TR200200548T2 - Kuinolin karbosiklik asit türevlerinin üretimi için ara maddeler - Google Patents

Kuinolin karbosiklik asit türevlerinin üretimi için ara maddeler

Info

Publication number
TR200200548T2
TR200200548T2 TR2002/00548T TR200200548T TR200200548T2 TR 200200548 T2 TR200200548 T2 TR 200200548T2 TR 2002/00548 T TR2002/00548 T TR 2002/00548T TR 200200548 T TR200200548 T TR 200200548T TR 200200548 T2 TR200200548 T2 TR 200200548T2
Authority
TR
Turkey
Prior art keywords
production
acid derivatives
quinoline
intermediates
carbocyclic acid
Prior art date
Application number
TR2002/00548T
Other languages
English (en)
Inventor
John Grinter Trevor
Howie Simon
Original Assignee
Sb Pharmco Puerto Rico Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sb Pharmco Puerto Rico Inc filed Critical Sb Pharmco Puerto Rico Inc
Publication of TR200200548T2 publication Critical patent/TR200200548T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

Antibaktiyarel faaliyeti olan kuinolon karbosiklik asit türevlerinin üretiminde faydali olan kimyasal ara maddeler.
TR2002/00548T 1999-09-03 2000-09-01 Kuinolin karbosiklik asit türevlerinin üretimi için ara maddeler TR200200548T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9920919.9A GB9920919D0 (en) 1999-09-03 1999-09-03 Novel compound

Publications (1)

Publication Number Publication Date
TR200200548T2 true TR200200548T2 (tr) 2002-09-23

Family

ID=10860355

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2002/00548T TR200200548T2 (tr) 1999-09-03 2000-09-01 Kuinolin karbosiklik asit türevlerinin üretimi için ara maddeler

Country Status (30)

Country Link
US (3) US6703512B1 (tr)
EP (1) EP1212321B1 (tr)
JP (1) JP4208463B2 (tr)
KR (1) KR100705363B1 (tr)
CN (1) CN1255402C (tr)
AR (1) AR029452A1 (tr)
AT (1) ATE270671T1 (tr)
AU (1) AU773698B2 (tr)
BR (1) BRPI0013750B8 (tr)
CA (1) CA2383751C (tr)
CO (1) CO5180620A1 (tr)
CZ (1) CZ2002759A3 (tr)
DE (1) DE60012028T2 (tr)
DK (1) DK1212321T3 (tr)
ES (1) ES2223570T3 (tr)
GB (1) GB9920919D0 (tr)
HK (1) HK1046908B (tr)
HU (1) HU229391B1 (tr)
IL (2) IL148441A0 (tr)
MX (1) MXPA02002356A (tr)
MY (1) MY126789A (tr)
NO (1) NO322501B1 (tr)
NZ (1) NZ517601A (tr)
PL (1) PL206491B1 (tr)
PT (1) PT1212321E (tr)
SI (1) SI1212321T1 (tr)
TR (1) TR200200548T2 (tr)
TW (1) TWI264435B (tr)
WO (1) WO2001017961A2 (tr)
ZA (1) ZA200201779B (tr)

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CA2281817C (en) * 1999-06-29 2008-07-29 Smithkline Beecham Corporation Methods of use of fluoroquinolone compounds against maxillary sinus pathogenic bacteria
GB9920919D0 (en) * 1999-09-03 1999-11-10 Sb Pharmco Inc Novel compound
GB9920917D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel process
ES2314082T3 (es) 2001-08-02 2009-03-16 Lg Life Sciences Limited Procedimientos para la produccion de derivados amino protegidos de 4-aminometilenpirrolidin-3-ona, gemifloxacina y sus sales.
KR100517638B1 (ko) 2002-04-08 2005-09-28 주식회사 엘지생명과학 게미플록사신 산염의 새로운 제조방법
WO2004007623A1 (en) * 2002-07-17 2004-01-22 Ciba Specialty Chemicals Holding Inc. Oxidation process for preparing quinacridone pigments
KR100653334B1 (ko) 2003-03-07 2006-12-04 주식회사 엘지생명과학 4-아미노메틸-3-알콕시이미노피롤리딘 메탄설폰산염의 신규한 제조 방법
US8822934B2 (en) * 2006-11-03 2014-09-02 Accuray Incorporated Collimator changer
CN104693088B (zh) * 2013-12-06 2018-01-05 常州市勇毅生物药业有限公司 一种吉米沙星侧链的制备方法

Family Cites Families (27)

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Publication number Priority date Publication date Assignee Title
JPS57134482A (en) 1981-02-13 1982-08-19 Dainippon Pharmaceut Co Ltd 1-ethyl-6-fluoro-1,4-dihydro-4-oxo-7-(1-piperazinyl)-1,8- naphthyridine-3-carboxylic acid-3/2 hydrate and its preparation
IN162769B (tr) 1984-11-13 1988-07-09 Kyorin Seiyaku Kk
NZ222047A (en) 1986-10-08 1991-01-29 Bristol Myers Co Quinoline - or naphthyridine - carboxylic acid anti-bacterial agents
JPH01100165A (ja) 1987-10-13 1989-04-18 Shionogi & Co Ltd オキシムまたはヒドロキシアミン誘導体系抗菌剤
US4920120A (en) 1988-01-25 1990-04-24 Warner-Lambert Company Antibacterial agents
JPH0356479A (ja) 1989-07-24 1991-03-12 Takeshi Yokota 水溶性キノロン誘導体のp‐トルエンスルホン酸塩
PL166381B1 (pl) 1989-08-16 1995-05-31 Pfizer Sposób wytwarzania nowych podstawionych kwasów 7-azabicyklochinolonokarboksylowych PL PL PL PL
US5137892A (en) 1990-12-12 1992-08-11 Abbott Laboratories Quinoline, naphthyridine and pyridobenzoxazine derivatives
EP0541086A1 (en) 1991-11-08 1993-05-12 Kaken Pharmaceutical Co., Ltd. Antibacterial 6-fluoro-quinolones having an oxime group on the substituent in position 7
JPH0673056A (ja) 1992-08-26 1994-03-15 Kaken Pharmaceut Co Ltd キノリンカルボン酸誘導体およびその塩
US5776944A (en) 1994-06-16 1998-07-07 Lg Chemical Ltd. 7-(4-aminomethyl-3-methyloxyiminopyrroplidin-1-yl)-1-cyclopropyl-6-flu oro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof
DK0688772T3 (da) 1994-06-16 1999-11-01 Lg Chemical Ltd Quinolincarboxylsyrederivater med 7-(4-aminomethyl-3-oxim)-pyrrolidinsubstituenter og fremgangsmåde til deres fremstilling
JP3449658B2 (ja) 1994-12-21 2003-09-22 杏林製薬株式会社 安定性に優れた8−アルコキシキノロンカルボン酸水和物並びにその製造方法
DE69503066T2 (de) 1995-06-06 1998-10-15 Pfizer Inc., New York, N.Y. KRISTALLFORM VON WASSERFREIEN 7-((1a,5a,6a)-6-AMINO-3-AZABICYCLO (3.1.0.) HEX-3-YL)-6-FLUORO-1-(2,4-DIFLUOROPHENYL)-1,4-DIHYDRO-4-OXO-1,8-NAPHTHYRIDIN-CARBONSÄURE METHANESULFONSÄURE SALZ
IL122649A (en) 1995-08-11 2001-08-26 Pfizer (1s, 2s) - 1- (4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)-1-propanol methanesulfonate trihydrate, its use in the preparation of medicaments and pharmaceutical compositions comprising same
UA49880C2 (uk) 1996-03-29 2002-10-15 Смітклайн Бічам Корпорейшн Дигідрат ерпоcартану, фармацевтична композиція, спосіб отримання твердої дозованої форми, спосіб блокування рецепторів ангіотензину іі
MA24500A1 (fr) 1997-03-21 1998-10-01 Lg Life Sciences Ltd Derive du sel d'acide carboxylique de naphthyridine .
KR100286874B1 (ko) 1998-03-04 2001-04-16 성재갑 보호된 4-아미노메틸-피롤리딘-3-온의 제조방법
EP1082300B1 (en) 1998-05-29 2003-09-10 PHARMACIA & UPJOHN COMPANY 3-[(1'-n-methylamino)ethyl-n-benzyl]pyrrolidine monomethanesulfonate
GB9820405D0 (en) 1998-09-18 1998-11-11 Smithkline Beecham Plc Process
DK1223935T3 (da) 1999-06-29 2008-02-04 Lg Life Sciences Ltd Anvendelse af gemifloxacinforbindelser mod bakterier
AU6947900A (en) 1999-09-01 2001-03-26 Smithkline Beecham Corporation Methods of use of fluoroquinolone compounds against bacteria
GB9920917D0 (en) 1999-09-03 1999-11-10 Sb Pharmco Inc Novel process
GB9920919D0 (en) * 1999-09-03 1999-11-10 Sb Pharmco Inc Novel compound
EP1242079A4 (en) 1999-09-22 2003-01-22 Smithkline Beecham Methods of anti-bacterial use of fluoroquinolonic compounds
KR20010091379A (ko) 2000-03-15 2001-10-23 성재갑 7-(4-아미노메틸-3-옥심)피롤리딘 치환체를 갖는 퀴놀린카르복실산 유도체의 신규 제조방법
KR20020018560A (ko) 2000-09-01 2002-03-08 성재갑 3-아미노메틸-4-z-메톡시이미노피롤리딘의 신규 제조방법

Also Published As

Publication number Publication date
NO322501B1 (no) 2006-10-16
WO2001017961A2 (en) 2001-03-15
US20050033064A1 (en) 2005-02-10
HK1046908A1 (en) 2003-01-30
US6803467B2 (en) 2004-10-12
CN1372558A (zh) 2002-10-02
PL354725A1 (en) 2004-02-09
DE60012028D1 (de) 2004-08-12
BR0013750A (pt) 2002-05-21
IL148441A (en) 2007-03-08
HUP0202733A3 (en) 2005-12-28
ZA200201779B (en) 2003-08-27
JP2003508517A (ja) 2003-03-04
US20040138292A1 (en) 2004-07-15
AU6857300A (en) 2001-04-10
TWI264435B (en) 2006-10-21
CZ2002759A3 (cs) 2002-06-12
KR20020041423A (ko) 2002-06-01
DE60012028T2 (de) 2005-08-18
EP1212321A2 (en) 2002-06-12
BR0013750B1 (pt) 2014-06-17
HK1046908B (en) 2005-05-27
PT1212321E (pt) 2004-10-29
SI1212321T1 (en) 2004-12-31
CO5180620A1 (es) 2002-07-30
BRPI0013750B8 (pt) 2021-05-25
NO20021043D0 (no) 2002-03-01
EP1212321B1 (en) 2004-07-07
HUP0202733A2 (hu) 2003-01-28
CN1255402C (zh) 2006-05-10
ATE270671T1 (de) 2004-07-15
JP4208463B2 (ja) 2009-01-14
DK1212321T3 (da) 2004-10-25
US6703512B1 (en) 2004-03-09
IL148441A0 (en) 2002-09-12
NZ517601A (en) 2003-08-29
HU229391B1 (hu) 2013-11-28
GB9920919D0 (en) 1999-11-10
CA2383751C (en) 2010-06-29
ES2223570T3 (es) 2005-03-01
AU773698B2 (en) 2004-06-03
NO20021043L (no) 2002-03-01
MXPA02002356A (es) 2002-07-30
PL206491B1 (pl) 2010-08-31
WO2001017961A3 (en) 2001-09-20
AR029452A1 (es) 2003-07-02
MY126789A (en) 2006-10-31
CA2383751A1 (en) 2001-03-15
KR100705363B1 (ko) 2007-04-10

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