NO971513L - Fremgangsmåte for fremstilling av enantiomert, rene cykloalkanoindol- og azaindol- og pyrimido£1,2a|-indolkarboksylsyrer og deres aktiverte derivater - Google Patents

Fremgangsmåte for fremstilling av enantiomert, rene cykloalkanoindol- og azaindol- og pyrimido£1,2a|-indolkarboksylsyrer og deres aktiverte derivater

Info

Publication number: NO971513L
Authority: NO; Norway
Prior art keywords: cycloalkanoindole; azaindole; pyrimido; preparation; enantiomeric pure
Prior art date: 1996-04-04

Application number

NO971513A

Other languages

English (en)

Other versions

NO308301B1 (no

NO971513D0 (no

Inventor

Jan-Bernd Lenfers

Peter Fey

Paul Naab

Kai Van Laak

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-04-04

Filing date

1997-04-03

Publication date

1997-10-06

1997-04-03 Application filed by Bayer Ag filed Critical Bayer Ag

1997-04-03 Publication of NO971513D0 publication Critical patent/NO971513D0/no

1997-10-06 Publication of NO971513L publication Critical patent/NO971513L/no

2000-08-28 Publication of NO308301B1 publication Critical patent/NO308301B1/no

Links

BAXOFTOLAUCFNW-UHFFFAOYSA-N 1H-indazole Chemical compound C1=CC=C2C=NNC2=C1 BAXOFTOLAUCFNW-UHFFFAOYSA-N 0.000 title 1
HCUARRIEZVDMPT-UHFFFAOYSA-N Indole-2-carboxylic acid Chemical class C1=CC=C2NC(C(=O)O)=CC2=C1 HCUARRIEZVDMPT-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/612—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety
- C07C69/616—Esters of carboxylic acids having a carboxyl group bound to an acyclic carbon atom and having a six-membered aromatic ring in the acid moiety polycyclic
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/62—Halogen-containing esters
- C07C69/65—Halogen-containing esters of unsaturated acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

NO971513A 1996-04-04 1997-04-03 FremgangsmÕte for fremstilling av enantiomer-rene cykloalkanoindol- og azaindol- og pyrimido[1,2a]- indolkarboksylsyrer og deres aktiverte derivater, mellomprodukter samt anvendelse av disse NO308301B1 (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19613549A DE19613549A1 (de)	1996-04-04	1996-04-04	Verfahren zur Herstellung von enantiomerenreinen Cycloalkano-indol- und azaindol-carbonsäuren und deren aktivierte Derivate

Publications (3)

Publication Number	Publication Date
NO971513D0 NO971513D0 (no)	1997-04-03
NO971513L true NO971513L (no)	1997-10-06
NO308301B1 NO308301B1 (no)	2000-08-28

Family

ID=7790501

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
NO971513A NO308301B1 (no)	1996-04-04	1997-04-03	FremgangsmÕte for fremstilling av enantiomer-rene cykloalkanoindol- og azaindol- og pyrimido[1,2a]- indolkarboksylsyrer og deres aktiverte derivater, mellomprodukter samt anvendelse av disse
NO20003784A NO20003784D0 (no)	1996-04-04	2000-07-24	FremgangsmÕte for fremstilling av enansiomert rene cykloalkanoindolkarboksylsyre og azaindolkarboksylsyrer og pyrimido 1,2a indolkarboksylsyrer og derivater derav

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
NO20003784A NO20003784D0 (no)	1996-04-04	2000-07-24	FremgangsmÕte for fremstilling av enansiomert rene cykloalkanoindolkarboksylsyre og azaindolkarboksylsyrer og pyrimido 1,2a indolkarboksylsyrer og derivater derav

Country Status (27)

Country	Link
US (1)	US5952498A (no)
EP (1)	EP0799829B1 (no)
JP (2)	JP4235268B2 (no)
KR (1)	KR970069988A (no)
CN (2)	CN1067394C (no)
AR (2)	AR006544A1 (no)
AT (1)	ATE246193T1 (no)
AU (1)	AU722592B2 (no)
BR (1)	BR9701672A (no)
CA (1)	CA2201435C (no)
CZ (1)	CZ102197A3 (no)
DE (2)	DE19613549A1 (no)
DZ (1)	DZ2202A1 (no)
EE (1)	EE9700079A (no)
ES (1)	ES2202506T3 (no)
HR (1)	HRP970178A2 (no)
HU (1)	HU218494B (no)
ID (1)	ID16794A (no)
IL (1)	IL120591A (no)
MA (1)	MA24130A1 (no)
NO (2)	NO308301B1 (no)
NZ (1)	NZ314498A (no)
PL (1)	PL319269A1 (no)
SG (1)	SG60050A1 (no)
SK (1)	SK42897A3 (no)
TN (1)	TNSN97060A1 (no)
ZA (1)	ZA972831B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4435477A1 (de)	1994-10-04	1996-04-11	Bayer Ag	Cycloalkano-indol- und -azaindol-derivate
AU2001244635A1 (en) *	2000-03-30	2001-10-15	Yamanouchi Pharmaceutical Co..Ltd.	Hydrazide derivatives
WO2005051382A1 (ja) *	2003-11-28	2005-06-09	Astellas Pharma Inc.	脂質低下作用増強剤
KR101494067B1 (ko)	2004-03-05	2015-02-16	더 트러스티스 오브 더 유니버시티 오브 펜실바니아	부작용을 최소화하면서 과지질혈증 및 과콜레스테롤혈증과 연관된 질환 또는 질병의 치료 방법
AU2005230397B2 (en) *	2004-04-09	2010-04-08	Elanco Animal Health Ireland Limited	Intermittent dosing regimen for the treatment of overweight with MTP-inhibitors
AU2006304689A1 (en) *	2005-10-18	2007-04-26	Aegerion Pharmaceuticals	Compositions for lowering serum cholesterol and/or triglycerides
US20080051427A1 (en) *	2006-05-18	2008-02-28	Fritz Schuckler	Pharmaceutical Compositions and Methods of Using Same
JP2010513534A (ja) *	2006-12-21	2010-04-30	エージェリオンファーマシューティカルズ，インコーポレイテッド	Ｍｔｐインヒビターおよびコレステロール吸収インヒビターを含む組み合わせを用いて肥満症を処置する方法
WO2008124384A2 (en) *	2007-04-03	2008-10-16	Aegerion Pharmaceuticals, Inc.	Combinations of mtp inhibitors with cholesterol absorption inhibitors or interferon for treating hepatitis c
PT2968284T (pt)	2013-03-14	2021-06-28	Osteoqc Inc	Derivados alquilamina de harmina para promoção de crescimento ósseo
AU2019320773B2 (en)	2018-08-14	2024-12-05	Ossifi Therapeutics Llc	Fluoro β-carboline compounds
US10947236B2 (en)	2018-08-14	2021-03-16	Osteoqc Inc.	Pyrrolo-dipyridine compounds
CA3186856A1 (en)	2020-07-29	2022-02-03	Ruth NALLEN	Lomitapide for use in methods of treating hyperlipidemia and hypercholesterolemia in pediatric patients

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3900261A1 (de) *	1988-05-31	1989-12-07	Bayer Ag	Substituierte 4-(chinolin-2-yl-methoxy) phenyl-essigsaeure-derivate
DE4200954A1 (de) *	1991-04-26	1992-10-29	Bayer Ag	Heterocyclisch substituierte phenylessigsaeurederivate
DE4208051A1 (de) *	1992-03-13	1993-09-16	Bayer Ag	Substituierte phenylessigsaeureamide
DE4302956A1 (de) *	1993-02-03	1994-08-04	Bayer Ag	Substituierte Imidazo(4,5-b)pyridine und Benzimidazole
DE4435477A1 (de) *	1994-10-04	1996-04-11	Bayer Ag	Cycloalkano-indol- und -azaindol-derivate

1996
- 1996-04-04 DE DE19613549A patent/DE19613549A1/de not_active Withdrawn
1997
- 1997-03-24 AT AT97104941T patent/ATE246193T1/de not_active IP Right Cessation
- 1997-03-24 ES ES97104941T patent/ES2202506T3/es not_active Expired - Lifetime
- 1997-03-24 DE DE59710487T patent/DE59710487D1/de not_active Expired - Lifetime
- 1997-03-24 EP EP97104941A patent/EP0799829B1/de not_active Expired - Lifetime
- 1997-03-27 AU AU16602/97A patent/AU722592B2/en not_active Ceased
- 1997-03-27 NZ NZ314498A patent/NZ314498A/en unknown
- 1997-03-28 HR HR19613549.4A patent/HRP970178A2/xx not_active Application Discontinuation
- 1997-03-31 US US08/829,566 patent/US5952498A/en not_active Expired - Lifetime
- 1997-03-31 ID IDP971060A patent/ID16794A/id unknown
- 1997-04-01 SG SG1997001028A patent/SG60050A1/en unknown
- 1997-04-01 CA CA002201435A patent/CA2201435C/en not_active Expired - Fee Related
- 1997-04-01 JP JP09635197A patent/JP4235268B2/ja not_active Expired - Fee Related
- 1997-04-01 MA MA24543A patent/MA24130A1/fr unknown
- 1997-04-02 TN TNTNSN97060A patent/TNSN97060A1/fr unknown
- 1997-04-02 IL IL12059197A patent/IL120591A/xx not_active IP Right Cessation
- 1997-04-02 DZ DZ970049A patent/DZ2202A1/fr active
- 1997-04-03 KR KR1019970012291A patent/KR970069988A/ko not_active Withdrawn
- 1997-04-03 HU HU9700698A patent/HU218494B/hu not_active IP Right Cessation
- 1997-04-03 NO NO971513A patent/NO308301B1/no not_active IP Right Cessation
- 1997-04-03 ZA ZA9702831A patent/ZA972831B/xx unknown
- 1997-04-03 PL PL97319269A patent/PL319269A1/xx unknown
- 1997-04-03 CZ CZ971021A patent/CZ102197A3/cs unknown
- 1997-04-03 SK SK428-97A patent/SK42897A3/sk unknown
- 1997-04-03 EE EE9700079A patent/EE9700079A/xx unknown
- 1997-04-04 BR BR9701672A patent/BR9701672A/pt active Search and Examination
- 1997-04-04 AR ARP970101366A patent/AR006544A1/es unknown
- 1997-04-04 CN CN97110276A patent/CN1067394C/zh not_active Expired - Fee Related
1998
- 1998-03-06 AR ARP980101029A patent/AR012048A2/es unknown
2000
- 2000-07-24 NO NO20003784A patent/NO20003784D0/no not_active Application Discontinuation
- 2000-10-12 CN CN00133103A patent/CN1330065A/zh active Pending
2008
- 2008-01-31 JP JP2008021569A patent/JP2008169218A/ja active Pending

Also Published As

Publication number	Publication date
AU1660297A (en)	1997-10-09
CN1067394C (zh)	2001-06-20
PL319269A1 (en)	1997-10-13
CN1330065A (zh)	2002-01-09
NO20003784L (no)	1997-10-06
DZ2202A1 (fr)	2002-12-03
HRP970178A2 (en)	1998-04-30
CN1184109A (zh)	1998-06-10
NZ314498A (en)	1999-09-29
SK42897A3 (en)	1997-10-08
AU722592B2 (en)	2000-08-10
CZ102197A3 (en)	1997-10-15
ATE246193T1 (de)	2003-08-15
MX9702446A (es)	1997-10-31
CA2201435C (en)	2006-12-12
US5952498A (en)	1999-09-14
JPH1045759A (ja)	1998-02-17
KR970069988A (ko)	1997-11-07
IL120591A0 (en)	1997-08-14
CA2201435A1 (en)	1997-10-04
NO20003784D0 (no)	2000-07-24
ID16794A (id)	1997-11-13
DE59710487D1 (de)	2003-09-04
HU9700698D0 (en)	1997-05-28
IL120591A (en)	2000-11-21
AR006544A1 (es)	1999-09-08
MA24130A1 (fr)	1997-10-01
TNSN97060A1 (fr)	2005-03-15
AR012048A2 (es)	2000-09-27
EP0799829B1 (de)	2003-07-30
JP2008169218A (ja)	2008-07-24
ES2202506T3 (es)	2004-04-01
HU218494B (hu)	2000-09-28
NO308301B1 (no)	2000-08-28
NO971513D0 (no)	1997-04-03
EP0799829A1 (de)	1997-10-08
HUP9700698A1 (hu)	1998-01-28
SG60050A1 (en)	1999-02-22
EE9700079A (et)	1997-10-15
DE19613549A1 (de)	1997-10-09
ZA972831B (en)	1997-10-31
BR9701672A (pt)	1998-11-03
JP4235268B2 (ja)	2009-03-11

Legal Events

Date	Code	Title	Description
2002-12-09	MM1K	Lapsed by not paying the annual fees	Free format text: LAPSED IN OCTOBER 2002

Publication	Publication Date	Title
EG25852A (en)	2012-09-10	Teracyclic derivatives process of preparation
NO971513L (no)	1997-10-06	Fremgangsmåte for fremstilling av enantiomert, rene cykloalkanoindol- og azaindol- og pyrimido£1,2a\|-indolkarboksylsyrer og deres aktiverte derivater
AP9400706A0 (en)	1995-01-31	Indole derivatives, method of preparation and use
NO970212D0 (no)	1997-01-17	Fremgangsmåte for fremstilling av enantiomerene av O-demetyltramadol
AU2713297A (en)	1998-03-06	Process for stereoselective preparation of trans-azetidinones
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NO990697L (no)	1999-02-15	FremgangsmÕte for fremstilling av N-[(1-n-butyl-4-piperidyl)metyl]-3,4-dihydro-2H-[1,3]oksazino[3,2-a]indol-10-karboksamid og salter og mellomprodukter i fremgangsmÕten
PL309645A1 (en)	1995-10-30	Method of obtaining substituted indolone derivatives
PL330281A1 (en)	1999-05-10	Method of obtaining derivatives of phenoxypropinic acid
AU5472990A (en)	1990-11-15	Indole derivative and method of production thereof
NO993845D0 (no)	1999-08-10	Fremgangsmåte for fremstilling av smörsyrederivater
NO984206D0 (no)	1998-09-11	Fremgangsmåte for fremstilling av N-beskyttende D-prolinderivater
GR3033714T3 (en)	2000-10-31	Process for the preparation of o-chloro-methyl-phenylglyoxylic acid derivatives
PL326699A1 (en)	1998-10-26	Method of obtaining derivatives of 3-phenyl-1-methylenedioxyphenyl-indane 2-carboxylic acids
IL120747A0 (en)	1997-09-30	Efficient and highly enantioselective process for the preparation of enantiomerically pure cyclopentane-beta-amino acids
AU4596097A (en)	1998-04-17	Improved therapeutic uses of 4-quinoline-carboxylic acid derivatives
NO991098L (no)	1999-05-05	FremgangsmÕte for fremstilling av 2-fenyl-3-naftylpropionsyrederivater
IL136922A0 (en)	2001-06-14	Process for the preparation of enantiomerically pure indolecarboxylic acid derivatives and some such new compounds
AU1733597A (en)	1997-09-10	Process for the preparation of alpha-alkoxyphenylacetic acid derivatives
NO915055D0 (no)	1991-12-20	Fremgangsmaate for fremstilling av enantiomerisk rene tienopyranderivater
PL319445A1 (en)	1998-10-12	Method of obtaining substituted derivatives of indole
PL293174A1 (en)	1993-11-02	Method of obtaining 3,7-disubstituted indole derivatives
PL303257A1 (en)	1995-10-30	Method of obtaining novel 3-acyl derivatives of 1-phenylimidazolidine
ZA9713B (en)	1997-07-17	Process for the preparation of o-chloromethyl-phenyl-glyoxylic acid derivatives
AU5654098A (en)	1998-06-29	Process for the racemization of substituted 4-ketocarboxylic acids