ATA24995A - Verfahren zur herstellung von 3-(2-(4-(6-fluor- benzo(d)isoxazol-3-yl)piperidin-1-yl)-ethyl) - 2-methyl-6,7,8,9-tetrahydro-4h- pyrido(1,2-a)pyrimidin-4-on - Google Patents

Verfahren zur herstellung von 3-(2-(4-(6-fluor- benzo(d)isoxazol-3-yl)piperidin-1-yl)-ethyl) - 2-methyl-6,7,8,9-tetrahydro-4h- pyrido(1,2-a)pyrimidin-4-on

Info

Publication number: ATA24995A
Authority: AT; Austria
Prior art keywords: isoxazol; pyrido; pyrimidin; benzo; tetrahydro
Prior art date: 1994-02-11

Application number

AT0024995A

Other languages

English (en)

Other versions

AT405401B (de

Original Assignee

Vita Invest Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-02-11

Filing date

1995-02-10

Publication date

1998-12-15

1995-02-10 Application filed by Vita Invest Sa filed Critical Vita Invest Sa

1998-12-15 Publication of ATA24995A publication Critical patent/ATA24995A/de

1999-08-25 Application granted granted Critical

1999-08-25 Publication of AT405401B publication Critical patent/AT405401B/de

Links

RAPZEAPATHNIPO-UHFFFAOYSA-N risperidone Chemical compound FC1=CC=C2C(C3CCN(CC3)CCC=3C(=O)N4CCCCC4=NC=3C)=NOC2=C1 RAPZEAPATHNIPO-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

AT0024995A 1994-02-11 1995-02-10 Verfahren zur herstellung von 3-(2-(4-(6-fluor- benzo(d)isoxazol-3-yl)piperidin-1-yl)-ethyl) - 2-methyl-6,7,8,9-tetrahydro-4h- pyrido(1,2-a)pyrimidin-4-on AT405401B (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
ES09400252A ES2074966B1 (es)	1994-02-11	1994-02-11	Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il)piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a)pirimidin-4-ona.

Publications (2)

Publication Number	Publication Date
ATA24995A true ATA24995A (de)	1998-12-15
AT405401B AT405401B (de)	1999-08-25

Family

ID=8285178

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT0024995A AT405401B (de)	1994-02-11	1995-02-10	Verfahren zur herstellung von 3-(2-(4-(6-fluor- benzo(d)isoxazol-3-yl)piperidin-1-yl)-ethyl) - 2-methyl-6,7,8,9-tetrahydro-4h- pyrido(1,2-a)pyrimidin-4-on

Country Status (14)

Country	Link
KR (1)	KR100221108B1 (de)
AT (1)	AT405401B (de)
CZ (1)	CZ286398B6 (de)
EG (1)	EG20877A (de)
ES (1)	ES2074966B1 (de)
FI (1)	FI110000B (de)
GR (1)	GR1002344B (de)
HU (1)	HU222110B1 (de)
IS (1)	IS1766B (de)
NO (1)	NO306022B1 (de)
PL (1)	PL181420B1 (de)
PT (1)	PT101654B (de)
RU (1)	RU2123004C1 (de)
SK (1)	SK281752B6 (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2101646B1 (es) *	1995-04-12	1998-04-01	Ferrer Int	Nuevo compuesto derivado del cromeno.
ES2144355B1 (es) *	1997-12-30	2001-01-01	Ferrer Int	Compuestos derivados del cromeno.
DE60009959T2 (de) *	2000-05-05	2005-03-31	Rpg Life Sciences Limited	Verfahren zur herstellung von antipsychotischem 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-a]pyrimidin-4-on
PL365608A1 (en)	2000-08-14	2005-01-10	Teva Pharmaceutical Industries Ltd.	Preparation of risperidone
ES2197801B1 (es) *	2002-03-05	2005-03-16	Ferrer Internacional,S.A	Procedimiento de obtencion de la 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il) piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a ) pirimidin-4-ona.
KR20040034996A (ko)	2002-10-18	2004-04-29	한미약품 주식회사	리스페리돈의 개선된 제조방법
CN100390146C (zh)	2002-11-13	2008-05-28	斯索恩有限公司	制备利培酮的方法和用于该方法的中间体
RU2310653C1 (ru) *	2006-07-17	2007-11-20	Государственное образовательное учреждение высшего профессионального образования "Кубанский государственный технологический университет" (ГОУВПО "КубГТУ")	СПОСОБ ПОЛУЧЕНИЯ ПРОИЗВОДНЫХ 2-МЕТИЛ-5-(5-МЕТИЛ-2-ФУРИЛ)-4,10-ДИГИДРО-3H-ПИРИДАЗИНО[1,6-b]ИЗОХИНОЛИН-10-ОНА (ВАРИАНТЫ)
BRPI0809837A2 (pt) *	2007-04-19	2014-11-11	Youxin Li	"composto para tratamento de distúrbios mentais, saldo do composto para tratamento de distúrbios mentais, composição farmacéutica e uso do composto para tratamento de distúrbios mentais"

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AT327199B (de) *	1971-10-14	1976-01-26	Sumitomo Chemical Co	Verfahren zur herstellung von neuen nitrochinazolinonen
US4352811A (en) *	1981-11-12	1982-10-05	Hoechst-Roussel Pharmaceuticals Inc.	3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4485107A (en) *	1982-11-01	1984-11-27	Janssen Pharmaceutica N.V.	[[Bis(aryl)methylene]-1-piperidinyl]alkyl-pyrimidinones
US4804663A (en) *	1985-03-27	1989-02-14	Janssen Pharmaceutica N.V.	3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) *	1987-07-13	1990-12-25	Hoechst-Roussel Pharmaceuticals Inc.	N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

1994
- 1994-02-11 ES ES09400252A patent/ES2074966B1/es not_active Expired - Fee Related
1995
- 1995-02-01 GR GR950100035A patent/GR1002344B/el not_active IP Right Cessation
- 1995-02-07 SK SK156-95A patent/SK281752B6/sk not_active IP Right Cessation
- 1995-02-08 IS IS4259A patent/IS1766B/is unknown
- 1995-02-08 CZ CZ1995329A patent/CZ286398B6/cs not_active IP Right Cessation
- 1995-02-09 EG EG11595A patent/EG20877A/xx active
- 1995-02-09 PT PT101654A patent/PT101654B/pt active IP Right Grant
- 1995-02-09 NO NO950501A patent/NO306022B1/no not_active IP Right Cessation
- 1995-02-10 AT AT0024995A patent/AT405401B/de not_active IP Right Cessation
- 1995-02-10 PL PL95307200A patent/PL181420B1/pl not_active IP Right Cessation
- 1995-02-10 FI FI950579A patent/FI110000B/fi not_active IP Right Cessation
- 1995-02-10 RU RU95101859/04A patent/RU2123004C1/ru not_active IP Right Cessation
- 1995-02-10 HU HU9500418A patent/HU222110B1/hu not_active IP Right Cessation
- 1995-02-11 KR KR1019950002516A patent/KR100221108B1/ko not_active Expired - Fee Related

Also Published As

Publication number	Publication date
CZ32995A3 (en)	1995-09-13
NO950501L (no)	1995-08-14
PT101654B (pt)	2002-01-30
KR950032196A (ko)	1995-12-20
FI950579A0 (fi)	1995-02-10
ES2074966A1 (es)	1995-09-16
EG20877A (en)	2000-05-31
ES2074966B1 (es)	1996-06-16
SK281752B6 (sk)	2001-07-10
FI950579L (fi)	1995-08-12
GR1002344B (el)	1996-05-24
PL181420B1 (pl)	2001-07-31
IS1766B (is)	2001-03-15
AT405401B (de)	1999-08-25
FI110000B (fi)	2002-11-15
HU9500418D0 (en)	1995-03-28
HUT70169A (en)	1995-09-28
SK15695A3 (en)	1995-10-11
CZ286398B6 (en)	2000-04-12
NO306022B1 (no)	1999-09-06
RU2123004C1 (ru)	1998-12-10
RU95101859A (ru)	1997-03-20
PT101654A (pt)	1995-09-12
IS4259A (is)	1995-08-12
HU222110B1 (hu)	2003-04-28
PL307200A1 (en)	1995-08-21
NO950501D0 (no)	1995-02-09
KR100221108B1 (ko)	1999-09-15

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Legal Events

Date	Code	Title
2005-03-15	EIH	Change in the person of patent owner
2008-01-15	EIH	Change in the person of patent owner
2010-05-15	EIH	Change in the person of patent owner
2011-08-15	ELJ	Ceased due to non-payment of the annual fee