NO20083480L - Piperidinoylpyrrolidiner som melanokortin type 4 reseptor agonister - Google Patents

Piperidinoylpyrrolidiner som melanokortin type 4 reseptor agonister

Info

Publication number
NO20083480L
NO20083480L NO20083480A NO20083480A NO20083480L NO 20083480 L NO20083480 L NO 20083480L NO 20083480 A NO20083480 A NO 20083480A NO 20083480 A NO20083480 A NO 20083480A NO 20083480 L NO20083480 L NO 20083480L
Authority
NO
Norway
Prior art keywords
piperidinoylpyrrolidines
receptor agonists
melanocortin
melanocortin type
type
Prior art date
Application number
NO20083480A
Other languages
English (en)
Norwegian (no)
Inventor
Mark David Andrews
Alan Daniel Brown
Mark Ian Landsdell
Nicholas William Summerhill
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of NO20083480L publication Critical patent/NO20083480L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO20083480A 2006-02-23 2008-08-11 Piperidinoylpyrrolidiner som melanokortin type 4 reseptor agonister NO20083480L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US77629506P 2006-02-23 2006-02-23
US88784007P 2007-02-02 2007-02-02
PCT/IB2007/000456 WO2007096763A2 (fr) 2006-02-23 2007-02-19 Pipéridinoylpyrrolidines en tant qu'agonistes du récepteur de la mélanocortine de type 4

Publications (1)

Publication Number Publication Date
NO20083480L true NO20083480L (no) 2008-09-10

Family

ID=38169450

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20083480A NO20083480L (no) 2006-02-23 2008-08-11 Piperidinoylpyrrolidiner som melanokortin type 4 reseptor agonister

Country Status (21)

Country Link
US (1) US8138188B2 (fr)
EP (1) EP1989196B1 (fr)
KR (1) KR101036981B1 (fr)
AP (1) AP2008004602A0 (fr)
AU (1) AU2007219236B2 (fr)
BR (1) BRPI0708264A2 (fr)
CA (1) CA2642922C (fr)
CR (1) CR10219A (fr)
DK (1) DK1989196T3 (fr)
EA (1) EA200801738A1 (fr)
EC (1) ECSP088688A (fr)
ES (1) ES2402581T3 (fr)
IL (1) IL193279A (fr)
MA (1) MA30228B1 (fr)
ME (1) MEP6808A (fr)
MX (1) MX2008010899A (fr)
NO (1) NO20083480L (fr)
RS (1) RS20080371A (fr)
SG (1) SG185849A1 (fr)
TN (1) TNSN08337A1 (fr)
WO (1) WO2007096763A2 (fr)

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US8848656B2 (en) 2007-11-16 2014-09-30 Qualcomm Incorporated Utilizing broadcast signals to convey restricted association information
EP2103614A1 (fr) * 2008-03-18 2009-09-23 Santhera Pharmaceuticals (Schweiz) AG Dérivés d'imidazopyrimidine, d'imidazopyrazine et d' imidazopyridazine substitués en tant que modulateur de récepteur de la mélanocortine-4
US8588773B2 (en) 2008-08-04 2013-11-19 Qualcomm Incorporated System and method for cell search and selection in a wireless communication system
UA99555C2 (en) 2008-11-12 2012-08-27 Элджи Лайф Саенсез Лтд. Melanocortin receptor agonists
EP2722045B1 (fr) 2009-11-18 2016-07-06 Helsinn Healthcare SA Compositions pour traiter les nausées et vomissements à médiation centrale
HRP20140759T1 (hr) * 2009-11-18 2014-10-24 Helsinn Healthcare S.A. Kompozicije za lijeäśenje središnje posredovane muäśnine i povraä†anja
US8828994B2 (en) 2011-03-08 2014-09-09 Sanofi Di- and tri-substituted oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
US8710050B2 (en) 2011-03-08 2014-04-29 Sanofi Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
EP2683704B1 (fr) 2011-03-08 2014-12-17 Sanofi Dérivés oxathiazine ramifiés, procédé pour leur préparation, utilisation en tant que médicament, agents pharmaceutiques contenant ces dérivés et leur utilisation
EP2766349B1 (fr) 2011-03-08 2016-06-01 Sanofi Dérivés d'oxathiazine substitués par des carbocycles ou des hétérocycles, leur procédé de préparation, médicaments contenant ces composés et leur utilisation
US8871758B2 (en) 2011-03-08 2014-10-28 Sanofi Tetrasubstituted oxathiazine derivatives, method for producing them, their use as medicine and drug containing said derivatives and the use thereof
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EP3870292A4 (fr) 2018-10-26 2022-11-09 The Research Foundation for The State University of New York Combinaison d'un inhibiteur de réabsorption spécifique de la sérotonine et d'un agoniste partiel du récepteur de la sérotonine 1a pour réduire la dyskinésie induite par l-dopa
PT4161927T (pt) 2020-06-09 2024-10-08 Pfizer Compostos de espiro como antagonistas do recetor de melanocortina 4 e utilizações dos mesmos
CA3241470A1 (fr) 2021-12-06 2023-06-15 Pfizer Inc. Antagonistes du recepteur 4 de la melanocortine et leurs utilisations
WO2025228895A1 (fr) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Indazoles et benzimidazoles à substitution hétaryle utilisés en tant qu'antagonistes de sting et leur utilisation en tant que médicament
WO2025228889A1 (fr) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Composés hétérocycliques monoaryliques utilisés en tant qu'antagonistes de sting et leur utilisation en tant que médicament
WO2025228900A1 (fr) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Indazoles substitués par arylamide et leur utilisation en tant que médicament
WO2025228902A1 (fr) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Acides hétérocycliques en tant qu'antagonistes de sting et leur utilisation en tant que médicament
US20250333398A1 (en) 2024-04-30 2025-10-30 Boehringer Ingelheim International Gmbh Monoaryl and hetaryl substituted indazoles and benzimidazoles as sting antagonists and the use thereof as medicament
WO2025228899A1 (fr) 2024-04-30 2025-11-06 Boehringer Ingelheim International Gmbh Autres composés hétérocycliques utilisés en tant qu'antagonistes de sting et leur utilisation en tant que médicament

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Also Published As

Publication number Publication date
ES2402581T3 (es) 2013-05-06
KR20080095918A (ko) 2008-10-29
KR101036981B1 (ko) 2011-05-25
DK1989196T3 (da) 2013-04-15
ECSP088688A (es) 2008-10-31
EP1989196A2 (fr) 2008-11-12
IL193279A0 (en) 2009-02-11
CA2642922C (fr) 2011-08-02
IL193279A (en) 2012-12-31
RS20080371A (sr) 2009-07-15
MX2008010899A (es) 2008-11-27
WO2007096763A2 (fr) 2007-08-30
WO2007096763A3 (fr) 2007-10-18
HK1126489A1 (en) 2009-09-04
EP1989196B1 (fr) 2013-02-13
EA200801738A1 (ru) 2008-12-30
US8138188B2 (en) 2012-03-20
MA30228B1 (fr) 2009-02-02
CR10219A (es) 2008-09-23
AU2007219236A1 (en) 2007-08-30
AP2008004602A0 (en) 2008-10-31
TNSN08337A1 (fr) 2009-12-29
AU2007219236B2 (en) 2012-06-21
BRPI0708264A2 (pt) 2011-05-24
SG185849A1 (en) 2012-12-28
MEP6808A (xx) 2010-02-10
CA2642922A1 (fr) 2007-08-30
US20090036459A1 (en) 2009-02-05

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