NO832107L - Fremgangsmaate ved fremstilling av dynorfinderivater - Google Patents

Fremgangsmaate ved fremstilling av dynorfinderivater

Info

Publication number
NO832107L
NO832107L NO832107A NO832107A NO832107L NO 832107 L NO832107 L NO 832107L NO 832107 A NO832107 A NO 832107A NO 832107 A NO832107 A NO 832107A NO 832107 L NO832107 L NO 832107L
Authority
NO
Norway
Prior art keywords
dynorphin
morphine
arg
animals
analgesia
Prior art date
Application number
NO832107A
Other languages
English (en)
Norwegian (no)
Inventor
Nancy M Lee
Jaw-Kang Chang
Horace H Loh
Original Assignee
Univ California
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ California filed Critical Univ California
Publication of NO832107L publication Critical patent/NO832107L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Zoology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Toxicology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Polyamides (AREA)
NO832107A 1982-06-10 1983-06-09 Fremgangsmaate ved fremstilling av dynorfinderivater NO832107L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/387,005 US4462941A (en) 1982-06-10 1982-06-10 Dynorphin amide analogs

Publications (1)

Publication Number Publication Date
NO832107L true NO832107L (no) 1983-12-12

Family

ID=23528034

Family Applications (1)

Application Number Title Priority Date Filing Date
NO832107A NO832107L (no) 1982-06-10 1983-06-09 Fremgangsmaate ved fremstilling av dynorfinderivater

Country Status (15)

Country Link
US (1) US4462941A (cs)
EP (1) EP0096592B1 (cs)
JP (1) JPS5925365A (cs)
KR (1) KR840005080A (cs)
AT (1) ATE22449T1 (cs)
AU (1) AU1448983A (cs)
CA (1) CA1241645A (cs)
DE (1) DE3366428D1 (cs)
DK (1) DK262683A (cs)
FI (1) FI832095A7 (cs)
IL (1) IL68825A0 (cs)
IS (1) IS2812A7 (cs)
NO (1) NO832107L (cs)
PT (1) PT76860B (cs)
ZA (1) ZA834189B (cs)

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US4481191A (en) * 1983-03-30 1984-11-06 The Regents Of The University Of California Method for controlling blood pressure
US4900811A (en) * 1983-07-21 1990-02-13 Scripps Clinic And Research Foundation Synthetic polypeptides corresponding to portions of proteinoids translated from brain-specific mRNAs, receptors, methods and diagnostics using the same
US5242798A (en) * 1983-07-21 1993-09-07 Scripps Clinic And Research Foundation Synthetic polypeptides corresponding to portions of proteinoids translated from brain-specific mRNAs, receptors, methods and diagnostics using the same
EP0147194B1 (en) * 1983-12-22 1989-07-19 Yoshio Hosobuchi Compositions for treating cerebral ischemia
JPH0680079B2 (ja) * 1984-11-09 1994-10-12 エーザイ株式会社 ポリペプチド
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US5482930A (en) * 1993-06-09 1996-01-09 The Regents Of The University Of California Anti-inflammatory composition and method with des-Tyr dynorphin and analogues
US6184208B1 (en) 1994-06-29 2001-02-06 Immunotech Developments Inc. Peptide, a method for its preparation and a pharmaceutical composition containing the peptide
AU7637394A (en) * 1994-08-26 1996-03-22 Avram Goldstein Analgesic method with dynorphin analogues truncated at the n-terminus
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US20070048228A1 (en) 2003-08-06 2007-03-01 Elisabeth Arkenau-Maric Abuse-proofed dosage form
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US20090099074A1 (en) * 2007-01-10 2009-04-16 Conjuchem Biotechnologies Inc. Modulating food intake
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US9617274B1 (en) 2011-08-26 2017-04-11 Demerx, Inc. Synthetic noribogaine
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US9150584B2 (en) 2012-01-25 2015-10-06 Demerx, Inc. Indole and benzofuran fused isoquinuclidene derivatives and processes for preparing them
BR112014019988A8 (pt) 2012-02-28 2017-07-11 Gruenenthal Gmbh Forma de dosagem resistente a socamento compreendendo um composto farmacologicamente ativo e um polímero aniônico
LT2838512T (lt) 2012-04-18 2018-11-12 GrĆ¼nenthal GmbH Pažeidimui atspari ir dozės atpalaidavimo nuokrypiui atspari farmacinė vaisto forma
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US10428115B2 (en) 2013-05-24 2019-10-01 Arizona Board Of Regents On Behalf Of The University Of Arizona Dynorphin A analogs with bradykinin receptors specificity for modulation of neuropathic pain
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Family Cites Families (4)

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Publication number Priority date Publication date Assignee Title
JPS5572153A (en) * 1978-11-26 1980-05-30 Shionogi & Co Ltd Undecapeptide
US4396606A (en) * 1979-11-05 1983-08-02 Addiction Research Foundation Novel polypeptide analgesics
US4361553A (en) * 1981-05-18 1982-11-30 Regents Of The University Of California Therapeutic uses of dynorphin
JPS5815946A (ja) 1981-07-21 1983-01-29 Eisai Co Ltd 新規ヘプタデカペプタイド

Also Published As

Publication number Publication date
JPS5925365A (ja) 1984-02-09
IS2812A7 (is) 1983-10-07
KR840005080A (ko) 1984-11-03
EP0096592A1 (en) 1983-12-21
FI832095A0 (fi) 1983-06-10
DE3366428D1 (en) 1986-10-30
DK262683A (da) 1983-12-11
ZA834189B (en) 1984-02-29
FI832095L (fi) 1983-12-11
ATE22449T1 (de) 1986-10-15
JPH0427995B2 (cs) 1992-05-13
FI832095A7 (fi) 1983-12-11
US4462941A (en) 1984-07-31
PT76860A (en) 1983-07-01
EP0096592B1 (en) 1986-09-24
AU1448983A (en) 1983-12-15
IL68825A0 (en) 1983-09-30
PT76860B (en) 1986-01-27
DK262683D0 (da) 1983-06-09
CA1241645A (en) 1988-09-06

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