NO950501L - Fremgangsmåte til å oppnå 3-æ2[4-(6-fluoro-benzo[dÅisoxazol-3-yl)piperidin-1-ylÅ-etylå-2-metyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-aÅpyrimidin-4-on - Google Patents

Fremgangsmåte til å oppnå 3-æ2[4-(6-fluoro-benzo[dÅisoxazol-3-yl)piperidin-1-ylÅ-etylå-2-metyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-aÅpyrimidin-4-on

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Publication number
NO950501L
NO950501L NO950501A NO950501A NO950501L NO 950501 L NO950501 L NO 950501L NO 950501 A NO950501 A NO 950501A NO 950501 A NO950501 A NO 950501A NO 950501 L NO950501 L NO 950501L
Authority
NO
Norway
Prior art keywords
daisoxazol
aåpyrimidin
pyrido
piperidin
benzo
Prior art date
Application number
NO950501A
Other languages
English (en)
Other versions
NO306022B1 (no
NO950501D0 (no
Inventor
Pere Dalmases Barjoan
Francisco Marquillas Olondritz
Joan Huguet Clotet
Ana Bosch Rovira
Juan Carlos Del Castillo Nieto
Jose Maria Caldero Ges
Original Assignee
Vita Invest Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vita Invest Sa filed Critical Vita Invest Sa
Publication of NO950501D0 publication Critical patent/NO950501D0/no
Publication of NO950501L publication Critical patent/NO950501L/no
Publication of NO306022B1 publication Critical patent/NO306022B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO950501A 1994-02-11 1995-02-09 Fremgangsmåte til å oppnå 3-{2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidin-1-yl]-etyl}-2-metyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-on NO306022B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES09400252A ES2074966B1 (es) 1994-02-11 1994-02-11 Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il)piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a)pirimidin-4-ona.

Publications (3)

Publication Number Publication Date
NO950501D0 NO950501D0 (no) 1995-02-09
NO950501L true NO950501L (no) 1995-08-14
NO306022B1 NO306022B1 (no) 1999-09-06

Family

ID=8285178

Family Applications (1)

Application Number Title Priority Date Filing Date
NO950501A NO306022B1 (no) 1994-02-11 1995-02-09 Fremgangsmåte til å oppnå 3-{2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidin-1-yl]-etyl}-2-metyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-on

Country Status (14)

Country Link
KR (1) KR100221108B1 (no)
AT (1) AT405401B (no)
CZ (1) CZ286398B6 (no)
EG (1) EG20877A (no)
ES (1) ES2074966B1 (no)
FI (1) FI110000B (no)
GR (1) GR1002344B (no)
HU (1) HU222110B1 (no)
IS (1) IS1766B (no)
NO (1) NO306022B1 (no)
PL (1) PL181420B1 (no)
PT (1) PT101654B (no)
RU (1) RU2123004C1 (no)
SK (1) SK281752B6 (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2101646B1 (es) * 1995-04-12 1998-04-01 Ferrer Int Nuevo compuesto derivado del cromeno.
ES2144355B1 (es) * 1997-12-30 2001-01-01 Ferrer Int Compuestos derivados del cromeno.
ATE264329T1 (de) * 2000-05-05 2004-04-15 Rpg Life Sciences Ltd Verfahren zur herstellung von antipsychotischem 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-
ATE401313T1 (de) 2000-08-14 2008-08-15 Teva Pharma Herstellung von risperidon
ES2197801B1 (es) * 2002-03-05 2005-03-16 Ferrer Internacional,S.A Procedimiento de obtencion de la 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il) piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a ) pirimidin-4-ona.
KR20040034996A (ko) 2002-10-18 2004-04-29 한미약품 주식회사 리스페리돈의 개선된 제조방법
EP1560814A1 (en) 2002-11-13 2005-08-10 Synthon B.V. Process for making risperidone and intermediates therefor
RU2310653C1 (ru) * 2006-07-17 2007-11-20 Государственное образовательное учреждение высшего профессионального образования "Кубанский государственный технологический университет" (ГОУВПО "КубГТУ") СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ 2-МЕТИЛ-5-(5-МЕТИЛ-2-ФУРИЛ)-4,10-ДИГИДРО-3H-ПИРИДАЗИНО[1,6-b]ИЗОХИНОЛИН-10-ОНА (ВАРИАНТЫ)
US8314110B2 (en) * 2007-04-19 2012-11-20 Youxin Li Compounds for treating mental disorders, and preparation and uses thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT327199B (de) * 1971-10-14 1976-01-26 Sumitomo Chemical Co Verfahren zur herstellung von neuen nitrochinazolinonen
US4352811A (en) * 1981-11-12 1982-10-05 Hoechst-Roussel Pharmaceuticals Inc. 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4485107A (en) * 1982-11-01 1984-11-27 Janssen Pharmaceutica N.V. [[Bis(aryl)methylene]-1-piperidinyl]alkyl-pyrimidinones
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) * 1987-07-13 1990-12-25 Hoechst-Roussel Pharmaceuticals Inc. N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

Also Published As

Publication number Publication date
FI950579A0 (fi) 1995-02-10
HUT70169A (en) 1995-09-28
IS4259A (is) 1995-08-12
PT101654B (pt) 2002-01-30
KR950032196A (ko) 1995-12-20
CZ32995A3 (en) 1995-09-13
PT101654A (pt) 1995-09-12
HU9500418D0 (en) 1995-03-28
ES2074966B1 (es) 1996-06-16
FI110000B (fi) 2002-11-15
PL307200A1 (en) 1995-08-21
KR100221108B1 (ko) 1999-09-15
RU2123004C1 (ru) 1998-12-10
IS1766B (is) 2001-03-15
NO306022B1 (no) 1999-09-06
FI950579L (fi) 1995-08-12
RU95101859A (ru) 1997-03-20
SK15695A3 (en) 1995-10-11
ATA24995A (de) 1998-12-15
HU222110B1 (hu) 2003-04-28
GR1002344B (el) 1996-05-24
CZ286398B6 (en) 2000-04-12
EG20877A (en) 2000-05-31
SK281752B6 (sk) 2001-07-10
ES2074966A1 (es) 1995-09-16
PL181420B1 (pl) 2001-07-31
AT405401B (de) 1999-08-25
NO950501D0 (no) 1995-02-09

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