NO20060319L - 3,5-disubstituerte indazolforbindelser, farmasoytiske blandinger og fremgangsmater for a mediere eller inhibere celleproliferasjon - Google Patents
3,5-disubstituerte indazolforbindelser, farmasoytiske blandinger og fremgangsmater for a mediere eller inhibere celleproliferasjonInfo
- Publication number
- NO20060319L NO20060319L NO20060319A NO20060319A NO20060319L NO 20060319 L NO20060319 L NO 20060319L NO 20060319 A NO20060319 A NO 20060319A NO 20060319 A NO20060319 A NO 20060319A NO 20060319 L NO20060319 L NO 20060319L
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- cell proliferation
- mediate
- methods
- inhibit cell
- Prior art date
Links
- 230000004663 cell proliferation Effects 0.000 title abstract 4
- 238000000034 method Methods 0.000 title abstract 2
- -1 3,5-Disubstituted Indazole Compounds Chemical class 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 206010012689 Diabetic retinopathy Diseases 0.000 abstract 1
- 208000010412 Glaucoma Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000001253 Protein Kinase Human genes 0.000 abstract 1
- 201000004681 Psoriasis Diseases 0.000 abstract 1
- 230000033115 angiogenesis Effects 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 230000001419 dependent effect Effects 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 125000003453 indazolyl group Chemical class N1N=C(C2=C1C=CC=C2)* 0.000 abstract 1
- 201000003142 neovascular glaucoma Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 230000003449 preventive effect Effects 0.000 abstract 1
- 108060006633 protein kinase Proteins 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US49147403P | 2003-07-30 | 2003-07-30 | |
| US49207303P | 2003-07-31 | 2003-07-31 | |
| PCT/IB2004/002441 WO2005009997A1 (en) | 2003-07-30 | 2004-07-19 | 3,5 disubstituted indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20060319L true NO20060319L (no) | 2006-02-24 |
Family
ID=34108010
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20060319A NO20060319L (no) | 2003-07-30 | 2006-01-20 | 3,5-disubstituerte indazolforbindelser, farmasoytiske blandinger og fremgangsmater for a mediere eller inhibere celleproliferasjon |
Country Status (24)
| Country | Link |
|---|---|
| US (2) | US7008953B2 (es) |
| EP (1) | EP1658284A1 (es) |
| JP (1) | JP3920914B2 (es) |
| KR (1) | KR20060030914A (es) |
| AR (1) | AR045143A1 (es) |
| AU (1) | AU2004259531A1 (es) |
| BR (1) | BRPI0413051A (es) |
| CA (1) | CA2532908A1 (es) |
| CO (1) | CO5650247A2 (es) |
| EA (1) | EA200600123A1 (es) |
| EC (1) | ECSP066335A (es) |
| IL (1) | IL172924A0 (es) |
| IS (1) | IS8214A (es) |
| MA (1) | MA27937A1 (es) |
| MX (1) | MXPA06001193A (es) |
| NL (1) | NL1026761C2 (es) |
| NO (1) | NO20060319L (es) |
| OA (1) | OA13196A (es) |
| PA (1) | PA8608201A1 (es) |
| PE (1) | PE20050330A1 (es) |
| TN (1) | TNSN06038A1 (es) |
| TW (1) | TW200521124A (es) |
| UY (1) | UY28442A1 (es) |
| WO (1) | WO2005009997A1 (es) |
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| US12419865B2 (en) | 2018-12-06 | 2025-09-23 | Arisan Therapeutics Inc. | Compounds for the treatment of arenavirus infection |
| WO2020150545A1 (en) | 2019-01-17 | 2020-07-23 | Samumed, Llc | Pyrazole derivatives as modulators of the wnt/b-catenin signaling pathway |
| WO2021168341A1 (en) | 2020-02-21 | 2021-08-26 | Samumed, Llc | Solid forms of 1-(5-(3-(7-(3-fluorophenyl)-3h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridin-5-yl)pyridin-3-yl)-n,n-dimethylmethanamine |
| JP2025530213A (ja) | 2022-09-09 | 2025-09-11 | ミリックス ファーマ リミテッド | Ｎｍｔ阻害剤を含む抗体薬物コンジュゲート及びその使用 |
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| GB1376600A (en) | 1971-02-15 | 1974-12-04 | Agfa Gevaert | Photographic developer compositions |
| FR2265739B1 (es) | 1974-03-29 | 1976-12-17 | Ugine Kuhlmann | |
| JPS5615287A (en) | 1979-07-16 | 1981-02-14 | Chugai Pharmaceut Co Ltd | Pyrazoloindazole derivative and its preparation |
| JPS57109787A (en) | 1980-12-26 | 1982-07-08 | Chugai Pharmaceut Co Ltd | Pyrazoloindazole derivative |
| JPS59228248A (ja) | 1983-06-08 | 1984-12-21 | Konishiroku Photo Ind Co Ltd | 直接ポジ用ハロゲン化銀写真感光材料 |
| JPS604184A (ja) | 1983-06-23 | 1985-01-10 | Chugai Pharmaceut Co Ltd | ピラゾロインダゾ−ル誘導体 |
| DE3842091A1 (de) | 1987-12-14 | 1989-07-13 | Fuji Photo Film Co Ltd | Bilderzeugungsverfahren |
| US5208248A (en) | 1991-01-11 | 1993-05-04 | Merck Sharpe & Dohme, Ltd. | Indazole-substituted five-membered heteroaromatic compounds |
| EP0494774A1 (en) | 1991-01-11 | 1992-07-15 | MERCK SHARP & DOHME LTD. | Indazole-substituted fivemembered heteroaromatic compounds |
| NZ243065A (en) | 1991-06-13 | 1995-07-26 | Lundbeck & Co As H | Piperidine derivatives and pharmaceutical compositions |
| ZA951822B (en) | 1994-12-23 | 1996-09-26 | Glaxo Group Ltd | Chemical compounds |
| DE69624081T2 (de) | 1995-12-20 | 2003-06-12 | Agouron Pharmaceuticals, Inc. | Matrix-metalloprotease Inhibitoren |
| EP0818442A3 (en) | 1996-07-12 | 1998-12-30 | Pfizer Inc. | Cyclic sulphone derivatives as inhibitors of metalloproteinases and of the production of tumour necrosis factor |
| HRP970371A2 (en) | 1996-07-13 | 1998-08-31 | Kathryn Jane Smith | Heterocyclic compounds |
| EP0973767A1 (en) | 1997-03-31 | 2000-01-26 | Dupont Pharmaceuticals Company | Indazoles of cyclic ureas useful as hiv protease inhibitors |
| FR2767475A1 (fr) | 1997-08-25 | 1999-02-26 | Oreal | Compositions de teinture des fibres keratiniques contenant des derives d'indazoles et procede |
| BR9916536A (pt) | 1998-12-23 | 2002-01-02 | Searle & Co | Método para o tratamento ou prevenção de um distúrbio de neoplasia em um mamìfero em necessidade deste tratamento ou prevenção, e, combinação |
| GB2345486A (en) | 1999-01-11 | 2000-07-12 | Glaxo Group Ltd | Heteroaromatic protein tyrosine kinase inhibitors |
| YU54202A (sh) | 2000-01-18 | 2006-01-16 | Agouron Pharmaceuticals Inc. | Jedinjenja indazola, farmaceutske smeše i postupci za stimulisanje i inhibiranje ćelijske proliferacije |
| KR100423899B1 (ko) | 2000-05-10 | 2004-03-24 | 주식회사 엘지생명과학 | 세포 증식 억제제로 유용한 1,1-디옥소이소티아졸리딘을갖는 인다졸 |
| US6897231B2 (en) | 2000-07-31 | 2005-05-24 | Signal Pharmaceuticals, Inc. | Indazole derivatives as JNK inhibitors and compositions and methods related thereto |
| US7064215B2 (en) | 2001-07-03 | 2006-06-20 | Chiron Corporation | Indazole benzimidazole compounds |
| FR2831536A1 (fr) | 2001-10-26 | 2003-05-02 | Aventis Pharma Sa | Nouveaux derives de benzimidazoles, leur procede de preparation, leur application a titre de medicament, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de kdr |
| US7008953B2 (en) * | 2003-07-30 | 2006-03-07 | Agouron Pharmaceuticals, Inc. | 3, 5 Disubstituted indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation |
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- 2004-07-19 AU AU2004259531A patent/AU2004259531A1/en not_active Abandoned
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- 2004-07-19 EA EA200600123A patent/EA200600123A1/ru unknown
- 2004-07-19 CA CA002532908A patent/CA2532908A1/en not_active Abandoned
- 2004-07-19 EP EP04744094A patent/EP1658284A1/en not_active Withdrawn
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- 2004-07-19 JP JP2006521699A patent/JP3920914B2/ja not_active Expired - Fee Related
- 2004-07-19 OA OA1200600024A patent/OA13196A/fr unknown
- 2004-07-19 WO PCT/IB2004/002441 patent/WO2005009997A1/en not_active Ceased
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- 2006-01-30 EC EC2006006335A patent/ECSP066335A/es unknown
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| IS8214A (is) | 2005-12-30 |
| WO2005009997A1 (en) | 2005-02-03 |
| US20050026960A1 (en) | 2005-02-03 |
| CO5650247A2 (es) | 2006-06-30 |
| AR045143A1 (es) | 2005-10-19 |
| MXPA06001193A (es) | 2006-04-11 |
| AU2004259531A1 (en) | 2005-02-03 |
| JP2007500183A (ja) | 2007-01-11 |
| US20060142345A1 (en) | 2006-06-29 |
| ECSP066335A (es) | 2006-07-28 |
| NL1026761C2 (nl) | 2005-10-18 |
| MA27937A1 (fr) | 2006-06-01 |
| US7008953B2 (en) | 2006-03-07 |
| UY28442A1 (es) | 2005-02-28 |
| PA8608201A1 (es) | 2005-03-03 |
| NL1026761A1 (nl) | 2005-02-01 |
| CA2532908A1 (en) | 2005-02-03 |
| IL172924A0 (en) | 2006-06-11 |
| KR20060030914A (ko) | 2006-04-11 |
| BRPI0413051A (pt) | 2006-10-17 |
| EP1658284A1 (en) | 2006-05-24 |
| PE20050330A1 (es) | 2005-05-16 |
| OA13196A (en) | 2006-12-13 |
| TW200521124A (en) | 2005-07-01 |
| TNSN06038A1 (fr) | 2007-10-03 |
| EA200600123A1 (ru) | 2006-06-30 |
| JP3920914B2 (ja) | 2007-05-30 |
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