PT98919A - Metodo para a obtencao de um efeito analgesico e/ou anti-inflamatorio intensificado num ser humano ou animal de pequeno porte mediante a administracao de uma composicao compreendendo um acido carboxilico e uma ou mais aminas simpatomimeticas - Google Patents

Metodo para a obtencao de um efeito analgesico e/ou anti-inflamatorio intensificado num ser humano ou animal de pequeno porte mediante a administracao de uma composicao compreendendo um acido carboxilico e uma ou mais aminas simpatomimeticas Download PDF

Info

Publication number: PT98919A
Authority: PT; Portugal
Prior art keywords: carbon atoms; pharmaceutically acceptable; human; acceptable salts; analgesic
Prior art date: 1990-09-11

Application number

PT98919A

Other languages

English (en)

Portuguese (pt)

Inventor

James Vincent Sorrentino

Original Assignee

Richardson Vicks Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-09-11

Filing date

1991-09-10

Publication date

1992-07-31

1991-09-10 Application filed by Richardson Vicks Inc filed Critical Richardson Vicks Inc

1992-07-31 Publication of PT98919A publication Critical patent/PT98919A/pt

Links

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125000003261 o-tolyl group Chemical group [H]C1=C([H])C(*)=C(C([H])=C1[H])C([H])([H])[H] 0.000 description 1
150000007530 organic bases Chemical class 0.000 description 1
201000008482 osteoarthritis Diseases 0.000 description 1
125000001037 p-tolyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1*)C([H])([H])[H] 0.000 description 1
125000000913 palmityl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 description 1
229960005489 paracetamol Drugs 0.000 description 1
239000008188 pellet Substances 0.000 description 1
210000001428 peripheral nervous system Anatomy 0.000 description 1
239000000546 pharmaceutical excipient Substances 0.000 description 1
230000000144 pharmacologic effect Effects 0.000 description 1
229960003893 phenacetin Drugs 0.000 description 1
229960002895 phenylbutazone Drugs 0.000 description 1
VYMDGNCVAMGZFE-UHFFFAOYSA-N phenylbutazonum Chemical compound O=C1C(CCCC)C(=O)N(C=2C=CC=CC=2)N1C1=CC=CC=C1 VYMDGNCVAMGZFE-UHFFFAOYSA-N 0.000 description 1
IZRPKIZLIFYYKR-UHFFFAOYSA-N phenyltoloxamine Chemical compound CN(C)CCOC1=CC=CC=C1CC1=CC=CC=C1 IZRPKIZLIFYYKR-UHFFFAOYSA-N 0.000 description 1
230000035790 physiological processes and functions Effects 0.000 description 1
239000006187 pill Substances 0.000 description 1
229920000768 polyamine Polymers 0.000 description 1
239000011591 potassium Substances 0.000 description 1
229910052700 potassium Inorganic materials 0.000 description 1
230000003389 potentiating effect Effects 0.000 description 1
239000000843 powder Substances 0.000 description 1
MFDFERRIHVXMIY-UHFFFAOYSA-N procaine Chemical compound CCN(CC)CCOC(=O)C1=CC=C(N)C=C1 MFDFERRIHVXMIY-UHFFFAOYSA-N 0.000 description 1
229960004919 procaine Drugs 0.000 description 1
125000004368 propenyl group Chemical group C(=CC)* 0.000 description 1
QELSKZZBTMNZEB-UHFFFAOYSA-N propylparaben Chemical compound CCCOC(=O)C1=CC=C(O)C=C1 QELSKZZBTMNZEB-UHFFFAOYSA-N 0.000 description 1
230000003236 psychic effect Effects 0.000 description 1
239000012629 purifying agent Substances 0.000 description 1
150000003212 purines Chemical class 0.000 description 1
230000005855 radiation Effects 0.000 description 1
239000011347 resin Substances 0.000 description 1
229920005989 resin Polymers 0.000 description 1
230000000241 respiratory effect Effects 0.000 description 1
206010039073 rheumatoid arthritis Diseases 0.000 description 1
229960002052 salbutamol Drugs 0.000 description 1
150000003902 salicylic acid esters Chemical class 0.000 description 1
FSYKKLYZXJSNPZ-UHFFFAOYSA-N sarcosine Chemical compound C[NH2+]CC([O-])=O FSYKKLYZXJSNPZ-UHFFFAOYSA-N 0.000 description 1
125000002914 sec-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(*)C([H])([H])[H] 0.000 description 1
239000000932 sedative agent Substances 0.000 description 1
230000001624 sedative effect Effects 0.000 description 1
238000000926 separation method Methods 0.000 description 1
239000011734 sodium Substances 0.000 description 1
229910052708 sodium Inorganic materials 0.000 description 1
WXMKPNITSTVMEF-UHFFFAOYSA-M sodium benzoate Chemical compound [Na+].[O-]C(=O)C1=CC=CC=C1 WXMKPNITSTVMEF-UHFFFAOYSA-M 0.000 description 1
239000004299 sodium benzoate Substances 0.000 description 1
235000010234 sodium benzoate Nutrition 0.000 description 1
239000002904 solvent Substances 0.000 description 1
230000000638 stimulation Effects 0.000 description 1
125000001424 substituent group Chemical group 0.000 description 1
238000013268 sustained release Methods 0.000 description 1
239000012730 sustained-release form Substances 0.000 description 1
239000003765 sweetening agent Substances 0.000 description 1
230000008961 swelling Effects 0.000 description 1
208000024891 symptom Diseases 0.000 description 1
201000004415 tendinitis Diseases 0.000 description 1
210000002435 tendon Anatomy 0.000 description 1
229960004559 theobromine Drugs 0.000 description 1
229960000278 theophylline Drugs 0.000 description 1
229940124597 therapeutic agent Drugs 0.000 description 1
239000002562 thickening agent Substances 0.000 description 1
230000001960 triggered effect Effects 0.000 description 1
229960001128 triprolidine Drugs 0.000 description 1
CBEQULMOCCWAQT-WOJGMQOQSA-N triprolidine Chemical compound C1=CC(C)=CC=C1C(\C=1N=CC=CC=1)=C/CN1CCCC1 CBEQULMOCCWAQT-WOJGMQOQSA-N 0.000 description 1
YFTHZRPMJXBUME-UHFFFAOYSA-N tripropylamine Chemical compound CCCN(CCC)CCC YFTHZRPMJXBUME-UHFFFAOYSA-N 0.000 description 1
XPFJYKARVSSRHE-UHFFFAOYSA-K trisodium;2-hydroxypropane-1,2,3-tricarboxylate;2-hydroxypropane-1,2,3-tricarboxylic acid Chemical compound [Na+].[Na+].[Na+].OC(=O)CC(O)(C(O)=O)CC(O)=O.[O-]C(=O)CC(O)(CC([O-])=O)C([O-])=O XPFJYKARVSSRHE-UHFFFAOYSA-K 0.000 description 1
125000002948 undecyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 description 1
229930195735 unsaturated hydrocarbon Natural products 0.000 description 1
230000008728 vascular permeability Effects 0.000 description 1
208000009935 visceral pain Diseases 0.000 description 1
125000005023 xylyl group Chemical group 0.000 description 1
239000011701 zinc Substances 0.000 description 1
229910052725 zinc Inorganic materials 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Pain & Pain Management (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Pyrane Compounds (AREA)

PT98919A 1990-09-11 1991-09-10 Metodo para a obtencao de um efeito analgesico e/ou anti-inflamatorio intensificado num ser humano ou animal de pequeno porte mediante a administracao de uma composicao compreendendo um acido carboxilico e uma ou mais aminas simpatomimeticas PT98919A (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US58068590A	1990-09-11	1990-09-11

Publications (1)

Publication Number	Publication Date
PT98919A true PT98919A (pt)	1992-07-31

Family

ID=24322117

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT98919A PT98919A (pt)	1990-09-11	1991-09-10	Metodo para a obtencao de um efeito analgesico e/ou anti-inflamatorio intensificado num ser humano ou animal de pequeno porte mediante a administracao de uma composicao compreendendo um acido carboxilico e uma ou mais aminas simpatomimeticas

Country Status (9)

Country	Link
JP (1)	JPH06500784A (fr)
KR (1)	KR930701994A (fr)
AU (1)	AU662297B2 (fr)
CA (1)	CA2090234C (fr)
IE (1)	IE913185A1 (fr)
MA (1)	MA22277A1 (fr)
MX (1)	MX9101045A (fr)
PT (1)	PT98919A (fr)
WO (1)	WO1992004021A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1994028872A1 (fr) *	1993-06-04	1994-12-22	Warner-Lambert Company	Medication sans alcool contre les rhumes et pour les sinus
US5626831A (en) *	1995-12-20	1997-05-06	Van Moerkerken; Arthur	Method for relief and prevention of common cold, and compositions
JP4549618B2 (ja) *	2001-11-22	2010-09-22	第一三共ヘルスケア株式会社	鼻炎用組成物
TWI313598B (en) *	2002-12-18	2009-08-21	Wyeth Corp	Compositions of non-steroidal anti-inflammatory drugs, decongestants and anti-histamines

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4558051A (en) *	1983-10-11	1985-12-10	Richardson-Vicks, Inc.	Analgesic and anti-inflammatory compositions comprising xanthines and methods of using same
US4522826A (en) *	1984-02-08	1985-06-11	Richardson-Vicks Inc.	Analgesic and anti-inflammatory compositions comprising diphenhydramine and methods of using same
US4552899A (en) *	1984-04-09	1985-11-12	Analgesic Associates	Cough/cold mixtures comprising non-steroidal anti-inflammatory drugs

1991
- 1991-09-09 KR KR1019930700724A patent/KR930701994A/ko not_active Ceased
- 1991-09-09 WO PCT/US1991/006398 patent/WO1992004021A1/fr not_active Ceased
- 1991-09-09 AU AU85384/91A patent/AU662297B2/en not_active Ceased
- 1991-09-09 CA CA002090234A patent/CA2090234C/fr not_active Expired - Fee Related
- 1991-09-09 JP JP3515360A patent/JPH06500784A/ja active Pending
- 1991-09-10 PT PT98919A patent/PT98919A/pt not_active Application Discontinuation
- 1991-09-10 MA MA22558A patent/MA22277A1/fr unknown
- 1991-09-10 IE IE318591A patent/IE913185A1/en unknown
- 1991-09-11 MX MX9101045A patent/MX9101045A/es unknown

Also Published As

Publication number	Publication date
KR930701994A (ko)	1993-09-08
MA22277A1 (fr)	1992-04-01
CA2090234C (fr)	1998-08-11
WO1992004021A1 (fr)	1992-03-19
AU662297B2 (en)	1995-08-31
JPH06500784A (ja)	1994-01-27
CA2090234A1 (fr)	1992-03-12
AU8538491A (en)	1992-03-30
MX9101045A (es)	1992-05-04
IE913185A1 (en)	1992-03-11

Legal Events

Date	Code	Title	Description
1992-07-31	BB1A	Laying open of patent application	Effective date: 19920327
1999-02-26	FC3A	Refusal	Effective date: 19981106

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EP0185420B1 (fr)	1991-05-29	Compositions pharmaceutiques de dihydrocodéine/ibuprofène et méthode
JP2000508341A (ja)	2000-07-04	片頭痛の治療法及び薬効の強化組成物
WO1995007103A1 (fr)	1995-03-16	Compositions contenant un sel d'acide amine d'un agent anti-inflammatoire non steroidien a base d'acide propionique et au moins un decongestionnant ou un expectorant ou un antihistaminique ou un antitussif
EP0186241A1 (fr)	1986-07-02	Compositions pharmaceutiques d'hydrocodone/ibuprofène et méthode
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CA2090234C (fr)	1998-08-11	Methode permettant d'obtenir un effet analgesique ameliore
EP0841947A1 (fr)	1998-05-20	Compositions contenant des analgesiques et des antihistaminiques et procedes de traitement d'affections respiratoires
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