IS8147A - Nýjar línkómýsín afleiður sem búa yfir örverueyðandi virkni - Google Patents

Nýjar línkómýsín afleiður sem búa yfir örverueyðandi virkni

Info

Publication number: IS8147A
Authority: IS; Iceland
Prior art keywords: new; antimicrobial activity; derivatives possessing; lincomycin derivatives; possessing antimicrobial
Prior art date: 2003-06-17

Application number

IS8147A

Other languages

English (en)

Icelandic (is)

Inventor

Gustaf Lewis Jason

Anandan Sampath-Kumar

Fremont

O'dowd Hardwin

Federovich Gordeev Mikhail

Original Assignee

Vicuron Pharmaceuticals Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-06-17

Filing date

2005-11-24

Publication date

2005-11-24

2003-08-15 Priority claimed from US10/642,807 external-priority patent/US7164011B2/en

2004-02-11 Priority claimed from US10/777,455 external-priority patent/US7199105B2/en

2005-11-24 Application filed by Vicuron Pharmaceuticals Inc. filed Critical Vicuron Pharmaceuticals Inc.

2005-11-24 Publication of IS8147A publication Critical patent/IS8147A/is

Links

230000000845 anti-microbial effect Effects 0.000 title 1
OJMMVQQUTAEWLP-KIDUDLJLSA-N lincomycin Chemical class CN1C[C@H](CCC)C[C@H]1C(=O)N[C@H]([C@@H](C)O)[C@@H]1[C@H](O)[C@H](O)[C@@H](O)[C@@H](SC)O1 OJMMVQQUTAEWLP-KIDUDLJLSA-N 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
- C07H15/16—Lincomycin; Derivatives thereof

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Genetics & Genomics (AREA)
Epidemiology (AREA)
Biotechnology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Crystallography & Structural Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Saccharide Compounds (AREA)

IS8147A 2003-06-17 2005-11-24 Nýjar línkómýsín afleiður sem búa yfir örverueyðandi virkni IS8147A (is)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
US47950203P	2003-06-17	2003-06-17
US47929603P	2003-06-17	2003-06-17
US10/642,807 US7164011B2 (en)	2002-08-15	2003-08-15	Lincomycin derivatives possessing antibacterial activity
US10/777,455 US7199105B2 (en)	2002-08-15	2004-02-11	Lincomycin derivatives possessing antibacterial activity
PCT/US2004/019689 WO2005012320A2 (en)	2003-06-17	2004-06-17	Novel lincomycin derivatives possessing antimicrobial activity

Publications (1)

Publication Number	Publication Date
IS8147A true IS8147A (is)	2005-11-24

Family

ID=40203032

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS8147A IS8147A (is)	2003-06-17	2005-11-24	Nýjar línkómýsín afleiður sem búa yfir örverueyðandi virkni

Country Status (16)

Country	Link
EP (1)	EP1644393A2 (sr)
JP (1)	JP2007516172A (sr)
KR (1)	KR20060091050A (sr)
AU (1)	AU2004261550A1 (sr)
BR (1)	BRPI0411534A (sr)
CA (1)	CA2528592A1 (sr)
EC (1)	ECSP056233A (sr)
GE (1)	GEP20084437B (sr)
IL (1)	IL172183A0 (sr)
IS (1)	IS8147A (sr)
MA (1)	MA27860A1 (sr)
MX (1)	MXPA05013915A (sr)
NO (1)	NO20055893L (sr)
OA (1)	OA13179A (sr)
RS (1)	RS20050931A (sr)
WO (1)	WO2005012320A2 (sr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1529052A2 (en)	2002-08-15	2005-05-11	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
US7199105B2 (en)	2002-08-15	2007-04-03	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
US7199106B2 (en)	2003-06-17	2007-04-03	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antimicrobial activity
US7256177B2 (en)	2003-06-17	2007-08-14	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
EP1654268A2 (en) *	2003-06-17	2006-05-10	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
US7361743B2 (en)	2004-02-11	2008-04-22	Pfizer Inc	Lincomycin derivatives possessing antibacterial activity
JP2009507793A (ja) *	2005-08-31	2009-02-26	ワイス	グリシルサイクリンの９−アミノカルボニル置換誘導体
US7871982B2 (en)	2005-12-09	2011-01-18	Meiji Seika Kaisha, Ltd.	Lincomycin derivatives and antimicrobial agents comprising the same as active ingredient
US7879808B2 (en)	2007-05-31	2011-02-01	Meiji Seika Kaisha, Ltd.	Lincomycin derivatives and antimicrobial agents comprising the same as active ingredient
WO2008146919A1 (ja)	2007-05-31	2008-12-04	Meiji Seika Kaisha, Ltd.	リンコサミド誘導体及びこれを有効成分とする抗菌剤
US20130267699A1 (en)	2011-06-24	2013-10-10	California Institute Of Technology	Quaternary heteroatom containing compounds
US8822679B2 (en) *	2011-06-24	2014-09-02	California Institute Of Technology	Quaternary heteroatom containing compounds
US10421696B2 (en)	2014-12-18	2019-09-24	California Institute Of Technology	Enantioselective synthesis of α-quaternary mannich adducts by palladium-catalyzed allylic alkylation
CN107922373A (zh)	2015-03-27	2018-04-17	加利福尼亚技术学院	使用低催化剂浓度和稳定的预催化剂的不对称催化脱羧烷基烷基化
EP3426391A4 (en)	2016-03-11	2019-08-28	California Institute of Technology	COMPOSITIONS AND METHODS FOR ACYLATING LACTAMEN
EP3480190B1 (en)	2017-11-01	2023-01-04	California Institute of Technology	Methods for enantioselective allylic alkylation of esters, lactones, and lactams with unactivated allylic alcohols
EP3699173A1 (en)	2018-10-18	2020-08-26	California Institute of Technology	Gem-disubstituted pyrrolidines, piperazines, and diazepanes, and compositions and methods of making the same
CN110357839A (zh) *	2019-08-29	2019-10-22	重庆经致制药技术开发有限公司	布瓦西坦手性中间体的制备方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3268556A (en) *	1964-04-13	1966-08-23	Upjohn Co	Novel lincomycin derivatives
NL128232C (sr) *	1964-04-13
NL146501C (sr) *	1964-07-01
US3282917A (en) *	1964-08-17	1966-11-01	Upjohn Co	Methyl n-(1-alkyl-4-alkoxy-prolyl)-alpha-thiolincosaminide compounds and process therefor
NL140527B (nl) *	1965-02-08	1973-12-17	Upjohn Co	Werkwijze ter bereiding van aan lincomycine verwante verbindingen.
US3496163A (en) *	1965-02-08	1970-02-17	Upjohn Co	7-halo-7-deoxylincomycins and process for preparing the same
US3555007A (en) *	1968-07-22	1971-01-12	Upjohn Co	7-deoxy-7-halo lincomycin d derivatives
US3549615A (en) *	1968-10-17	1970-12-22	Upjohn Co	Lincomycin derivatives and process for producing the same
DE2118636A1 (de) *	1970-04-20	1971-11-04	The Upjohn Co., Kalamazoo, Mich. (V.StA.)	3-Nucleotide von Lincomycin und deren Analogen, Verfahren zu ihrer Herstellung und ihre Verwendung in therapeutischen Präparaten
US3787390A (en) *	1971-06-23	1974-01-22	Upjohn Co	Analogs of lincomycin and process
US3849396A (en) *	1973-01-08	1974-11-19	Upjohn Co	Lincomycin and clindamycin 1-o-ethers
US3923602A (en) *	1973-10-25	1975-12-02	Upjohn Co	Composition of matter and process
JPS5641239A (en) *	1979-09-13	1981-04-17	Hitachi Cable Ltd	Flame-retardant composition
US4278789A (en) *	1979-11-23	1981-07-14	The Upjohn Company	Lincomycin compounds
EP1529052A2 (en) *	2002-08-15	2005-05-11	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
JP2007528360A (ja) *	2003-06-17	2007-10-11	ビキュロン・ファーマシューティカルズ・インコーポレイテッド	抗菌活性を有するリンコマイシン誘導体

2004
- 2004-06-17 RS YUP-2005/0931A patent/RS20050931A/sr unknown
- 2004-06-17 KR KR1020057024291A patent/KR20060091050A/ko not_active Ceased
- 2004-06-17 BR BRPI0411534-1A patent/BRPI0411534A/pt not_active IP Right Cessation
- 2004-06-17 OA OA1200500364A patent/OA13179A/en unknown
- 2004-06-17 EP EP04776816A patent/EP1644393A2/en not_active Withdrawn
- 2004-06-17 JP JP2006517464A patent/JP2007516172A/ja active Pending
- 2004-06-17 MX MXPA05013915A patent/MXPA05013915A/es unknown
- 2004-06-17 WO PCT/US2004/019689 patent/WO2005012320A2/en not_active Ceased
- 2004-06-17 GE GEAP20049117A patent/GEP20084437B/en unknown
- 2004-06-17 AU AU2004261550A patent/AU2004261550A1/en not_active Abandoned
- 2004-06-17 CA CA002528592A patent/CA2528592A1/en not_active Abandoned
2005
- 2005-11-24 IL IL172183A patent/IL172183A0/en unknown
- 2005-11-24 IS IS8147A patent/IS8147A/is unknown
- 2005-12-12 NO NO20055893A patent/NO20055893L/no not_active Application Discontinuation
- 2005-12-16 EC EC2005006233A patent/ECSP056233A/es unknown
- 2005-12-16 MA MA28672A patent/MA27860A1/fr unknown

Also Published As

Publication number	Publication date
MA27860A1 (fr)	2006-04-03
WO2005012320A3 (en)	2005-10-20
WO2005012320A2 (en)	2005-02-10
IL172183A0 (en)	2011-08-01
KR20060091050A (ko)	2006-08-17
BRPI0411534A (pt)	2006-08-22
JP2007516172A (ja)	2007-06-21
HK1090061A1 (zh)	2006-12-15
GEP20084437B (en)	2008-07-25
CA2528592A1 (en)	2005-02-10
EP1644393A2 (en)	2006-04-12
ECSP056233A (es)	2006-04-19
MXPA05013915A (es)	2006-07-03
OA13179A (en)	2006-12-13
NO20055893L (no)	2006-03-14
RS20050931A (sr)	2008-04-04
AU2004261550A1 (en)	2005-02-10

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DK1644024T3 (da)	2019-10-07	Antimikrobielle skylleopløsninger
DE60332094D1 (de)	2010-05-27	Aktive pulsspektrophotometrie
EP1618087A4 (en)	2007-01-31	ANTIBACTERIAL AGENTS
IS8322A (is)	2006-02-22	Tálmar Akt virkni
PL379212A1 (pl)	2006-08-07	Kompozycje bakteriobójcze, sposoby i układy
EP1560556A4 (en)	2011-07-06	ANTIMICROBIAL COMPOSITIONS
PT3127553T (pt)	2022-01-24	Conjugados de derivado da caliqueamicina - transportador
ATE383771T1 (de)	2008-02-15	Fungizide wirkstoffkombinationen
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EP1970377A4 (en)	2013-02-27	LINCOMYCIN DERIVATIVE AND ANTIBACTERIAL AGENT CONTAINING THIS AS AN ACTIVE SUBSTANCE
ATE392813T1 (de)	2008-05-15	Fungizide wirkstoffkombination
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IL172183A0 (en)	2011-08-01	Novel lincomycin derivatives possessing antimicrobial activity
DE502004005409D1 (de)	2007-12-20	Sprühfeuchtwerk
PT1556377E (pt)	2006-10-31	Ciclopropil-tienil-carboxamidas como fungicidas
PT1381609E (pt)	2005-05-31	5-halogeno-6-fenil-7-fluoroalquilamino-triazolopirimidinas como fungicidas
IL166476A0 (en)	2006-01-15	Lincomycin derivatives possessing antibacterial activity
IS7795A (is)	2005-04-11	Pyrrólafleiður sem efnasambönd gegn sveppagerlum
GB0303683D0 (en)	2003-03-19	Antimicrobial agents
BRPI0400485B1 (pt)	2013-12-17	Revestimento antimicrobiano
ITMI20020161A0 (it)	2002-01-31	Filtro attivo
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EP1483253A4 (en)	2007-03-21	ANTIMICROBIAL MEDIUM