-01	Lg Life Sciences Ltd	Derive du sel d'acide carboxylique de naphthyridine .
KR100286874B1 (ko)	1998-03-04	2001-04-16	성재갑	보호된 4-아미노메틸-피롤리딘-3-온의 제조방법
PT1082300E (pt)	1998-05-29	2004-02-27	Upjohn Co	Monometanossulfonato de 3-¬(1'-n-metilamino)etil-n-benzil\|pirrolidina
GB9820405D0 (en)	1998-09-18	1998-11-11	Smithkline Beecham Plc	Process
PT1223935E (pt)	1999-06-29	2008-04-03	Lg Life Sciences Ltd	Utilização de compostos de gemifloxacina contra bactérias
AU6947900A (en)	1999-09-01	2001-03-26	Smithkline Beecham Corporation	Methods of use of fluoroquinolone compounds against bacteria
GB9920919D0 (en)	1999-09-03	1999-11-10	Sb Pharmco Inc	Novel compound
GB9920917D0 (en)	1999-09-03	1999-11-10	Sb Pharmco Inc	Novel process
EP1242079A4 (en)	1999-09-22	2003-01-22	Smithkline Beecham	Methods of anti-bacterial use of fluoroquinolonic compounds
KR20010091379A (ko)	2000-03-15	2001-10-23	성재갑	7-(4-아미노메틸-3-옥심)피롤리딘 치환체를 갖는 퀴놀린카르복실산 유도체의 신규 제조방법
KR20020018560A (ko)	2000-09-01	2002-03-08	성재갑	3-아미노메틸-4-ｚ-메톡시이미노피롤리딘의 신규 제조방법

1999
- 1999-09-03 GB GBGB9920919.9A patent/GB9920919D0/en not_active Ceased
2000
- 2000-09-01 AT AT00956706T patent/ATE270671T1/de active
- 2000-09-01 TR TR2002/00548T patent/TR200200548T2/xx unknown
- 2000-09-01 HK HK02108460.2A patent/HK1046908B/en not_active IP Right Cessation
- 2000-09-01 CZ CZ2002759A patent/CZ2002759A3/cs unknown
- 2000-09-01 KR KR1020027002876A patent/KR100705363B1/ko not_active Expired - Lifetime
- 2000-09-01 AU AU68573/00A patent/AU773698B2/en not_active Ceased
- 2000-09-01 US US10/088,149 patent/US6703512B1/en not_active Expired - Lifetime
- 2000-09-01 DE DE60012028T patent/DE60012028T2/de not_active Expired - Lifetime
- 2000-09-01 ES ES00956706T patent/ES2223570T3/es not_active Expired - Lifetime
- 2000-09-01 PT PT00956706T patent/PT1212321E/pt unknown
- 2000-09-01 CA CA2383751A patent/CA2383751C/en not_active Expired - Lifetime
- 2000-09-01 HU HU0202733A patent/HU229391B1/hu not_active IP Right Cessation
- 2000-09-01 CN CNB008123292A patent/CN1255402C/zh not_active Expired - Lifetime
- 2000-09-01 JP JP2001521708A patent/JP4208463B2/ja not_active Expired - Fee Related
- 2000-09-01 IL IL14844100A patent/IL148441A0/xx active IP Right Grant
- 2000-09-01 EP EP00956706A patent/EP1212321B1/en not_active Expired - Lifetime
- 2000-09-01 MY MYPI20004053 patent/MY126789A/en unknown
- 2000-09-01 NZ NZ517601A patent/NZ517601A/en not_active IP Right Cessation
- 2000-09-01 WO PCT/GB2000/003358 patent/WO2001017961A2/en not_active Ceased
- 2000-09-01 SI SI200030481T patent/SI1212321T1/xx unknown
- 2000-09-01 BR BRPI0013750A patent/BRPI0013750B8/pt not_active IP Right Cessation
- 2000-09-01 DK DK00956706T patent/DK1212321T3/da active
- 2000-09-01 CO CO00065923A patent/CO5180620A1/es active IP Right Grant
- 2000-09-01 MX MXPA02002356A patent/MXPA02002356A/es active IP Right Grant
- 2000-09-01 AR ARP000104596A patent/AR029452A1/es active IP Right Grant
- 2000-09-01 PL PL354725A patent/PL206491B1/pl not_active IP Right Cessation
- 2000-09-29 TW TW089120154A patent/TWI264435B/zh not_active IP Right Cessation
2002
- 2002-02-28 IL IL148441A patent/IL148441A/en unknown
- 2002-03-01 NO NO20021043A patent/NO322501B1/no not_active IP Right Cessation
- 2002-03-04 ZA ZA200201779A patent/ZA200201779B/xx unknown
2003
- 2003-12-23 US US10/742,797 patent/US6803467B2/en not_active Expired - Lifetime
2004
- 2004-09-08 US US10/935,357 patent/US20050033064A1/en not_active Abandoned

Also Published As

Publication number	Publication date
CA2383751C (en)	2010-06-29
ES2223570T3 (es)	2005-03-01
NO322501B1 (no)	2006-10-16
WO2001017961A2 (en)	2001-03-15
US6703512B1 (en)	2004-03-09
PT1212321E (pt)	2004-10-29
GB9920919D0 (en)	1999-11-10
IL148441A0 (en)	2002-09-12
DE60012028D1 (de)	2004-08-12
JP2003508517A (ja)	2003-03-04
CN1372558A (zh)	2002-10-02
ZA200201779B (en)	2003-08-27
HUP0202733A3 (en)	2005-12-28
PL354725A1 (en)	2004-02-09
EP1212321B1 (en)	2004-07-07
KR20020041423A (ko)	2002-06-01
HK1046908A1 (en)	2003-01-30
CA2383751A1 (en)	2001-03-15
BR0013750A (pt)	2002-05-21
TWI264435B (en)	2006-10-21
DE60012028T2 (de)	2005-08-18
HUP0202733A2 (hu)	2003-01-28
BRPI0013750B8 (pt)	2021-05-25
AU773698B2 (en)	2004-06-03
NZ517601A (en)	2003-08-29
HK1046908B (en)	2005-05-27
EP1212321A2 (en)	2002-06-12
TR200200548T2 (tr)	2002-09-23
US20040138292A1 (en)	2004-07-15
HU229391B1 (hu)	2013-11-28
NO20021043D0 (no)	2002-03-01
US20050033064A1 (en)	2005-02-10
SI1212321T1 (en)	2004-12-31
CZ2002759A3 (cs)	2002-06-12
BR0013750B1 (pt)	2014-06-17
WO2001017961A3 (en)	2001-09-20
KR100705363B1 (ko)	2007-04-10
NO20021043L (no)	2002-03-01
ATE270671T1 (de)	2004-07-15
MY126789A (en)	2006-10-31
AU6857300A (en)	2001-04-10
CN1255402C (zh)	2006-05-10
CO5180620A1 (es)	2002-07-30
JP4208463B2 (ja)	2009-01-14
IL148441A (en)	2007-03-08
AR029452A1 (es)	2003-07-02
MXPA02002356A (es)	2002-07-30
PL206491B1 (pl)	2010-08-31
US6803467B2 (en)	2004-10-12

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