DK545786A - Hidtil ukendte insulinderivater og farmaceutiske praeparater, som indeholder disse derivater - Google Patents

Hidtil ukendte insulinderivater og farmaceutiske praeparater, som indeholder disse derivater

Info

Publication number
DK545786A
DK545786A DK545786A DK545786A DK545786A DK 545786 A DK545786 A DK 545786A DK 545786 A DK545786 A DK 545786A DK 545786 A DK545786 A DK 545786A DK 545786 A DK545786 A DK 545786A
Authority
DK
Denmark
Prior art keywords
derivatives
pharmaceutical preparations
preparations containing
insulin derivatives
unknown
Prior art date
Application number
DK545786A
Other languages
English (en)
Other versions
DK159856B (da
DK159856C (da
DK545786D0 (da
Inventor
Per Balschmidt
Finn Benned Hansen
Original Assignee
Nordisk Gentofte
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nordisk Gentofte filed Critical Nordisk Gentofte
Priority to DK545786A priority Critical patent/DK159856C/da
Publication of DK545786A publication Critical patent/DK545786A/da
Publication of DK545786D0 publication Critical patent/DK545786D0/da
Publication of DK159856B publication Critical patent/DK159856B/da
Application granted granted Critical
Publication of DK159856C publication Critical patent/DK159856C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/62Insulins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Toxicology (AREA)
  • Endocrinology (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Zoology (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Diabetes (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK545786A 1985-03-15 1986-11-14 Humaninsulinderivater og farmaceutiske praeparater, som indeholder disse derivater DK159856C (da)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DK545786A DK159856C (da) 1985-03-15 1986-11-14 Humaninsulinderivater og farmaceutiske praeparater, som indeholder disse derivater

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
DK119785A DK119785D0 (da) 1985-03-15 1985-03-15 Insulinpraeparat
DK119785 1985-03-15
PCT/DK1986/000023 WO1986005497A1 (en) 1985-03-15 1986-03-14 Novel insulin derivatives and pharmaceutical preparations containing these derivatives
DK8600023 1986-03-14
DK545786A DK159856C (da) 1985-03-15 1986-11-14 Humaninsulinderivater og farmaceutiske praeparater, som indeholder disse derivater
DK545786 1986-11-14

Publications (4)

Publication Number Publication Date
DK545786A true DK545786A (da) 1986-11-14
DK545786D0 DK545786D0 (da) 1986-11-14
DK159856B DK159856B (da) 1990-12-17
DK159856C DK159856C (da) 1991-05-06

Family

ID=8102063

Family Applications (3)

Application Number Title Priority Date Filing Date
DK119785A DK119785D0 (da) 1985-03-15 1985-03-15 Insulinpraeparat
DK545786A DK159856C (da) 1985-03-15 1986-11-14 Humaninsulinderivater og farmaceutiske praeparater, som indeholder disse derivater
DK545686A DK545686D0 (da) 1985-03-15 1986-11-14 Insulinderivater og farmaceutiske praeparater, som indeholder disse derivater

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK119785A DK119785D0 (da) 1985-03-15 1985-03-15 Insulinpraeparat

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK545686A DK545686D0 (da) 1985-03-15 1986-11-14 Insulinderivater og farmaceutiske praeparater, som indeholder disse derivater

Country Status (11)

Country Link
US (1) US5028586A (da)
EP (2) EP0216833B1 (da)
JP (2) JPS62502538A (da)
AT (2) ATE56022T1 (da)
AU (2) AU5622686A (da)
DE (2) DE3687500T2 (da)
DK (3) DK119785D0 (da)
FI (2) FI864559L (da)
IL (2) IL78161A0 (da)
NO (2) NO864555D0 (da)
WO (2) WO1986005497A1 (da)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK347086D0 (da) * 1986-07-21 1986-07-21 Novo Industri As Novel peptides
DK113585D0 (da) * 1985-03-12 1985-03-12 Novo Industri As Nye peptider
US5157021A (en) * 1985-03-15 1992-10-20 Novo Nordisk A/S Insulin derivatives and pharmaceutical preparations containing these derivatives
DK437786D0 (da) * 1986-09-12 1986-09-12 Nordisk Gentofte Insulinprecursorer
IE62879B1 (en) * 1987-02-25 1995-03-08 Novo Nordisk As Novel insulin derivatives
BR8803345A (pt) * 1988-06-30 1990-02-13 Biobras Bioquimica Do Brasil S Processo aperfeicoado para producao em larga escala de cristais de insulina humana purificada
BR8803346A (pt) * 1988-06-30 1990-02-13 Biobras Bioquimica Do Brasil S Processo aperfeicoado para producao em larga escala de cristais de insulina purificada
JPH03506023A (ja) * 1988-07-20 1991-12-26 ノボ ノルデイスク アクツイエセルスカプ ポリペプチド
US5716927A (en) * 1988-12-23 1998-02-10 Novo Nordisk A/S Insulin analogs having a modified B-chain
DK134189D0 (da) * 1989-03-20 1989-03-20 Nordisk Gentofte Insulinforbindelser
WO1992010284A2 (en) 1990-12-07 1992-06-25 Cnc Development, Inc. Catalytic chemical reactor
DK33591D0 (da) * 1991-02-27 1991-02-27 Novo Nordisk As
SG49239A1 (en) * 1991-05-24 1998-05-18 Amylin Pharmaceuticals Inc Amylin and possibly insulin containing composition for the treatment of aneroxia and related states
US5461031A (en) * 1994-06-16 1995-10-24 Eli Lilly And Company Monomeric insulin analog formulations
AUPO269996A0 (en) * 1996-10-01 1996-10-24 Walter And Eliza Hall Institute Of Medical Research, The A method of prophylaxis and treatment
US5898067A (en) * 1997-02-07 1999-04-27 Novo Nordisk A/S Crystallization of proteins
CA2503723A1 (en) * 2002-11-01 2004-05-21 Antares Pharma, Inc. Administration of insulin by jet injection
ES2642214T3 (es) 2004-01-21 2017-11-15 Novo Nordisk Health Care Ag Conjugación de péptidos mediante transglutaminasa
US7833513B2 (en) 2004-12-03 2010-11-16 Rhode Island Hospital Treatment of Alzheimer's Disease
US20090069216A1 (en) * 2006-02-21 2009-03-12 Novo Nordisk A/S Single-Chain Insulin Analogues and Pharmaceutical Formulations Thereof
EP2249853A4 (en) * 2008-01-30 2012-12-26 Univ Indiana Res & Tech Corp ESTER BASED PEPTIDE PRODRUGS
WO2010080605A1 (en) * 2008-12-19 2010-07-15 Indiana University Research And Technology Corporation Dipeptide linked medicinal agents
PE20120332A1 (es) 2008-12-19 2012-04-14 Univ Indiana Res & Tech Corp Profarmacos de peptido de la superfamilia de glucagon basado en amida
EP2585102B1 (en) 2010-06-24 2015-05-06 Indiana University Research and Technology Corporation Amide-based insulin prodrugs
BR112014015156A2 (pt) 2011-12-20 2020-10-27 Indiana University Research And Technology Corporation análogos de insulina à base de ctp, seus métodos de produção e uso no tratamento de hiperglicemia, bem como sequência de ácido nucleico e célula hospedeira
EP3395358B1 (en) 2012-09-26 2019-11-06 Indiana University Research and Technology Corporation Insulin analog dimers
JP6538645B2 (ja) 2013-03-14 2019-07-03 インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションIndiana University Research And Technology Corporation インスリン‐インクレチン複合物
JP6701208B2 (ja) 2014-09-24 2020-05-27 インディアナ ユニヴァーシティ リサーチ アンド テクノロジー コーポレイション 脂質化アミド系インスリンプロドラッグ
CN108271356A (zh) 2014-09-24 2018-07-10 印第安纳大学研究及科技有限公司 肠降血糖素-胰岛素缀合物

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3903068A (en) * 1972-12-26 1975-09-02 Us Health Education & Welfare Facile synthesis of human insulin by modification of porcine insulin
NO153061C (no) * 1979-04-13 1986-01-08 Shionogi & Co Fremgangsmaate for fremstilling av et b30-threonininsulin
JPS55138391A (en) * 1979-04-13 1980-10-29 Shionogi & Co Ltd New synthetic method of peptide derivative
JPS55138393A (en) * 1979-04-13 1980-10-29 Shionogi & Co Ltd Semisynthesis of insulin
DK147437A (en) * 1980-02-11 1900-01-01 Process for preparing human insulin or threonine B30 esters of human insulin, or a salt or complex thereof
US4421685A (en) * 1980-03-27 1983-12-20 Eli Lilly And Company Process for producing an insulin
DK319780A (da) * 1980-07-24 1982-01-25 Forenede Bryggerier As Fremgangsmaade til enzymatisk udskiftning af b-30 aminosyren i insuliner
IE52768B1 (en) * 1981-04-06 1988-02-17 Boots Co Ltd 1-arylcyclobutylalkylamine compounds useful as therapeutic agents
DE3327709A1 (de) * 1983-07-29 1985-02-07 Hoechst Ag, 6230 Frankfurt Insulin-derivat-kristallsuspensionen, verfahren zu deren herstellung und deren verwendung
DK113585D0 (da) * 1985-03-12 1985-03-12 Novo Industri As Nye peptider

Also Published As

Publication number Publication date
WO1986005496A1 (en) 1986-09-25
FI864560L (fi) 1986-11-10
FI93460B (fi) 1994-12-30
NO864555L (no) 1986-11-14
IL78160A (en) 1991-06-10
IL78161A0 (en) 1986-07-31
IL78160A0 (en) 1986-07-31
AU596968B2 (en) 1990-05-24
AU5622686A (en) 1986-10-13
WO1986005497A1 (en) 1986-09-25
DK119785D0 (da) 1985-03-15
EP0216833B1 (en) 1993-01-13
NO174278B (no) 1994-01-03
DE3687500T2 (de) 1993-07-01
DK545686A (da) 1986-11-14
DE3673737D1 (de) 1990-10-04
FI93460C (fi) 1995-04-10
EP0216832A1 (en) 1987-04-08
DK159856B (da) 1990-12-17
JPS62502538A (ja) 1987-10-01
NO174278C (no) 1994-04-13
EP0216833A1 (en) 1987-04-08
DK159856C (da) 1991-05-06
DK545786D0 (da) 1986-11-14
EP0216832B1 (en) 1990-08-29
NO864556D0 (no) 1986-11-14
US5028586A (en) 1991-07-02
ATE56022T1 (de) 1990-09-15
DK545686D0 (da) 1986-11-14
FI864559A0 (fi) 1986-11-10
FI864559A7 (fi) 1986-11-10
ATE84546T1 (de) 1993-01-15
FI864559L (fi) 1986-11-10
DE3687500D1 (de) 1993-02-25
JPS62502196A (ja) 1987-08-27
FI864560A0 (fi) 1986-11-10
AU5622786A (en) 1986-10-13
NO864555D0 (no) 1986-11-14
NO864556L (no) 1986-11-14

Similar Documents

Publication Publication Date Title
DK545786A (da) Hidtil ukendte insulinderivater og farmaceutiske praeparater, som indeholder disse derivater
DK164868C (da) Imidazooe4,5-baaquinolin-2-on-derivater, fremgangsmaade til fremstilling deraf samt farmaceutiske praeparater indeholdende disse
DK214090D0 (da) 5-aminosulfonylalkyl-indolderivater, fremgangsmaade og mellemprodukt til fremstilling deraf samt farmaceutiske praeparater indeholdende disse
DK163991C (da) Dichloranilinderivater, fremgangsmaade til fremstilling af disse, samt farmaceutiske praeparater indeholdende derivaterne
DK553988A (da) 4-aminopyridin-derivater og farmaceutiske praeparater indeholdende disse
DK642588D0 (da) Indanderivater, fremgangsmaade til fremstilling deraf samt farmaceutiske praeparater indeholdende samme
DK188286D0 (da) Phenylalkyl-2,3-dihydrobenzofuraner og analoge heraf samt praeparater indeholdende disse forbindelser
DK191086D0 (da) Benzisoselenazolonylderivater, fremgangsmaade til fremstilling deraf samt farmaceutiske praeparater indeholdende disse
DK163127C (da) Antibiotiske antitumormidler og antibiotiske midler, fremgangsmaade til fremstilling deraf samt farmaceutiske praeparater indeholdende disse
DK131188D0 (da) 3-(2-halogenalkyl)-1,4-oxathiiner og 2(2-halogenalkyl)-1,4-dithiiner, samt farmaceutiske praeparater indeholdende disse til behandling af leukaemi og tumorer
NO862917D0 (no) Dihydrokinolinon-derivater, fremgangsmaate til deres fremstilling, legemidler som inneholder disse og deres anvendelse, samt mellomprodukter til deres fremstilling.
DK157007C (da) Vitamin d3 derivater, farmaceutiske praeparater indeholdende disse forbindelser, samt anvendelse af disse forbindelser til fremstilling af farmaceutiske praeparater til behandling af neoplastiske sygdomme eller til induktion af differentiering i maligne celler
NO903967L (no) Dihydrocaffeinsyrederivater og farmasoeytiske preparater som inneholder disse.
NO872223D0 (no) Bakteriociner og preparater inneholdende disse for anti-virus behandling.
DK488688A (da) Azolidindion-derivater og farmaceutiske praeparater indeholdende disse
DK511687A (da) Farmaceutisk praeparat, samt fremstilling og anvendelse heraf
DK22286A (da) 1,4-dihydropyridin-derivater og farmaceutiske praeparater indeholdende disse
DK157925C (da) 2,3,4,5-tetrahydro-1h-3-benzazepinderivater og farmaceutiske praeparater indeholdende disse
DK163511C (da) Imidazooe1,5-aaaquinoxalinforbindelser og farmaceutiske praeparater indeholdende disse
NO900698D0 (no) Gem-dihalo-1,8-diamino-4-aza-octanderivater, og diagnostiske midler inneholdende disse.
DK179489D0 (da) Oxazolopyridinderivater, fremgangsmaade til fremstilling heraf samt farmaceutiske midler indeholdende disse
NO900699L (no) Gem-dihalo- eller tetrahalo-1,12-diamino-4,9-diazadodecan-derivater, og diagnostiske midler inneholdende disse.
NO860828L (no) Mikrokuler som ikke er radioaktivt merket og anvendelse derav for mÿling av blodstrÿmmen.
DK155941C (da) Benzodiazepinderivater og farmaceutiske praeparater indeholdende disse

Legal Events

Date Code Title Description
PBP Patent lapsed