|
US3169967A
(en)
|
1957-11-14 |
1965-02-16 |
Ciba Geigy Corp |
Methyl o-lower alkanoyl-reserpates
|
|
US3037980A
(en)
|
1955-08-18 |
1962-06-05 |
Burroughs Wellcome Co |
Pyrrolopyrimidine vasodilators and method of making them
|
|
US3506643A
(en)
|
1966-12-09 |
1970-04-14 |
Max Thiel |
N**6-aralkyl-adenosine derivatives
|
|
DE2139107A1
(de)
|
1971-08-04 |
1973-02-15 |
Merck Patent Gmbh |
Heterocyclisch substituierte adenosinverbindungen
|
|
US3962443A
(en)
|
1972-08-14 |
1976-06-08 |
Dainippon Pharmaceutical Co., Ltd. |
Antibacterial pharmaceutical compositions and processes for preparation thereof
|
|
DE2248232A1
(de)
|
1972-10-02 |
1974-04-11 |
Basf Ag |
4-thiopyrimido eckige klammer auf 4,5-d eckige klammer zu pyrimidine
|
|
AR204003A1
(es)
|
1973-04-03 |
1975-11-12 |
Dainippon Pharmaceutical Co |
Procedimiento para preparar compuestos derivados del acido 2-(1-piperazinil)-5-oxopirido-(2,3-d)pirimidino-6-carboxilico y sus sales farmaceuticamente aceptables
|
|
US3936454A
(en)
|
1973-08-14 |
1976-02-03 |
Warner-Lambert Company |
5-Amino-4-chloro-6-(substituted amino)-pyrimidines
|
|
US3862189A
(en)
|
1973-08-14 |
1975-01-21 |
Warner Lambert Co |
Aralkyl-substituted purines and pyrimidines as antianginal bronchodilator agents
|
|
DK3375A
(fr)
|
1974-01-25 |
1975-09-15 |
Ciba Geigy Ag |
|
|
JPS587626B2
(ja)
|
1974-02-13 |
1983-02-10 |
大日本製薬株式会社 |
ナフチリジン オヨビ キノリンユウドウタイノセイホウ
|
|
JPS5359663A
(en)
|
1976-11-09 |
1978-05-29 |
Sumitomo Chem Co Ltd |
2-halogeno methyl indole derivatives and process for praparation of the same
|
|
JPS5392767A
(en)
|
1977-01-27 |
1978-08-15 |
Sumitomo Chem Co Ltd |
Preparation of 2-phthalimidomethylindole derivatives
|
|
JPS5625234A
(en)
|
1979-08-02 |
1981-03-11 |
Hitachi Denshi Ltd |
Dropout display system
|
|
JPS56123981A
(en)
|
1981-02-23 |
1981-09-29 |
Dainippon Pharmaceut Co Ltd |
Preparation of 1,4-disubstituted piperazine
|
|
JPS5883698A
(ja)
|
1981-11-13 |
1983-05-19 |
Takeda Chem Ind Ltd |
キノン化合物およびその製造法
|
|
JPS58162949A
(ja)
|
1982-03-20 |
1983-09-27 |
Konishiroku Photo Ind Co Ltd |
ハロゲン化銀カラ−写真感光材料
|
|
JPS6067709U
(ja)
|
1983-10-14 |
1985-05-14 |
三洋電機株式会社 |
ヘア−ドライヤ−
|
|
JPS6190153A
(ja)
|
1984-10-09 |
1986-05-08 |
Fuji Photo Film Co Ltd |
ハロゲン化銀写真感光材料の処理方法
|
|
JPS6263591U
(fr)
|
1985-06-29 |
1987-04-20 |
|
|
|
JPS62103640A
(ja)
|
1985-07-18 |
1987-05-14 |
Fuji Photo Film Co Ltd |
ハロゲン化銀カラ−写真感光材料
|
|
JPS635783Y2
(fr)
|
1985-10-17 |
1988-02-17 |
|
|
|
JPH07119970B2
(ja)
|
1986-04-18 |
1995-12-20 |
富士写真フイルム株式会社 |
画像形成方法
|
|
JPS6310746A
(ja)
|
1986-07-01 |
1988-01-18 |
Tanabe Seiyaku Co Ltd |
ナフタレン誘導体
|
|
CA1324609C
(fr)
|
1986-07-30 |
1993-11-23 |
Eastman Kodak Company |
Element et processus photographiques
|
|
JPS6427257U
(fr)
|
1987-08-11 |
1989-02-16 |
|
|
|
US4861701A
(en)
|
1987-10-05 |
1989-08-29 |
Eastman Kodak Company |
Photographic element and process comprising a compound which comprises two timing groups in sequence
|
|
AT388372B
(de)
|
1987-10-08 |
1989-06-12 |
Tanabe Seiyaku Co |
Neue naphthalinderivate und sie enthaltende pharmazeutika
|
|
JPH01250316A
(ja)
|
1987-12-28 |
1989-10-05 |
Tanabe Seiyaku Co Ltd |
抗脂血剤
|
|
EP0364598A4
(en)
|
1988-03-02 |
1992-01-15 |
Yoshitomi Pharmaceutical Industries, Ltd. |
3,4-dihydrothieno 2,3-d¨pyrimidine compounds and pharmaceutical application thereof
|
|
US5208250A
(en)
|
1988-05-25 |
1993-05-04 |
Warner-Lambert Company |
Known and selected novel arylmethylenyl derivatives of thiazolidinones, imidazolidinones and oxazolidinones useful as antiallergy agents and anti-inflammatory agents
|
|
ES2149761T3
(es)
|
1990-04-25 |
2000-11-16 |
Nissan Chemical Ind Ltd |
Derivado de piridazinona.
|
|
SU1712359A1
(ru)
|
1990-05-07 |
1992-02-15 |
Уфимский Нефтяной Институт |
Гидрохлорид 8 @ -гидроксихинолинового эфира 8-гидроксихинолин-7-карбоновой кислоты, в качестве бактерицида дл подавлени сульфатвосстанавливающих бактерий и культур РSеUDомоNаS и АRтнRовастеR
|
|
EP0464612B1
(fr)
|
1990-06-28 |
1998-05-13 |
Fuji Photo Film Co., Ltd. |
Matériaux photographiques à l'halogénure d'argent
|
|
EP0481614A1
(fr)
|
1990-10-01 |
1992-04-22 |
Merck & Co. Inc. |
Pyridopyrimidinones substituées et hétérocyles apparantés comme antagonistes de la angiotensine II
|
|
US5480883A
(en)
|
1991-05-10 |
1996-01-02 |
Rhone-Poulenc Rorer Pharmaceuticals Inc. |
Bis mono- and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase
|
|
AU1625192A
(en)
|
1991-05-31 |
1992-12-03 |
Zeneca Limited |
Heterocyclic derivatives
|
|
JP3108483B2
(ja)
|
1991-09-30 |
2000-11-13 |
日清製粉株式会社 |
インドール誘導体およびこれを有効成分とする抗潰瘍薬
|
|
HUT64064A
(en)
|
1992-02-13 |
1993-11-29 |
Chinoin Gyogyszer Es Vegyeszet |
Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient
|
|
US5521184A
(en)
|
1992-04-03 |
1996-05-28 |
Ciba-Geigy Corporation |
Pyrimidine derivatives and processes for the preparation thereof
|
|
AU3933493A
(en)
|
1992-04-24 |
1993-11-29 |
E.I. Du Pont De Nemours And Company |
Arthropodicidal and fungicidal aminopyrimidines
|
|
TW229140B
(fr)
|
1992-06-05 |
1994-09-01 |
Shell Internat Res Schappej B V |
|
|
FR2714907B1
(fr)
|
1994-01-07 |
1996-03-29 |
Union Pharma Scient Appl |
Nouveaux dérivés de l'Adénosine, leurs procédés de préparation, compositions pharmaceutiques les contenant.
|
|
US6342501B1
(en)
|
1994-02-25 |
2002-01-29 |
The Regents Of The University Of Michigan |
Pyrrolo[2,3-d] pyrimidines as antiviral agents
|
|
JPH09176162A
(ja)
|
1995-12-22 |
1997-07-08 |
Toubishi Yakuhin Kogyo Kk |
チアゾリジンジオン誘導体及びその製造法並びにそれを含む医薬組成物
|
|
JPH1025294A
(ja)
|
1996-03-26 |
1998-01-27 |
Akira Matsuda |
縮合ヘテロ環誘導体、その製造法及びそれを含有する悪性腫瘍治療剤
|
|
CA2258728C
(fr)
|
1996-06-19 |
2011-09-27 |
Rhone Poulenc Rorer Limited |
Composes azabicycliques substitues et leur utilisation en tant qu'inhibiteurs de la production de tnf et de la photodiesterase cyclique d'amp
|
|
JP4667543B2
(ja)
|
1996-07-03 |
2011-04-13 |
大日本住友製薬株式会社 |
新規プリン誘導体
|
|
US5866702A
(en)
|
1996-08-02 |
1999-02-02 |
Cv Therapeutics, Incorporation |
Purine inhibitors of cyclin dependent kinase 2
|
|
US6630496B1
(en)
|
1996-08-26 |
2003-10-07 |
Genetics Institute Llc |
Inhibitors of phospholipase enzymes
|
|
JPH10231297A
(ja)
|
1997-02-20 |
1998-09-02 |
Japan Energy Corp |
新規なアデニン−1−n−オキシド誘導体およびその医薬用途
|
|
DE69824632T2
(de)
|
1997-11-12 |
2005-06-09 |
Mitsubishi Chemical Corp. |
Purinderivate und medikamente, welche dieselben als aktiven bestandteil enthalten
|
|
TW572758B
(en)
|
1997-12-22 |
2004-01-21 |
Sumitomo Pharma |
Type 2 helper T cell-selective immune response inhibitors comprising purine derivatives
|
|
EE200000522A
(et)
|
1998-02-25 |
2002-02-15 |
Genetics Institute, Inc. |
Fosfolipaas A2 ensüümi inhibiitor, seda sisaldav farmatseutiline kompositsioon ning meetod fosfolipaasensüümi toime pärssimiseks
|
|
ID27280A
(id)
|
1998-02-25 |
2001-03-22 |
Genetics Inst |
Inhibitor-inhibitor dari enzim-enzim fosfolipase
|
|
US6828344B1
(en)
|
1998-02-25 |
2004-12-07 |
Genetics Institute, Llc |
Inhibitors of phospholipase enzymes
|
|
US6479487B1
(en)
|
1998-02-26 |
2002-11-12 |
Aventis Pharmaceuticals Inc. |
6, 9-disubstituted 2-[trans-(4-aminocyclohexyl)amino] purines
|
|
SK16352000A3
(sk)
|
1998-05-04 |
2002-07-02 |
Zentaris Ag |
Indolové deriváty, spôsob ich výroby, ich použitie na liečivá obsahujúce tieto zlúčeniny
|
|
ATE482945T1
(de)
|
1998-05-26 |
2010-10-15 |
Chugai Pharmaceutical Co Ltd |
Heterozyklische indolderivate und mono- oder diazaindol-derivate
|
|
JP3997651B2
(ja)
|
1998-06-24 |
2007-10-24 |
コニカミノルタホールディングス株式会社 |
新規色素及び画像記録材料及び感熱転写材料及びインクジェット記録液
|
|
ES2342240T3
(es)
|
1998-08-11 |
2010-07-02 |
Novartis Ag |
Derivados de isoquinolina con actividad que inhibe la angiogenia.
|
|
IL141513A0
(en)
|
1998-08-25 |
2002-03-10 |
Uab Research Foundation |
Inhibitors of bacterial nad synthetase
|
|
ATE228375T1
(de)
*
|
1998-09-04 |
2002-12-15 |
Univ Michigan |
THIOMOLYBDAT VERBUNDEN MIT MINDESTENS EINEM KOHLENHYDRAT, UND SEINE VERWENDUNG ZUR VORBEUGUNG UND BEHANDLUNG VON ERKRANKUNGEN, DIE DURCH EINE ANORMALE VASKULARISIERUNG GEKENNZEICHNET SIND, WIE Z.B. KREBS, ßFEUCHTEß MAKULADEGENERATION, RHEUMATOIDE ARTHRITIS
|
|
US6133031A
(en)
|
1999-08-19 |
2000-10-17 |
Isis Pharmaceuticals Inc. |
Antisense inhibition of focal adhesion kinase expression
|
|
IL144675A0
(en)
|
1999-02-01 |
2002-05-23 |
Cv Therapeutics Inc |
PURINE INHIBITORS OF CYCLIN DEPENDENT KINASE 2 AND IkB-α
|
|
GB9905075D0
(en)
|
1999-03-06 |
1999-04-28 |
Zeneca Ltd |
Chemical compounds
|
|
JP2000281654A
(ja)
|
1999-03-26 |
2000-10-10 |
Tanabe Seiyaku Co Ltd |
イソキノリン誘導体
|
|
DE19932571A1
(de)
|
1999-07-13 |
2001-01-18 |
Clariant Gmbh |
Verfahren zur Herstellung von Biarylen unter Palladophosphacyclobutan-Katalyse
|
|
JP2001151771A
(ja)
|
1999-09-10 |
2001-06-05 |
Kyowa Hakko Kogyo Co Ltd |
含窒素芳香族複素環誘導体
|
|
GB0004890D0
(en)
|
2000-03-01 |
2000-04-19 |
Astrazeneca Uk Ltd |
Chemical compounds
|
|
US6436965B1
(en)
|
2000-03-02 |
2002-08-20 |
Merck Frosst Canada & Co. |
PDE IV inhibiting amides, compositions and methods of treatment
|
|
EP1138328A1
(fr)
|
2000-03-29 |
2001-10-04 |
Eli Lilly And Company Limited |
Dérivés du naphthalène comme médicaments du SNC
|
|
US6667300B2
(en)
|
2000-04-25 |
2003-12-23 |
Icos Corporation |
Inhibitors of human phosphatidylinositol 3-kinase delta
|
|
EP1294358B1
(fr)
|
2000-06-28 |
2004-08-18 |
Smithkline Beecham Plc |
Procede de broyage par voie humide
|
|
CN1331340A
(zh)
|
2000-06-30 |
2002-01-16 |
上海博德基因开发有限公司 |
一种新的多肽——人拓扑异构酶12.1和编码这种多肽的多核苷酸
|
|
PT1300398E
(pt)
|
2000-07-05 |
2006-07-31 |
Astellas Pharma Inc |
Processos e composicoes para terapias do cancro, utilizando genes que codificam o interferao-beta
|
|
FR2814073B1
(fr)
|
2000-09-21 |
2005-06-24 |
Yang Ji Chemical Company Ltd |
Composition pharmaceutique antifongique et/ou antiparasitaire et nouveaux derives de l'indole a titre de principes actifs d'une telle composition
|
|
DOP2002000334A
(es)
|
2001-02-14 |
2002-08-30 |
Warner Lambert Co |
Pirimidinas biciclicas como inhibidores de metaloproteinasas de matriz
|
|
SE0100568D0
(sv)
|
2001-02-20 |
2001-02-20 |
Astrazeneca Ab |
Compounds
|
|
CN1659143A
(zh)
|
2001-03-01 |
2005-08-24 |
盐野义制药株式会社 |
具有hiv整合酶抑制活性的含氮杂芳基化合物
|
|
UA76977C2
(en)
|
2001-03-02 |
2006-10-16 |
Icos Corp |
Aryl- and heteroaryl substituted chk1 inhibitors and their use as radiosensitizers and chemosensitizers
|
|
EP1372643A1
(fr)
|
2001-03-30 |
2004-01-02 |
Smithkline Beecham Corporation |
Pyralopyridines, leur procede de preparation et leur utilisation en tant que composes therapeutiques
|
|
WO2002078701A1
(fr)
|
2001-03-30 |
2002-10-10 |
Smithkline Beecham Corporation |
Utilisation de pyrazolopyridines comme composes therapeutiques
|
|
AU2002305143A1
(en)
|
2001-04-27 |
2002-11-11 |
Smithkline Beecham Corporation |
Pyrazolo'1,5-a!pyridine derivatives
|
|
CZ294535B6
(cs)
|
2001-08-02 |
2005-01-12 |
Ústav Experimentální Botaniky Avčr |
Heterocyklické sloučeniny na bázi N6-substituovaného adeninu, způsoby jejich přípravy, jejich použití pro přípravu léčiv, kosmetických přípravků a růstových regulátorů, farmaceutické přípravky, kosmetické přípravky a růstové regulátory tyto sloučeniny obsahující
|
|
GB0121033D0
(en)
|
2001-08-30 |
2001-10-24 |
Novartis Ag |
Organic compounds
|
|
US8124625B2
(en)
|
2001-09-14 |
2012-02-28 |
Shionogi & Co., Ltd. |
Method of enhancing the expression of apolipoprotein AI using olefin derivatives
|
|
CN100391958C
(zh)
|
2001-09-19 |
2008-06-04 |
安万特医药股份有限公司 |
化合物
|
|
BR0212829A
(pt)
|
2001-09-26 |
2004-08-03 |
Bayer Pharmaceuticals Corp |
Derivados de 1,8-naftiridina e seu uso para tratar diabetes e distúrbios relacionados
|
|
US7217710B2
(en)
|
2001-10-02 |
2007-05-15 |
Smithkline Beecham Corporation |
Substituted pyrazolopyrimidines
|
|
PT1441737E
(pt)
|
2001-10-30 |
2006-12-29 |
Dana Farber Cancer Inst Inc |
Derivados de estrutura como inibidores da actividade do receptor de tirosina cinase flt3
|
|
US7262164B2
(en)
|
2001-11-09 |
2007-08-28 |
Enzon, Inc. |
Polymeric thiol-linked prodrugs employing benzyl elimination systems
|
|
EP1314733A1
(fr)
|
2001-11-22 |
2003-05-28 |
Aventis Pharma Deutschland GmbH |
Indole-2-carboxamides comme inhibiteurs du facteur Xa
|
|
ATE372341T1
(de)
|
2001-12-06 |
2007-09-15 |
Merck & Co Inc |
Inhibitoren von mitotischem kinesin
|
|
ATE424388T1
(de)
|
2001-12-06 |
2009-03-15 |
Merck & Co Inc |
Mitotische kinesinhemmer
|
|
TW200301135A
(en)
|
2001-12-27 |
2003-07-01 |
Otsuka Maryland Res Inst Inc |
Pharmaceutical compositions comprising a multifunctional phosphodiesterase inhibitor and an adenosine uptake inhibitor
|
|
US7402595B2
(en)
|
2002-02-13 |
2008-07-22 |
Takeda Pharmaceutical Company Limited |
JNK inhibitor
|
|
AU2003225668A1
(en)
|
2002-03-01 |
2003-09-16 |
Pintex Pharmaceutical, Inc. |
Pin1-modulating compounds and methods of use thereof
|
|
AU2003222106A1
(en)
|
2002-04-03 |
2003-10-20 |
Bristol-Myers Squibb Company |
Thiopene-based tricyclic compounds and pharmaceutical compositions comprising same
|
|
BR0309581A
(pt)
|
2002-05-06 |
2005-03-29 |
Genelabs Tech Inc |
Derivados de nucleosìdeo para tratamento de infecção por vìrus de hepatite c
|
|
PE20040522A1
(es)
|
2002-05-29 |
2004-09-28 |
Novartis Ag |
Derivados de diarilurea dependientes de la cinasa de proteina
|
|
GB0215676D0
(en)
|
2002-07-05 |
2002-08-14 |
Novartis Ag |
Organic compounds
|
|
ATE404537T1
(de)
|
2002-08-13 |
2008-08-15 |
Shionogi & Co |
Heterocyclische verbindungen mit hiv-integrase- hemmender wirkung
|
|
CA2497765A1
(fr)
|
2002-09-27 |
2004-04-08 |
Sumitomo Pharmaceuticals Co., Ltd. |
Nouveau compose d'adenine et son application
|
|
AR042052A1
(es)
|
2002-11-15 |
2005-06-08 |
Vertex Pharma |
Diaminotriazoles utiles como inhibidores de proteinquinasas
|
|
DK2316831T3
(da)
|
2002-11-21 |
2013-06-10 |
Novartis Ag |
2-(Morpholin-4-yl)pyrimidiner som phosphotidylinositol (PI)-3-kinaseinhibitorer samt deres anvendelse ved behandling af cancer
|
|
US7494987B2
(en)
|
2002-11-25 |
2009-02-24 |
Mochida Pharmaceutical Co., Ltd. |
Agent for treating respiratory diseases containing 4-hydroxypiperidine derivative as active ingredient
|
|
UA80767C2
(en)
|
2002-12-20 |
2007-10-25 |
Pfizer Prod Inc |
Pyrimidine derivatives for the treatment of abnormal cell growth
|
|
CA2512000C
(fr)
|
2002-12-26 |
2011-08-09 |
Eisai Co., Ltd. |
Modulateurs selectifs des recepteurs d'oestrogene
|
|
CZ294538B6
(cs)
|
2002-12-30 |
2005-01-12 |
Ústav Experimentální Botaniky Akademie Vědčeské Re |
Substituční deriváty N6-benzyladenosinu, způsob jejich přípravy, jejich použití pro přípravu léčiv, kosmetických přípravků a růstových regulátorů, farmaceutické přípravky, kosmetické přípravky a růstové regulátory tyto sloučeniny obsahující
|
|
RU2233842C1
(ru)
|
2003-01-13 |
2004-08-10 |
Петров Владимир Иванович |
Производные пурина, обладающие противовирусной активностью
|
|
AR043692A1
(es)
|
2003-02-06 |
2005-08-10 |
Novartis Ag |
2-cianopirrolopirimidinas y sus usos farmaceuticos
|
|
GB0304640D0
(en)
|
2003-02-28 |
2003-04-02 |
Novartis Ag |
Organic compounds
|
|
GB0305929D0
(en)
|
2003-03-14 |
2003-04-23 |
Novartis Ag |
Organic compounds
|
|
SE0300908D0
(sv)
|
2003-03-31 |
2003-03-31 |
Astrazeneca Ab |
Azaindole derivatives, preparations thereof, uses thereof and compositions containing them
|
|
US7129264B2
(en)
|
2003-04-16 |
2006-10-31 |
Bristol-Myers Squibb Company |
Biarylmethyl indolines and indoles as antithromboembolic agents
|
|
EP1619948A4
(fr)
|
2003-05-05 |
2007-02-14 |
Neurogen Corp |
Derives d'imidazolopyrazine et de triazolopyrazine substitues: des ligands des recepteurs gabaa
|
|
ES2339862T3
(es)
|
2003-06-20 |
2010-05-26 |
Novartis Vaccines And Diagnostics, Inc. |
Compuestos de piridino 1,2-a-pirimidin-4-ona como agentes anticancerosos.
|
|
WO2005000309A2
(fr)
|
2003-06-27 |
2005-01-06 |
Ionix Pharmaceuticals Limited |
Composes chimiques
|
|
JP4570015B2
(ja)
|
2003-07-14 |
2010-10-27 |
クミアイ化学工業株式会社 |
2−イソオキサゾリン誘導体及びそれを有効成分として含有する除草剤
|
|
JP2007502776A
(ja)
|
2003-08-15 |
2007-02-15 |
アイアールエム・リミテッド・ライアビリティ・カンパニー |
Rtk阻害剤としての6−置換アニリノプリン類
|
|
NZ546611A
(en)
|
2003-09-18 |
2010-02-26 |
Conforma Therapeutics Corp |
Novel heterocyclic compounds as HSP90-inhibitors
|
|
US7709476B2
(en)
|
2003-09-23 |
2010-05-04 |
Merck Sharp & Dohme Corp. |
Isoquinolinone potassium channel inhibitors
|
|
PE20050952A1
(es)
|
2003-09-24 |
2005-12-19 |
Novartis Ag |
Derivados de isoquinolina como inhibidores de b-raf
|
|
WO2005074603A2
(fr)
|
2004-02-03 |
2005-08-18 |
Abbott Laboratories |
Utilisation d'aminobenzoxazoles comme agents therapeutiques
|
|
WO2005077948A1
(fr)
|
2004-02-16 |
2005-08-25 |
Daiichi Pharmaceutical Co., Ltd. |
Composes heterocycliques fongicides
|
|
CN1560035A
(zh)
|
2004-03-12 |
2005-01-05 |
沈阳药科大学 |
5-羟基吲哚-3-羧酸脂类衍生物
|
|
WO2005091857A2
(fr)
|
2004-03-12 |
2005-10-06 |
Bayer Pharmaceuticals Corporation |
Derives de 1,6-naphtyridine et 1,8-naphtyridine et leur utilisation pour le traitement du diabete et de troubles associes
|
|
WO2005092892A1
(fr)
|
2004-03-26 |
2005-10-06 |
Dainippon Sumitomo Pharma Co., Ltd. |
Compose 8-oxoadenine
|
|
AU2005231440B9
(en)
|
2004-04-02 |
2012-02-23 |
Dogwood Pharmaceuticals, Inc. |
Selective antagonists of A2A adenosine receptors
|
|
LT2612862T
(lt)
|
2004-05-13 |
2017-01-25 |
Icos Corporation |
Chinazolinonai kaip žmogaus fosfatidilinozitol-3-kinazės delta inhibitoriai
|
|
MXPA06013250A
(es)
|
2004-05-14 |
2007-02-28 |
Abbott Lab |
Inhibidores de quinasa como agentes terapeuticos.
|
|
MXPA06014247A
(es)
|
2004-06-10 |
2007-03-12 |
Irm Llc |
Compuestos y composiciones como inhibidores de la proteina quinasa.
|
|
US20070287703A1
(en)
|
2004-07-22 |
2007-12-13 |
Astrazeneca Ab |
Fused Pyrimidones Useful in the Treatment and the Prevention of Cancer
|
|
DE102004044221A1
(de)
|
2004-09-14 |
2006-03-16 |
Boehringer Ingelheim Pharma Gmbh & Co. Kg |
Neue 3-Methyl-7-butinyl-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
|
|
GB0420719D0
(en)
|
2004-09-17 |
2004-10-20 |
Addex Pharmaceuticals Sa |
Novel allosteric modulators
|
|
EP1807399A2
(fr)
|
2004-10-19 |
2007-07-18 |
Novartis Vaccines and Diagnostics, Inc. |
Derives d'indole et de benzimidazole
|
|
EP1807417A2
(fr)
|
2004-11-04 |
2007-07-18 |
Neurogen Corporation |
Dérivés hétéroaryles de pyrazolylméthyle
|
|
US9512125B2
(en)
|
2004-11-19 |
2016-12-06 |
The Regents Of The University Of California |
Substituted pyrazolo[3.4-D] pyrimidines as anti-inflammatory agents
|
|
RU2007123675A
(ru)
|
2004-11-24 |
2008-12-27 |
Новартис АГ (CH) |
Комбинации ингибиторов jak
|
|
US20080287469A1
(en)
|
2005-02-17 |
2008-11-20 |
Diacovo Thomas G |
Phosphoinositide 3-Kinase Inhibitors for Inhibiting Leukocyte Accumulation
|
|
DE602006015658D1
(de)
|
2005-06-27 |
2010-09-02 |
Amgen Inc |
Entzündungshemmende arylnitrilverbindungen
|
|
FR2889192A1
(fr)
|
2005-07-27 |
2007-02-02 |
Cytomics Systems Sa |
Composes antifongiques, compositions contenant ces composes et leurs utilisations
|
|
JP2009504769A
(ja)
|
2005-08-16 |
2009-02-05 |
ジェンザイム・コーポレーション |
ケモカイン受容体結合化合物
|
|
US7642270B2
(en)
|
2005-09-14 |
2010-01-05 |
Janssen Pharmaceutica N.V. |
5-oxo-5,8-dihydro-pyrido-pyrimidine as inhibitors of c-fms kinase
|
|
EP1939202A4
(fr)
|
2005-09-22 |
2010-06-16 |
Dainippon Sumitomo Pharma Co |
Nouveau composé de l'adénine
|
|
GB0520657D0
(en)
|
2005-10-11 |
2005-11-16 |
Ludwig Inst Cancer Res |
Pharmaceutical compounds
|
|
WO2007053452A1
(fr)
|
2005-11-01 |
2007-05-10 |
Targegen, Inc. |
Inhibiteurs de kinase de type biaryl-méta-pyrimidine
|
|
EP1783114A1
(fr)
|
2005-11-03 |
2007-05-09 |
Novartis AG |
Dérivés de N-(hétéro)aryle indole comme pesticides
|
|
ATE486875T1
(de)
|
2005-11-10 |
2010-11-15 |
Chemocentryx Inc |
Substituierte chinolone und verwendungsverfahren
|
|
HUE028588T2
(hu)
|
2005-12-13 |
2016-12-28 |
Incyte Holdings Corp |
Heteroaril-szubsztituált pirrolo[2,3-b]piridinek és pirrolo[2,3-b]pirimidinek mint Janus-kináz inhibitorok
|
|
US7989461B2
(en)
|
2005-12-23 |
2011-08-02 |
Amgen Inc. |
Substituted quinazolinamine compounds for the treatment of cancer
|
|
WO2007087548A2
(fr)
|
2006-01-25 |
2007-08-02 |
Smithkline Beecham Corporation |
Composés chimiques
|
|
PE20071025A1
(es)
|
2006-01-31 |
2007-10-17 |
Mitsubishi Tanabe Pharma Corp |
Compuesto amina trisustituido
|
|
PE20070978A1
(es)
|
2006-02-14 |
2007-11-15 |
Novartis Ag |
COMPUESTOS HETEROCICLICOS COMO INHIBIDORES DE FOSFATIDILINOSITOL 3-QUINASAS (PI3Ks)
|
|
US20090069304A1
(en)
|
2006-03-03 |
2009-03-12 |
Shionogi & Co., Ltd. |
Mmp-13 selective inhibitor
|
|
US20100273776A1
(en)
|
2006-03-29 |
2010-10-28 |
FOLDRx PHARMACEUTICALS, INC |
Inhibition of alpha-synuclein toxicity
|
|
KR20150038395A
(ko)
|
2006-04-04 |
2015-04-08 |
더 리젠트스 오브 더 유니이버시티 오브 캘리포니아 |
키나제 길항물질
|
|
CA2656067C
(fr)
|
2006-06-23 |
2014-08-12 |
Radius Health, Inc. |
Traitement de symptomes vasomoteurs par des modulateurs des recepteurs d'oestrogene selectifs
|
|
US20080004253A1
(en)
|
2006-06-30 |
2008-01-03 |
Bryan James Branstetter |
Thiazolopyrimidine modulators of TRPV1
|
|
US20080009508A1
(en)
|
2006-07-10 |
2008-01-10 |
Lucie Szucova |
6,9-Disubstituted Purine Derivatives And Their Use For Treating Skin
|
|
AU2007272009A1
(en)
|
2006-07-12 |
2008-01-17 |
Syngenta Limited |
Triazolopyridine derivatives as herbicides
|
|
AU2007282535B9
(en)
|
2006-08-08 |
2013-06-20 |
Chugai Seiyaku Kabushiki Kaisha |
Pyrimidine derivative as PI3K inhibitor and use thereof
|
|
JP5336375B2
(ja)
|
2006-08-30 |
2013-11-06 |
セルゾーム リミテッド |
キナーゼ阻害剤としてのトリアゾール誘導体
|
|
WO2008032033A1
(fr)
|
2006-09-14 |
2008-03-20 |
Astrazeneca Ab |
Dérivés de 4-benzimidazolyl-2-morpholino-6-pipérazinylpyrimidine utilisés en tant que pi3k et inhibiteurs de mtor destinés au traitement de troubles prolifératifs
|
|
EP1972631A1
(fr)
|
2007-03-23 |
2008-09-24 |
Novartis AG |
Imidazopyridazines comme inhibiteurs de kinase lipide PI3K
|
|
US20080114007A1
(en)
|
2006-10-31 |
2008-05-15 |
Player Mark R |
5-oxo-5,8-dihydro-pyrido-pyrimidines as inhibitors of c-fms kinase
|
|
EP2441768A1
(fr)
|
2006-11-13 |
2012-04-18 |
Eli Lilly & Co. |
Thiénopyrimidinones destinées au traitement de troubles inflammatoires et de cancers
|
|
GEP20125658B
(en)
|
2006-11-22 |
2012-10-10 |
Incyte Corp |
Imidazotriazines and imidazo pyrimidines as kinase inhibitors
|
|
CA2672960A1
(fr)
|
2006-12-20 |
2008-07-10 |
Schering Corporation |
Nouveaux inhibiteurs de jnk
|
|
PT2125827E
(pt)
|
2006-12-29 |
2010-11-22 |
Hoffmann La Roche |
Derivados azaespiro
|
|
CA2677493A1
(fr)
|
2007-02-05 |
2008-08-14 |
Xenon Pharmaceuticals Inc. |
Composes de pyridopyrimidinone utiles dans le traitement de maladies ou d'affections vehiculees par les canaux sodiques
|
|
EP2134683A2
(fr)
|
2007-02-12 |
2009-12-23 |
Intermune, Inc. |
Nouveaux inhibiteurs de réplication du virus de l'hépatite c
|
|
TW200902018A
(en)
|
2007-03-20 |
2009-01-16 |
Dainippon Sumitomo Pharma Co |
Novel adenine compound
|
|
US20080233127A1
(en)
|
2007-03-21 |
2008-09-25 |
Wyeth |
Imidazolopyrimidine analogs and their use as pi3 kinase and mtor inhibitors
|
|
CA2680783C
(fr)
|
2007-03-23 |
2012-04-24 |
Amgen Inc. |
Composes heterocycliques et leurs utilisations
|
|
HRP20160350T1
(hr)
|
2007-03-23 |
2016-05-06 |
Amgen Inc. |
Heterociklički spojevi i njihove uporabe
|
|
US8039505B2
(en)
|
2007-04-11 |
2011-10-18 |
University Of Utah Research Foundation |
Compounds for modulating T-cells
|
|
US8633186B2
(en)
|
2007-06-08 |
2014-01-21 |
Senomyx Inc. |
Modulation of chemosensory receptors and ligands associated therewith
|
|
US9603848B2
(en)
|
2007-06-08 |
2017-03-28 |
Senomyx, Inc. |
Modulation of chemosensory receptors and ligands associated therewith
|
|
EP2740731B1
(fr)
|
2007-06-13 |
2016-03-23 |
Incyte Holdings Corporation |
Sels cristallines de l'inhibiteur de janus kinase (r)-3-(4- (7h-pyrrolo [2,3-d] pyrimidin-4-yl)-1h-pyrazol-1-yl) -3-cyclopentylpropanenitrile
|
|
CL2008001709A1
(es)
|
2007-06-13 |
2008-11-03 |
Incyte Corp |
Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras.
|
|
JP2010531304A
(ja)
|
2007-06-18 |
2010-09-24 |
ユニバーシティ オブ ルイビル リサーチ ファウンデーション、インコーポレイテッド |
抗悪性腫瘍活性を有するpfkfb3阻害物質ファミリー
|
|
EP2170888B1
(fr)
|
2007-06-29 |
2015-04-22 |
Gilead Sciences, Inc. |
Dérivés de purine et leur utilisation comme modulateurs du récepteur de type toll-7
|
|
WO2009042294A2
(fr)
|
2007-08-10 |
2009-04-02 |
Burnham Institute For Medical Research |
Activateurs de la phosphatase alcaline non spécifique des tissus (tnap) et leurs utilisations
|
|
WO2009026701A1
(fr)
|
2007-08-29 |
2009-03-05 |
Methylgene Inc. |
Inhibiteurs de sirtuine
|
|
JP2009076865A
(ja)
|
2007-08-29 |
2009-04-09 |
Fujifilm Corp |
有機電界発光素子
|
|
WO2009034386A1
(fr)
|
2007-09-13 |
2009-03-19 |
Astrazeneca Ab |
Dérivés de l'adénine et de la 8-aza-adénine et leurs utilisations
|
|
JP2009080233A
(ja)
|
2007-09-26 |
2009-04-16 |
Kyocera Mita Corp |
電子写真感光体
|
|
CZ300774B6
(cs)
|
2007-10-05 |
2009-08-05 |
Univerzita Palackého |
Substituované 6-(alkylbenzylamino)purinové deriváty pro použití jako antagonisté cytokininových receptoru a prípravky obsahující tyto slouceniny
|
|
WO2009062118A2
(fr)
|
2007-11-07 |
2009-05-14 |
Foldrx Pharmaceuticals, Inc. |
Régulation du trafic de protéines
|
|
WO2009063235A1
(fr)
|
2007-11-13 |
2009-05-22 |
Astrazeneca Ab |
Dérivés de 1,9-dihydro-6h-purin-6-one et leurs utilisations -018
|
|
JP2009120686A
(ja)
|
2007-11-14 |
2009-06-04 |
Toyo Ink Mfg Co Ltd |
光重合開始剤、重合性組成物、および重合物の製造方法。
|
|
US7820665B2
(en)
|
2007-12-19 |
2010-10-26 |
Amgen Inc. |
Imidazopyridazine inhibitors of PI3 kinase for cancer treatment
|
|
WO2009081105A2
(fr)
|
2007-12-21 |
2009-07-02 |
Ucb Pharma S.A. |
Dérivés de quinoxaline et de quinoléine en tant qu'inhibiteurs de kinase
|
|
AU2008345225A1
(en)
|
2007-12-21 |
2009-07-09 |
University Of Rochester |
Method for altering the lifespan of eukaryotic organisms
|
|
WO2009086123A1
(fr)
|
2007-12-21 |
2009-07-09 |
Wyeth |
Composés d'imidazo[1,2-a]pyridine
|
|
WO2009082845A1
(fr)
|
2007-12-28 |
2009-07-09 |
Topharman Shanghai Co., Ltd. |
N-{1-[3-(2-éthoxy-5-(4-éthylpipérazinyl)benzènesulfonyl)-4,5-dihydro-5-oxo-1,2,4-triazin-6-yl]éthyl}butyramide, son procédé de préparation et son utilisation
|
|
US7960397B2
(en)
|
2007-12-28 |
2011-06-14 |
Institute Of Experimental Botany, Academy Of Sciences Of The Czech Republic |
6,9-disubstituted purine derivatives and their use as cosmetics and cosmetic compositions
|
|
US8193182B2
(en)
|
2008-01-04 |
2012-06-05 |
Intellikine, Inc. |
Substituted isoquinolin-1(2H)-ones, and methods of use thereof
|
|
KR20100116607A
(ko)
|
2008-01-11 |
2010-11-01 |
낫코 파마 리미티드 |
항암제로서의 신규한 피라졸로[3,4-d]피리미딘 유도체
|
|
US9089572B2
(en)
|
2008-01-17 |
2015-07-28 |
California Institute Of Technology |
Inhibitors of p97
|
|
JP5608099B2
(ja)
|
2008-01-30 |
2014-10-15 |
ジェネンテック, インコーポレイテッド |
ピラゾロピリミジンpi3k阻害剤化合物および使用方法
|
|
US20110105457A1
(en)
|
2008-04-18 |
2011-05-05 |
Shionogi & Co., Ltd. |
Heterocyclic compound having inhibitory activity on pi3k
|
|
US8119647B2
(en)
|
2008-04-23 |
2012-02-21 |
Glenmark Pharmaceuticals S.A. |
Fused pyrimidineone compounds as TRPV3 modulators
|
|
WO2009140215A2
(fr)
|
2008-05-11 |
2009-11-19 |
Geraghty, Erin |
Procédé pour traiter des infections bactériennes résistant au médicament et d'autres infections par du clioquinol, de la phanquinone et des composés apparentés
|
|
EP2300005A4
(fr)
|
2008-05-28 |
2011-07-13 |
Us Of America As Represented By The Secretary Of The Army On Behalf Of U S Army Medical Res And Mate |
Inhibiteurs à petites molécules de neurotoxines botuliniques
|
|
BRPI0914891A2
(pt)
|
2008-06-20 |
2015-11-24 |
Metabolex Inc |
agonistas de aril gpr119 e usos dos mesmos
|
|
US8026271B2
(en)
|
2008-07-11 |
2011-09-27 |
National Health Research Institutes |
Formulations of indol-3-yl-2-oxoacetamide compounds
|
|
WO2010018458A2
(fr)
|
2008-08-12 |
2010-02-18 |
Crystalgenomics, Inc. |
Dérivés de phénol et leurs procédés d'utilisation
|
|
WO2010036380A1
(fr)
|
2008-09-26 |
2010-04-01 |
Intellikine, Inc. |
Inhibiteurs hétérocycliques de kinases
|
|
CL2009001884A1
(es)
|
2008-10-02 |
2010-05-14 |
Incyte Holdings Corp |
Uso de 3-ciclopentil-3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)propanonitrilo, inhibidor de janus quinasa, y uso de una composición que lo comprende para el tratamiento del ojo seco.
|
|
KR20170060179A
(ko)
|
2008-11-13 |
2017-05-31 |
길리아드 칼리스토가 엘엘씨 |
혈액 종양에 대한 요법
|
|
US20110245209A1
(en)
|
2008-12-16 |
2011-10-06 |
Schering Corporation |
Pyridopyrimidine derivatives and methods of use thereof
|
|
AU2009330821B2
(en)
|
2008-12-24 |
2015-06-11 |
Bial - Portela & Ca, S.A. |
Pharmaceutical compounds
|
|
EP2387575B1
(fr)
|
2009-01-15 |
2013-09-04 |
Anvyl, LLC |
Modulateurs allostériques des récepteurs nicotiniques de l'acétylcholine de type alpha7, leurs dérivés et leurs utilisations
|
|
WO2010083283A2
(fr)
|
2009-01-15 |
2010-07-22 |
Incyte Corporation |
Procédés de préparation d'inhibiteurs des jak et composés intermédiaires apparentés
|
|
US8513284B2
(en)
|
2009-02-13 |
2013-08-20 |
Ucb Pharma, S.A. |
Fused pyridine and pyrazine derivatives as kinase inhibitors
|
|
TW201100428A
(en)
|
2009-03-31 |
2011-01-01 |
Arqule Inc |
Substituted indolo-piperidine compounds
|
|
WO2010118367A2
(fr)
|
2009-04-10 |
2010-10-14 |
Progenics Pharmaceuticals, Inc. |
Pyrimidines antivirales
|
|
JP2012524126A
(ja)
|
2009-04-20 |
2012-10-11 |
ギリアド カリストガ リミテッド ライアビリティ カンパニー |
固形腫瘍の治療方法
|
|
CA2702567A1
(fr)
|
2009-04-28 |
2010-10-28 |
Katch Kan Holdings Ltd. |
Appareil et methode de vidange de solides et de fluides d'un train de tiges servant au forage ou a l'entretien de puits
|
|
WO2010127208A1
(fr)
|
2009-04-30 |
2010-11-04 |
Forest Laboratories Holdings Limited |
Inhibiteurs de l'acétyl-coa carboxylase
|
|
JP5789252B2
(ja)
|
2009-05-07 |
2015-10-07 |
インテリカイン, エルエルシー |
複素環式化合物およびその使用
|
|
BRPI1012108B8
(pt)
|
2009-05-22 |
2021-05-25 |
Incyte Corp |
composto 3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il]octa no- ou heptano-nitrila, sua composição, seus usos e processo para preparar um sal de ácido fosfórico
|
|
NZ596479A
(en)
|
2009-05-22 |
2014-01-31 |
Incyte Corp |
N-(hetero)aryl-pyrrolidine derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines and pyrrol-3-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
|
|
CA2781865A1
(fr)
|
2009-06-25 |
2010-12-29 |
Amgen Inc. |
Derives polycycliques de pyridine et leur utilisation dans le traitement, entre autres, de l'arthrite rhumatoide et de troubles similaires
|
|
JP2012531435A
(ja)
|
2009-06-25 |
2012-12-10 |
アムジエン・インコーポレーテツド |
PI3K阻害剤としての4H−ピリド[1,2−a]ピリミジン−4−オン誘導体
|
|
AR077252A1
(es)
|
2009-06-29 |
2011-08-10 |
Xenon Pharmaceuticals Inc |
Enantiomeros de compuestos de espirooxindol y sus usos como agentes terapeuticos
|
|
FR2947269B1
(fr)
|
2009-06-29 |
2013-01-18 |
Sanofi Aventis |
Nouveaux composes anticancereux
|
|
PE20120693A1
(es)
|
2009-06-29 |
2012-07-04 |
Agios Pharmaceuticals Inc |
Compuestos heterociclos como moduladores de la piruvato cinasa m2 (pkm2)
|
|
EP2448938B9
(fr)
|
2009-06-29 |
2015-06-10 |
Incyte Corporation |
Pyrimidinones comme inhibiteurs de pi3k
|
|
CA2768843A1
(fr)
|
2009-07-21 |
2011-01-27 |
Gilead Calistoga Llc |
Traitement de troubles du foie par des inhibiteurs de pi3k
|
|
AR077974A1
(es)
|
2009-08-28 |
2011-10-05 |
Takeda Pharmaceutical |
Compuestos de hexahidrooxazinopterina para uso como inhibidores de mtor
|
|
TW201113285A
(en)
|
2009-09-01 |
2011-04-16 |
Incyte Corp |
Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
|
|
EA022120B1
(ru)
|
2009-10-20 |
2015-11-30 |
Целльзом Лимитид |
Аналоги гетероциклил пиразолопиримидина в качестве ингибиторов jak
|
|
BR112012009329A2
(pt)
|
2009-10-22 |
2016-06-07 |
Gilead Sciences Inc |
derivados de purina ou deazapurina úteis para o tratamento de infecções virais (inter alia)
|
|
LT2496567T
(lt)
|
2009-11-05 |
2017-11-27 |
Rhizen Pharmaceuticals S.A. |
Nauji benzopirano kinazės moduliatoriai
|
|
UA102336C2
(uk)
|
2009-11-10 |
2013-06-25 |
Пфайзер Інк. |
N1-ПІРАЗОЛСПІРОКЕТОНИ ЯК ІНГІБІТОРИ АЦЕТИЛ-СоА-КАРБОКСИЛАЗ
|
|
WO2011058113A1
(fr)
|
2009-11-12 |
2011-05-19 |
Ucb Pharma S.A. |
Dérivés de pyridine et de pyrazine bicycliques condensés comme inhibiteurs de kinases
|
|
WO2011058111A1
(fr)
|
2009-11-12 |
2011-05-19 |
Ucb Pharma S.A. |
Dérivés d'aminopurine en tant qu'inhibiteurs de kinase
|
|
CN102812033B
(zh)
|
2009-12-10 |
2015-11-25 |
中国医学科学院药物研究所 |
N6-取代腺苷衍生物和n6-取代腺嘌呤衍生物及其用途
|
|
WO2011075630A1
(fr)
|
2009-12-18 |
2011-06-23 |
Incyte Corporation |
Dérivés substitués d'aryles et d'hétéroaryles fusionnés au titre d'inhibiteurs de pi3k
|
|
US8633313B2
(en)
|
2009-12-18 |
2014-01-21 |
Amgen Inc. |
Heterocyclic compounds and their uses
|
|
WO2011075643A1
(fr)
|
2009-12-18 |
2011-06-23 |
Incyte Corporation |
Dérivés condensés d'hétéroaryles substitués à titre d'inhibiteurs de pi3k
|
|
JP2011136925A
(ja)
|
2009-12-28 |
2011-07-14 |
Dainippon Sumitomo Pharma Co Ltd |
含窒素二環性化合物
|
|
RU2547721C2
(ru)
|
2010-01-07 |
2015-04-10 |
ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи |
ТИАЗОЛО [5, 4-d] ПИРИМИДИНЫ И ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ АГРОХИМИЧЕСКИХ СРЕДСТВ
|
|
US8633183B2
(en)
|
2010-01-26 |
2014-01-21 |
Boehringer Ingelheim International Gmbh |
5-alkynyl-pyrimidines
|
|
US20110207754A1
(en)
|
2010-02-18 |
2011-08-25 |
Incyte Corporation |
Cyclobutane and methylcyclobutane derivatives as janus kinase inhibitors
|
|
CA2792508C
(fr)
|
2010-03-10 |
2018-01-16 |
Incyte Corporation |
Derives de piperidin-4-yl azetidine en tant qu'inhibiteurs de jak1
|
|
KR20130028081A
(ko)
|
2010-03-22 |
2013-03-18 |
그렌마크 파머수티칼스 에스. 아. |
피리미딘온 유도체를 포함하는 약제학적 조성물
|
|
UY33304A
(es)
|
2010-04-02 |
2011-10-31 |
Amgen Inc |
Compuestos heterocíclicos y sus usos
|
|
EP2558463A1
(fr)
|
2010-04-14 |
2013-02-20 |
Incyte Corporation |
Dérivés condensés en tant qu'inhibiteurs de i3
|
|
JP5951600B2
(ja)
|
2010-05-21 |
2016-07-13 |
インフィニティー ファーマシューティカルズ, インコーポレイテッド |
キナーゼ調節のための、化合物、組成物および方法
|
|
EA202091303A3
(ru)
|
2010-05-21 |
2021-05-31 |
Инсайт Холдингс Корпорейшн |
Композиция ингибитора jak для местного применения
|
|
WO2011156759A1
(fr)
|
2010-06-11 |
2011-12-15 |
Calistoga Pharmaceuticals, Inc. |
Méthodes de traitement de troubles hématologiques par des composés quinazolinone chez des patients sélectionnés
|
|
US9062055B2
(en)
|
2010-06-21 |
2015-06-23 |
Incyte Corporation |
Fused pyrrole derivatives as PI3K inhibitors
|
|
JP2013530236A
(ja)
|
2010-07-01 |
2013-07-25 |
アムジエン・インコーポレーテツド |
Pi3k活性の阻害剤としての複素環式化合物およびその用途
|
|
MX2012015135A
(es)
|
2010-07-01 |
2013-05-06 |
Amgen Inc |
Compuestos heterociclicos y su uso como inhibidores de la actividad pi3k.
|
|
JP2013533884A
(ja)
|
2010-07-02 |
2013-08-29 |
アムジエン・インコーポレーテツド |
Pi3k活性阻害剤としての複素環化合物およびそれらの使用
|
|
US20130324561A1
(en)
|
2010-09-24 |
2013-12-05 |
Gilead Calistroga Llc. |
Atropisomers of p13k-inhibiting compounds
|
|
US20140031355A1
(en)
|
2010-11-04 |
2014-01-30 |
Amgen Inc. |
Heterocyclic compounds and their uses
|
|
WO2012064973A2
(fr)
|
2010-11-10 |
2012-05-18 |
Infinity Pharmaceuticals, Inc. |
Composés hétérocycliques et utilisations de ceux-ci
|
|
WO2012068343A1
(fr)
|
2010-11-17 |
2012-05-24 |
Amgen Inc. |
Dérivés de quinoléine en tant qu'inhibiteurs de pi3k
|
|
ES2536415T3
(es)
|
2010-11-19 |
2015-05-25 |
Incyte Corporation |
Pirrolopiridinas y pirrolopirimidinas sustituidas heterocíclicas como inhibidores de JAK
|
|
CA2818542A1
(fr)
|
2010-11-19 |
2012-05-24 |
Incyte Corporation |
Derives pyrrolopyridine et pyrrolopyrimidine a substitution cyclobutyle utilises comme inhibiteurs des jak
|
|
EP2651405A2
(fr)
|
2010-12-14 |
2013-10-23 |
Electrophoretics Limited |
Inhibiteurs de caséine kinase 1 (ck1 )
|
|
JP5961187B2
(ja)
|
2010-12-20 |
2016-08-02 |
インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation |
Pi3k阻害剤としてのn−(1−(置換フェニル)エチル)−9h−プリン−6−アミン
|
|
MX2013007261A
(es)
|
2010-12-23 |
2013-11-04 |
Amgen Inc |
Compuestos heterociclicos y sus usos.
|
|
EP3238722B1
(fr)
|
2011-01-10 |
2019-03-13 |
Infinity Pharmaceuticals, Inc. |
Formes solides d'isoquinolinones
|
|
USRE47009E1
(en)
|
2011-02-01 |
2018-08-28 |
The Children's Hospital Of Philadelphia |
HDAC inhibitors and therapeutic methods using the same
|
|
US9108984B2
(en)
|
2011-03-14 |
2015-08-18 |
Incyte Corporation |
Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors
|
|
US9126948B2
(en)
|
2011-03-25 |
2015-09-08 |
Incyte Holdings Corporation |
Pyrimidine-4,6-diamine derivatives as PI3K inhibitors
|
|
US8691807B2
(en)
|
2011-06-20 |
2014-04-08 |
Incyte Corporation |
Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors
|
|
EP2734520B1
(fr)
|
2011-07-19 |
2016-09-14 |
Infinity Pharmaceuticals, Inc. |
Composés hétérocycliques et leurs utilisations
|
|
WO2013023119A1
(fr)
|
2011-08-10 |
2013-02-14 |
Novartis Pharma Ag |
Polythérapie par jak p13k/mtor
|
|
TW201313721A
(zh)
|
2011-08-18 |
2013-04-01 |
Incyte Corp |
作為jak抑制劑之環己基氮雜環丁烷衍生物
|
|
MX389479B
(es)
|
2011-09-02 |
2025-03-20 |
Incyte Holdings Corp |
Heterociclilaminas como inhibidores de fosfoinositida 3-cinasas (pi3k)
|
|
UA111854C2
(uk)
|
2011-09-07 |
2016-06-24 |
Інсайт Холдінгс Корпорейшн |
Способи і проміжні сполуки для отримання інгібіторів jak
|
|
EP2763994A4
(fr)
|
2011-10-04 |
2015-08-26 |
Gilead Calistoga Llc |
Nouveaux inhibiteurs de quinoxaline de la voie pi3k
|
|
US20140343128A1
(en)
|
2011-11-15 |
2014-11-20 |
Novartis Ag |
Combination of a phosphoinositide 3-kinase inhibitor and a modulator of the Janus Kinase 2 - Signal Transducer and Activator of Transcription 5 pathway
|
|
AR090548A1
(es)
|
2012-04-02 |
2014-11-19 |
Incyte Corp |
Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
|
|
TW201406761A
(zh)
|
2012-05-18 |
2014-02-16 |
Incyte Corp |
做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物
|
|
CA2888816A1
(fr)
|
2012-11-01 |
2014-05-08 |
Incyte Corporation |
Derives de thiophene condenses tricycliques a titre d'inhibiteurs de jak
|
|
KR102242077B1
(ko)
|
2012-11-15 |
2021-04-20 |
인사이트 홀딩스 코포레이션 |
룩솔리티니브의 서방성 제형
|
|
WO2014130587A1
(fr)
|
2013-02-19 |
2014-08-28 |
Roger Linington |
Nouveaux inhibiteurs à petites molécules de la formation de biofilms et nouvelle utilisation des composés précédemment identifiés pour inhiber la formation de biofilms et applications de thérapie médicamenteuse et de revêtement de dispositifs médicaux
|
|
TWI736135B
(zh)
|
2013-03-01 |
2021-08-11 |
美商英塞特控股公司 |
吡唑并嘧啶衍生物治療PI3Kδ相關病症之用途
|
|
EP3489239B1
(fr)
|
2013-03-06 |
2021-09-15 |
Incyte Holdings Corporation |
Procédés et intermédiaires pour fabriquer un inhibiteur de jak
|
|
CR20190156A
(es)
|
2013-05-17 |
2019-05-16 |
Incyte Corp |
Derivados de bipirazol como inhibidores jak
|
|
MX376856B
(es)
|
2013-08-07 |
2025-03-07 |
Incyte Holdings Corp |
Formas de dosificacion de liberacion prolongada para un inhibidor de jak 1 (cinasa de janus 1).
|
|
EA201690421A1
(ru)
|
2013-08-20 |
2016-06-30 |
Инсайт Корпорейшн |
Положительный эффект в форме увеличения продолжительности жизни у больных с солидными опухолями с повышенными уровнями c-реактивного белка
|
|
SG11201607083VA
(en)
|
2014-02-28 |
2016-09-29 |
Incyte Corp |
Jak1 inhibitors for the treatment of myelodysplastic syndromes
|
|
CA3158254C
(fr)
|
2014-04-08 |
2024-05-21 |
Incyte Corporation |
Traitement des malignites de cellules b par une combinaison d'inhibiteurs de jak et de pi3k
|
|
SG11201609016VA
(en)
|
2014-04-30 |
2016-11-29 |
Incyte Corp |
Processes of preparing a jak1 inhibitor and new forms thereto
|
|
WO2015184305A1
(fr)
|
2014-05-30 |
2015-12-03 |
Incyte Corporation |
Traitement de la leucémie neutrophile chronique (cnl) et de la leucémie myéloïde chronique atypique (acml) par des inhibiteurs de jak1
|
|
US10077277B2
(en)
|
2014-06-11 |
2018-09-18 |
Incyte Corporation |
Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
|
|
SG10201912302VA
(en)
|
2015-02-27 |
2020-02-27 |
Incyte Corp |
Salts of pi3k inhibitor and processes for their preparation
|
|
US20160362424A1
(en)
|
2015-05-11 |
2016-12-15 |
Incyte Corporation |
Salts of (s)-7-(1-(9h-purin-6-ylamino)ethyl)-6-(3-fluorophenyl)-3-methyl-5h-thiazolo[3,2-a]pyrimidin-5-one
|
|
US9988401B2
(en)
|
2015-05-11 |
2018-06-05 |
Incyte Corporation |
Crystalline forms of a PI3K inhibitor
|
|
WO2016183060A1
(fr)
|
2015-05-11 |
2016-11-17 |
Incyte Corporation |
Procédé de synthèse d'un inhibiteur de phospho-inositide 3-kinases
|
|
JP6785804B2
(ja)
*
|
2015-06-23 |
2020-11-18 |
ギリアド サイエンシズ, インコーポレイテッド |
B細胞悪性腫瘍を治療するための組合せ療法
|
|
IL278889B2
(en)
|
2018-06-01 |
2025-11-01 |
Incyte Corp |
Dosing regimen for the treatment of pi3k related disorders
|