EG24415A - Quinoline derivatives - Google Patents

Quinoline derivatives

Info

Publication number: EG24415A
Authority: EG; Egypt
Prior art keywords: quinoline derivatives; quinoline; derivatives
Prior art date: 2002-03-07

Application number

EG2003030215A

Other languages

English (en)

Inventor

Peter Gull

Esteban Pombo Villar

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-03-07

Filing date

2003-03-03

Publication date

2009-05-25

2003-03-03 Application filed by Novartis Ag filed Critical Novartis Ag

2009-05-25 Application granted granted Critical

2009-05-25 Publication of EG24415A publication Critical patent/EG24415A/xx

Links

229940027991 antiseptic and disinfectant quinoline derivative Drugs 0.000 title 1
125000002943 quinolinyl group Chemical class N1=C(C=CC2=CC=CC=C12)* 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/10—Ophthalmic agents for accommodation disorders, e.g. myopia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Ophthalmology & Optometry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

EG2003030215A 2002-03-07 2003-03-03 Quinoline derivatives EG24415A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP02005115		2002-03-07
EP02005117		2002-03-07

Publications (1)

Publication Number	Publication Date
EG24415A true EG24415A (en)	2009-05-25

Family

ID=27790094

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EG2003030215A EG24415A (en)	2002-03-07	2003-03-03	Quinoline derivatives

Country Status (28)

Country	Link
US (2)	US7399768B2 (pl)
EP (1)	EP1480970B1 (pl)
JP (2)	JP2005519117A (pl)
KR (1)	KR101027977B1 (pl)
CN (2)	CN1939915A (pl)
AR (1)	AR038730A1 (pl)
AU (1)	AU2003219023B2 (pl)
BR (1)	BR0308201A (pl)
CA (2)	CA2706618A1 (pl)
CO (1)	CO5611196A2 (pl)
CY (1)	CY1106409T1 (pl)
DE (1)	DE60311233T2 (pl)
DK (1)	DK1480970T3 (pl)
EC (1)	ECSP045271A (pl)
EG (1)	EG24415A (pl)
ES (1)	ES2279100T3 (pl)
IL (1)	IL163769A0 (pl)
MX (1)	MXPA04008666A (pl)
MY (1)	MY134325A (pl)
NO (1)	NO20044117L (pl)
NZ (1)	NZ534732A (pl)
PE (1)	PE20030927A1 (pl)
PL (2)	PL210336B1 (pl)
PT (1)	PT1480970E (pl)
RU (1)	RU2345991C2 (pl)
SI (1)	SI1480970T1 (pl)
TW (1)	TW200406401A (pl)
WO (1)	WO2003074511A1 (pl)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PT1757601E (pt) *	2002-03-07	2009-10-23	Novartis Ag	Derivados de quinolina e sua utilização em glaucoma e miopia
CR20200225A (es)	2017-11-24	2020-07-25	H Lundbeck As	Nuevos fármacos de catecolamina para uso en el tratamiento de la enfermedad de parkinson
US11104697B2 (en)	2019-05-20	2021-08-31	H. Lundbeck A/S	Process for the manufacture of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4AR,10AR)-7-hydroxy-1- propyl-1,2,3,4,4A,5,10,10A-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11130775B2 (en)	2019-05-20	2021-09-28	H. Lundbeck A/S	Solid forms of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4aR,10aR)-7-hydroxy-1-propyl-1,2,3,4,4A,5,10,10A-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11111263B2 (en)	2019-05-20	2021-09-07	H. Lundbeck A/S	Process for the manufacture of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4aR,10aR)-7-hydroxy-1-propyl-1,2,3,4,4a,5,10,10a-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11168056B2 (en)	2019-05-20	2021-11-09	H. Lundbeck A/S	Process for the manufacturing of (6aR,10aR)-7-propyl-6,6a,7,8,9,10,10a,11-octahydro-[1,3]dioxolo[4′,5′:5,6]benzo[1,2-G]quinoline and (4aR,10aR)-1-propyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[G]quinoline-6,7-diol
JP7641234B2 (ja)	2019-05-21	2025-03-06	ハー・ルンドベック・アクチエゼルスカベット	パーキンソン病の治療に使用するための新規なカテコールアミンプロドラッグ
EP3972600B1 (en)	2019-05-21	2026-02-18	H. Lundbeck A/S	Catecholamine carbamate prodrugs for use in the treatment of parkinson s disease
JP7562562B2 (ja)	2019-05-21	2024-10-07	ハー・ルンドベック・アクチエゼルスカベット	パーキンソン病の治療に使用するための新規なカテコールアミンプロドラッグ
EP3972971A1 (en)	2019-05-21	2022-03-30	H. Lundbeck A/S	New catecholamine prodrugs for use in the treatment of parkinson's diseases

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL100555A (en) *	1991-02-07	2000-08-31	Hoechst Marion Roussel Inc	N-substituted quinoline derivatives their preparation their use for the preparation of medicaments and the pharmaceutical compositions containing them
GB9326010D0 (en) *	1993-12-21	1994-02-23	Sandoz Ltd	Improvements in or relating to organic compounds
TW378209B (en) *	1996-07-08	2000-01-01	Novartis Ag	Benzo[g]quinoline derivatives, their preparation and the pharmaceutical composition containing them
PE20030240A1 (es) *	2001-07-09	2003-04-16	Novartis Ag	DERIVADOS DE BENZO [g] QUINOLINA

2003
- 2003-03-03 EG EG2003030215A patent/EG24415A/xx active
- 2003-03-05 AR ARP030100740A patent/AR038730A1/es unknown
- 2003-03-05 TW TW092104671A patent/TW200406401A/zh unknown
- 2003-03-05 PE PE2003000212A patent/PE20030927A1/es not_active Application Discontinuation
- 2003-03-06 NZ NZ534732A patent/NZ534732A/en unknown
- 2003-03-06 DK DK03714784T patent/DK1480970T3/da active
- 2003-03-06 CN CNA2006101357990A patent/CN1939915A/zh active Pending
- 2003-03-06 CN CNB038053608A patent/CN1293070C/zh not_active Expired - Fee Related
- 2003-03-06 PL PL370915A patent/PL210336B1/pl unknown
- 2003-03-06 EP EP03714784A patent/EP1480970B1/en not_active Expired - Lifetime
- 2003-03-06 WO PCT/EP2003/002321 patent/WO2003074511A1/en not_active Ceased
- 2003-03-06 SI SI200330755T patent/SI1480970T1/sl unknown
- 2003-03-06 US US10/506,232 patent/US7399768B2/en not_active Expired - Fee Related
- 2003-03-06 DE DE60311233T patent/DE60311233T2/de not_active Expired - Lifetime
- 2003-03-06 RU RU2004129767/04A patent/RU2345991C2/ru not_active IP Right Cessation
- 2003-03-06 PT PT03714784T patent/PT1480970E/pt unknown
- 2003-03-06 IL IL16376903A patent/IL163769A0/xx unknown
- 2003-03-06 ES ES03714784T patent/ES2279100T3/es not_active Expired - Lifetime
- 2003-03-06 JP JP2003572979A patent/JP2005519117A/ja active Pending
- 2003-03-06 MX MXPA04008666A patent/MXPA04008666A/es active IP Right Grant
- 2003-03-06 PL PL394208A patent/PL215012B1/pl unknown
- 2003-03-06 CA CA2706618A patent/CA2706618A1/en not_active Abandoned
- 2003-03-06 BR BR0308201-6A patent/BR0308201A/pt not_active Application Discontinuation
- 2003-03-06 KR KR1020047012409A patent/KR101027977B1/ko not_active Expired - Fee Related
- 2003-03-06 CA CA2477720A patent/CA2477720C/en not_active Expired - Fee Related
- 2003-03-06 AU AU2003219023A patent/AU2003219023B2/en not_active Ceased
- 2003-03-07 MY MYPI20030808A patent/MY134325A/en unknown
2004
- 2004-09-02 EC EC2004005271A patent/ECSP045271A/es unknown
- 2004-09-15 CO CO04091781A patent/CO5611196A2/es not_active Application Discontinuation
- 2004-09-28 NO NO20044117A patent/NO20044117L/no not_active Application Discontinuation
2007
- 2007-03-22 CY CY20071100405T patent/CY1106409T1/el unknown
2008
- 2008-06-12 US US12/137,819 patent/US20080255176A1/en not_active Abandoned
2010
- 2010-02-04 JP JP2010022863A patent/JP2010095550A/ja active Pending

Also Published As

Publication number	Publication date
DE60311233T2 (de)	2007-11-15
SI1480970T1 (sl)	2007-06-30
EP1480970B1 (en)	2007-01-17
ECSP045271A (es)	2004-10-26
ES2279100T3 (es)	2007-08-16
DE60311233D1 (de)	2007-03-08
KR20040089615A (ko)	2004-10-21
CA2477720A1 (en)	2003-09-12
CN1293070C (zh)	2007-01-03
DK1480970T3 (da)	2007-03-05
RU2345991C2 (ru)	2009-02-10
AU2003219023A1 (en)	2003-09-16
US7399768B2 (en)	2008-07-15
WO2003074511A1 (en)	2003-09-12
NZ534732A (en)	2006-05-26
CO5611196A2 (es)	2006-02-28
CA2477720C (en)	2010-09-21
PL210336B1 (pl)	2012-01-31
BR0308201A (pt)	2005-01-04
AU2003219023B2 (en)	2006-11-30
PT1480970E (pt)	2007-03-30
PL394208A1 (pl)	2011-08-16
PL370915A1 (pl)	2005-06-13
TW200406401A (en)	2004-05-01
HK1071364A1 (en)	2005-07-15
EP1480970A1 (en)	2004-12-01
JP2005519117A (ja)	2005-06-30
NO20044117L (no)	2004-09-28
MY134325A (en)	2007-12-31
MXPA04008666A (es)	2004-12-06
CN1639148A (zh)	2005-07-13
RU2004129767A (ru)	2005-06-27
US20080255176A1 (en)	2008-10-16
PE20030927A1 (es)	2003-12-26
PL215012B1 (pl)	2013-10-31
CY1106409T1 (el)	2011-10-12
AR038730A1 (es)	2005-01-26
CN1939915A (zh)	2007-04-04
IL163769A0 (en)	2005-12-18
CA2706618A1 (en)	2003-09-12
KR101027977B1 (ko)	2011-04-13
US20050234085A1 (en)	2005-10-20
JP2010095550A (ja)	2010-04-30

Publication	Publication Date	Title
IL164324A0 (en)	2005-12-18	Quinolinone derivatives
AP2006003619A0 (en)	2006-06-30	Novel quinoline derivatives
AP1850A (en)	2008-05-26	Spiroindolineplperidine derivatives
EG24050A (en)	2008-04-13	Heterocylocarboxamide derivatives
PL374718A1 (pl)	2005-10-31	Azolidynono-winylowe pochodne skondensowanego benzenu
IL166121A0 (en)	2006-01-15	Indole-3-sulphur derivatives
EP1522540A4 (en)	2011-08-10	AZAARENE DERIVATIVES
PL376475A1 (pl)	2005-12-27	Pochodne N-podstawionej 2-oksodihydropirydyny
IL159288A0 (en)	2004-06-01	Tetrahydroquinoline derivatives
GB0219896D0 (en)	2002-10-02	Dihydropyridine derivatives
IL166426A0 (en)	2006-01-15	N-biarylmethyl aminocycloalkanecarboxamide derivatives
PL376997A1 (pl)	2006-01-23	Pochodne tetrahydrochinoliny
PL373697A1 (pl)	2005-09-05	Pochodne izochinoliny
IL165572A0 (en)	2006-01-15	1-Ä(indoÜ-3-yl)carbonylÜpiperazine derivatives
PL377318A1 (pl)	2006-01-23	Pochodne tetrahydrochinoliny
GB0104422D0 (en)	2001-04-11	Quinoline derivative
PL371216A1 (pl)	2005-06-13	Pochodne izochinoliny
AU2003222659A8 (en)	2003-11-03	23-o-substituted 5-o-mycaminosyltylonide derivatives
IL163769A0 (en)	2005-12-18	Quinoline derivatives
AU2003274551A1 (en)	2004-06-03	Quinoline derivatives
AU2003252333A1 (en)	2004-02-23	Novel tetrahydroquinoline derivatives
EP1531854A4 (en)	2006-06-28	O-DERIVATED NOCATHIACIN DERIVATIVES
GB0213488D0 (en)	2002-07-24	2-Naphthamide derivatives
AU2003243397A8 (en)	2003-12-19	Homo-camptothecin derivatives
AU2003290095A8 (en)	2004-07-14	Quinolizidine derivatives