NO20081075L - Macrocykliske inhibitorer av hepatitt C virus - Google Patents

Macrocykliske inhibitorer av hepatitt C virus

Info

Publication number
NO20081075L
NO20081075L NO20081075A NO20081075A NO20081075L NO 20081075 L NO20081075 L NO 20081075L NO 20081075 A NO20081075 A NO 20081075A NO 20081075 A NO20081075 A NO 20081075A NO 20081075 L NO20081075 L NO 20081075L
Authority
NO
Norway
Prior art keywords
alkylene
alkyl
carbocyclyl
hydrogen
heterocyclyl
Prior art date
Application number
NO20081075A
Other languages
English (en)
Norwegian (no)
Inventor
Herman Augustinus De Kock
Hans Wallberg
Pierre Jean-Marie Raboisson
Kenneth Alan Simmen
Lili Hu
Karl Magnus Nilsson
Bengt Bertil Samuelsson
Asa Annicka Kristina Rosenquist
Anna Karin Gertrud Linnea Belfrage
Mats Stefan Lindstrom
Pia Cecilia Kahnberg
Karin Charlotta Lindquist
Horst Juergen Wahling
Sven Christer Sahlberg
Bjorn Olof Classon
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37708968&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20081075(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of NO20081075L publication Critical patent/NO20081075L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D245/00Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
    • C07D245/04Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20081075A 2005-07-29 2008-02-29 Macrocykliske inhibitorer av hepatitt C virus NO20081075L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05107057 2005-07-29
EP06113097 2006-04-25
PCT/EP2006/064822 WO2007014927A2 (fr) 2005-07-29 2006-07-28 Inhibiteurs macrocycliques du virus de l'hepatite c

Publications (1)

Publication Number Publication Date
NO20081075L true NO20081075L (no) 2008-04-25

Family

ID=37708968

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20081075A NO20081075L (no) 2005-07-29 2008-02-29 Macrocykliske inhibitorer av hepatitt C virus

Country Status (31)

Country Link
US (1) US7659245B2 (fr)
EP (1) EP1912981B1 (fr)
JP (1) JP5230418B2 (fr)
KR (1) KR101083631B1 (fr)
AP (1) AP2585A (fr)
AR (1) AR057702A1 (fr)
AT (1) ATE455775T1 (fr)
AU (1) AU2006274866B2 (fr)
BR (1) BRPI0614153A2 (fr)
CA (1) CA2617103C (fr)
CY (1) CY1110008T1 (fr)
DE (1) DE602006011905D1 (fr)
DK (1) DK1912981T3 (fr)
EA (1) EA014188B1 (fr)
ES (1) ES2339702T3 (fr)
GT (1) GT200600343A (fr)
HR (1) HRP20100209T1 (fr)
IL (1) IL188320A (fr)
ME (1) ME01454B (fr)
MY (1) MY151026A (fr)
NO (1) NO20081075L (fr)
NZ (1) NZ564540A (fr)
PE (1) PE20070343A1 (fr)
PL (1) PL1912981T3 (fr)
PT (1) PT1912981E (fr)
RS (1) RS51227B (fr)
SI (1) SI1912981T1 (fr)
SV (1) SV2008002641A (fr)
TW (1) TWI387597B (fr)
UY (1) UY29704A1 (fr)
WO (1) WO2007014927A2 (fr)

Families Citing this family (58)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY140680A (en) 2002-05-20 2010-01-15 Bristol Myers Squibb Co Hepatitis c virus inhibitors
BRPI0506948B1 (pt) 2004-01-30 2018-09-18 Medivir Ab inibidores de serina protease ns-3 de hcv
PE20070211A1 (es) 2005-07-29 2007-05-12 Medivir Ab Compuestos macrociclicos como inhibidores del virus de hepatitis c
RU2436787C2 (ru) 2005-07-29 2011-12-20 Тиботек Фармасьютикалз Лтд. Макроциклические ингибиторы вируса гепатита с
JO2768B1 (en) * 2005-07-29 2014-03-15 تيبوتيك فارماسيوتيكالز ليمتد Large cyclic inhibitors of hepatitis C virus
WO2007014925A1 (fr) 2005-07-29 2007-02-08 Tibotec Pharmaceuticals Ltd. Inhibiteurs macrocycliques du virus de l'hépatite c
BRPI0617274A2 (pt) 2005-10-11 2011-07-19 Intermune Inc compostos e métodos para a inibição de replicação viral de hepatite c
US7741281B2 (en) 2005-11-03 2010-06-22 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
RU2008152171A (ru) 2006-07-05 2010-08-10 Интермьюн, Инк. (Us) Новые ингибиторы вирусной репликации гепатита с
US7935670B2 (en) 2006-07-11 2011-05-03 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
DK2041156T3 (en) 2006-07-13 2014-02-24 Achillion Pharmaceuticals Inc 4-AMINO-4-OXOBUTANOYL Peptides AS INHIBITORS OF VIRUS REPLICATION
US8343477B2 (en) 2006-11-01 2013-01-01 Bristol-Myers Squibb Company Inhibitors of hepatitis C virus
US7772180B2 (en) 2006-11-09 2010-08-10 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US7763584B2 (en) 2006-11-16 2010-07-27 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US8003604B2 (en) 2006-11-16 2011-08-23 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US7888464B2 (en) 2006-11-16 2011-02-15 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
ES2470568T3 (es) * 2006-11-17 2014-06-24 Janssen R&D Ireland Inhibidores macroc�clicos del virus de la hepatitis C
BRPI0806853B1 (pt) * 2007-02-01 2018-03-20 Janssen Sciences Ireland Uc Processos e intermediários para preparar um inibidor de protease macrocíclico de hcv
BRPI0807087A2 (pt) * 2007-02-08 2014-06-10 Tibotec Pharm Ltd Inibidores de hcv macrocíclicos substituídos de pirimidina
ITMI20071616A1 (it) 2007-08-03 2009-02-04 Cosmo Spa Processo enzimatico per l'ottenimento di 17-alfa monoesteri del cortexolone e/o suoi 9,11-deidroderivati.
WO2009042668A2 (fr) * 2007-09-24 2009-04-02 Achillion Pharmaceuticals, Inc. Peptides contenant de l'urée en tant qu'inhibiteurs de la réplication virale
US8383583B2 (en) 2007-10-26 2013-02-26 Enanta Pharmaceuticals, Inc. Macrocyclic, pyridazinone-containing hepatitis C serine protease inhibitors
US8426360B2 (en) * 2007-11-13 2013-04-23 Enanta Pharmaceuticals, Inc. Carbocyclic oxime hepatitis C virus serine protease inhibitors
US8263549B2 (en) 2007-11-29 2012-09-11 Enanta Pharmaceuticals, Inc. C5-substituted, proline-derived, macrocyclic hepatitis C serine protease inhibitors
US8202996B2 (en) 2007-12-21 2012-06-19 Bristol-Myers Squibb Company Crystalline forms of N-(tert-butoxycarbonyl)-3-methyl-L-valyl-(4R)-4-((7-chloro-4-methoxy-1-isoquinolinyl)oxy)-N- ((1R,2S)-1-((cyclopropylsulfonyl)carbamoyl)-2-vinylcyclopropyl)-L-prolinamide
EP2226315A4 (fr) 2007-12-28 2012-01-25 Carna Biosciences Inc Dérivé de 2-aminoquinazoline
CA2719008A1 (fr) 2008-03-20 2009-09-24 Enanta Pharmaceuticals, Inc. Composes macrocycliques fluores en tant qu'inhibiteurs du virus de l'hepatite c
US8163921B2 (en) 2008-04-16 2012-04-24 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
EP2300491B1 (fr) 2008-05-29 2016-01-06 Bristol-Myers Squibb Company Inhibiteurs du virus de l hépatite c
US7964560B2 (en) 2008-05-29 2011-06-21 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US8207341B2 (en) 2008-09-04 2012-06-26 Bristol-Myers Squibb Company Process or synthesizing substituted isoquinolines
UY32099A (es) * 2008-09-11 2010-04-30 Enanta Pharm Inc Inhibidores macrocíclicos de serina proteasas de hepatitis c
US8563505B2 (en) 2008-09-29 2013-10-22 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US8044087B2 (en) 2008-09-29 2011-10-25 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
AU2009324643B2 (en) 2008-12-10 2014-08-28 Achillion Pharmaceuticals, Inc. New 4-amino-4-oxobutanoyl peptides as inhibitors of viral replication
US8283310B2 (en) 2008-12-15 2012-10-09 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
LT2401272T (lt) 2009-02-27 2017-03-27 Janssen Pharmaceuticals, Inc. Hcv makrociklinio slopiklio amorfinė druska
WO2010118078A1 (fr) 2009-04-08 2010-10-14 Idenix Pharmaceuticals, Inc. Inhibiteurs macrocycliques de la sérine protéase
NZ596546A (en) * 2009-05-29 2012-12-21 Syngenta Participations Ag Substituted quinazolines as fungicides
TW201117812A (en) 2009-08-05 2011-06-01 Idenix Pharmaceuticals Inc Macrocyclic serine protease inhibitors
CA2822556A1 (fr) 2010-12-30 2012-07-05 Enanta Pharmaceuticals, Inc Inhibiteurs macrocycliques de serine protease d'hepatite c
US8951964B2 (en) 2010-12-30 2015-02-10 Abbvie Inc. Phenanthridine macrocyclic hepatitis C serine protease inhibitors
WO2012109398A1 (fr) 2011-02-10 2012-08-16 Idenix Pharmaceuticals, Inc. Inhibiteurs macrocycliques de sérine protéase, compositions pharmaceutiques les contenant et leur utilisation pour le traitement des infections par le vhc
US8957203B2 (en) 2011-05-05 2015-02-17 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US10201584B1 (en) 2011-05-17 2019-02-12 Abbvie Inc. Compositions and methods for treating HCV
US8691757B2 (en) 2011-06-15 2014-04-08 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
CA2858659A1 (fr) 2011-12-28 2013-07-04 Janssen R&D Ireland Derives heterobicycliques en tant qu'inhibiteurs de vhc
NZ707115A (en) * 2012-10-15 2018-03-23 Albemarle Corp Processes for the synthesis of 2-amino-4,6-dimethoxybenzamide and other benzamide compounds
BR112015007879A2 (pt) 2012-10-19 2017-07-04 Bristol Myers Squibb Co inibidores do vírus da hepatite c
EP2914613B1 (fr) 2012-11-02 2017-11-22 Bristol-Myers Squibb Company Inhibiteurs du virus de l'hépatite c
US9334279B2 (en) 2012-11-02 2016-05-10 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US9643999B2 (en) 2012-11-02 2017-05-09 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US9409943B2 (en) 2012-11-05 2016-08-09 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
EP2964664B1 (fr) 2013-03-07 2017-01-11 Bristol-Myers Squibb Company Inhibiteurs du virus de l'hépatite c
US9006423B2 (en) 2013-03-15 2015-04-14 Achillion Pharmaceuticals Inc. Process for making a 4-amino-4-oxobutanoyl peptide cyclic analogue, an inhibitor of viral replication, and intermediates thereof
US9085607B2 (en) 2013-03-15 2015-07-21 Achillion Pharmaceuticals, Inc. ACH-0142684 sodium salt polymorph, composition including the same, and method of manufacture thereof
WO2015103490A1 (fr) 2014-01-03 2015-07-09 Abbvie, Inc. Formes galéniques antivirales solides
EP3108879A1 (fr) 2015-06-25 2016-12-28 Cassiopea S.p.A. Formulation à concentration élevée

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6323180B1 (en) 1998-08-10 2001-11-27 Boehringer Ingelheim (Canada) Ltd Hepatitis C inhibitor tri-peptides
UA74546C2 (en) * 1999-04-06 2006-01-16 Boehringer Ingelheim Ca Ltd Macrocyclic peptides having activity relative to hepatitis c virus, a pharmaceutical composition and use of the pharmaceutical composition
US6867185B2 (en) * 2001-12-20 2005-03-15 Bristol-Myers Squibb Company Inhibitors of hepatitis C virus
NZ575692A (en) 2002-04-11 2009-10-30 Vertex Pharma Inhibitors of Serine Proteases, Particularly Hepatitis C Virus NS3-NS4 Protease
MY140680A (en) 2002-05-20 2010-01-15 Bristol Myers Squibb Co Hepatitis c virus inhibitors
US20050075279A1 (en) * 2002-10-25 2005-04-07 Boehringer Ingelheim International Gmbh Macrocyclic peptides active against the hepatitis C virus
US20040180815A1 (en) * 2003-03-07 2004-09-16 Suanne Nakajima Pyridazinonyl macrocyclic hepatitis C serine protease inhibitors
WO2004072243A2 (fr) * 2003-02-07 2004-08-26 Enanta Pharmaceuticals, Inc. Inhibiteurs macrocycliques de la serine protease de l'hepatite c
EP1629000B1 (fr) * 2003-04-16 2009-02-18 Bristol-Myers Squibb Company Peptide d'isoquinoleine macrocyclique inhibiteurs du virus de l'hepatite c
US7125845B2 (en) * 2003-07-03 2006-10-24 Enanta Pharmaceuticals, Inc. Aza-peptide macrocyclic hepatitis C serine protease inhibitors
UY28525A1 (es) * 2003-09-22 2005-04-29 Boehringer Ingelheim Int Péptidos macrociclicos activos contra en virus de la hepatitis c
BRPI0506948B1 (pt) * 2004-01-30 2018-09-18 Medivir Ab inibidores de serina protease ns-3 de hcv
PE20070211A1 (es) * 2005-07-29 2007-05-12 Medivir Ab Compuestos macrociclicos como inhibidores del virus de hepatitis c
TWI393723B (zh) * 2005-07-29 2013-04-21 Tibotec Pharm Ltd C型肝炎病毒之大環抑制劑(九)
US7700552B2 (en) * 2005-07-29 2010-04-20 Medivir Ab Macrocyclic inhibitors of hepatitis C virus
TWI383980B (zh) * 2005-07-29 2013-02-01 Tibotec Pharm Ltd C型肝炎病毒之大環抑制劑

Also Published As

Publication number Publication date
JP2009502890A (ja) 2009-01-29
DK1912981T3 (da) 2010-05-25
TW200745116A (en) 2007-12-16
SV2008002641A (es) 2008-07-23
HK1116488A1 (en) 2008-12-24
EA014188B1 (ru) 2010-10-29
WO2007014927A3 (fr) 2007-11-29
RS51227B (sr) 2010-12-31
ATE455775T1 (de) 2010-02-15
DE602006011905D1 (de) 2010-03-11
KR20080033475A (ko) 2008-04-16
WO2007014927A2 (fr) 2007-02-08
TWI387597B (zh) 2013-03-01
AU2006274866B2 (en) 2012-04-12
AR057702A1 (es) 2007-12-12
IL188320A (en) 2014-07-31
BRPI0614153A2 (pt) 2011-03-15
CA2617103A1 (fr) 2007-02-08
SI1912981T1 (sl) 2010-05-31
MY151026A (en) 2014-03-31
PL1912981T3 (pl) 2010-07-30
EP1912981A2 (fr) 2008-04-23
EP1912981B1 (fr) 2010-01-20
IL188320A0 (en) 2008-04-13
KR101083631B1 (ko) 2011-11-16
AP2585A (en) 2013-02-04
NZ564540A (en) 2010-03-26
PE20070343A1 (es) 2007-05-12
CY1110008T1 (el) 2015-01-14
US20090118312A1 (en) 2009-05-07
HRP20100209T1 (hr) 2010-05-31
JP5230418B2 (ja) 2013-07-10
EA200800482A1 (ru) 2008-06-30
GT200600343A (es) 2007-08-06
ES2339702T3 (es) 2010-05-24
ME01454B (me) 2014-04-20
UY29704A1 (es) 2007-05-31
AU2006274866A1 (en) 2007-02-08
CA2617103C (fr) 2015-01-06
US7659245B2 (en) 2010-02-09
PT1912981E (pt) 2010-04-16

Similar Documents

Publication Publication Date Title
NO20081075L (no) Macrocykliske inhibitorer av hepatitt C virus
NO20080879L (no) HCV-NS3-proteaseinhibitorer
NO20090595L (no) Ny pyridazinforbindelse og anvendelse derav
TNSN07252A1 (en) Indole derivatives for treating viral infections
IN2012DN00999A (fr)
MX2012007420A (es) Analogos para el tratamiento o prevencion de infecciones de flavivirus.
MX2012008443A (es) Nucleosidos antiviricos.
PE20090478A1 (es) Compuestos de indol macrociclicos como inhibidores de la proteasa del virus de la hepatitis c
MY140729A (en) Amide derivatives
WO2007103550A3 (fr) Derives d'aminothiazole substitues presentant une activite anti-hcv
WO2010062821A8 (fr) Composés antiviraux, compositions, et procédés d’utilisation
WO2010063996A3 (fr) Composés antibactériens
TW200732336A (en) Alyphactic heterocyclic compounds
NO20063407L (no) Benzenforbindelser disubstituert med cykliske grupper i 1- og 2-posisjoner
DE60112933D1 (de) N-phenyl-4-(4-pyridyl)-2-pyrimidinamine-derivate
NO20076680L (no) Utvalgte CGRP-antagonister, metoder for fremstilling av disse og deres anvendelse som medikamenter
MY140868A (en) Amide derivatives
TW200640879A (en) Amide derivatives
NO20053570L (no) Termostabilt, vannopploselig polymer som er tverrbindbar ved hoye temperaturer
NO20084804L (no) Disazosyre-fargestoffer
TW200728291A (en) Amide derivatives
NO20076389L (no) Sammenstninger og metoder for behandling av HIV-infeksjon med cupredoxin og cytokrom C
CO5630031A2 (es) Derivados de benzotiazol como ligandos del receptor adenosina
TW200609228A (en) Substituted n-acyl-2-aminothiazoles
NO20081083L (no) Antitumorforbindelser

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application