MA28798B1 - Dérivés de triazolopyridinylsufanyle servant d'inhibiteurs de kinase MAP P38 - Google Patents

Dérivés de triazolopyridinylsufanyle servant d'inhibiteurs de kinase MAP P38

Info

Publication number
MA28798B1
MA28798B1 MA29676A MA29676A MA28798B1 MA 28798 B1 MA28798 B1 MA 28798B1 MA 29676 A MA29676 A MA 29676A MA 29676 A MA29676 A MA 29676A MA 28798 B1 MA28798 B1 MA 28798B1
Authority
MA
Morocco
Prior art keywords
triazolopyridinylsufanyl
map
derivatives
kinase inhibitors
kinase
Prior art date
Application number
MA29676A
Other languages
English (en)
Inventor
John Paul Mathias
David Simon Millan
Russell Andrew Lewthwaite
Christopher Phillips
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0418015A external-priority patent/GB0418015D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of MA28798B1 publication Critical patent/MA28798B1/fr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Virology (AREA)
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  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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MA29676A 2004-08-12 2007-02-12 Dérivés de triazolopyridinylsufanyle servant d'inhibiteurs de kinase MAP P38 MA28798B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0418015A GB0418015D0 (en) 2004-08-12 2004-08-12 New compounds
US69155905P 2005-06-17 2005-06-17

Publications (1)

Publication Number Publication Date
MA28798B1 true MA28798B1 (fr) 2007-08-01

Family

ID=35783420

Family Applications (1)

Application Number Title Priority Date Filing Date
MA29676A MA28798B1 (fr) 2004-08-12 2007-02-12 Dérivés de triazolopyridinylsufanyle servant d'inhibiteurs de kinase MAP P38

Country Status (34)

Country Link
US (2) US7511057B2 (fr)
EP (1) EP1778686B9 (fr)
JP (1) JP4084836B2 (fr)
AP (1) AP2326A (fr)
AR (1) AR050692A1 (fr)
AT (1) ATE412652T1 (fr)
AU (1) AU2005273612B2 (fr)
BR (1) BRPI0514255A (fr)
CA (1) CA2576297C (fr)
CR (1) CR8918A (fr)
CU (1) CU23497A3 (fr)
CY (1) CY1108788T1 (fr)
DE (1) DE602005010714D1 (fr)
DK (1) DK1778686T3 (fr)
EA (1) EA012119B1 (fr)
EC (1) ECSP077232A (fr)
ES (1) ES2314690T3 (fr)
GE (1) GEP20104973B (fr)
GT (1) GT200500218A (fr)
HN (1) HN2005000418A (fr)
HR (1) HRP20080608T3 (fr)
IL (1) IL181047A (fr)
MA (1) MA28798B1 (fr)
MX (1) MX2007001759A (fr)
MY (1) MY140021A (fr)
NL (1) NL1029726C2 (fr)
NO (1) NO339320B1 (fr)
NZ (1) NZ552868A (fr)
PL (1) PL1778686T3 (fr)
PT (1) PT1778686E (fr)
SI (1) SI1778686T1 (fr)
SV (1) SV2006002193A (fr)
TN (1) TNSN07050A1 (fr)
WO (1) WO2006018718A2 (fr)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7572807B2 (en) * 2005-06-09 2009-08-11 Bristol-Myers Squibb Company Heteroaryl 11-beta-hydroxysteroid dehydrogenase type I inhibitors
US7579360B2 (en) * 2005-06-09 2009-08-25 Bristol-Myers Squibb Company Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors
US20090012079A1 (en) * 2006-02-09 2009-01-08 Russell Andrew Lewthwaite Triazolopyridine Compounds
JP5244369B2 (ja) * 2006-11-10 2013-07-24 富士フイルム株式会社 ５−アミノピラゾール誘導体の製造方法、アゾ色素
EP1992344A1 (fr) 2007-05-18 2008-11-19 Institut Curie P38 alpha comme cible therapeutique pour les maladies associées á une mutation de FGFR3
US8119658B2 (en) * 2007-10-01 2012-02-21 Bristol-Myers Squibb Company Triazolopyridine 11-beta hydroxysteroid dehydrogenase type I inhibitors
CA2712574C (fr) 2008-02-04 2014-01-07 Pfizer Limited Forme polymorphe
US8498729B2 (en) 2008-08-29 2013-07-30 Smp Logic Systems Llc Manufacturing execution system for use in manufacturing baby formula
CA2736913A1 (fr) * 2008-09-12 2010-03-18 Dorothee Viemann Moyens et procedes pour evaluer une therapie avec un inhibiteur de map-kinase p38
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