OA12916A - Novel benzoimidazole derivatives useful as antiproliferative agents. - Google Patents

Novel benzoimidazole derivatives useful as antiproliferative agents. Download PDF

Info

Publication number: OA12916A
Authority: OA; OAPI
Prior art keywords: compound; group; formula; benzoimidazol; optionally substituted
Prior art date: 2002-08-28

Application number

OA1200500059A

Other languages

English (en)

Inventor

John Charles Kath

Huifen Faye Wang

Joseph Peter Lyssikatos

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-08-28

Filing date

2003-08-14

Publication date

2006-10-13

2003-08-14 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2006-10-13 Publication of OA12916A publication Critical patent/OA12916A/en

Links

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- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
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Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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Communicable Diseases (AREA)
Oncology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

OA1200500059A 2002-08-28 2003-08-14 Novel benzoimidazole derivatives useful as antiproliferative agents. OA12916A (en)

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US40652402P	2002-08-28	2002-08-28
US41704702P	2002-10-08	2002-10-08

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CN (1)	CN1319966C (is)
AP (1)	AP2005003237A0 (is)
AR (1)	AR041055A1 (is)
AT (1)	ATE445610T1 (is)
AU (1)	AU2003250499B2 (is)
BR (1)	BRPI0313942C1 (is)
CA (1)	CA2495577C (is)
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GE (1)	GEP20064005B (is)
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HR (1)	HRP20050191B1 (is)
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MA (1)	MA27389A1 (is)
MX (1)	MXPA05001256A (is)
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NO (1)	NO20051303L (is)
NZ (1)	NZ538427A (is)
OA (1)	OA12916A (is)
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UY (1)	UY27952A1 (is)
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Also Published As

Publication number	Publication date
WO2004020431A3 (en)	2004-05-13
SI1594858T1 (sl)	2010-01-29
NO20051303L (no)	2005-05-18
PE20050131A1 (es)	2005-03-21
AP2005003237A0 (en)	2005-03-31
EA008448B1 (ru)	2007-06-29
MY139357A (en)	2009-09-30
ES2333219T3 (es)	2010-02-18
AR041055A1 (es)	2005-04-27
HRP20050191B1 (hr)	2013-12-20
CY1110580T1 (el)	2015-04-29
BRPI0313942B8 (pt)	2020-08-04
AU2003250499B2 (en)	2009-04-23
DE60329715D1 (de)	2009-11-26
PL377678A1 (pl)	2006-02-06
IS2738B (is)	2011-06-15
JP2006501309A (ja)	2006-01-12
HN2003000257A (es)	2004-12-01
NZ538427A (en)	2007-04-27
CN1319966C (zh)	2007-06-06
ATE445610T1 (de)	2009-10-15
MA27389A1 (fr)	2005-06-01
WO2004020431A2 (en)	2004-03-11
HK1078571A1 (en)	2006-03-17
IS7660A (is)	2005-01-20
BRPI0313942B1 (pt)	2019-06-04
GEP20064005B (en)	2006-12-25
TW200407131A (en)	2004-05-16
IL166832A (en)	2011-03-31
KR20070086768A (ko)	2007-08-27
US7071337B2 (en)	2006-07-04
UY27952A1 (es)	2004-03-31
PA8580301A1 (es)	2005-05-24
EP1594858B1 (en)	2009-10-14
BRPI0313942C1 (pt)	2021-05-25
DOP2003000694A (es)	2004-02-29
CR7698A (es)	2007-11-23
ECSP055633A (es)	2005-04-18
KR100816166B1 (ko)	2008-03-21
DK1594858T3 (da)	2009-12-14
RS20050180A (sr)	2007-08-03
CA2495577C (en)	2010-06-15
KR20050036984A (ko)	2005-04-20
MXPA05001256A (es)	2005-06-08
BR0313942A (pt)	2005-07-12
CN1678604A (zh)	2005-10-05
EA200500174A1 (ru)	2005-08-25
JP4551771B2 (ja)	2010-09-29
CA2495577A1 (en)	2004-03-11
US20050124599A1 (en)	2005-06-09
HRP20050191A2 (en)	2005-10-31
HRP20050191A9 (hr)	2013-11-22
AU2003250499A1 (en)	2004-03-19
CU23413B7 (es)	2009-09-08
PT1594858E (pt)	2009-12-14
EP1594858A2 (en)	2005-11-16

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ZA200501353B (en)	2006-09-27	Novel benzoimidazole derivatives useful as antiproliferative agents
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