MA24130A1 - PROCEDE DE PREPARATION D'ENANTIOMERES PURS D'ACIDES CYCLO-ALCANO-INDOLAZAINDOL ET PYRIMIDO-(1,2a) INDOL - CARBOCYCLIQUES ET LEURS DERIVES - Google Patents

PROCEDE DE PREPARATION D'ENANTIOMERES PURS D'ACIDES CYCLO-ALCANO-INDOLAZAINDOL ET PYRIMIDO-(1,2a) INDOL - CARBOCYCLIQUES ET LEURS DERIVES

Info

Publication number: MA24130A1
Authority: MA; Morocco
Prior art keywords: indolazaindol; carbocyclics; alkano; pyrimido; indol
Prior art date: 1996-04-04

Application number

MA24543A

Other languages

English (en)

Inventor

Van Laak Kai

Lenfers Jan-Bernd

Naab Paul

Fey Peter

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-04-04

Filing date

1997-04-01

Publication date

1997-10-01

1997-04-01 Application filed by Bayer Ag filed Critical Bayer Ag

1997-10-01 Publication of MA24130A1 publication Critical patent/MA24130A1/fr

Links

HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical compound C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 title 1
SIKJAQJRHWYJAI-UHFFFAOYSA-N Indole Chemical compound C1=CC=C2NC=CC2=C1 SIKJAQJRHWYJAI-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
- C07C69/616—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety polycyclic
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/62—Halogen-containing esters
- C07C69/65—Halogen-containing esters of unsaturated acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

MA24543A 1996-04-04 1997-04-01 PROCEDE DE PREPARATION D'ENANTIOMERES PURS D'ACIDES CYCLO-ALCANO-INDOLAZAINDOL ET PYRIMIDO-(1,2a) INDOL - CARBOCYCLIQUES ET LEURS DERIVES MA24130A1 (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19613549A DE19613549A1 (de)	1996-04-04	1996-04-04	Verfahren zur Herstellung von enantiomerenreinen Cycloalkano-indol- und azaindol-carbonsäuren und deren aktivierte Derivate

Publications (1)

Publication Number	Publication Date
MA24130A1 true MA24130A1 (fr)	1997-10-01

Family

ID=7790501

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
MA24543A MA24130A1 (fr)	1996-04-04	1997-04-01	PROCEDE DE PREPARATION D'ENANTIOMERES PURS D'ACIDES CYCLO-ALCANO-INDOLAZAINDOL ET PYRIMIDO-(1,2a) INDOL - CARBOCYCLIQUES ET LEURS DERIVES

Country Status (27)

Country	Link
US (1)	US5952498A (fr)
EP (1)	EP0799829B1 (fr)
JP (2)	JP4235268B2 (fr)
KR (1)	KR970069988A (fr)
CN (2)	CN1067394C (fr)
AR (2)	AR006544A1 (fr)
AT (1)	ATE246193T1 (fr)
AU (1)	AU722592B2 (fr)
BR (1)	BR9701672A (fr)
CA (1)	CA2201435C (fr)
CZ (1)	CZ102197A3 (fr)
DE (2)	DE19613549A1 (fr)
DZ (1)	DZ2202A1 (fr)
EE (1)	EE9700079A (fr)
ES (1)	ES2202506T3 (fr)
HR (1)	HRP970178A2 (fr)
HU (1)	HU218494B (fr)
ID (1)	ID16794A (fr)
IL (1)	IL120591A (fr)
MA (1)	MA24130A1 (fr)
NO (2)	NO308301B1 (fr)
NZ (1)	NZ314498A (fr)
PL (1)	PL319269A1 (fr)
SG (1)	SG60050A1 (fr)
SK (1)	SK42897A3 (fr)
TN (1)	TNSN97060A1 (fr)
ZA (1)	ZA972831B (fr)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4435477A1 (de)	1994-10-04	1996-04-11	Bayer Ag	Cycloalkano-indol- und -azaindol-derivate
AU2001244635A1 (en) *	2000-03-30	2001-10-15	Yamanouchi Pharmaceutical Co..Ltd.	Hydrazide derivatives
WO2005051382A1 (fr) *	2003-11-28	2005-06-09	Astellas Pharma Inc.	Agent renforçant l'effet hypolipidemiant
KR101494067B1 (ko)	2004-03-05	2015-02-16	더 트러스티스 오브 더 유니버시티 오브 펜실바니아	부작용을 최소화하면서 과지질혈증 및 과콜레스테롤혈증과 연관된 질환 또는 질병의 치료 방법
AU2005230397B2 (en) *	2004-04-09	2010-04-08	Elanco Animal Health Ireland Limited	Intermittent dosing regimen for the treatment of overweight with MTP-inhibitors
AU2006304689A1 (en) *	2005-10-18	2007-04-26	Aegerion Pharmaceuticals	Compositions for lowering serum cholesterol and/or triglycerides
US20080051427A1 (en) *	2006-05-18	2008-02-28	Fritz Schuckler	Pharmaceutical Compositions and Methods of Using Same
JP2010513534A (ja) *	2006-12-21	2010-04-30	エージェリオンファーマシューティカルズ，インコーポレイテッド	Ｍｔｐインヒビターおよびコレステロール吸収インヒビターを含む組み合わせを用いて肥満症を処置する方法
WO2008124384A2 (fr) *	2007-04-03	2008-10-16	Aegerion Pharmaceuticals, Inc.	Méthodes de traitement de l'hépatite c
PT2968284T (pt)	2013-03-14	2021-06-28	Osteoqc Inc	Derivados alquilamina de harmina para promoção de crescimento ósseo
AU2019320773B2 (en)	2018-08-14	2024-12-05	Ossifi Therapeutics Llc	Fluoro β-carboline compounds
US10947236B2 (en)	2018-08-14	2021-03-16	Osteoqc Inc.	Pyrrolo-dipyridine compounds
CA3186856A1 (fr)	2020-07-29	2022-02-03	Ruth NALLEN	Lomitapide destine a etre utilise dans des methodes de traitement de l'hyperlipidemie et de l'hypercholesterolemie chez des patients pediatriques

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3900261A1 (de) *	1988-05-31	1989-12-07	Bayer Ag	Substituierte 4-(chinolin-2-yl-methoxy) phenyl-essigsaeure-derivate
DE4200954A1 (de) *	1991-04-26	1992-10-29	Bayer Ag	Heterocyclisch substituierte phenylessigsaeurederivate
DE4208051A1 (de) *	1992-03-13	1993-09-16	Bayer Ag	Substituierte phenylessigsaeureamide
DE4302956A1 (de) *	1993-02-03	1994-08-04	Bayer Ag	Substituierte Imidazo(4,5-b)pyridine und Benzimidazole
DE4435477A1 (de) *	1994-10-04	1996-04-11	Bayer Ag	Cycloalkano-indol- und -azaindol-derivate

1996
- 1996-04-04 DE DE19613549A patent/DE19613549A1/de not_active Withdrawn
1997
- 1997-03-24 AT AT97104941T patent/ATE246193T1/de not_active IP Right Cessation
- 1997-03-24 ES ES97104941T patent/ES2202506T3/es not_active Expired - Lifetime
- 1997-03-24 DE DE59710487T patent/DE59710487D1/de not_active Expired - Lifetime
- 1997-03-24 EP EP97104941A patent/EP0799829B1/fr not_active Expired - Lifetime
- 1997-03-27 AU AU16602/97A patent/AU722592B2/en not_active Ceased
- 1997-03-27 NZ NZ314498A patent/NZ314498A/en unknown
- 1997-03-28 HR HR19613549.4A patent/HRP970178A2/xx not_active Application Discontinuation
- 1997-03-31 US US08/829,566 patent/US5952498A/en not_active Expired - Lifetime
- 1997-03-31 ID IDP971060A patent/ID16794A/id unknown
- 1997-04-01 SG SG1997001028A patent/SG60050A1/en unknown
- 1997-04-01 CA CA002201435A patent/CA2201435C/fr not_active Expired - Fee Related
- 1997-04-01 JP JP09635197A patent/JP4235268B2/ja not_active Expired - Fee Related
- 1997-04-01 MA MA24543A patent/MA24130A1/fr unknown
- 1997-04-02 TN TNTNSN97060A patent/TNSN97060A1/fr unknown
- 1997-04-02 IL IL12059197A patent/IL120591A/xx not_active IP Right Cessation
- 1997-04-02 DZ DZ970049A patent/DZ2202A1/fr active
- 1997-04-03 KR KR1019970012291A patent/KR970069988A/ko not_active Withdrawn
- 1997-04-03 HU HU9700698A patent/HU218494B/hu not_active IP Right Cessation
- 1997-04-03 NO NO971513A patent/NO308301B1/no not_active IP Right Cessation
- 1997-04-03 ZA ZA9702831A patent/ZA972831B/xx unknown
- 1997-04-03 PL PL97319269A patent/PL319269A1/xx unknown
- 1997-04-03 CZ CZ971021A patent/CZ102197A3/cs unknown
- 1997-04-03 SK SK428-97A patent/SK42897A3/sk unknown
- 1997-04-03 EE EE9700079A patent/EE9700079A/xx unknown
- 1997-04-04 BR BR9701672A patent/BR9701672A/pt active Search and Examination
- 1997-04-04 AR ARP970101366A patent/AR006544A1/es unknown
- 1997-04-04 CN CN97110276A patent/CN1067394C/zh not_active Expired - Fee Related
1998
- 1998-03-06 AR ARP980101029A patent/AR012048A2/es unknown
2000
- 2000-07-24 NO NO20003784A patent/NO20003784D0/no not_active Application Discontinuation
- 2000-10-12 CN CN00133103A patent/CN1330065A/zh active Pending
2008
- 2008-01-31 JP JP2008021569A patent/JP2008169218A/ja active Pending

Also Published As

Publication number	Publication date
AU1660297A (en)	1997-10-09
CN1067394C (zh)	2001-06-20
PL319269A1 (en)	1997-10-13
CN1330065A (zh)	2002-01-09
NO20003784L (no)	1997-10-06
DZ2202A1 (fr)	2002-12-03
HRP970178A2 (en)	1998-04-30
CN1184109A (zh)	1998-06-10
NZ314498A (en)	1999-09-29
SK42897A3 (en)	1997-10-08
AU722592B2 (en)	2000-08-10
CZ102197A3 (en)	1997-10-15
ATE246193T1 (de)	2003-08-15
MX9702446A (es)	1997-10-31
CA2201435C (fr)	2006-12-12
US5952498A (en)	1999-09-14
NO971513L (no)	1997-10-06
JPH1045759A (ja)	1998-02-17
KR970069988A (ko)	1997-11-07
IL120591A0 (en)	1997-08-14
CA2201435A1 (fr)	1997-10-04
NO20003784D0 (no)	2000-07-24
ID16794A (id)	1997-11-13
DE59710487D1 (de)	2003-09-04
HU9700698D0 (en)	1997-05-28
IL120591A (en)	2000-11-21
AR006544A1 (es)	1999-09-08
TNSN97060A1 (fr)	2005-03-15
AR012048A2 (es)	2000-09-27
EP0799829B1 (fr)	2003-07-30
JP2008169218A (ja)	2008-07-24
ES2202506T3 (es)	2004-04-01
HU218494B (hu)	2000-09-28
NO308301B1 (no)	2000-08-28
NO971513D0 (no)	1997-04-03
EP0799829A1 (fr)	1997-10-08
HUP9700698A1 (hu)	1998-01-28
SG60050A1 (en)	1999-02-22
EE9700079A (et)	1997-10-15
DE19613549A1 (de)	1997-10-09
ZA972831B (en)	1997-10-31
BR9701672A (pt)	1998-11-03
JP4235268B2 (ja)	2009-03-11

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MA24130A1 (fr)	1997-10-01	PROCEDE DE PREPARATION D'ENANTIOMERES PURS D'ACIDES CYCLO-ALCANO-INDOLAZAINDOL ET PYRIMIDO-(1,2a) INDOL - CARBOCYCLIQUES ET LEURS DERIVES
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NO985535D0 (no)	1998-11-27	FremgangsmÕte for fremstilling av 1,3-alkandioler
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MA23081A1 (fr)	1994-10-01	Procede de preparation de derives d'indolone
FI964429A7 (fi)	1996-11-04	Menetelmä 1-(3-trialkyylisilyylifenyyli)-2,2,2-trifluorimetyylietanoni n johdannaisten valmistamiseksi
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NO975961D0 (no)	1997-12-18	Fremgangsmåte for fremstilling av 1-(3-trialkylsilylfenyl)-2,2,2-trifluorometyl-ethanonderivater
FR2715167B1 (fr)	1996-04-12	Procédé de production de la L-carnitine par voie microbiologique.
EP0945433A4 (fr)	2004-09-01	Procede de preparation d'acides acyloxyalcanesulfoniques
FR2755689B1 (fr)	1998-12-18	Procede de preparation d'amines polyglycerylees, les amines ainsi obtenues et leurs derives
FR2736635B1 (fr)	1997-08-14	Procede de preparation d'alpha,omega-bromochloroalcanes