NO20003784D0 - FremgangsmÕte for fremstilling av enansiomert rene cykloalkanoindolkarboksylsyre og azaindolkarboksylsyrer og pyrimido 1,2a indolkarboksylsyrer og derivater derav - Google Patents

FremgangsmÕte for fremstilling av enansiomert rene cykloalkanoindolkarboksylsyre og azaindolkarboksylsyrer og pyrimido 1,2a indolkarboksylsyrer og derivater derav

Info

Publication number: NO20003784D0
Authority: NO; Norway
Prior art keywords: acids; enansiomerically; cycloalkanoindolecarboxylic; azaindolecarboxylic; pyrimido
Prior art date: 1996-04-04

Application number

NO20003784A

Other languages

English (en)

Other versions

NO20003784L (no

Inventor

Jan-Bernd Lenfers

Peter Fey

Paul Naab

Kai Van Laak

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-04-04

Filing date

2000-07-24

Publication date

2000-07-24

1997-10-06 Publication of NO20003784L publication Critical patent/NO20003784L/no

2000-07-24 Application filed by Bayer Ag filed Critical Bayer Ag

2000-07-24 Publication of NO20003784D0 publication Critical patent/NO20003784D0/no

Links

239000002253 acid Substances 0.000 title 2
HCUARRIEZVDMPT-UHFFFAOYSA-N Indole-2-carboxylic acid Chemical class C1=CC=C2NC(C(=O)O)=CC2=C1 HCUARRIEZVDMPT-UHFFFAOYSA-N 0.000 title 1
150000007513 acids Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
- C07C69/616—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety polycyclic
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/62—Halogen-containing esters
- C07C69/65—Halogen-containing esters of unsaturated acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

NO20003784A 1996-04-04 2000-07-24 FremgangsmÕte for fremstilling av enansiomert rene cykloalkanoindolkarboksylsyre og azaindolkarboksylsyrer og pyrimido 1,2a indolkarboksylsyrer og derivater derav NO20003784D0 (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19613549A DE19613549A1 (de)	1996-04-04	1996-04-04	Verfahren zur Herstellung von enantiomerenreinen Cycloalkano-indol- und azaindol-carbonsäuren und deren aktivierte Derivate

Publications (2)

Publication Number	Publication Date
NO20003784L NO20003784L (no)	1997-10-06
NO20003784D0 true NO20003784D0 (no)	2000-07-24

Family

ID=7790501

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
NO971513A NO308301B1 (no)	1996-04-04	1997-04-03	FremgangsmÕte for fremstilling av enantiomer-rene cykloalkanoindol- og azaindol- og pyrimido[1,2a]- indolkarboksylsyrer og deres aktiverte derivater, mellomprodukter samt anvendelse av disse
NO20003784A NO20003784D0 (no)	1996-04-04	2000-07-24	FremgangsmÕte for fremstilling av enansiomert rene cykloalkanoindolkarboksylsyre og azaindolkarboksylsyrer og pyrimido 1,2a indolkarboksylsyrer og derivater derav

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
NO971513A NO308301B1 (no)	1996-04-04	1997-04-03	FremgangsmÕte for fremstilling av enantiomer-rene cykloalkanoindol- og azaindol- og pyrimido[1,2a]- indolkarboksylsyrer og deres aktiverte derivater, mellomprodukter samt anvendelse av disse

Country Status (27)

Country	Link
US (1)	US5952498A (no)
EP (1)	EP0799829B1 (no)
JP (2)	JP4235268B2 (no)
KR (1)	KR970069988A (no)
CN (2)	CN1067394C (no)
AR (2)	AR006544A1 (no)
AT (1)	ATE246193T1 (no)
AU (1)	AU722592B2 (no)
BR (1)	BR9701672A (no)
CA (1)	CA2201435C (no)
CZ (1)	CZ102197A3 (no)
DE (2)	DE19613549A1 (no)
DZ (1)	DZ2202A1 (no)
EE (1)	EE9700079A (no)
ES (1)	ES2202506T3 (no)
HR (1)	HRP970178A2 (no)
HU (1)	HU218494B (no)
ID (1)	ID16794A (no)
IL (1)	IL120591A (no)
MA (1)	MA24130A1 (no)
NO (2)	NO308301B1 (no)
NZ (1)	NZ314498A (no)
PL (1)	PL319269A1 (no)
SG (1)	SG60050A1 (no)
SK (1)	SK42897A3 (no)
TN (1)	TNSN97060A1 (no)
ZA (1)	ZA972831B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4435477A1 (de) *	1994-10-04	1996-04-11	Bayer Ag	Cycloalkano-indol- und -azaindol-derivate
AU2001244635A1 (en) *	2000-03-30	2001-10-15	Yamanouchi Pharmaceutical Co..Ltd.	Hydrazide derivatives
WO2005051382A1 (ja) *	2003-11-28	2005-06-09	Astellas Pharma Inc.	脂質低下作用増強剤
PT1725234E (pt)	2004-03-05	2013-03-04	Univ Pennsylvania	Métodos com efeitos secundários reduzidos para tratamento de patologias ou doenças associadas a hiperlipidemia e hipercolesterolemia
EP1737460A2 (en) *	2004-04-09	2007-01-03	Janssen Pharmaceutica N.V.	Intermittent dosing regimen for the treatment of overweight with mtp-inhibitors
EP1951220A2 (en) *	2005-10-18	2008-08-06	Aegerion Pharmaceuticals	Compositions for lowering serum cholesterol and/or triglycerides
JP2009537505A (ja) *	2006-05-18	2009-10-29	バイエル・ヘルスケア・アクチェンゲゼルシャフト	インプリタピドを含む薬学的組成物およびこの薬学的組成物の使用方法
JP2010513534A (ja) *	2006-12-21	2010-04-30	エージェリオンファーマシューティカルズ，インコーポレイテッド	Ｍｔｐインヒビターおよびコレステロール吸収インヒビターを含む組み合わせを用いて肥満症を処置する方法
WO2008124384A2 (en) *	2007-04-03	2008-10-16	Aegerion Pharmaceuticals, Inc.	Combinations of mtp inhibitors with cholesterol absorption inhibitors or interferon for treating hepatitis c
SI2968284T1 (sl)	2013-03-14	2021-08-31	Osteoqc Inc.	Alkil-amin harmin derivati za pospeševanje rasti kosti
JP7695496B2 (ja)	2018-08-14	2025-06-19	オシフィセラピューティクスリミティドライアビリティカンパニー	フルオロβ－カルボリン化合物
EP3836923B1 (en)	2018-08-14	2024-10-16	OssiFi Therapeutics LLC	Pyrrolo - dipyridine compounds for the treatment of bone loss
BR112023000808A2 (pt)	2020-07-29	2023-02-07	Amryt Pharmaceuticals Inc	Lomitapida para uso em métodos para tratar hiperlipidemia e hipercolesterolemia em pacientes pediátricos

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3900261A1 (de) *	1988-05-31	1989-12-07	Bayer Ag	Substituierte 4-(chinolin-2-yl-methoxy) phenyl-essigsaeure-derivate
DE4200954A1 (de) *	1991-04-26	1992-10-29	Bayer Ag	Heterocyclisch substituierte phenylessigsaeurederivate
DE4208051A1 (de) *	1992-03-13	1993-09-16	Bayer Ag	Substituierte phenylessigsaeureamide
DE4302956A1 (de) *	1993-02-03	1994-08-04	Bayer Ag	Substituierte Imidazo(4,5-b)pyridine und Benzimidazole
DE4435477A1 (de) *	1994-10-04	1996-04-11	Bayer Ag	Cycloalkano-indol- und -azaindol-derivate

1996
- 1996-04-04 DE DE19613549A patent/DE19613549A1/de not_active Withdrawn
1997
- 1997-03-24 EP EP97104941A patent/EP0799829B1/de not_active Expired - Lifetime
- 1997-03-24 DE DE59710487T patent/DE59710487D1/de not_active Expired - Lifetime
- 1997-03-24 AT AT97104941T patent/ATE246193T1/de not_active IP Right Cessation
- 1997-03-24 ES ES97104941T patent/ES2202506T3/es not_active Expired - Lifetime
- 1997-03-27 AU AU16602/97A patent/AU722592B2/en not_active Ceased
- 1997-03-27 NZ NZ314498A patent/NZ314498A/en unknown
- 1997-03-28 HR HR19613549.4A patent/HRP970178A2/xx not_active Application Discontinuation
- 1997-03-31 US US08/829,566 patent/US5952498A/en not_active Expired - Lifetime
- 1997-03-31 ID IDP971060A patent/ID16794A/id unknown
- 1997-04-01 SG SG1997001028A patent/SG60050A1/en unknown
- 1997-04-01 CA CA002201435A patent/CA2201435C/en not_active Expired - Fee Related
- 1997-04-01 JP JP09635197A patent/JP4235268B2/ja not_active Expired - Fee Related
- 1997-04-01 MA MA24543A patent/MA24130A1/fr unknown
- 1997-04-02 DZ DZ970049A patent/DZ2202A1/fr active
- 1997-04-02 IL IL12059197A patent/IL120591A/xx not_active IP Right Cessation
- 1997-04-02 TN TNTNSN97060A patent/TNSN97060A1/fr unknown
- 1997-04-03 SK SK428-97A patent/SK42897A3/sk unknown
- 1997-04-03 ZA ZA9702831A patent/ZA972831B/xx unknown
- 1997-04-03 PL PL97319269A patent/PL319269A1/xx unknown
- 1997-04-03 HU HU9700698A patent/HU218494B/hu not_active IP Right Cessation
- 1997-04-03 CZ CZ971021A patent/CZ102197A3/cs unknown
- 1997-04-03 NO NO971513A patent/NO308301B1/no not_active IP Right Cessation
- 1997-04-03 EE EE9700079A patent/EE9700079A/xx unknown
- 1997-04-03 KR KR1019970012291A patent/KR970069988A/ko not_active Withdrawn
- 1997-04-04 BR BR9701672A patent/BR9701672A/pt active Search and Examination
- 1997-04-04 AR ARP970101366A patent/AR006544A1/es unknown
- 1997-04-04 CN CN97110276A patent/CN1067394C/zh not_active Expired - Fee Related
1998
- 1998-03-06 AR ARP980101029A patent/AR012048A2/es unknown
2000
- 2000-07-24 NO NO20003784A patent/NO20003784D0/no not_active Application Discontinuation
- 2000-10-12 CN CN00133103A patent/CN1330065A/zh active Pending
2008
- 2008-01-31 JP JP2008021569A patent/JP2008169218A/ja active Pending

Also Published As

Publication number	Publication date
AR012048A2 (es)	2000-09-27
JPH1045759A (ja)	1998-02-17
CN1330065A (zh)	2002-01-09
DZ2202A1 (fr)	2002-12-03
EE9700079A (et)	1997-10-15
IL120591A0 (en)	1997-08-14
US5952498A (en)	1999-09-14
CN1184109A (zh)	1998-06-10
HUP9700698A1 (hu)	1998-01-28
NZ314498A (en)	1999-09-29
JP4235268B2 (ja)	2009-03-11
DE19613549A1 (de)	1997-10-09
SG60050A1 (en)	1999-02-22
CN1067394C (zh)	2001-06-20
PL319269A1 (en)	1997-10-13
ES2202506T3 (es)	2004-04-01
NO971513L (no)	1997-10-06
BR9701672A (pt)	1998-11-03
IL120591A (en)	2000-11-21
AU722592B2 (en)	2000-08-10
TNSN97060A1 (fr)	2005-03-15
EP0799829B1 (de)	2003-07-30
MX9702446A (es)	1997-10-31
CA2201435C (en)	2006-12-12
NO971513D0 (no)	1997-04-03
MA24130A1 (fr)	1997-10-01
KR970069988A (ko)	1997-11-07
EP0799829A1 (de)	1997-10-08
NO308301B1 (no)	2000-08-28
ID16794A (id)	1997-11-13
CZ102197A3 (en)	1997-10-15
JP2008169218A (ja)	2008-07-24
ZA972831B (en)	1997-10-31
DE59710487D1 (de)	2003-09-04
HU9700698D0 (en)	1997-05-28
SK42897A3 (en)	1997-10-08
AR006544A1 (es)	1999-09-08
ATE246193T1 (de)	2003-08-15
HU218494B (hu)	2000-09-28
HRP970178A2 (en)	1998-04-30
AU1660297A (en)	1997-10-09
NO20003784L (no)	1997-10-06
CA2201435A1 (en)	1997-10-04

Legal Events

Date	Code	Title	Description
2001-11-19	FC2A	Withdrawal, rejection or dismissal of laid open patent application

Publication	Publication Date	Title
ZA9710038B (en)	1998-07-01	Method for the production of levulinic acid and its derivatives
NO961006D0 (no)	1996-03-12	Fosfonomononukleinsyrer, fremgangsmåter for fremstilling derav og anvendelse av forbindelsene
NO890921D0 (no)	1989-03-03	Fremgangsmaate for fremstilling av aminosyrederivater.
FI945776L (fi)	1995-06-11	Yhden astian menetelmä 3-kinolonikarboksyylihaapojohdannaisten valmistamiseksi
NO971513D0 (no)	1997-04-03	Fremgangsmåte for fremstilling av enantiomert, rene cykloalkanoindol- og azaindol- og pyrimido£1,2a\|-indolkarboksylsyrer og deres aktiverte derivater
NO982237L (no)	1998-07-10	FremgangsmÕte for fremstilling av fenylimidazolidinderivater
IL105100A0 (en)	1993-12-28	Glutamic acid derivatives and process for their preparation
FI900145L (fi)	1990-01-11	Menetelmä farmaseuttisesti käyttökelpoisten 1,1-diokso-kefem-4-karbotiolihappojohdannaisten valmistamiseksi
FI941149A0 (fi)	1994-03-10	2,4-diamino-3-hydroksikarboksyylihapon johdannaisia
NO308465B1 (no)	2000-09-18	FremgangsmÕte for fremstilling av karboksylsyrederivater
NO952713D0 (no)	1995-07-07	Fremgangsmåte for fremstilling av substituerte indolonderivater
ZA952759B (en)	1996-01-05	Process for the preparation of carboxyarenesulfonic acids and their carboxylic acid derivatives
NO942531D0 (no)	1994-07-05	Fremgangsmåte for fremstilling av 3-acylöstratriener og acylbenzener
IL119922A0 (en)	1997-03-18	Process for the preparation of omicron-chloromethyl-phenylglyoxylic acid derivatives
NO942381L (no)	1994-12-27	Fremgangsmåte for fremstilling av indoler
NO912167D0 (no)	1991-06-06	Fremgangsmaate for fremstilling av ftalsyreanhydrid-derivater.
NO972129D0 (no)	1997-05-07	Fremgangsmåte for fremstilling av 1-halo-3-trialkylsilanyl-benzenderivater
NO991098D0 (no)	1999-03-05	FremgangsmÕte for fremstilling av 2-fenyl-3-naftylpropionsyrederivater
NO982090L (no)	1998-07-07	FremgangsmÕte for fremstilling av 3-fenyl-1-metylendioksyfenyl-indan-2-karboksylsyrederivater
NO964519D0 (no)	1996-10-24	Fremgangsmåte for fremstilling av chitosanalkylderivater
AU2416295A (en)	1995-12-05	Acid amide derivatives and process for the preparation thereof
ZA9713B (en)	1997-07-17	Process for the preparation of o-chloromethyl-phenyl-glyoxylic acid derivatives
HU9700366D0 (en)	1997-03-28	Novel derivatives of 3-bromo- and 3,3 dibromo-4-oxo-1-azetidines, process for the preparation thereof and their use
HU9602052D0 (en)	1996-09-30	Process for the preparation of 2,4-dibromo-4- and -3-fluoro-buthane carboxylic acid and its derivatives
IL136922A0 (en)	2001-06-14	Process for the preparation of enantiomerically pure indolecarboxylic acid derivatives and some such new compounds