PL370915A1 - Pochodne chinoliny - Google Patents

Pochodne chinoliny

Info

Publication number: PL370915A1
Authority: PL; Poland
Prior art keywords: quinoline derivatives; quinoline; derivatives
Prior art date: 2002-03-07

Application number

PL03370915A

Other languages

English (en)

Other versions

PL210336B1 (pl

Inventor

Peter Gull

Villar Esteban Pombo

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-03-07

Filing date

2003-03-06

Publication date

2005-06-13

2003-03-06 Application filed by Novartis Ag filed Critical Novartis Ag

2005-06-13 Publication of PL370915A1 publication Critical patent/PL370915A1/pl

2012-01-31 Publication of PL210336B1 publication Critical patent/PL210336B1/pl

Links

229940027991 antiseptic and disinfectant quinoline derivative Drugs 0.000 title 1
125000002943 quinolinyl group Chemical class N1=C(C=CC2=CC=CC=C12)* 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/10—Ophthalmic agents for accommodation disorders, e.g. myopia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Ophthalmology & Optometry (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

PL370915A 2002-03-07 2003-03-06 Pochodna benzo(g)chinoliny, kompozycja farmaceutyczna zawierająca tę pochodną oraz zastosowanie tej pochodnej benzo(g)chinoliny PL210336B1 (pl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP02005117		2002-03-07
EP02005115		2002-03-07

Publications (2)

Publication Number	Publication Date
PL370915A1 true PL370915A1 (pl)	2005-06-13
PL210336B1 PL210336B1 (pl)	2012-01-31

Family

ID=27790094

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
PL394208A PL215012B1 (pl)	2002-03-07	2003-03-06	Nowe pochodne benzo[g]chinoliny, kompozycje farmaceutyczne je zawierajace oraz zastosowania farmaceutyczne tych zwiazków
PL370915A PL210336B1 (pl)	2002-03-07	2003-03-06	Pochodna benzo(g)chinoliny, kompozycja farmaceutyczna zawierająca tę pochodną oraz zastosowanie tej pochodnej benzo(g)chinoliny

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
PL394208A PL215012B1 (pl)	2002-03-07	2003-03-06	Nowe pochodne benzo[g]chinoliny, kompozycje farmaceutyczne je zawierajace oraz zastosowania farmaceutyczne tych zwiazków

Country Status (28)

Country	Link
US (2)	US7399768B2 (pl)
EP (1)	EP1480970B1 (pl)
JP (2)	JP2005519117A (pl)
KR (1)	KR101027977B1 (pl)
CN (2)	CN1939915A (pl)
AR (1)	AR038730A1 (pl)
AU (1)	AU2003219023B2 (pl)
BR (1)	BR0308201A (pl)
CA (2)	CA2477720C (pl)
CO (1)	CO5611196A2 (pl)
CY (1)	CY1106409T1 (pl)
DE (1)	DE60311233T2 (pl)
DK (1)	DK1480970T3 (pl)
EC (1)	ECSP045271A (pl)
EG (1)	EG24415A (pl)
ES (1)	ES2279100T3 (pl)
IL (1)	IL163769A0 (pl)
MX (1)	MXPA04008666A (pl)
MY (1)	MY134325A (pl)
NO (1)	NO20044117L (pl)
NZ (1)	NZ534732A (pl)
PE (1)	PE20030927A1 (pl)
PL (2)	PL215012B1 (pl)
PT (1)	PT1480970E (pl)
RU (1)	RU2345991C2 (pl)
SI (1)	SI1480970T1 (pl)
TW (1)	TW200406401A (pl)
WO (1)	WO2003074511A1 (pl)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SI1757601T1 (sl) *	2002-03-07	2009-12-31	Novartis Ag	Kinolinski derivati in njihova uporaba pri glavkomu in miopiji
PT3713933T (pt)	2017-11-24	2026-05-19	H Lundbeck As	Novos profrmacos de catecolamina para utilizao no tratamento de doena de parkinson
US11104697B2 (en)	2019-05-20	2021-08-31	H. Lundbeck A/S	Process for the manufacture of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4AR,10AR)-7-hydroxy-1- propyl-1,2,3,4,4A,5,10,10A-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11130775B2 (en)	2019-05-20	2021-09-28	H. Lundbeck A/S	Solid forms of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4aR,10aR)-7-hydroxy-1-propyl-1,2,3,4,4A,5,10,10A-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11168056B2 (en)	2019-05-20	2021-11-09	H. Lundbeck A/S	Process for the manufacturing of (6aR,10aR)-7-propyl-6,6a,7,8,9,10,10a,11-octahydro-[1,3]dioxolo[4′,5′:5,6]benzo[1,2-G]quinoline and (4aR,10aR)-1-propyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[G]quinoline-6,7-diol
US11111263B2 (en)	2019-05-20	2021-09-07	H. Lundbeck A/S	Process for the manufacture of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4aR,10aR)-7-hydroxy-1-propyl-1,2,3,4,4a,5,10,10a-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
EP3972600B1 (en)	2019-05-21	2026-02-18	H. Lundbeck A/S	Catecholamine carbamate prodrugs for use in the treatment of parkinson s disease
JP7641234B2 (ja)	2019-05-21	2025-03-06	ハー・ルンドベック・アクチエゼルスカベット	パーキンソン病の治療に使用するための新規なカテコールアミンプロドラッグ
US12391650B2 (en)	2019-05-21	2025-08-19	H. Lundbeck A/S	Catecholamine prodrugs for use in the treatment of Parkinson's disease
WO2020234275A1 (en)	2019-05-21	2020-11-26	H. Lundbeck A/S	New catecholamine prodrugs for use in the treatment of parkinson's diseases

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL100555A (en) *	1991-02-07	2000-08-31	Hoechst Marion Roussel Inc	N-substituted quinoline derivatives their preparation their use for the preparation of medicaments and the pharmaceutical compositions containing them
GB9326010D0 (en) *	1993-12-21	1994-02-23	Sandoz Ltd	Improvements in or relating to organic compounds
TW378209B (en) *	1996-07-08	2000-01-01	Novartis Ag	Benzo[g]quinoline derivatives, their preparation and the pharmaceutical composition containing them
PE20030240A1 (es) *	2001-07-09	2003-04-16	Novartis Ag	DERIVADOS DE BENZO [g] QUINOLINA

2003
- 2003-03-03 EG EG2003030215A patent/EG24415A/xx active
- 2003-03-05 PE PE2003000212A patent/PE20030927A1/es not_active Application Discontinuation
- 2003-03-05 AR ARP030100740A patent/AR038730A1/es unknown
- 2003-03-05 TW TW092104671A patent/TW200406401A/zh unknown
- 2003-03-06 SI SI200330755T patent/SI1480970T1/sl unknown
- 2003-03-06 DK DK03714784T patent/DK1480970T3/da active
- 2003-03-06 ES ES03714784T patent/ES2279100T3/es not_active Expired - Lifetime
- 2003-03-06 KR KR1020047012409A patent/KR101027977B1/ko not_active Expired - Fee Related
- 2003-03-06 EP EP03714784A patent/EP1480970B1/en not_active Expired - Lifetime
- 2003-03-06 DE DE60311233T patent/DE60311233T2/de not_active Expired - Lifetime
- 2003-03-06 CN CNA2006101357990A patent/CN1939915A/zh active Pending
- 2003-03-06 IL IL16376903A patent/IL163769A0/xx unknown
- 2003-03-06 RU RU2004129767/04A patent/RU2345991C2/ru not_active IP Right Cessation
- 2003-03-06 PL PL394208A patent/PL215012B1/pl unknown
- 2003-03-06 WO PCT/EP2003/002321 patent/WO2003074511A1/en not_active Ceased
- 2003-03-06 US US10/506,232 patent/US7399768B2/en not_active Expired - Fee Related
- 2003-03-06 BR BR0308201-6A patent/BR0308201A/pt not_active Application Discontinuation
- 2003-03-06 JP JP2003572979A patent/JP2005519117A/ja active Pending
- 2003-03-06 CA CA2477720A patent/CA2477720C/en not_active Expired - Fee Related
- 2003-03-06 AU AU2003219023A patent/AU2003219023B2/en not_active Ceased
- 2003-03-06 NZ NZ534732A patent/NZ534732A/en unknown
- 2003-03-06 CA CA2706618A patent/CA2706618A1/en not_active Abandoned
- 2003-03-06 PL PL370915A patent/PL210336B1/pl unknown
- 2003-03-06 CN CNB038053608A patent/CN1293070C/zh not_active Expired - Fee Related
- 2003-03-06 PT PT03714784T patent/PT1480970E/pt unknown
- 2003-03-06 MX MXPA04008666A patent/MXPA04008666A/es active IP Right Grant
- 2003-03-07 MY MYPI20030808A patent/MY134325A/en unknown
2004
- 2004-09-02 EC EC2004005271A patent/ECSP045271A/es unknown
- 2004-09-15 CO CO04091781A patent/CO5611196A2/es not_active Application Discontinuation
- 2004-09-28 NO NO20044117A patent/NO20044117L/no not_active Application Discontinuation
2007
- 2007-03-22 CY CY20071100405T patent/CY1106409T1/el unknown
2008
- 2008-06-12 US US12/137,819 patent/US20080255176A1/en not_active Abandoned
2010
- 2010-02-04 JP JP2010022863A patent/JP2010095550A/ja active Pending

Also Published As

Publication number	Publication date
CN1639148A (zh)	2005-07-13
CA2477720A1 (en)	2003-09-12
CN1293070C (zh)	2007-01-03
CA2706618A1 (en)	2003-09-12
CN1939915A (zh)	2007-04-04
CY1106409T1 (el)	2011-10-12
US7399768B2 (en)	2008-07-15
HK1071364A1 (en)	2005-07-15
ECSP045271A (es)	2004-10-26
IL163769A0 (en)	2005-12-18
JP2005519117A (ja)	2005-06-30
CA2477720C (en)	2010-09-21
AU2003219023B2 (en)	2006-11-30
DE60311233T2 (de)	2007-11-15
JP2010095550A (ja)	2010-04-30
NO20044117L (no)	2004-09-28
PL210336B1 (pl)	2012-01-31
US20050234085A1 (en)	2005-10-20
RU2345991C2 (ru)	2009-02-10
PL394208A1 (pl)	2011-08-16
WO2003074511A1 (en)	2003-09-12
KR20040089615A (ko)	2004-10-21
MY134325A (en)	2007-12-31
EP1480970B1 (en)	2007-01-17
BR0308201A (pt)	2005-01-04
ES2279100T3 (es)	2007-08-16
MXPA04008666A (es)	2004-12-06
PT1480970E (pt)	2007-03-30
AU2003219023A1 (en)	2003-09-16
DK1480970T3 (da)	2007-03-05
KR101027977B1 (ko)	2011-04-13
PL215012B1 (pl)	2013-10-31
DE60311233D1 (de)	2007-03-08
RU2004129767A (ru)	2005-06-27
PE20030927A1 (es)	2003-12-26
AR038730A1 (es)	2005-01-26
TW200406401A (en)	2004-05-01
US20080255176A1 (en)	2008-10-16
CO5611196A2 (es)	2006-02-28
EG24415A (en)	2009-05-25
EP1480970A1 (en)	2004-12-01
NZ534732A (en)	2006-05-26
SI1480970T1 (sl)	2007-06-30

Publication	Publication Date	Title
IL164324A0 (en)	2005-12-18	Quinolinone derivatives
ZA200603657B (en)	2007-08-29	Novel quinoline derivatives
AP1850A (en)	2008-05-26	Spiroindolineplperidine derivatives
EG24050A (en)	2008-04-13	Heterocylocarboxamide derivatives
PL374718A1 (pl)	2005-10-31	Azolidynono-winylowe pochodne skondensowanego benzenu
IL166121A0 (en)	2006-01-15	Indole-3-sulphur derivatives
EP1522540A4 (en)	2011-08-10	AZAARENE DERIVATIVES
PL376475A1 (pl)	2005-12-27	Pochodne N-podstawionej 2-oksodihydropirydyny
IL159288A0 (en)	2004-06-01	Tetrahydroquinoline derivatives
GB0219896D0 (en)	2002-10-02	Dihydropyridine derivatives
IL166426A0 (en)	2006-01-15	N-biarylmethyl aminocycloalkanecarboxamide derivatives
PL376997A1 (pl)	2006-01-23	Pochodne tetrahydrochinoliny
PL373697A1 (pl)	2005-09-05	Pochodne izochinoliny
IL165572A0 (en)	2006-01-15	1-Ä(indoÜ-3-yl)carbonylÜpiperazine derivatives
PL377318A1 (pl)	2006-01-23	Pochodne tetrahydrochinoliny
GB0104422D0 (en)	2001-04-11	Quinoline derivative
PL371216A1 (pl)	2005-06-13	Pochodne izochinoliny
AU2003222659A8 (en)	2003-11-03	23-o-substituted 5-o-mycaminosyltylonide derivatives
EG24415A (en)	2009-05-25	Quinoline derivatives
AU2003274551A1 (en)	2004-06-03	Quinoline derivatives
AU2003252333A1 (en)	2004-02-23	Novel tetrahydroquinoline derivatives
EP1531854A4 (en)	2006-06-28	O-DERIVATED NOCATHIACIN DERIVATIVES
GB0213488D0 (en)	2002-07-24	2-Naphthamide derivatives
AU2003243397A8 (en)	2003-12-19	Homo-camptothecin derivatives
AU2003290095A8 (en)	2004-07-14	Quinolizidine derivatives