NO323751B1 - 13-substituerte milbemycinderivater, preparater omfattende disse og anvendelse av dem mot insekter og andre skadedyr - Google Patents

13-substituerte milbemycinderivater, preparater omfattende disse og anvendelse av dem mot insekter og andre skadedyr Download PDF

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Publication number
NO323751B1
NO323751B1 NO20025141A NO20025141A NO323751B1 NO 323751 B1 NO323751 B1 NO 323751B1 NO 20025141 A NO20025141 A NO 20025141A NO 20025141 A NO20025141 A NO 20025141A NO 323751 B1 NO323751 B1 NO 323751B1
Authority
NO
Norway
Prior art keywords
group
groups
carbon atoms
atoms
optionally
Prior art date
Application number
NO20025141A
Other languages
English (en)
Norwegian (no)
Other versions
NO20025141D0 (no
NO20025141L (no
Inventor
Toshimitsu Toyama
Akio Saito
Yoko Sugiyama
Toshihiko Nanba
Original Assignee
Sankyo Lifetech Company Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Lifetech Company Ltd filed Critical Sankyo Lifetech Company Ltd
Publication of NO20025141D0 publication Critical patent/NO20025141D0/no
Publication of NO20025141L publication Critical patent/NO20025141L/no
Publication of NO323751B1 publication Critical patent/NO323751B1/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

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  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Wood Science & Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20025141A 2000-04-27 2002-10-25 13-substituerte milbemycinderivater, preparater omfattende disse og anvendelse av dem mot insekter og andre skadedyr NO323751B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000127209 2000-04-27
PCT/JP2001/003656 WO2001083500A1 (en) 2000-04-27 2001-04-26 13-substituted milbemycin derivatives, their preparation and their use against insects and other pests

Publications (3)

Publication Number Publication Date
NO20025141D0 NO20025141D0 (no) 2002-10-25
NO20025141L NO20025141L (no) 2002-12-16
NO323751B1 true NO323751B1 (no) 2007-07-02

Family

ID=18636847

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20025141A NO323751B1 (no) 2000-04-27 2002-10-25 13-substituerte milbemycinderivater, preparater omfattende disse og anvendelse av dem mot insekter og andre skadedyr

Country Status (23)

Country Link
US (1) US6653342B2 (de)
EP (1) EP1276748B1 (de)
KR (1) KR100711931B1 (de)
CN (1) CN1247607C (de)
AR (1) AR029250A1 (de)
AT (1) ATE315573T1 (de)
AU (2) AU5261301A (de)
BR (1) BR0110385A (de)
CA (1) CA2407611A1 (de)
CZ (1) CZ20023565A3 (de)
DE (1) DE60116615T2 (de)
DK (1) DK1276748T3 (de)
ES (1) ES2254400T3 (de)
HU (1) HUP0301040A3 (de)
IL (1) IL152449A0 (de)
MX (1) MXPA02010587A (de)
NO (1) NO323751B1 (de)
NZ (1) NZ522247A (de)
PL (1) PL357598A1 (de)
RU (1) RU2226531C1 (de)
TW (1) TWI285206B (de)
WO (1) WO2001083500A1 (de)
ZA (1) ZA200208630B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20040047962A (ko) * 2001-10-25 2004-06-05 상꾜 라이프테크 가부시키가이샤 기생충 구제 조성물
AR045142A1 (es) 2003-07-30 2005-10-19 Novartis Ag Composicion veterinaria masticable ductil de buen sabor
US20090281175A1 (en) * 2006-09-28 2009-11-12 Galderma S.A. Avermectin compounds and treatment of dermatological disorders in humans therewith
TWI457347B (zh) 2008-12-04 2014-10-21 Merial Ltd 二聚合的阿佛菌素（ａｖｅｒｍｅｃｔｉｎ）及密倍脈心（ｍｉｌｂｅｍｙｃｉｎ）衍生物
RU2413513C2 (ru) * 2009-04-06 2011-03-10 Государственное образовательное учреждение высшего профессионального образования "Казанский государственный университет им. В.И. Ульянова-Ленина" Антигельминтная композиция на основе соли четвертичного фосфония и замещенного динитробензофуроксана
US8980896B2 (en) 2009-12-17 2015-03-17 Merial, Inc. Compositions comprising macrocyclic lactone compounds and spirodioxepinoindoles
MX379693B (es) 2011-12-02 2025-03-11 Merial Ltd Formulaciones de moxidectina inyectables de larga acción y formas de cristal de moxidectina novedosas.
PL2983712T3 (pl) 2013-04-12 2021-05-31 Zoetis Services Llc Kompozycja makrocyklicznych laktonów, lewamizolu, aminocukru i dodatkowego środka przeciwpasożytniczego
CA3123852A1 (en) * 2018-12-21 2020-06-25 Bayer Healthcare Llc Parasiticidal formulations and use thereof

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4201861A (en) 1977-10-03 1980-05-06 Merck & Co., Inc. Acyl derivatives of C-076 compounds
US4206205A (en) 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
NZ188459A (en) 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
US4171314A (en) 1977-12-19 1979-10-16 Merck & Co., Inc. 13-Halo and 13-deoxy C-076 compounds
US4173571A (en) 1977-12-19 1979-11-06 Merck & Co., Inc. 13-Halo and 13-deoxy derivatives of C-076 compounds
US4203976A (en) 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4200581A (en) 1978-08-04 1980-04-29 Merck & Co., Inc. Alkyl derivatives of C-076 compounds
US4289760A (en) 1980-05-02 1981-09-15 Merck & Co., Inc. 23-Keto derivatives of C-076 compounds
JPS57120589A (en) 1981-01-20 1982-07-27 Sankyo Co Ltd 5-methoxy and 5-lower alkanoyloxy derivative, its preparation and acaricide and parasiticide
IT1144368B (it) 1981-05-20 1986-10-29 Gaudino Di P Gaudino & C Sas O Perfezionamenti nei laminatoi con almeno un campo di stiro per la filatura diretta di pettinato e semipettinato
US4457920A (en) 1981-09-03 1984-07-03 Merck & Co., Inc. 4a-Substituted avermectin compounds
US4423209A (en) 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
JPS5916894A (ja) 1982-07-21 1984-01-28 Sankyo Co Ltd ミルベマイシンｄの５−アシルオキシ誘導体
JPS5920285A (ja) 1982-07-23 1984-02-01 Sankyo Co Ltd ミルベマイシンｄの５−二塩基酸エステル誘導体及びその塩
JPS59108785A (ja) 1982-11-25 1984-06-23 Sankyo Co Ltd ミルベマイシン類の５−オキシム誘導体
US4469682A (en) 1983-01-28 1984-09-04 Merck & Co., Inc. Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
US4579864A (en) 1984-06-11 1986-04-01 Merck & Co., Inc. Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives
US4547491A (en) 1984-07-18 1985-10-15 Merck & Co., Inc. C-8A-Oxo-avermectin and milbemycin derivatives, pharmaceutical compositions and method of use
EP0180539A1 (de) 1984-09-18 1986-05-07 Ciba-Geigy Ag 13-Halo- und 13-Hydroximilbemycine
US4696922A (en) 1984-11-26 1987-09-29 Ciba-Geigy Corporation 5-azolylacetoxymilbemycins as ecto- and endoparasites
JPS6289685A (ja) 1985-05-31 1987-04-24 Sankyo Co Ltd １３−ハロゲンミルベマイシン誘導体
RU2024527C1 (ru) 1986-03-25 1994-12-15 Санкио Компани Лимитед Способ получения макролидных соединений
US5614470A (en) * 1994-04-01 1997-03-25 Sankyo Company, Limited 13-substituted milbemycin derivatives, their preparation and their use
PT765879E (pt) 1995-09-29 2001-05-31 Sankyo Co Derivados 13-substituidos de milbemicina-5-oxima sua preparacao e utilizacao contra insectos e outras pragas

Also Published As

Publication number Publication date
DE60116615D1 (de) 2006-04-06
ATE315573T1 (de) 2006-02-15
US6653342B2 (en) 2003-11-25
RU2226531C1 (ru) 2004-04-10
PL357598A1 (en) 2004-07-26
NZ522247A (en) 2004-07-30
DE60116615T2 (de) 2006-09-07
ES2254400T3 (es) 2006-06-16
CA2407611A1 (en) 2001-11-08
KR20020087987A (ko) 2002-11-23
MXPA02010587A (es) 2003-03-10
IL152449A0 (en) 2003-05-29
CN1439016A (zh) 2003-08-27
EP1276748A1 (de) 2003-01-22
US20030139601A1 (en) 2003-07-24
RU2002131794A (ru) 2004-02-27
KR100711931B1 (ko) 2007-05-02
CN1247607C (zh) 2006-03-29
NO20025141D0 (no) 2002-10-25
TWI285206B (en) 2007-08-11
WO2001083500A1 (en) 2001-11-08
BR0110385A (pt) 2003-02-04
EP1276748B1 (de) 2006-01-11
HUP0301040A2 (hu) 2003-08-28
ZA200208630B (en) 2004-02-12
HUP0301040A3 (en) 2005-11-28
NO20025141L (no) 2002-12-16
HK1057757A1 (en) 2004-04-16
DK1276748T3 (da) 2006-03-20
CZ20023565A3 (cs) 2003-04-16
WO2001083500A8 (en) 2003-05-08
AR029250A1 (es) 2003-06-18
AU5261301A (en) 2001-11-12
AU2001252613B2 (en) 2004-05-13

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