DK1981506T3 - Langtidsbehandling af HIV-infektion med TMC278 - Google Patents
Langtidsbehandling af HIV-infektion med TMC278Info
- Publication number
- DK1981506T3 DK1981506T3 DK07712053.3T DK07712053T DK1981506T3 DK 1981506 T3 DK1981506 T3 DK 1981506T3 DK 07712053 T DK07712053 T DK 07712053T DK 1981506 T3 DK1981506 T3 DK 1981506T3
- Authority
- DK
- Denmark
- Prior art keywords
- tmc278
- long
- hiv infection
- term treatment
- term
- Prior art date
Links
- 208000031886 HIV Infections Diseases 0.000 title 1
- 208000037357 HIV infectious disease Diseases 0.000 title 1
- 208000033519 human immunodeficiency virus infectious disease Diseases 0.000 title 1
- 238000011866 long-term treatment Methods 0.000 title 1
- YIBOMRUWOWDFLG-ONEGZZNKSA-N rilpivirine Chemical compound CC1=CC(\C=C\C#N)=CC(C)=C1NC1=CC=NC(NC=2C=CC(=CC=2)C#N)=N1 YIBOMRUWOWDFLG-ONEGZZNKSA-N 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Organic Chemistry (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06100677 | 2006-01-20 | ||
| PCT/EP2007/050516 WO2007082922A2 (en) | 2006-01-20 | 2007-01-19 | Long term treatment of hiv- infection with tcm278 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK1981506T3 true DK1981506T3 (da) | 2013-06-24 |
| DK1981506T6 DK1981506T6 (da) | 2021-06-14 |
Family
ID=36446113
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK07712053.3T DK1981506T6 (da) | 2006-01-20 | 2007-01-19 | Langtidsbehandling af hiv-infektion med tcm278 |
Country Status (27)
| Country | Link |
|---|---|
| US (4) | USRE50189E1 (da) |
| EP (1) | EP1981506B3 (da) |
| JP (2) | JP5754005B2 (da) |
| KR (2) | KR101501475B1 (da) |
| CN (2) | CN103877091A (da) |
| AP (1) | AP2936A (da) |
| AR (1) | AR059097A1 (da) |
| AU (1) | AU2007206901B2 (da) |
| BR (1) | BRPI0707179A2 (da) |
| CA (1) | CA2636436C (da) |
| CY (1) | CY1114089T1 (da) |
| DK (1) | DK1981506T6 (da) |
| EA (1) | EA014914B1 (da) |
| ES (1) | ES2414982T7 (da) |
| HR (1) | HRP20130544T4 (da) |
| IL (1) | IL192132A (da) |
| ME (1) | ME01617B (da) |
| MY (1) | MY150717A (da) |
| NZ (1) | NZ569347A (da) |
| PL (1) | PL1981506T6 (da) |
| PT (1) | PT1981506E (da) |
| RS (1) | RS52821B2 (da) |
| SG (1) | SG170073A1 (da) |
| SI (1) | SI1981506T1 (da) |
| TW (1) | TWI458483B (da) |
| UA (1) | UA96436C2 (da) |
| WO (1) | WO2007082922A2 (da) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY169670A (en) | 2003-09-03 | 2019-05-08 | Tibotec Pharm Ltd | Combinations of a pyrimidine containing nnrti with rt inhibitors |
| TW201414495A (zh) * | 2005-04-04 | 2014-04-16 | Tibotec Pharm Ltd | Hiv-感染之預防 |
| UA96436C2 (ru) | 2006-01-20 | 2011-11-10 | Тиботек Фармасьютикелз Лтд. | Долгосрочное лечение вич-инфекции |
| AU2016219555B2 (en) * | 2006-06-23 | 2017-08-10 | Janssen Sciences Ireland Uc | Aqueous suspensions of TMC278 |
| AU2014200819B2 (en) * | 2006-06-23 | 2016-05-26 | Janssen Sciences Ireland Uc | Aqueous suspensions of TMC278 |
| EA021700B1 (ru) * | 2006-06-23 | 2015-08-31 | Тиботек Фармасьютикалз Лтд. | Фармацевтическая композиция, содержащая 4-[[4-[[4-(2-цианоэтенил)-2,6-диметилфенил]амино]-2-пиримидинил]амино]бензонитрил (тмс278) в форме суспензии микро- или наночастиц, способ ее получения и ее применение для длительного лечения или профилактики вич-инфекции |
| AR065720A1 (es) | 2007-03-14 | 2009-06-24 | Tibotec Pharm Ltd | Polvos para reconstitucion que comprenden rilpivirina dispersos en ciertos polimeros. uso. proceso. |
| RU2546529C2 (ru) * | 2008-12-24 | 2015-04-10 | Тиботек Фармасьютикалз | Имплантируемые устройства для лечения вич |
| PL2480220T3 (pl) * | 2009-09-22 | 2015-10-30 | Janssen Sciences Ireland Uc | Leczenie i zapobieganie zakażeniu HIV |
| SG181759A1 (en) | 2009-12-21 | 2012-07-30 | Janssen R & D Ireland | Degradable removable implant for the sustained release of an active compound |
| LT2932970T (lt) | 2010-01-27 | 2018-06-25 | Viiv Healthcare Company | Antivirusinė terapija |
| TWI577377B (zh) | 2010-09-16 | 2017-04-11 | Viiv醫療保健公司 | 醫藥組合物 |
| US9266824B2 (en) | 2014-01-13 | 2016-02-23 | Warsaw Orthopedic, Inc. | Methods and compositions for making an amino acid triisocyanate |
| EP3377039B1 (en) * | 2015-11-16 | 2024-01-03 | Evonik Operations GmbH | Injection solution comprising a non-nucleoside reverse-transcriptase inhibitor and poly(lactide-co-glycolide) |
| US20190163877A1 (en) * | 2017-11-27 | 2019-05-30 | International Business Machines Corporation | Decision support for effective long-term drug therapy |
| WO2022079739A1 (en) | 2020-10-14 | 2022-04-21 | Cipla Limited | Fixed dose compositions of cabotegravir and rilpivirine |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5145684A (en) | 1991-01-25 | 1992-09-08 | Sterling Drug Inc. | Surface modified drug nanoparticles |
| JPH06316524A (ja) | 1992-09-11 | 1994-11-15 | Naoyuki Inoue | 抗エイズウイルス剤 |
| US6045829A (en) | 1997-02-13 | 2000-04-04 | Elan Pharma International Limited | Nanocrystalline formulations of human immunodeficiency virus (HIV) protease inhibitors using cellulosic surface stabilizers |
| UA72189C2 (uk) | 1997-11-17 | 2005-02-15 | Янссен Фармацевтика Н.В. | Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот |
| US6258932B1 (en) | 1999-08-09 | 2001-07-10 | Tripep Ab | Peptides that block viral infectivity and methods of use thereof |
| AU7984200A (en) | 1999-09-21 | 2001-04-24 | Skyepharma Canada Inc. | Surface modified particulate compositions of biologically active substances |
| EE200200564A (et) | 2000-03-30 | 2004-06-15 | Bristol-Myers Squibb Company | Stavudiini sisaldavad toimeainet aeglustatult vabastavad graanulid |
| US20040115268A1 (en) | 2000-04-26 | 2004-06-17 | Control Delivery Systems, Inc. | Systemic delivery of antiviral agents |
| MY169670A (en) * | 2003-09-03 | 2019-05-08 | Tibotec Pharm Ltd | Combinations of a pyrimidine containing nnrti with rt inhibitors |
| JO3429B1 (ar) * | 2001-08-13 | 2019-10-20 | Janssen Pharmaceutica Nv | مشتقات برميدينات مثبطة فيروس الايدز |
| US7638522B2 (en) | 2001-08-13 | 2009-12-29 | Janssen Pharmaceutica N.V. | Salt of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl]amino] benzonitrile |
| CA2465779A1 (en) | 2001-11-20 | 2003-05-30 | Advanced Inhalation Research, Inc. | Compositions for sustained action product delivery |
| US6568805B1 (en) * | 2001-11-26 | 2003-05-27 | Dan L. Dietz Trust | Magnetic buckle for eyeglasses |
| AU2003210659A1 (en) * | 2002-01-24 | 2003-09-02 | Sangstat Medical Corporation | Combination therapy for treatment of hiv infection |
| WO2004043433A2 (en) | 2002-11-08 | 2004-05-27 | Glaxo Group Limited | Pharmaceutical antiviral compositions |
| ES2477118T3 (es) | 2002-11-18 | 2014-07-15 | Polaris Group | Método para inhibir la replicaci�n viral in vivo |
| JP5602333B2 (ja) | 2003-02-07 | 2014-10-08 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | Hiv感染の予防のためのピリミジン誘導体 |
| EP1603546A1 (en) | 2003-02-21 | 2005-12-14 | Tripep AB | Glycinamide derivative for inhibiting hiv replication |
| ES2371442T7 (es) * | 2004-09-02 | 2022-05-12 | Janssen Pharmaceutica Nv | Sal de 4-[[4-[[4-(2-cianoetenil)-2,6-dimetilfenil]amino]-2-pirimidinil]amino]benzonitrilo |
| WO2006024668A1 (en) * | 2004-09-02 | 2006-03-09 | Janssen Pharmaceutica N.V. | Hydrochloride of 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2-pyrimidinyl] amino]benzonitrile |
| KR20130030305A (ko) | 2004-11-16 | 2013-03-26 | 엘란 파마 인터내셔널 리미티드 | 주사가능한 나노입자형 올란자핀 제형 |
| TW201414495A (zh) * | 2005-04-04 | 2014-04-16 | Tibotec Pharm Ltd | Hiv-感染之預防 |
| UA96436C2 (ru) | 2006-01-20 | 2011-11-10 | Тиботек Фармасьютикелз Лтд. | Долгосрочное лечение вич-инфекции |
| EA021700B1 (ru) | 2006-06-23 | 2015-08-31 | Тиботек Фармасьютикалз Лтд. | Фармацевтическая композиция, содержащая 4-[[4-[[4-(2-цианоэтенил)-2,6-диметилфенил]амино]-2-пиримидинил]амино]бензонитрил (тмс278) в форме суспензии микро- или наночастиц, способ ее получения и ее применение для длительного лечения или профилактики вич-инфекции |
| WO2009007441A2 (en) | 2007-07-12 | 2009-01-15 | Tibotec Pharmaceuticals Ltd. | Crystalline form of (e) 4-[[4-[[4-(2-cyanoethenyl)-2,6-dimethylphenyl]amino]-2 pyrimidinyl]amino]benzonitrile |
-
2007
- 2007-01-19 UA UAA200809750A patent/UA96436C2/ru unknown
- 2007-01-19 BR BRPI0707179-5A patent/BRPI0707179A2/pt not_active Application Discontinuation
- 2007-01-19 RS RS20130258A patent/RS52821B2/sr unknown
- 2007-01-19 CN CN201410126123.XA patent/CN103877091A/zh active Pending
- 2007-01-19 CA CA2636436A patent/CA2636436C/en active Active
- 2007-01-19 KR KR1020087018888A patent/KR101501475B1/ko active Active
- 2007-01-19 EA EA200870183A patent/EA014914B1/ru unknown
- 2007-01-19 PT PT77120533T patent/PT1981506E/pt unknown
- 2007-01-19 EP EP07712053.3A patent/EP1981506B3/en active Active
- 2007-01-19 TW TW096101983A patent/TWI458483B/zh active
- 2007-01-19 SG SG201101585-6A patent/SG170073A1/en unknown
- 2007-01-19 CN CNA2007800024269A patent/CN101370504A/zh active Pending
- 2007-01-19 NZ NZ569347A patent/NZ569347A/en unknown
- 2007-01-19 AU AU2007206901A patent/AU2007206901B2/en active Active
- 2007-01-19 ES ES07712053T patent/ES2414982T7/es active Active
- 2007-01-19 AR ARP070100247A patent/AR059097A1/es not_active Application Discontinuation
- 2007-01-19 JP JP2008550764A patent/JP5754005B2/ja active Active
- 2007-01-19 HR HRP20130544TT patent/HRP20130544T4/hr unknown
- 2007-01-19 US US17/473,424 patent/USRE50189E1/en active Active
- 2007-01-19 DK DK07712053.3T patent/DK1981506T6/da active
- 2007-01-19 US US12/161,445 patent/US10953009B2/en not_active Ceased
- 2007-01-19 KR KR1020147030400A patent/KR101562943B1/ko active Active
- 2007-01-19 SI SI200731253T patent/SI1981506T1/sl unknown
- 2007-01-19 ME MEP-2013-66A patent/ME01617B/me unknown
- 2007-01-19 PL PL07712053T patent/PL1981506T6/pl unknown
- 2007-01-19 AP AP2008004535A patent/AP2936A/xx active
- 2007-01-19 WO PCT/EP2007/050516 patent/WO2007082922A2/en not_active Ceased
- 2007-01-19 MY MYPI20082697 patent/MY150717A/en unknown
-
2008
- 2008-06-12 IL IL192132A patent/IL192132A/en active IP Right Grant
-
2013
- 2013-01-28 JP JP2013013118A patent/JP5836983B2/ja active Active
- 2013-06-27 CY CY20131100521T patent/CY1114089T1/el unknown
-
2021
- 2021-03-01 US US17/188,850 patent/US20210177843A1/en not_active Abandoned
-
2023
- 2023-08-22 US US18/236,734 patent/US20240226099A1/en not_active Abandoned
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