PH20906A - Substituted anthra (1,9-cd) pyrazol-6(2h)-ones - Google Patents

Substituted anthra (1,9-cd) pyrazol-6(2h)-ones

Info

Publication number: PH20906A
Authority: PH; Philippines
Prior art keywords: pyrazol; ones; substituted anthra; anthra; substituted
Prior art date: 1982-07-23

Application number

PH29268A

Other languages

English (en)

Inventor

Showalter Howard Daniel Hollis

Leslie M Werbel

Edward F Elslager

Judith L Johnson

Original Assignee

Warner Lambert Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-07-23

Filing date

1983-07-22

Publication date

1987-05-27

1983-06-28 Priority claimed from US06/507,961 external-priority patent/US4556654A/en

1983-07-22 Application filed by Warner Lambert Co filed Critical Warner Lambert Co

1987-05-27 Publication of PH20906A publication Critical patent/PH20906A/en

Links

ACPOUJIDANTYHO-UHFFFAOYSA-N anthra[1,9-cd]pyrazol-6(2H)-one Chemical class C1=CC(C(=O)C=2C3=CC=CC=2)=C2C3=NNC2=C1 ACPOUJIDANTYHO-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
- C09B—ORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
- C09B5/00—Dyes with an anthracene nucleus condensed with one or more heterocyclic rings with or without carbocyclic rings
- C09B5/02—Dyes with an anthracene nucleus condensed with one or more heterocyclic rings with or without carbocyclic rings the heterocyclic ring being only condensed in peri position
- C09B5/16—Benz-diazabenzanthrones, e.g. anthrapyrimidones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/205—Radicals derived from carbonic acid

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Hematology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

PH29268A 1982-07-23 1983-07-22 Substituted anthra (1,9-cd) pyrazol-6(2h)-ones PH20906A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US40115782A	1982-07-23	1982-07-23
US06/507,961 US4556654A (en)	1983-06-28	1983-06-28	Antimicrobial substituted anthra[1,9-cd]pyrazol-6(2H)-ones

Publications (1)

Publication Number	Publication Date
PH20906A true PH20906A (en)	1987-05-27

Family

ID=27017319

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PH29268A PH20906A (en)	1982-07-23	1983-07-22	Substituted anthra (1,9-cd) pyrazol-6(2h)-ones

Country Status (18)

Country	Link
EP (1)	EP0103381B1 (es)
JP (2)	JPH072719B2 (es)
KR (1)	KR900005026B1 (es)
AR (1)	AR240315A1 (es)
AU (1)	AU549659B2 (es)
CA (1)	CA1230115A (es)
DE (1)	DE3373811D1 (es)
DK (3)	DK159429C (es)
ES (3)	ES8504731A1 (es)
FI (1)	FI82932C (es)
GR (1)	GR79610B (es)
HU (1)	HU195779B (es)
IE (1)	IE56782B1 (es)
IL (1)	IL69211A (es)
NO (1)	NO160000C (es)
NZ (1)	NZ205001A (es)
PH (1)	PH20906A (es)
PT (1)	PT77088B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1251451A (en) *	1984-06-29	1989-03-21	Ellen M. Berman	Benzoseleno¬4,3,2-cd\|indazole compositions and methods for their production and use
CA1251450A (en) *	1984-06-29	1989-03-21	David B. Capps	Benzopyrano¬4,3,2-cd\|indazole compositions and methods for their production and use
US4608439A (en) *	1985-04-26	1986-08-26	Warner-Lambert Company	Process for preparing substituted anthra[1,9-cd]pyrazol-6(2H)-ones
US4672129A (en) *	1986-05-05	1987-06-09	Warner-Lambert Company	Process for preparing substituted anthra[1,9-cd]pyrazol-6(2H)-ones
GB9107843D0 (en) *	1991-04-12	1991-05-29	Patterson Laurence H	Anti-cancer compounds
GB9107852D0 (en) *	1991-04-12	1991-05-29	Patterson Laurence H	Anti-cancer compounds
DE69330131T2 (de) *	1992-09-08	2001-08-30	Novuspharma S.P.A., Mailand/Milano	2-aminoalkyl-5-aminoalkylamino substituierte isochinoindazole-6 (2h)-on mit antitumorwirkung
US5393886A (en) *	1993-05-05	1995-02-28	The Du Pont Merck Pharmaceutical Company	Intermediates for the synthesis of anthrapyrazolone anticancer agents
US5596097A (en) *	1994-03-08	1997-01-21	The University Of Vermont	Hetero-annulated indazoles
IT1277576B1 (it) *	1995-09-13	1997-11-11	Boehringer Mannheim Italia	2-2-(2-idrossietil) ammino etil -5- 2-metilammino etil ammino indazolo 4,3-gh isochinolin-6 (2h)-one come agente antitumorale
US20100233689A1 (en)	2007-03-22	2010-09-16	The General Hospital Corporation	Pyrazoloanthrone and derivatives thereof for the treatment of cancer expressing 'mullerian inhibiting substance' type ii receptor (misrii) and of excess androgen states

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH191142A (de) *	1936-02-07	1937-05-31	Chem Ind Basel	Verfahren zur Herstellung eines Anthrachinonderivates.
GB470475A (en) *	1936-02-14	1937-08-16	Of Chemical Industry Soc	Manufacture of dyestuffs and intermediate products
US2518150A (en) *	1946-02-01	1950-08-08	Ciba Ltd	Vat dyestuffs
DE2558812C2 (de) *	1975-12-27	1987-04-30	Hoechst Ag, 6230 Frankfurt	Photopolymerisierbares Gemisch

1983
- 1983-07-12 IE IE1622/83A patent/IE56782B1/en not_active IP Right Cessation
- 1983-07-12 IL IL69211A patent/IL69211A/xx unknown
- 1983-07-13 AU AU16810/83A patent/AU549659B2/en not_active Expired
- 1983-07-18 CA CA000432584A patent/CA1230115A/en not_active Expired
- 1983-07-18 DK DK329683A patent/DK159429C/da not_active IP Right Cessation
- 1983-07-19 GR GR71970A patent/GR79610B/el unknown
- 1983-07-20 FI FI832638A patent/FI82932C/fi not_active IP Right Cessation
- 1983-07-21 NO NO832659A patent/NO160000C/no not_active IP Right Cessation
- 1983-07-22 HU HU832603A patent/HU195779B/hu unknown
- 1983-07-22 PH PH29268A patent/PH20906A/en unknown
- 1983-07-22 JP JP58132981A patent/JPH072719B2/ja not_active Expired - Lifetime
- 1983-07-22 PT PT77088A patent/PT77088B/pt unknown
- 1983-07-22 AR AR293692A patent/AR240315A1/es active
- 1983-07-22 DE DE8383304264T patent/DE3373811D1/de not_active Expired
- 1983-07-22 NZ NZ205001A patent/NZ205001A/en unknown
- 1983-07-22 ES ES524380A patent/ES8504731A1/es not_active Expired
- 1983-07-22 EP EP83304264A patent/EP0103381B1/en not_active Expired
- 1983-07-23 KR KR1019830003410A patent/KR900005026B1/ko not_active Expired
1984
- 1984-02-09 ES ES529577A patent/ES8507502A1/es not_active Expired
- 1984-02-09 ES ES529578A patent/ES8507503A1/es not_active Expired
1989
- 1989-08-31 DK DK430289A patent/DK160251C/da not_active IP Right Cessation
- 1989-08-31 DK DK430389A patent/DK159849C/da not_active IP Right Cessation
1994
- 1994-07-19 JP JP6166780A patent/JPH07110829B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
IE56782B1 (en)	1991-12-18
KR840005431A (ko)	1984-11-12
NO160000C (no)	1989-03-01
FI82932C (fi)	1991-05-10
NZ205001A (en)	1986-09-10
AU1681083A (en)	1984-01-26
DE3373811D1 (en)	1987-10-29
PT77088A (en)	1983-08-01
DK430289A (da)	1989-08-31
DK160251C (da)	1991-07-22
NO832659L (no)	1984-01-24
ES529577A0 (es)	1985-09-01
CA1251442C (es)	1989-03-21
DK430289D0 (da)	1989-08-31
HU195779B (en)	1988-07-28
JPS5951268A (ja)	1984-03-24
ES529578A0 (es)	1985-09-01
FI832638A0 (fi)	1983-07-20
DK159849C (da)	1991-05-13
JPH07179389A (ja)	1995-07-18
FI82932B (fi)	1991-01-31
DK160251B (da)	1991-02-18
DK329683D0 (da)	1983-07-18
CA1230115A (en)	1987-12-08
JPH072719B2 (ja)	1995-01-18
IE831622L (en)	1984-01-23
KR900005026B1 (ko)	1990-07-18
ES8507503A1 (es)	1985-09-01
DK430389A (da)	1989-08-31
IL69211A0 (en)	1983-11-30
DK430389D0 (da)	1989-08-31
AU549659B2 (en)	1986-02-06
DK159429B (da)	1990-10-15
AR240315A1 (es)	1990-03-30
DK159849B (da)	1990-12-17
ES524380A0 (es)	1985-04-16
EP0103381B1 (en)	1987-09-23
PT77088B (en)	1986-02-12
ES8504731A1 (es)	1985-04-16
EP0103381A1 (en)	1984-03-21
DK329683A (da)	1984-01-24
FI832638A7 (fi)	1984-01-24
IL69211A (en)	1987-01-30
GR79610B (es)	1984-10-31
JPH07110829B2 (ja)	1995-11-29
ES8507502A1 (es)	1985-09-01
DK159429C (da)	1991-03-18
NO160000B (no)	1988-11-21

Publication	Publication Date	Title
DE3268733D1 (en)	1986-03-13	3,5-di-tert-butyl-4-hydroxyphenyl-substituted heterocyclic compounds
DE3373811D1 (en)	1987-10-29	Substituted anthra(1,9-cd)pyrazol-6(2h)-ones
GB2082581B (en)	1985-02-13	4h-1,2,4-triazole derivatives
EP0096061A4 (en)	1985-10-28	DEMULTIPLEXING CIRCUIT.
ES523282A0 (es)	1985-02-16	Un compuesto de pirazol (3,4-b) piridina.
PH18982A (en)	1985-11-29	1- 3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl-4-hydroxy-4-phenylpiperidines
ZA835333B (en)	1984-03-28	Substituted anthra(1,9-cd)pyrazol-6(2h)-ones
AU561700B2 (en)	1987-05-14	2h(1)benzoxepino(5,4-b)1,4-oxazines
FI871945L (fi)	1987-11-06	Menetelmä substituoitujen antra(1,9-cd) pyratsol-6(2H)-onien valmistamiseksi
ATE29876T1 (de)	1987-10-15	Anthra(1,9-cd)pyrazol-6(2h)-one.
GB8315303D0 (en)	1983-07-06	Alpha-(1-triazolyl)-keto-derivatives
GB8301383D0 (en)	1983-02-23	3,3-dialkyl-and 3,3-alkylene-indoline derivatives
IL79383A0 (en)	1986-10-31	Substituted anthra(1,9-cd)pyrazol-6(2h)-ones and pharmaceutical compositions containing them
DE3368070D1 (en)	1987-01-15	Stabilization of poly-(alkadiene-1,3)
PH20407A (en)	1987-01-05	Substituted 4,5-dihydro-6-vinyl-3(2h)-pyridazinones
GB2104520B (en)	1985-01-09	Decarboxylase-inhibiting fluorinated alkane diamine derivatives
SU1088330A1 (ru)	1995-10-10	4-замещенные 11-нитро-1,4,7,9-тетраазатрицикло 7,3,1,1тетрадекан-2,6-дионы
IL70942A0 (en)	1984-05-31	2h-(1)benzoxepino(5,4-b)-1,4-oxazine derivatives
EG14280A (en)	1983-09-30	Amino-substituted 4,5,6,7-tetrahydro-1 h (or 2h) indazoles
ZA841012B (en)	1984-09-26	2h-(1)benzoxepino(5,4-b)1,4-oxazine derivatives
GB2125032B (en)	1984-08-01	1-methoxy-6, 10, 11-trihydroxy-7, 8, 9, 10 tetrahydro-5, 12-naphthacene derivatives
IL68335A0 (en)	1983-07-31	1,3,5-triacrylylhexahydro-s-triazine derivatives
IE812628L (en)	1983-05-09	1,2,4-triazole derivatives
IE822728L (en)	1983-05-17	HERBICIDAL THIAZOLO- AND £1,3\| THIAZINO-£2,3-c\|£1,2,4\|¹THIAZINONES
CS381584A2 (en)	1985-12-16	Zpusob vyroby novych derivatu thieno l3,2 c ppyridinu