NO985253L - Ny isomeriseringsfremgangsmÕte for metylradikalet i 10-stilling pÕ erytromycinderivater - Google Patents

Ny isomeriseringsfremgangsmÕte for metylradikalet i 10-stilling pÕ erytromycinderivater

Info

Publication number: NO985253L
Authority: NO; Norway
Prior art keywords: radical; pct; methyl radical; nar; hydrogen atom
Prior art date: 1996-05-14

Application number

NO985253A

Other languages

English (en)

Other versions

NO310823B1 (no

NO985253D0 (no

Inventor

Yannick Benedetti

Jacques Lagouardat

Jacques Scholl

Original Assignee

Hoechst Marion Roussel Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-05-14

Filing date

1998-11-10

Publication date

1998-11-10

1998-11-10 Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc

1998-11-10 Publication of NO985253D0 publication Critical patent/NO985253D0/no

1998-11-10 Publication of NO985253L publication Critical patent/NO985253L/no

2001-09-03 Publication of NO310823B1 publication Critical patent/NO310823B1/no

Links

238000006317 isomerization reaction Methods 0.000 title abstract 2
238000000034 method Methods 0.000 title abstract 2
WCYWZMWISLQXQU-UHFFFAOYSA-N methyl Chemical compound [CH3] WCYWZMWISLQXQU-UHFFFAOYSA-N 0.000 title abstract 2
ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 title 1
-1 NH2 radical Chemical class 0.000 abstract 3
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
150000001875 compounds Chemical class 0.000 abstract 2
150000003254 radicals Chemical class 0.000 abstract 2
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
239000003795 chemical substances by application Substances 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Engineering & Computer Science (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

NO19985253A 1996-05-14 1998-11-10 Ny isomeriseringsfremgangsmåte for metylradikalet i 10- stilling på erytromycinderivater NO310823B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9605966A FR2748746B1 (fr)	1996-05-14	1996-05-14	Nouveau procede d'isomerisation du radical methyle en 10 de derives de l'erythromycine
PCT/FR1997/000840 WO1997043297A1 (fr)	1996-05-14	1997-05-13	Nouveau procede d'isomerisation du radical methyle en 10 de derives de l'erythromycine

Publications (3)

Publication Number	Publication Date
NO985253D0 NO985253D0 (no)	1998-11-10
NO985253L true NO985253L (no)	1998-11-10
NO310823B1 NO310823B1 (no)	2001-09-03

Family

ID=9492104

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO19985253A NO310823B1 (no)	1996-05-14	1998-11-10	Ny isomeriseringsfremgangsmåte for metylradikalet i 10- stilling på erytromycinderivater

Country Status (28)

Country	Link
US (1)	US6022965A (no)
EP (1)	EP0912591B1 (no)
JP (1)	JP3304098B2 (no)
KR (1)	KR100457757B1 (no)
CN (1)	CN1160366C (no)
AT (1)	ATE213251T1 (no)
AU (1)	AU720721B2 (no)
BG (1)	BG62699B1 (no)
BR (1)	BR9709243A (no)
CA (1)	CA2254795C (no)
CZ (1)	CZ289644B6 (no)
DE (1)	DE69710468T2 (no)
DK (1)	DK0912591T3 (no)
EA (1)	EA000939B1 (no)
ES (1)	ES2171943T3 (no)
FR (1)	FR2748746B1 (no)
GE (1)	GEP20012418B (no)
HU (1)	HU226676B1 (no)
IL (1)	IL126796A0 (no)
NO (1)	NO310823B1 (no)
NZ (1)	NZ332411A (no)
PL (1)	PL183467B1 (no)
PT (1)	PT912591E (no)
SK (1)	SK283649B6 (no)
TR (1)	TR199802297T2 (no)
UA (1)	UA55412C2 (no)
WO (1)	WO1997043297A1 (no)
YU (1)	YU49500B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2243066T3 (es)	1998-09-22	2005-11-16	Pfizer Products Inc.	Antibioticos de carbamato y carbazato cetolida.
CA2359708C (en)	1999-01-27	2005-10-25	Pfizer Products Inc.	Ketolide antibiotics
ATE340183T1 (de)	1999-04-16	2006-10-15	Kosan Biosciences Inc	Antiinfektiöse makrolidderivate
US6939861B2 (en)	1999-04-16	2005-09-06	Kosan Biosciences, Inc.	Amido macrolides
US6590083B1 (en)	1999-04-16	2003-07-08	Ortho-Mcneil Pharmaceutical, Inc.	Ketolide antibacterials
US6451768B1 (en)	1999-04-16	2002-09-17	Kosan Biosciences, Inc.	Macrolide antiinfective agents
US6514944B2 (en)	1999-04-16	2003-02-04	Kosan Biosciences, Inc.	Macrolide antiinfective agents
HUP0201516A3 (en) *	1999-05-24	2003-03-28	Pfizer Prod Inc	13-methyl-erythromycin derivatives, process for their preparation and pharmaceutical compositions containing them
EP1146051A3 (en) *	2000-04-10	2001-10-31	Pfizer Products Inc.	Erythromycin A derivatives
US20020115621A1 (en) *	2000-08-07	2002-08-22	Wei-Gu Su	Macrolide antibiotics
EP1723159B1 (en) *	2004-02-27	2019-06-12	Melinta Therapeutics, Inc.	Macrocyclic compounds and methods of making and using the same
UA85937C2 (uk) *	2004-12-21	2009-03-10	Пфайзер Продактс Інк.	Макроліди
EP1934237A2 (en)	2005-08-24	2008-06-25	Rib-X Pharmaceuticals, Inc.	Triazole compounds and methods of making and using the same

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2718450B1 (fr) *	1994-04-08	1997-01-10	Roussel Uclaf	Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

1996
- 1996-05-14 FR FR9605966A patent/FR2748746B1/fr not_active Expired - Lifetime
1997
- 1997-05-13 CZ CZ19983557A patent/CZ289644B6/cs not_active IP Right Cessation
- 1997-05-13 HU HU9901158A patent/HU226676B1/hu unknown
- 1997-05-13 SK SK1530-98A patent/SK283649B6/sk not_active IP Right Cessation
- 1997-05-13 KR KR10-1998-0709175A patent/KR100457757B1/ko not_active Expired - Lifetime
- 1997-05-13 EA EA199801008A patent/EA000939B1/ru not_active IP Right Cessation
- 1997-05-13 NZ NZ332411A patent/NZ332411A/xx not_active IP Right Cessation
- 1997-05-13 UA UA98126445A patent/UA55412C2/uk unknown
- 1997-05-13 GE GEAP19974602A patent/GEP20012418B/en unknown
- 1997-05-13 US US09/180,641 patent/US6022965A/en not_active Expired - Lifetime
- 1997-05-13 PT PT97924078T patent/PT912591E/pt unknown
- 1997-05-13 AU AU29663/97A patent/AU720721B2/en not_active Expired
- 1997-05-13 DE DE69710468T patent/DE69710468T2/de not_active Expired - Lifetime
- 1997-05-13 DK DK97924078T patent/DK0912591T3/da active
- 1997-05-13 IL IL12679697A patent/IL126796A0/xx not_active IP Right Cessation
- 1997-05-13 JP JP54059497A patent/JP3304098B2/ja not_active Expired - Lifetime
- 1997-05-13 AT AT97924078T patent/ATE213251T1/de active
- 1997-05-13 EP EP97924078A patent/EP0912591B1/fr not_active Expired - Lifetime
- 1997-05-13 PL PL97329809A patent/PL183467B1/pl unknown
- 1997-05-13 CN CNB971963835A patent/CN1160366C/zh not_active Expired - Lifetime
- 1997-05-13 ES ES97924078T patent/ES2171943T3/es not_active Expired - Lifetime
- 1997-05-13 BR BR9709243A patent/BR9709243A/pt not_active Application Discontinuation
- 1997-05-13 TR TR1998/02297T patent/TR199802297T2/xx unknown
- 1997-05-13 YU YU50398A patent/YU49500B/sh unknown
- 1997-05-13 CA CA002254795A patent/CA2254795C/fr not_active Expired - Lifetime
- 1997-05-13 WO PCT/FR1997/000840 patent/WO1997043297A1/fr not_active Ceased
1998
- 1998-11-10 NO NO19985253A patent/NO310823B1/no not_active IP Right Cessation
- 1998-11-13 BG BG102925A patent/BG62699B1/bg unknown

Also Published As

Publication number	Publication date
JP3304098B2 (ja)	2002-07-22
KR100457757B1 (ko)	2004-12-16
NO310823B1 (no)	2001-09-03
GEP20012418B (en)	2001-04-25
CZ289644B6 (cs)	2002-03-13
KR20000011025A (ko)	2000-02-25
SK283649B6 (sk)	2003-11-04
FR2748746B1 (fr)	1998-08-14
EA000939B1 (ru)	2000-06-26
AU720721B2 (en)	2000-06-08
ATE213251T1 (de)	2002-02-15
PL329809A1 (en)	1999-04-12
YU49500B (sh)	2006-08-17
PL183467B1 (pl)	2002-06-28
TR199802297T2 (xx)	1999-02-22
NO985253D0 (no)	1998-11-10
HU226676B1 (en)	2009-06-29
ES2171943T3 (es)	2002-09-16
BR9709243A (pt)	1999-08-10
CA2254795A1 (fr)	1997-11-20
FR2748746A1 (fr)	1997-11-21
BG62699B1 (bg)	2000-05-31
PT912591E (pt)	2002-07-31
CN1225097A (zh)	1999-08-04
DK0912591T3 (da)	2002-07-08
DE69710468D1 (de)	2002-03-21
CZ355798A3 (cs)	1999-02-17
CA2254795C (fr)	2004-07-20
CN1160366C (zh)	2004-08-04
BG102925A (en)	1999-08-31
EP0912591A1 (fr)	1999-05-06
HUP9901158A1 (hu)	1999-08-30
JP2000510142A (ja)	2000-08-08
YU50398A (en)	1999-11-22
SK153098A3 (en)	1999-05-07
HUP9901158A3 (en)	1999-11-29
DE69710468T2 (de)	2002-08-22
UA55412C2 (uk)	2003-04-15
EP0912591B1 (fr)	2002-02-13
WO1997043297A1 (fr)	1997-11-20
US6022965A (en)	2000-02-08
EA199801008A1 (ru)	1999-04-29
IL126796A0 (en)	1999-08-17
AU2966397A (en)	1997-12-05
NZ332411A (en)	1999-07-29

Legal Events

Date	Code	Title	Description
2017-05-22	MK1K	Patent expired

Publication	Publication Date	Title
NO985253L (no)	1998-11-10	Ny isomeriseringsfremgangsmÕte for metylradikalet i 10-stilling pÕ erytromycinderivater
IE860083L (en)	1986-07-14	New steroids substituted at position 10
DK0595851T3 (da)	1996-02-12	Fremgangsmåde til fremstilling af sertralin-mellemprodukter
HUP0001192A2 (hu)	2000-11-28	Topiramát és származékainak alkalmazása elhízás kezelésére használható gyógyszerkészítmények előállítására
SE9100342D0 (sv)	1991-02-04	Novel steroid esters
ES2134801T3 (es)	1999-10-16	Monohidrato de hidrocloruro de tiagabina cristalina, su preparacion y su uso.
ATE323495T1 (de)	2006-05-15	Steroid-3-o-sulfamat-derivate als estronsulfatase-hemmer
GB2331987B (en)	2002-11-27	Polycyclic sulphamate inhibitors of oestrone sulphatase
ES2028871T3 (es)	1992-07-16	Un procedimiento para la preparacion de un glicosido de antraciclina. .
PT93071A (pt)	1990-08-31	Processo para a preparacao de novas 4`-epi-4`-amino-antraciclinas e de composicoes farmaceuticas que as contem
DE3885145D1 (de)	1993-12-02	3-Methylen-4-androsten-17-one, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Präparate.
ES2129661T3 (es)	1999-06-16	Agente de aclarado para la limpieza a maquina de superficies duras.
FI932446A0 (fi)	1993-05-28	2b,19-metylaminobrosteroider som aromatasinhibitorer
IT1262974B (it)	1996-07-23	Composti azoici, loro preparazione e loro impiego come coloranti dispersi.
ATE42957T1 (de)	1989-05-15	Waessrige kristallsuspension von steroidglykoestern.
ES2186127T3 (es)	2003-05-01	Sintesis de derivados de nucleosidos aciclicos.
ES2135716T3 (es)	1999-11-01	Nuevos derivados de glicina, sus compuestos intermedios y composiciones limpiadoras que los comprenden.
ES2071832T3 (es)	1995-07-01	Procedimiento para la preparacion de derivados de 21-bromo-4-pregneno-3,20-diona.
AR004776A1 (es)	1999-03-10	Derivados de 2-tioxo-imidazolidin-4-ona
IT8434937U1 (it)	1986-05-23	Bide' ad elevata versatilità di applicazione per i rispettivi accessori
MX9605046A (es)	1998-02-28	Derivados de adenosina.