NO20083462L - Nye tiofenderivater som S1P1/EDG1-reseptoragonister - Google Patents

Nye tiofenderivater som S1P1/EDG1-reseptoragonister

Info

Publication number
NO20083462L
NO20083462L NO20083462A NO20083462A NO20083462L NO 20083462 L NO20083462 L NO 20083462L NO 20083462 A NO20083462 A NO 20083462A NO 20083462 A NO20083462 A NO 20083462A NO 20083462 L NO20083462 L NO 20083462L
Authority
NO
Norway
Prior art keywords
thiophene derivatives
receptor agonists
edg1 receptor
new thiophene
new
Prior art date
Application number
NO20083462A
Other languages
English (en)
Inventor
Martin Bolli
Oliver Nayler
Claus Mueller
David Lehmann
Jorg Velker
Boris Mathys
Beat Steiner
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37908151&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20083462(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of NO20083462L publication Critical patent/NO20083462L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Diabetes (AREA)
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  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
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Abstract

Oppfinnelsen vedrører nye tiofenderivater, deres fremstilling og deres anvendelse som farmasøytisk active forbindelser. Forbindelsene virker spesielt som immunsuppressive midler.
NO20083462A 2006-01-11 2008-08-08 Nye tiofenderivater som S1P1/EDG1-reseptoragonister NO20083462L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IB2006050103 2006-01-11
PCT/IB2007/050070 WO2007080542A1 (en) 2006-01-11 2007-01-10 Novel thiophene derivatives as s1p1/edg1 receptor agonists

Publications (1)

Publication Number Publication Date
NO20083462L true NO20083462L (no) 2008-10-09

Family

ID=37908151

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20083462A NO20083462L (no) 2006-01-11 2008-08-08 Nye tiofenderivater som S1P1/EDG1-reseptoragonister

Country Status (17)

Country Link
US (1) US8003800B2 (no)
EP (1) EP1976512B1 (no)
JP (1) JP5114430B2 (no)
KR (1) KR101382710B1 (no)
CN (1) CN101370496B (no)
AR (1) AR058956A1 (no)
AU (1) AU2007204121B2 (no)
BR (1) BRPI0706476A2 (no)
CA (1) CA2635047C (no)
ES (1) ES2553345T3 (no)
IL (1) IL192657A (no)
MY (1) MY154909A (no)
NO (1) NO20083462L (no)
NZ (1) NZ570258A (no)
RU (1) RU2437877C2 (no)
TW (1) TWI404706B (no)
WO (1) WO2007080542A1 (no)

Families Citing this family (40)

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