IS1766B - Aðferð við að fá fram 3-{2-[4-(6-flúor-bensó[D]isoxasól-3-ýl)píperidín-1-ýl]-etýl}-2-metýl-6,7,8,9-fjórhýdró-4H-pýridó[1,2-A]pýrimidín-4-on - Google Patents

Aðferð við að fá fram 3-{2-[4-(6-flúor-bensó[D]isoxasól-3-ýl)píperidín-1-ýl]-etýl}-2-metýl-6,7,8,9-fjórhýdró-4H-pýridó[1,2-A]pýrimidín-4-on

Info

Publication number
IS1766B
IS1766B IS4259A IS4259A IS1766B IS 1766 B IS1766 B IS 1766B IS 4259 A IS4259 A IS 4259A IS 4259 A IS4259 A IS 4259A IS 1766 B IS1766 B IS 1766B
Authority
IS
Iceland
Prior art keywords
isoxazol
pyrido
pyrimidin
piperidin
benzo
Prior art date
Application number
IS4259A
Other languages
English (en)
Other versions
IS4259A (is
Inventor
Dalmases Barjoan Pere
Marquillas Olondriz Francisco
Huguet Clotet Joan
Bosch Rovira Ana
Carlos Del Castillo Nieto Juan
María Caldero Ges José
Original Assignee
Vita Cientifica
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vita Cientifica filed Critical Vita Cientifica
Publication of IS4259A publication Critical patent/IS4259A/is
Publication of IS1766B publication Critical patent/IS1766B/is

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IS4259A 1994-02-11 1995-02-08 Aðferð við að fá fram 3-{2-[4-(6-flúor-bensó[D]isoxasól-3-ýl)píperidín-1-ýl]-etýl}-2-metýl-6,7,8,9-fjórhýdró-4H-pýridó[1,2-A]pýrimidín-4-on IS1766B (is)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES09400252A ES2074966B1 (es) 1994-02-11 1994-02-11 Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il)piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a)pirimidin-4-ona.

Publications (2)

Publication Number Publication Date
IS4259A IS4259A (is) 1995-08-12
IS1766B true IS1766B (is) 2001-03-15

Family

ID=8285178

Family Applications (1)

Application Number Title Priority Date Filing Date
IS4259A IS1766B (is) 1994-02-11 1995-02-08 Aðferð við að fá fram 3-{2-[4-(6-flúor-bensó[D]isoxasól-3-ýl)píperidín-1-ýl]-etýl}-2-metýl-6,7,8,9-fjórhýdró-4H-pýridó[1,2-A]pýrimidín-4-on

Country Status (14)

Country Link
KR (1) KR100221108B1 (is)
AT (1) AT405401B (is)
CZ (1) CZ286398B6 (is)
EG (1) EG20877A (is)
ES (1) ES2074966B1 (is)
FI (1) FI110000B (is)
GR (1) GR1002344B (is)
HU (1) HU222110B1 (is)
IS (1) IS1766B (is)
NO (1) NO306022B1 (is)
PL (1) PL181420B1 (is)
PT (1) PT101654B (is)
RU (1) RU2123004C1 (is)
SK (1) SK281752B6 (is)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2101646B1 (es) * 1995-04-12 1998-04-01 Ferrer Int Nuevo compuesto derivado del cromeno.
ES2144355B1 (es) * 1997-12-30 2001-01-01 Ferrer Int Compuestos derivados del cromeno.
DE60009959T2 (de) * 2000-05-05 2005-03-31 Rpg Life Sciences Limited Verfahren zur herstellung von antipsychotischem 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-a]pyrimidin-4-on
PL365608A1 (en) 2000-08-14 2005-01-10 Teva Pharmaceutical Industries Ltd. Preparation of risperidone
ES2197801B1 (es) * 2002-03-05 2005-03-16 Ferrer Internacional,S.A Procedimiento de obtencion de la 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il) piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a ) pirimidin-4-ona.
KR20040034996A (ko) 2002-10-18 2004-04-29 한미약품 주식회사 리스페리돈의 개선된 제조방법
CN100390146C (zh) 2002-11-13 2008-05-28 斯索恩有限公司 制备利培酮的方法和用于该方法的中间体
RU2310653C1 (ru) * 2006-07-17 2007-11-20 Государственное образовательное учреждение высшего профессионального образования "Кубанский государственный технологический университет" (ГОУВПО "КубГТУ") СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ 2-МЕТИЛ-5-(5-МЕТИЛ-2-ФУРИЛ)-4,10-ДИГИДРО-3H-ПИРИДАЗИНО[1,6-b]ИЗОХИНОЛИН-10-ОНА (ВАРИАНТЫ)
BRPI0809837A2 (pt) * 2007-04-19 2014-11-11 Youxin Li "composto para tratamento de distúrbios mentais, saldo do composto para tratamento de distúrbios mentais, composição farmacéutica e uso do composto para tratamento de distúrbios mentais"

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT327199B (de) * 1971-10-14 1976-01-26 Sumitomo Chemical Co Verfahren zur herstellung von neuen nitrochinazolinonen
US4352811A (en) * 1981-11-12 1982-10-05 Hoechst-Roussel Pharmaceuticals Inc. 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4485107A (en) * 1982-11-01 1984-11-27 Janssen Pharmaceutica N.V. [[Bis(aryl)methylene]-1-piperidinyl]alkyl-pyrimidinones
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) * 1987-07-13 1990-12-25 Hoechst-Roussel Pharmaceuticals Inc. N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

Also Published As

Publication number Publication date
CZ32995A3 (en) 1995-09-13
NO950501L (no) 1995-08-14
PT101654B (pt) 2002-01-30
KR950032196A (ko) 1995-12-20
FI950579A0 (fi) 1995-02-10
ES2074966A1 (es) 1995-09-16
EG20877A (en) 2000-05-31
ES2074966B1 (es) 1996-06-16
SK281752B6 (sk) 2001-07-10
FI950579L (fi) 1995-08-12
GR1002344B (el) 1996-05-24
PL181420B1 (pl) 2001-07-31
AT405401B (de) 1999-08-25
FI110000B (fi) 2002-11-15
HU9500418D0 (en) 1995-03-28
HUT70169A (en) 1995-09-28
SK15695A3 (en) 1995-10-11
CZ286398B6 (en) 2000-04-12
NO306022B1 (no) 1999-09-06
RU2123004C1 (ru) 1998-12-10
RU95101859A (ru) 1997-03-20
PT101654A (pt) 1995-09-12
IS4259A (is) 1995-08-12
ATA24995A (de) 1998-12-15
HU222110B1 (hu) 2003-04-28
PL307200A1 (en) 1995-08-21
NO950501D0 (no) 1995-02-09
KR100221108B1 (ko) 1999-09-15

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