DK2081955T3 - Metastinderivater og anvendelse deraf - Google Patents

Metastinderivater og anvendelse deraf Download PDF

Info

Publication number: DK2081955T3
Authority: DK; Denmark
Prior art keywords: metastin derivatives; metastin; derivatives
Prior art date: 2006-10-25

Application number

DK07830903.6T

Other languages

English (en)

Inventor

Taiji Asami

Naoki Nishizawa

Original Assignee

Takeda Pharmaceutical

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-10-25

Filing date

2007-10-24

Publication date

2015-06-15

2007-10-24 Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical

2015-06-15 Application granted granted Critical

2015-06-15 Publication of DK2081955T3 publication Critical patent/DK2081955T3/da

Links

KAHDONZOCXSKII-NJVVDGNHSA-N kisspeptin Chemical class C([C@@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](C)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CCC(N)=O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC=1C=CC=CC=1)C(N)=O)NC(=O)[C@H]1N(CCC1)C(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H]1N(CCC1)C(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H]1N(CCC1)C(=O)[C@H]1N(CCC1)C(=O)[C@H]1N(CCC1)C(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)CN)[C@@H](C)O)C1=CN=CN1 KAHDONZOCXSKII-NJVVDGNHSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
- C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
- C07K14/4701—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
- C07K14/4702—Regulators; Modulating activity
- C07K14/4703—Inhibitors; Suppressors
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
- C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
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- A61K38/1703—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Diabetes (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Endocrinology (AREA)
Gastroenterology & Hepatology (AREA)
Hematology (AREA)
Immunology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Reproductive Health (AREA)
Zoology (AREA)
Rheumatology (AREA)
Physical Education & Sports Medicine (AREA)
Pulmonology (AREA)
Toxicology (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Gynecology & Obstetrics (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Orthopedic Medicine & Surgery (AREA)
Oncology (AREA)
Urology & Nephrology (AREA)
Obesity (AREA)
Psychiatry (AREA)

DK07830903.6T 2006-10-25 2007-10-24 Metastinderivater og anvendelse deraf DK2081955T3 (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
JP2006290536		2006-10-25
JP2007021387		2007-01-31
JP2007221911		2007-08-28
PCT/JP2007/071169 WO2008050897A1 (en)	2006-10-25	2007-10-24	Metastin derivatives and use thereof

Publications (1)

Publication Number	Publication Date
DK2081955T3 true DK2081955T3 (da)	2015-06-15

Family

ID=38925530

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK07830903.6T DK2081955T3 (da)	2006-10-25	2007-10-24	Metastinderivater og anvendelse deraf

Country Status (33)

Country	Link
US (2)	US8765909B2 (da)
EP (1)	EP2081955B1 (da)
JP (2)	JP2010507565A (da)
KR (1)	KR101424306B1 (da)
AR (1)	AR063367A1 (da)
AU (1)	AU2007309969B2 (da)
BR (1)	BRPI0717441B8 (da)
CA (1)	CA2667537C (da)
CL (1)	CL2007003053A1 (da)
CR (1)	CR10799A (da)
CY (1)	CY1116627T1 (da)
DK (1)	DK2081955T3 (da)
EC (1)	ECSP099279A (da)
ES (1)	ES2539430T3 (da)
GE (1)	GEP20125568B (da)
HR (1)	HRP20150819T1 (da)
HU (1)	HUE025291T2 (da)
IL (1)	IL198046A (da)
JO (1)	JO3048B1 (da)
MA (1)	MA30887B1 (da)
ME (1)	ME00786B (da)
MX (1)	MX2009004148A (da)
MY (1)	MY145975A (da)
NO (1)	NO341584B1 (da)
NZ (1)	NZ576375A (da)
PE (1)	PE20081469A1 (da)
PL (1)	PL2081955T3 (da)
PT (1)	PT2081955E (da)
RS (1)	RS54083B1 (da)
SI (1)	SI2081955T1 (da)
TN (1)	TN2009000140A1 (da)
TW (1)	TWI404726B (da)
WO (1)	WO2008050897A1 (da)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20060241051A1 (en)	2002-12-26	2006-10-26	Chieko Kitada	Metastin derivatives and use thereof
AR049938A1 (es) *	2004-06-25	2006-09-13	Takeda Pharmaceutical	Derivados de metastina y utilizacion de los mismos
US20090093615A1 (en) *	2005-12-22	2009-04-09	Takeda Pharmaceutical Company Limited	Metastin derivatives and use thereof
US8404643B2 (en)	2005-12-22	2013-03-26	Takeda Pharmaceutical Company Limited	Metastin derivatives and use thereof
TWI386417B (zh)	2005-12-22	2013-02-21	Takeda Pharmaceutical	轉移抑素衍生物及其用途
US20090099334A1 (en) *	2005-12-22	2009-04-16	Takeda Pharmaceutical Company Limited	Metastin derivatives and use thereof
WO2007125619A1 (ja) *	2006-04-26	2007-11-08	Kyoto University	Ｇｐｒ５４アゴニスト活性を有する新規化合物
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Also Published As

Publication number	Publication date
KR101424306B1 (ko)	2014-08-01
ES2539430T3 (es)	2015-06-30
BRPI0717441A2 (pt)	2013-11-19
ECSP099279A (es)	2009-06-30
GEP20125568B (en)	2012-07-10
SI2081955T1 (sl)	2015-06-30
HK1130500A1 (en)	2009-12-31
CA2667537A1 (en)	2008-05-02
PL2081955T3 (pl)	2015-10-30
RS54083B1 (sr)	2015-10-30
ME00786B (me)	2011-12-20
MX2009004148A (es)	2009-05-01
WO2008050897A1 (en)	2008-05-02
IL198046A (en)	2014-06-30
MA30887B1 (fr)	2009-11-02
JP5686825B2 (ja)	2015-03-18
CY1116627T1 (el)	2017-03-15
US7786083B2 (en)	2010-08-31
PE20081469A1 (es)	2008-12-25
AU2007309969A2 (en)	2009-06-04
TN2009000140A1 (en)	2010-10-18
EP2081955A1 (en)	2009-07-29
HUE025291T2 (en)	2016-02-29
US20110059888A1 (en)	2011-03-10
PT2081955E (pt)	2015-07-10
JO3048B1 (ar)	2016-09-05
JP2010507565A (ja)	2010-03-11
TW200823232A (en)	2008-06-01
CL2007003053A1 (es)	2008-08-08
NO20091487L (no)	2009-07-07
HRP20150819T1 (hr)	2015-09-11
NO341584B1 (no)	2017-12-11
US20090215700A1 (en)	2009-08-27
AR063367A1 (es)	2009-01-21
BRPI0717441B8 (pt)	2021-05-25
TWI404726B (zh)	2013-08-11
CR10799A (es)	2009-06-09
NZ576375A (en)	2011-07-29
EP2081955B1 (en)	2015-05-06
IL198046A0 (en)	2011-08-01
JP2013075913A (ja)	2013-04-25
AU2007309969B2 (en)	2012-04-19
KR20090090315A (ko)	2009-08-25
CA2667537C (en)	2017-01-17
BRPI0717441B1 (pt)	2019-07-02
US8765909B2 (en)	2014-07-01
MY145975A (en)	2012-05-31
AU2007309969A1 (en)	2008-05-02

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