DK1283839T3 - Adenosin A2a-receptorantagonister - Google Patents

Adenosin A2a-receptorantagonister

Info

Publication number
DK1283839T3
DK1283839T3 DK01945991T DK01945991T DK1283839T3 DK 1283839 T3 DK1283839 T3 DK 1283839T3 DK 01945991 T DK01945991 T DK 01945991T DK 01945991 T DK01945991 T DK 01945991T DK 1283839 T3 DK1283839 T3 DK 1283839T3
Authority
DK
Denmark
Prior art keywords
adenosine
receptor antagonists
antagonists
receptor
Prior art date
Application number
DK01945991T
Other languages
Danish (da)
English (en)
Inventor
Bernard R Neustadt
William J Greenlee
Deen Tulshian
Lisa S Silverman
Yan Xia
Craig D Boyle
Samuel Chackalamannil
Neil A Lindo
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Application granted granted Critical
Publication of DK1283839T3 publication Critical patent/DK1283839T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK01945991T 2000-05-26 2001-05-24 Adenosin A2a-receptorantagonister DK1283839T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20714300P 2000-05-26 2000-05-26
PCT/US2001/016954 WO2001092264A1 (fr) 2000-05-26 2001-05-24 Antagonistes du recepteur adenosine a2a
EP01945991A EP1283839B1 (fr) 2000-05-26 2001-05-24 Antagonistes du recepteur adenosine a2a

Publications (1)

Publication Number Publication Date
DK1283839T3 true DK1283839T3 (da) 2005-07-25

Family

ID=22769372

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01945991T DK1283839T3 (da) 2000-05-26 2001-05-24 Adenosin A2a-receptorantagonister

Country Status (31)

Country Link
US (4) US6630475B2 (fr)
EP (1) EP1283839B1 (fr)
JP (3) JP4574112B2 (fr)
KR (1) KR100520907B1 (fr)
CN (2) CN100384847C (fr)
AR (1) AR028621A1 (fr)
AT (1) ATE293627T1 (fr)
AU (2) AU6808901A (fr)
BR (1) BRPI0111015B8 (fr)
CA (1) CA2410237C (fr)
CZ (1) CZ303790B6 (fr)
DE (1) DE60110219T2 (fr)
DK (1) DK1283839T3 (fr)
EC (1) ECSP024364A (fr)
ES (1) ES2237576T3 (fr)
HK (1) HK1049007B (fr)
HU (1) HU230420B1 (fr)
IL (3) IL152726A0 (fr)
MX (1) MXPA02011625A (fr)
MY (1) MY132006A (fr)
NO (1) NO325008B1 (fr)
NZ (1) NZ522326A (fr)
PE (1) PE20020062A1 (fr)
PL (1) PL218764B1 (fr)
PT (1) PT1283839E (fr)
RU (1) RU2315053C2 (fr)
SI (1) SI1283839T1 (fr)
SK (1) SK287748B6 (fr)
TW (1) TWI288137B (fr)
WO (1) WO2001092264A1 (fr)
ZA (1) ZA200208898B (fr)

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CN112592354B (zh) 2019-07-30 2022-05-27 厦门宝太生物科技股份有限公司 一种异噁唑并嘧啶类杂环化合物的制备方法
CN111072675A (zh) * 2019-12-12 2020-04-28 广东东阳光药业有限公司 含氮稠合三环衍生物及其用途
CN113773327B (zh) * 2021-09-13 2022-07-15 八叶草健康产业研究院(厦门)有限公司 一种吡唑并嘧啶并三唑环类化合物的制备方法
CN117946123A (zh) * 2024-01-26 2024-04-30 北京脑重大疾病研究院 放射性三氮唑并嘧啶基衍生物及其制备方法和应用
CN118812544A (zh) * 2024-06-19 2024-10-22 厦门大学 一种腺苷a2ar靶向小分子化合物、核素标记探针及其制备方法、应用和药物组合物
CN118812539B (zh) * 2024-06-19 2025-11-28 苏州大学 一种5-氨基三唑并嘧啶衍生物及其制备方法

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DE60110219T2 (de) 2006-03-09
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DE60110219D1 (de) 2005-05-25
US6897216B2 (en) 2005-05-24
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