NO176568C - Analogifremgangsmåte for fremstilling av substituerte alkylamider av teikoplaninforbindelser - Google Patents

Analogifremgangsmåte for fremstilling av substituerte alkylamider av teikoplaninforbindelser

Info

Publication number: NO176568C
Authority: NO; Norway
Prior art keywords: substituted alkyl; alkyl amides; analogous process; preparing substituted; teicoplanin compounds
Prior art date: 1987-03-02

Application number

NO884821A

Other languages

English (en)

Norwegian (no)

Other versions

NO176568B (no

NO884821D0 (no

NO884821L (no

Inventor

Giorgio Tarzia

Adriano Malabarba

Original Assignee

Lepetit Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-03-02

Filing date

1988-10-28

Publication date

1995-04-26

1988-10-28 Application filed by Lepetit Spa filed Critical Lepetit Spa

1988-10-28 Publication of NO884821D0 publication Critical patent/NO884821D0/no

1988-10-28 Publication of NO884821L publication Critical patent/NO884821L/no

1995-01-16 Publication of NO176568B publication Critical patent/NO176568B/no

1995-04-26 Publication of NO176568C publication Critical patent/NO176568C/no

Links

DDTDNCYHLGRFBM-YZEKDTGTSA-N chembl2367892 Chemical class CC(=O)N[C@H]1[C@@H](O)[C@H](O)[C@H](CO)O[C@H]1O[C@@H]([C@H]1C(N[C@@H](C2=CC(O)=CC(O[C@@H]3[C@H]([C@H](O)[C@H](O)[C@@H](CO)O3)O)=C2C=2C(O)=CC=C(C=2)[C@@H](NC(=O)[C@@H]2NC(=O)[C@@H]3C=4C=C(O)C=C(C=4)OC=4C(O)=CC=C(C=4)[C@@H](N)C(=O)N[C@H](CC=4C=C(Cl)C(O5)=CC=4)C(=O)N3)C(=O)N1)C(O)=O)=O)C(C=C1Cl)=CC=C1OC1=C(O[C@H]3[C@H]([C@@H](O)[C@H](O)[C@H](CO)O3)NC(C)=O)C5=CC2=C1 DDTDNCYHLGRFBM-YZEKDTGTSA-N 0.000 title abstract 2
238000004519 manufacturing process Methods 0.000 title 1
-1 substituted alkyl amides Chemical class 0.000 title 1
DQJCDTNMLBYVAY-ZXXIYAEKSA-N (2S,5R,10R,13R)-16-{[(2R,3S,4R,5R)-3-{[(2S,3R,4R,5S,6R)-3-acetamido-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}-5-(ethylamino)-6-hydroxy-2-(hydroxymethyl)oxan-4-yl]oxy}-5-(4-aminobutyl)-10-carbamoyl-2,13-dimethyl-4,7,12,15-tetraoxo-3,6,11,14-tetraazaheptadecan-1-oic acid Chemical group NCCCC[C@H](C(=O)N[C@@H](C)C(O)=O)NC(=O)CC[C@H](C(N)=O)NC(=O)[C@@H](C)NC(=O)C(C)O[C@@H]1[C@@H](NCC)C(O)O[C@H](CO)[C@H]1O[C@H]1[C@H](NC(C)=O)[C@@H](O)[C@H](O)[C@@H](CO)O1 DQJCDTNMLBYVAY-ZXXIYAEKSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
- C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Biochemistry (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
General Chemical & Material Sciences (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
Communicable Diseases (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Peptides Or Proteins (AREA)
Luminescent Compositions (AREA)
Polyamides (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Saccharide Compounds (AREA)

NO884821A 1987-03-02 1988-10-28 Analogifremgangsmåte for fremstilling av substituerte alkylamider av teikoplaninforbindelser NO176568C (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB878704847A GB8704847D0 (en)	1987-03-02	1987-03-02	Substituted alkylamides of teicoplanin compounds
PCT/EP1988/000129 WO1988006600A1 (en)	1987-03-02	1988-02-23	Substituted alkylamides of teicoplanin compounds

Publications (4)

Publication Number	Publication Date
NO884821D0 NO884821D0 (no)	1988-10-28
NO884821L NO884821L (no)	1988-10-28
NO176568B NO176568B (no)	1995-01-16
NO176568C true NO176568C (no)	1995-04-26

Family

ID=10613186

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO884821A NO176568C (no)	1987-03-02	1988-10-28	Analogifremgangsmåte for fremstilling av substituerte alkylamider av teikoplaninforbindelser

Country Status (22)

Country	Link
US (1)	US5198418A (de)
EP (1)	EP0340245B1 (de)
JP (1)	JPH0776234B2 (de)
KR (1)	KR960014104B1 (de)
CN (1)	CN88101000A (de)
AT (1)	ATE79637T1 (de)
AU (1)	AU619460B2 (de)
DE (1)	DE3873907T2 (de)
DK (1)	DK543088D0 (de)
ES (1)	ES2009555A6 (de)
FI (1)	FI91765C (de)
GB (1)	GB8704847D0 (de)
GR (1)	GR1001625B (de)
HU (1)	HU205371B (de)
IE (1)	IE62860B1 (de)
IL (1)	IL85493A0 (de)
NO (1)	NO176568C (de)
NZ (1)	NZ223669A (de)
PH (1)	PH27406A (de)
PT (1)	PT86827B (de)
WO (1)	WO1988006600A1 (de)
ZA (1)	ZA881445B (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8522574D0 (en) *	1985-09-12	1985-10-16	Lepetit Spa	Amides of teicoplanin compounds
GB8827202D0 (en) *	1988-11-22	1988-12-29	Lepetit Spa	Process for preparing 63-carboxyamides of teicoplanin antibiotics
EP0376041B1 (de) *	1988-12-27	1996-02-28	GRUPPO LEPETIT S.p.A.	C63-Amidderivate von 34-de(acetylglucosaminyl)-34-deoxy-teicoplaninen
IE64155B1 (en) *	1989-03-29	1995-07-12	Lepetit Spa	New substituted alkylamide derivatives of teicoplanin
US5500410A (en) *	1989-03-29	1996-03-19	Gruppo Lepetit S.P.A.	Substituted alkylamide derivatives of teicoplanin
EP0391077A1 (de) *	1989-04-03	1990-10-10	GRUPPO LEPETIT S.p.A.	O56-Alkyl-Derivate von Aglycon und Pseudoaglycone von Teicoplanin
US5185320A (en) *	1989-04-03	1993-02-09	Gruppo Lepetit S.P.A.	O56 -alkyl derivatives of aglycone and pseudo aglycones of teicoplanin
AU647122B2 (en) *	1990-05-28	1994-03-17	Gruppo Lepetit S.P.A.	C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy- teicoplanin and their use as medicaments against bacteria resistant to glycopeptide antibiotics
HUT63860A (en) *	1990-12-05	1993-10-28	Lepetit Spa	Process for producing 39-decarboxy-38-(hydroxymethyl) derivatives of teikoplanin antibiotics
JPH06510281A (ja) *	1991-08-08	1994-11-17	アミリン・ファーマシューティカルズ，インコーポレイテッド	ペプチドアミドの製造
GB2278540A (en) *	1993-09-24	1994-12-07	Nick Andrew Lewis	Extendible garment hanger
US5679769A (en) *	1994-03-15	1997-10-21	Sloan-Kettering Institute For Cancer Research	Synthesis of asparagine-linked glycopeptides on a polymeric solid support
WO1997040067A1 (en)	1996-04-23	1997-10-30	Biosearch Italia S.P.A.	Improved chemical process for preparing amide derivatives of antibiotic a 40926
SG87877A1 (en) *	1998-12-23	2002-04-16	Advanced Medicine Inc	Glycopeptide derivatives and pharmaceutical compositions containing the same
DK1140993T3 (da)	1998-12-23	2003-10-06	Theravance Inc	Glycopeptidderivater og farmaceutiske præparater indeholdende dem
US6770621B2 (en)	2000-05-02	2004-08-03	Theravance, Inc.	Polyacid glycopeptide derivatives

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3981303A (en) *	1971-09-09	1976-09-21	Alza Corporation	Bioerodible ocular device
GB1496386A (en) *	1975-03-05	1977-12-30	Lepetit Spa	Antibiotics
US4604239A (en) *	1982-03-24	1986-08-05	Eli Lilly And Company	Antibiotics
GB8307847D0 (en) *	1983-03-22	1983-04-27	Lepetit Spa	Antibiotics l 17054 and l 17046
US4534969A (en) *	1983-09-19	1985-08-13	The Dow Chemical Company	Method for improving lactation in ruminant animals
AU579120B2 (en) *	1983-12-16	1988-11-17	Gruppo Lepetit S.P.A.	Chemical process for preparing antibiotic L 17392 (deglucoteicoplanin) and its salts
IT1173329B (it) *	1984-02-21	1987-06-24	Lepetit Spa	Procedimento per la trasformazione quantitativa di teicoplanina a2 fattore 1 in teicoplanina a2 fattore 3
GB8415092D0 (en) *	1984-06-13	1984-07-18	Lepetit Spa	Ester derivatives
GB8420405D0 (en) *	1984-08-10	1984-09-12	Lepetit Spa	Preparing antibiotic l 17046
GB8522574D0 (en) *	1985-09-12	1985-10-16	Lepetit Spa	Amides of teicoplanin compounds

1987
- 1987-03-02 GB GB878704847A patent/GB8704847D0/en active Pending
1988
- 1988-02-22 IL IL85493A patent/IL85493A0/xx not_active IP Right Cessation
- 1988-02-23 DE DE8888902122T patent/DE3873907T2/de not_active Expired - Fee Related
- 1988-02-23 JP JP63501993A patent/JPH0776234B2/ja not_active Expired - Lifetime
- 1988-02-23 AU AU13632/88A patent/AU619460B2/en not_active Ceased
- 1988-02-23 EP EP88902122A patent/EP0340245B1/de not_active Expired - Lifetime
- 1988-02-23 KR KR1019880701400A patent/KR960014104B1/ko not_active Expired - Lifetime
- 1988-02-23 HU HU881742A patent/HU205371B/hu not_active IP Right Cessation
- 1988-02-23 AT AT88902122T patent/ATE79637T1/de not_active IP Right Cessation
- 1988-02-23 WO PCT/EP1988/000129 patent/WO1988006600A1/en not_active Ceased
- 1988-02-25 PT PT86827A patent/PT86827B/pt not_active IP Right Cessation
- 1988-02-25 IE IE51388A patent/IE62860B1/en not_active IP Right Cessation
- 1988-02-26 NZ NZ223669A patent/NZ223669A/en unknown
- 1988-02-29 CN CN198888101000A patent/CN88101000A/zh active Pending
- 1988-03-01 ZA ZA881445A patent/ZA881445B/xx unknown
- 1988-03-01 GR GR880100118A patent/GR1001625B/el unknown
- 1988-03-01 ES ES8800594A patent/ES2009555A6/es not_active Expired
- 1988-03-02 PH PH36578A patent/PH27406A/en unknown
- 1988-09-29 DK DK543088A patent/DK543088D0/da not_active Application Discontinuation
- 1988-10-28 NO NO884821A patent/NO176568C/no unknown
1989
- 1989-08-31 FI FI894078A patent/FI91765C/fi not_active IP Right Cessation
1992
- 1992-01-21 US US07/826,198 patent/US5198418A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
WO1988006600A1 (en)	1988-09-07
FI894078A0 (fi)	1989-08-31
DE3873907T2 (de)	1993-01-14
PT86827A (pt)	1988-03-01
HUT51300A (en)	1990-04-28
NO176568B (no)	1995-01-16
JPH0776234B2 (ja)	1995-08-16
GB8704847D0 (en)	1987-04-08
DK543088A (da)	1988-09-29
CN88101000A (zh)	1988-09-14
PH27406A (en)	1993-06-21
ZA881445B (en)	1989-01-25
IE880513L (en)	1988-09-02
AU619460B2 (en)	1992-01-30
PT86827B (pt)	1992-05-29
GR880100118A (en)	1989-01-31
DE3873907D1 (de)	1992-09-24
FI894078L (fi)	1989-08-31
DK543088D0 (da)	1988-09-29
AU1363288A (en)	1988-09-26
JPH02502456A (ja)	1990-08-09
NZ223669A (en)	1990-12-21
KR960014104B1 (ko)	1996-10-14
IE62860B1 (en)	1995-03-08
ES2009555A6 (es)	1989-10-01
GR1001625B (el)	1994-07-29
HU205371B (en)	1992-04-28
US5198418A (en)	1993-03-30
NO884821D0 (no)	1988-10-28
EP0340245B1 (de)	1992-08-19
KR890700607A (ko)	1989-04-26
EP0340245A1 (de)	1989-11-08
ATE79637T1 (de)	1992-09-15
IL85493A0 (en)	1988-07-31
FI91765C (fi)	1994-08-10
NO884821L (no)	1988-10-28
FI91765B (fi)	1994-04-29

Publication	Publication Date	Title
NO176568C (no)	1995-04-26	Analogifremgangsmåte for fremstilling av substituerte alkylamider av teikoplaninforbindelser
FI914905L (fi)	1992-04-19	Menetelmä uusien terapeuttisesti käyttökelpoisten merkaptoasetyyliamidopyrrolo- ja -pyridobentsatsepiinijohdannaisten valmistamiseksi
FI925737A7 (fi)	1993-06-20	Menetelmä uusien terapeuttisesti käyttökelpoisten indol-3-yylialkyylipiperatsiinijohdannaisten valmistamiseksi
FI914174A7 (fi)	1992-03-06	Menetelmä piperidyylialkyyliamiinien valmistamiseksi
FI924569A7 (fi)	1992-10-09	Menetelmä fenyyli-isoseriinijohdannaisten enantioselektiiviseksi valmi stamiseksi
FI923527L (fi)	1992-08-05	Menetelmä terapeuttisesti käyttökelpoisten 3-piperidino-4-hydroksikromaanijohdannaisten valmistamiseksi
GR3030718T3 (en)	1999-11-30	Novel prostaglandin analogue.
TNSN88080A1 (fr)	1990-07-10	Procede pour la preparation de nouveaux derives aminoalcoxyphenyle
HUT64744A (en)	1994-02-28	Process for preparing 3-indolyl-thioacetate derivatives
EE03027B1 (et)	1997-08-15	Meetod 8-klorokinolooni derivaatide valmistamiseks
PT88432A (pt)	1989-07-31	Process for the preparation of 4-oxo-3-quinolinecarboxylic acids useful as antibacterial agents
FI912626A7 (fi)	1991-12-05	Menetelmä B-hydroksi-a-aminohappojen valmistamiseksi
PT87359A (pt)	1989-05-31	Process for the preparation of pyrrolidine derivatives
PT88431A (pt)	1989-07-31	Process for the preparation of 4-oxo-3-quinolinecarboxylic acids useful as antibacterial agents
FI913464A7 (fi)	1992-01-21	Menetelmä 1-hydroksimetyylipyratsolien valmistamiseksi
DE3470312D1 (de)	1988-05-11	Ether of n-propanolamine derivative
PL291199A1 (en)	1992-03-09	Method of synthesizing 6-/aminopropionyl substituted/ forskolin derivatives
FI923866A7 (fi)	1992-08-28	Menetelmä 1-hydroksialkyyli-5-nitroimidatsolien valmistamiseksi
FI97388B (fi)	1996-08-30	Menetelmä heterosyklisten NMDA-antagonistien valmistamiseksi
DE69208047D1 (de)	1996-03-14	Verfahren zur Herstellung von Alkyl-Adipaten
FI913656A7 (fi)	1992-02-01	Menetelmä alkyyli-6-pyridatsiinijohdannaisten valmistamiseksi
FI913414A7 (fi)	1992-01-18	Menetelmä 2-hydroksi-3-halogeeni-5-nitro-pyridiinien valmistamiseksi
FI942678A0 (fi)	1994-06-07	Menetelmä 3'-deoksi-3-'fluorimetyylinukleosidijohdannaisten valmistamiseksi
NO950203L (no)	1991-10-11	Fremgangsmåte for fremstilling av propargylazetidion-forbindelser