NO20072767L - Gabapentin prodrug vedvarende frigivelse orale doseringsformer - Google Patents

Gabapentin prodrug vedvarende frigivelse orale doseringsformer

Info

Publication number
NO20072767L
NO20072767L NO20072767A NO20072767A NO20072767L NO 20072767 L NO20072767 L NO 20072767L NO 20072767 A NO20072767 A NO 20072767A NO 20072767 A NO20072767 A NO 20072767A NO 20072767 L NO20072767 L NO 20072767L
Authority
NO
Norway
Prior art keywords
dosage forms
sustained release
oral dosage
release oral
gabapentin
Prior art date
Application number
NO20072767A
Other languages
English (en)
Other versions
NO338688B1 (no
Inventor
Kenneth C Cundy
Srikonda Sastry
Manshiu Leung
Balaji V Kadri
Paul E Stach
Original Assignee
Xenoport Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35929688&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20072767(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Xenoport Inc filed Critical Xenoport Inc
Publication of NO20072767L publication Critical patent/NO20072767L/no
Publication of NO338688B1 publication Critical patent/NO338688B1/no

Links

Classifications

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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
    • A61K31/225—Polycarboxylic acids
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    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
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    • A61K9/20—Pills, tablets, discs, rods
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    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Addiction (AREA)
  • Inorganic Chemistry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Anesthesiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychology (AREA)
  • Immunology (AREA)
  • Hospice & Palliative Care (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Vedvarende frigivelse oral doseringsformer av et gabapentin prodrug av 1-{[(a-isobutanoyloksyetoksy)karbonyl]aminometyl}-1-sykloheksan eddiksyre er beskrevet. Doseringsformene er anvendelige for forebygging av sykdommer og forstyrrelser hvor gabapentin er terapeutisk effektivt.
NO20072767A 2004-11-04 2007-05-31 Gabapentin prodrug vedvarende frigivelse orale doseringsformuleringer NO338688B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US62573704P 2004-11-04 2004-11-04
PCT/US2005/040127 WO2006050514A1 (en) 2004-11-04 2005-11-03 Gabapentin prodrug sustained release oral dosage forms

Publications (2)

Publication Number Publication Date
NO20072767L true NO20072767L (no) 2007-07-27
NO338688B1 NO338688B1 (no) 2016-10-03

Family

ID=35929688

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20072767A NO338688B1 (no) 2004-11-04 2007-05-31 Gabapentin prodrug vedvarende frigivelse orale doseringsformuleringer

Country Status (16)

Country Link
US (8) US8795725B2 (no)
EP (1) EP1811986B1 (no)
JP (2) JP2008518971A (no)
KR (1) KR101228399B1 (no)
CN (2) CN101068538A (no)
AU (1) AU2005301970B2 (no)
BR (1) BRPI0517227B8 (no)
CA (1) CA2584338C (no)
IL (1) IL182964A0 (no)
MX (1) MX2007005306A (no)
NO (1) NO338688B1 (no)
NZ (1) NZ554737A (no)
RU (1) RU2440112C2 (no)
TW (1) TWI377938B (no)
WO (1) WO2006050514A1 (no)
ZA (1) ZA200703571B (no)

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US8048917B2 (en) 2005-04-06 2011-11-01 Xenoport, Inc. Prodrugs of GABA analogs, compositions and uses thereof
US7025745B2 (en) * 2002-10-07 2006-04-11 Advanced Cardiovascular Systems, Inc. Method of making a catheter balloon using a tapered mandrel
KR20060119971A (ko) * 2003-09-11 2006-11-24 제노포트 인코포레이티드 Ｇａｂａ 유사체의 전구약물을 이용한 요실금의 치료및/또는 예방
NZ579515A (en) * 2003-09-17 2011-09-30 Xenoport Inc Treating or preventing restless legs syndrome using prodrugs of gaba analogs
SG147437A1 (en) 2003-10-14 2008-11-28 Xenoport Inc Crystalline form of gamma-aminobutyric acid analog
MX2007005306A (es) * 2004-11-04 2007-06-11 Xenoport Inc Formas de dosis oral de liberacion sostenida de la prodroga gabapentina.
US7351740B2 (en) * 2005-06-20 2008-04-01 Xenoport, Inc. Acyloxyalkyl carbamate prodrugs of tranexamic acid, methods of synthesis and use
WO2007027477A2 (en) * 2005-08-23 2007-03-08 Xenoport, Inc. Treating vulvodynia using prodrugs of gaba analogs
WO2007027476A2 (en) * 2005-08-26 2007-03-08 Xenoport, Inc. Treating premature ejaculation using gabapentin and pregabalin prodrugs
US20080161393A1 (en) * 2006-12-08 2008-07-03 Barrett Ronald W Use of prodrugs of GABA analogs for treating disease
TWI369982B (en) * 2007-01-11 2012-08-11 Xenoport Inc Sustained release oral dosage forms of a prodrug of r-baclofen and methods of treatment
WO2010101115A1 (ja) 2009-03-02 2010-09-10 アステラス製薬株式会社 固形製剤の包装体
KR20110117216A (ko) * 2009-03-03 2011-10-26 제노포트 인코포레이티드 Ｒ-바클로펜 전구약물의 서방형 경구 투약 형태
JP5580345B2 (ja) * 2009-03-06 2014-08-27 ゼノポート，インコーポレイティド 高充填量のガバペンチンプロドラッグを有する経口剤形
WO2011028234A1 (en) * 2009-09-04 2011-03-10 Xenoport, Inc. Uses of acyloxyalkyl carbamate prodrugs of tranexamic acid
WO2011091164A1 (en) * 2010-01-22 2011-07-28 Xenoport, Inc. Oral dosage forms having a high loading of a tranexamic acid prodrug
JP5936542B2 (ja) 2010-09-01 2016-06-22 アステラス製薬株式会社 包装体
CN104042597A (zh) * 2013-03-13 2014-09-17 苏州朗易生物医药研究有限公司 一种治疗神经痛的药物组合物及其制备方法
CA2999367C (en) 2015-09-23 2023-09-26 Xw Laboratories Inc. Prodrugs of gamma-hydroxybutyric acid, compositions and uses thereof
BR102017028213B1 (pt) 2017-12-27 2022-07-19 Loccitane Do Brasil S.A. Composição cosmética compreende óleo de licuri, uso da dita composição e método cosmético
WO2020165633A1 (en) * 2019-02-11 2020-08-20 Glenmark Pharmaceuticals Limited A pharmaceutical composition of gabapentin enacarbil or salt thereof
CN114306234A (zh) * 2021-12-23 2022-04-12 江苏百奥信康医药科技有限公司 一种含有加巴喷丁复合物的tpgs胶束口服液及其制备方法
CN114288246A (zh) * 2021-12-23 2022-04-08 江苏百奥信康医药科技有限公司 一种含有加巴喷丁复合物的聚合物胶束口服液及其制备方法
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US20140302140A1 (en) 2014-10-09
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US20180207117A1 (en) 2018-07-26
RU2007120570A (ru) 2008-12-10
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US20170071888A1 (en) 2017-03-16
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