ES2176209T3 - Preparacion farmaceutica oral liberable en el tracto digestivo inferior. - Google Patents
Preparacion farmaceutica oral liberable en el tracto digestivo inferior.Info
- Publication number
- ES2176209T3 ES2176209T3 ES93924185T ES93924185T ES2176209T3 ES 2176209 T3 ES2176209 T3 ES 2176209T3 ES 93924185 T ES93924185 T ES 93924185T ES 93924185 T ES93924185 T ES 93924185T ES 2176209 T3 ES2176209 T3 ES 2176209T3
- Authority
- ES
- Spain
- Prior art keywords
- pharmaceutical preparation
- digestive tract
- liberable
- lower digestive
- oral pharmaceutical
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- 210000001035 gastrointestinal tract Anatomy 0.000 title abstract 2
- 239000008183 oral pharmaceutical preparation Substances 0.000 title 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 229920006318 anionic polymer Polymers 0.000 abstract 1
- 239000011248 coating agent Substances 0.000 abstract 1
- 238000000576 coating method Methods 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 239000007787 solid Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Medicinal Preparation (AREA)
Abstract
SE PRESENTA UNA PREPARACION FARMACEUTICA PERORAL LIBERABLE EN EL TRACTO DIGESTIVO INFERIOR, QUE TIENE UNA ESTRUCTURA DE REVESTIMIENTO DE DOBLE CAPA EN LA QUE UNA DROGA SOLIDA QUE COMPRENDE UN NUCLEO QUE CONTIENE EL INGREDIENTE ACTIVO SE RECUBRE CON UNA CAPA INTERIOR QUE COMPRENDE UN POLIMERO CATIONICO Y UN CAPA EXTERIOR QUE COMPRENDE UN POLIMERO ANIONICO.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP32247892 | 1992-11-06 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2176209T3 true ES2176209T3 (es) | 2002-12-01 |
Family
ID=18144084
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES93924185T Expired - Lifetime ES2176209T3 (es) | 1992-11-06 | 1993-11-05 | Preparacion farmaceutica oral liberable en el tracto digestivo inferior. |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US5654004A (es) |
| EP (1) | EP0667148B1 (es) |
| KR (1) | KR0157280B1 (es) |
| AU (1) | AU5376894A (es) |
| CA (1) | CA2148465C (es) |
| DE (1) | DE69332082T2 (es) |
| DK (1) | DK0667148T3 (es) |
| ES (1) | ES2176209T3 (es) |
| WO (1) | WO1994010983A1 (es) |
Families Citing this family (59)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5514663A (en) * | 1993-10-19 | 1996-05-07 | The Procter & Gamble Company | Senna dosage form |
| US6117453A (en) * | 1995-04-14 | 2000-09-12 | Pharma Pass | Solid compositions containing polyethylene oxide and an active ingredient |
| SG80553A1 (en) | 1995-07-20 | 2001-05-22 | Tanabe Seiyaku Co | Pharmaceutical preparation in form of coated capsule releasable at lower part of digestive tract |
| US6214378B1 (en) * | 1996-08-02 | 2001-04-10 | Hisamitsu Pharmaceutical Co., Inc. | Capsules for oral preparations and capsule preparations for oral administration |
| JPH10152431A (ja) * | 1996-08-02 | 1998-06-09 | Hisamitsu Pharmaceut Co Inc | 経口製剤用カプセルと経口カプセル製剤 |
| US5891474A (en) | 1997-01-29 | 1999-04-06 | Poli Industria Chimica, S.P.A. | Time-specific controlled release dosage formulations and method of preparing same |
| KR100522248B1 (ko) * | 1997-05-29 | 2006-02-01 | 동아제약주식회사 | 이중제어방출막구조의경구서방성제제및그제조방법 |
| DE19726282A1 (de) | 1997-06-20 | 1998-12-24 | Inst Neue Mat Gemein Gmbh | Nanoskalige Teilchen mit einem von mindestens zwei Schalen umgebenen eisenoxid-haltigen Kern |
| JPH11246439A (ja) * | 1998-03-02 | 1999-09-14 | Hisamitsu Pharmaceut Co Inc | 経粘膜用吸収促進剤 |
| DE59915041D1 (de) * | 1998-03-19 | 2009-07-30 | Max Planck Gesellschaft | Verfahren zum Aufbringen mehrerer Schichten von Beschichtungssubstanzen auf Templatpartikel |
| EP0972563A1 (en) * | 1998-07-15 | 2000-01-19 | Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. | Fabrication of multilayer-coated particles and hollow shells via electrostatic self-assembly of nanocomposite multilayers on decomposable colloidal templates |
| DE69904307T2 (de) | 1998-03-19 | 2003-09-04 | Max-Planck-Gesellschaft Zur Foerderung Der Wissenschaften E.V. | Herstellung von mit mehrlagen gestrichenen partikeln und hohlen schalen durch elektrostatische selbstorganisierung von nanokompositmehrlagen auf zersetzbaren schablonen |
| US7101575B2 (en) | 1998-03-19 | 2006-09-05 | Max-Planck-Gesellschaft Zur Forderung Der Wissenschaften E.V. | Production of nanocapsules and microcapsules by layer-wise polyelectrolyte self-assembly |
| JPH11335269A (ja) * | 1998-05-19 | 1999-12-07 | Hisamitsu Pharmaceut Co Inc | 遺伝子関連医薬の経口投与固形製剤 |
| US6197347B1 (en) | 1998-06-29 | 2001-03-06 | Andrx Pharmaceuticals, Inc. | Oral dosage for the controlled release of analgesic |
| FR2781666B1 (fr) | 1998-07-30 | 2000-09-08 | Oreal | Composition cosmetique solide et ses utilisations |
| KR100336975B1 (ko) * | 1998-08-11 | 2002-08-22 | 한국화학연구원 | 약물방출제어용패취 |
| ATE293981T1 (de) * | 1998-09-21 | 2005-05-15 | Amato Pharm Prod Ltd | System zur oralen wirkstoffabgabe zur steigerung der bioverfügbarkeit von aktiviertem glycyrrhetin |
| AU3074700A (en) * | 1999-01-22 | 2000-08-07 | Yamanouchi Pharmaceutical Co., Ltd. | Medicinal compositions with improved oral absorption |
| US7658938B2 (en) | 1999-02-22 | 2010-02-09 | Merrion Reasearch III Limited | Solid oral dosage form containing an enhancer |
| US8119159B2 (en) | 1999-02-22 | 2012-02-21 | Merrion Research Iii Limited | Solid oral dosage form containing an enhancer |
| WO2000050012A1 (en) * | 1999-02-22 | 2000-08-31 | Elan Corporation, Plc | Solid oral dosage form containing an enhancer |
| JP2000247911A (ja) * | 1999-02-26 | 2000-09-12 | Hisamitsu Pharmaceut Co Inc | 大腸用吸収促進剤 |
| WO2001001964A2 (en) | 1999-06-23 | 2001-01-11 | Sedum Laboratories, Inc. | Ionically formulated biomolecule microcarriers |
| US6620834B1 (en) | 1999-07-02 | 2003-09-16 | Hisamitsu Pharmaceutical Co., Inc. | Medicinal compositions for treating colorectal cancer |
| DE19943420A1 (de) * | 1999-09-08 | 2001-03-15 | Beiersdorf Ag | Mascara und Augenbrauenstifte mit einem Gehalt an fluormodifizierten Kammpolymeren |
| US20020015730A1 (en) * | 2000-03-09 | 2002-02-07 | Torsten Hoffmann | Pharmaceutical formulations and method for making |
| US6551617B1 (en) | 2000-04-20 | 2003-04-22 | Bristol-Myers Squibb Company | Taste masking coating composition |
| WO2001080826A2 (en) | 2000-04-20 | 2001-11-01 | Bristol-Myers Squibb Company | Taste masking coating composition |
| KR100411195B1 (ko) * | 2000-09-26 | 2003-12-18 | 한국화학연구원 | 케토롤락 트로메타민이 함유된 서방형 펠렛 |
| CA2359812C (en) | 2000-11-20 | 2004-02-10 | The Procter & Gamble Company | Pharmaceutical dosage form with multiple coatings for reduced impact of coating fractures |
| PT1456380E (pt) * | 2001-11-02 | 2012-07-23 | Giuliani Int Ltd | Inibidores smad7 para o tratamento de doenças do snc |
| JP2003201256A (ja) * | 2001-12-28 | 2003-07-18 | Hisamitsu Pharmaceut Co Inc | 大腸送達性経口医薬製剤、大腸癌治療用経口医薬製剤および大腸炎治療用経口医薬製剤 |
| US7007417B2 (en) * | 2002-01-18 | 2006-03-07 | M.H. Segan Limited Partnership | Audio-visual display device for pictorial artwork |
| TWI355276B (en) * | 2003-01-14 | 2012-01-01 | Akira Tsuji | Gastrointestinal absorption enhancer mediated by p |
| FR2850577B1 (fr) * | 2003-02-03 | 2005-04-15 | Ethypharm Sa | Particules enrobees a gout masque, leur procede de preparation et comprimes orodispersibles contenant lesdites particules |
| US20060188563A1 (en) * | 2003-03-27 | 2006-08-24 | Hisamitsu Pharmaceutical Co., Inc. | Medicinal oral preparations for colon delivery, medicinal oral preparations for treating colon cancer and medicinal oral preparations for treating colitis |
| ITRM20030149A1 (it) | 2003-04-02 | 2004-10-03 | Giuliani Spa | Oligonucleotidi (odn) antisenso per smad7 e loro usi in campo medico |
| US7348399B2 (en) | 2003-08-29 | 2008-03-25 | Louisiana Tech University Foundation, Inc. | Nanofabricated polypeptide multilayer films, coatings, and microcapsules |
| US7544770B2 (en) | 2003-08-29 | 2009-06-09 | Louisiana Tech Foundation, Inc. | Multilayer films, coatings, and microcapsules comprising polypeptides |
| US7550557B2 (en) | 2003-08-29 | 2009-06-23 | Louisiana Tech University Foundation, Inc. | Multilayer films, coatings, and microcapsules comprising polypeptides |
| US7670624B2 (en) * | 2004-01-29 | 2010-03-02 | Astella Pharma Inc. | Gastrointestinal-specific multiple drug release system |
| DE102004013637A1 (de) | 2004-03-19 | 2005-10-13 | Capsulution Nanoscience Ag | Verfahren zur Herstellung von CS-Partikeln und Mikrokapseln unter Verwendung poröser Template sowie CS-Partikel und Mikrokapseln |
| JP4521554B2 (ja) * | 2004-03-31 | 2010-08-11 | マイラン製薬株式会社 | シクロスポリン製剤 |
| DE102004035936A1 (de) * | 2004-07-23 | 2006-03-16 | Röhm GmbH & Co. KG | Mehrschichtige Arzneiform |
| CN100486568C (zh) * | 2004-08-26 | 2009-05-13 | 复旦大学 | 洛索洛芬钠缓释制剂 |
| ES2426445T3 (es) | 2006-04-07 | 2013-10-23 | Merrion Research Iii Limited | Forma de dosificación oral sólida que contiene un potenciador |
| CN101259140B (zh) * | 2007-03-08 | 2012-08-22 | 重庆北碚现代应用药物研究所 | 一种治疗胃炎、胃溃疡及十二指肠溃疡的复方药物及其制备方法 |
| WO2008117814A1 (ja) * | 2007-03-26 | 2008-10-02 | Teikoku Seiyaku Co., Ltd. | 大腸送達用経口製剤 |
| WO2009048073A1 (ja) * | 2007-10-09 | 2009-04-16 | Takeda Pharmaceutical Company Limited | 顆粒の被覆方法 |
| DE102008003615A1 (de) | 2008-01-09 | 2009-07-16 | Magforce Nanotechnologies Ag | Magnetische Transducer |
| WO2009137080A1 (en) | 2008-05-07 | 2009-11-12 | Merrion Research Iii Limited | Compositions of gnrh related compounds and processes of preparation |
| EP2172193A1 (en) * | 2008-10-02 | 2010-04-07 | Capsulution Nanoscience AG | Improved nanoparticulate compositions of poorly soluble compounds |
| US9089484B2 (en) | 2010-03-26 | 2015-07-28 | Merrion Research Iii Limited | Pharmaceutical compositions of selective factor Xa inhibitors for oral administration |
| US8802114B2 (en) | 2011-01-07 | 2014-08-12 | Merrion Research Iii Limited | Pharmaceutical compositions of iron for oral administration |
| MX377929B (es) | 2011-08-10 | 2025-03-10 | Magforce Ag | Aglomeracion de nanoparticulas recubiertas con alcoxisilano magnetico. |
| ES2655622T3 (es) * | 2012-04-30 | 2018-02-20 | Tillotts Pharma Ag | Una formulación de fármaco de liberación retardada |
| US9763887B2 (en) | 2013-03-15 | 2017-09-19 | Allergan Pharmaceuticals International Limited | Mesalamine pharmaceutical composition with multiple dosage elements for reduced delivery variability |
| JP7211704B2 (ja) | 2015-01-29 | 2023-01-24 | ノヴォ ノルディスク アー/エス | Glp-1アゴニスト及び腸溶コーティングを含む錠剤 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2246037B2 (de) * | 1972-09-20 | 1975-02-27 | Taeschner & Co, 8831 Kipfenberg | Peroral anwendbares Arzneimittel mit verzögerter Resorbierbarkeit in Suspensionsform |
| FR2471186A1 (fr) * | 1979-12-10 | 1981-06-19 | Roussel Uclaf | Nouveaux comprimes a delitescence colique, ainsi que leur procede de preparation |
| ZA825384B (en) * | 1981-07-31 | 1983-05-25 | Tillott J B Ltd | Orally administrable pharmaceutical compositions |
| SE457505B (sv) * | 1984-01-10 | 1989-01-09 | Lejus Medical Ab | Laminatbelagd oral farmaceutisk komposition och foerfarande foer dess framstaellning |
| US4627851A (en) * | 1984-10-26 | 1986-12-09 | Alza Corporation | Colonic-therapeutic delivery system |
| FR2576213B1 (fr) * | 1985-01-21 | 1989-02-24 | Cortial | Nouveau procede d'obtention de formes pharmaceutiques a liberation prolongee |
| US4775536A (en) * | 1986-02-24 | 1988-10-04 | Bristol-Myers Company | Enteric coated tablet and process for making |
| US5296236A (en) * | 1988-09-16 | 1994-03-22 | Recordati S.A., Chemical And Pharmaceutical Company | Controlled release therapeutic system for a liquid pharmaceutical formulations |
| US4996047A (en) * | 1988-11-02 | 1991-02-26 | Richardson-Vicks, Inc. | Sustained release drug-resin complexes |
| JPH0813748B2 (ja) * | 1990-04-23 | 1996-02-14 | 帝國製薬株式会社 | 大腸崩壊性ポリペプチド系経口製剤 |
-
1993
- 1993-11-05 EP EP93924185A patent/EP0667148B1/en not_active Expired - Lifetime
- 1993-11-05 DE DE69332082T patent/DE69332082T2/de not_active Expired - Fee Related
- 1993-11-05 US US08/432,202 patent/US5654004A/en not_active Expired - Fee Related
- 1993-11-05 CA CA002148465A patent/CA2148465C/en not_active Expired - Fee Related
- 1993-11-05 KR KR1019950701773A patent/KR0157280B1/ko not_active Expired - Fee Related
- 1993-11-05 ES ES93924185T patent/ES2176209T3/es not_active Expired - Lifetime
- 1993-11-05 AU AU53768/94A patent/AU5376894A/en not_active Abandoned
- 1993-11-05 WO PCT/JP1993/001608 patent/WO1994010983A1/ja not_active Ceased
- 1993-11-05 DK DK93924185T patent/DK0667148T3/da active
Also Published As
| Publication number | Publication date |
|---|---|
| EP0667148A4 (en) | 1997-02-26 |
| EP0667148A1 (en) | 1995-08-16 |
| CA2148465A1 (en) | 1994-05-26 |
| EP0667148B1 (en) | 2002-07-03 |
| AU5376894A (en) | 1994-06-08 |
| DE69332082D1 (de) | 2002-08-08 |
| KR950703938A (ko) | 1995-11-17 |
| CA2148465C (en) | 1999-11-02 |
| KR0157280B1 (ko) | 1998-11-16 |
| DK0667148T3 (da) | 2002-07-22 |
| DE69332082T2 (de) | 2003-02-06 |
| US5654004A (en) | 1997-08-05 |
| WO1994010983A1 (fr) | 1994-05-26 |
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