SE9801526D0 - New compounds - Google Patents

New compounds

Info

Publication number
SE9801526D0
SE9801526D0 SE9801526A SE9801526A SE9801526D0 SE 9801526 D0 SE9801526 D0 SE 9801526D0 SE 9801526 A SE9801526 A SE 9801526A SE 9801526 A SE9801526 A SE 9801526A SE 9801526 D0 SE9801526 D0 SE 9801526D0
Authority
SE
Sweden
Prior art keywords
substituted
new compounds
imidazo pyridine
moiety
prevention
Prior art date
Application number
SE9801526A
Other languages
English (en)
Swedish (sv)
Inventor
Kosrat Amin
Mikael Dahlstroem
Peter Nordberg
Ingemar Starke
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Ab filed Critical Astra Ab
Priority to SE9801526A priority Critical patent/SE9801526D0/xx
Publication of SE9801526D0 publication Critical patent/SE9801526D0/xx
Priority to TW088106129A priority patent/TW490466B/zh
Priority to ARP990101776A priority patent/AR015768A1/es
Priority to TW088106128A priority patent/TWI250159B/zh
Priority to ARP990101777A priority patent/AR015769A1/es
Priority to ES99947038T priority patent/ES2252975T3/es
Priority to JP2000545865A priority patent/JP3692034B2/ja
Priority to BRPI9909995-0A priority patent/BR9909995B1/pt
Priority to UA2000106034A priority patent/UA66846C2/uk
Priority to HK01104064.2A priority patent/HK1033317B/en
Priority to IDW20002206A priority patent/ID26819A/id
Priority to HU0102313A priority patent/HUP0102313A3/hu
Priority to US09/319,890 priority patent/US6313136B1/en
Priority to RU2000127020/04A priority patent/RU2235725C2/ru
Priority to IL13920099A priority patent/IL139200A0/xx
Priority to EEP200000626A priority patent/EE04676B1/xx
Priority to EP04023091A priority patent/EP1491543B1/en
Priority to NZ507638A priority patent/NZ507638A/en
Priority to SK1492-2000A priority patent/SK285768B6/sk
Priority to TR2000/03176T priority patent/TR200003176T2/xx
Priority to NZ507639A priority patent/NZ507639A/en
Priority to SI9930868T priority patent/SI1073657T1/sl
Priority to CNB998077992A priority patent/CN1174980C/zh
Priority to AU43006/99A priority patent/AU769108B2/en
Priority to KR1020007012028A priority patent/KR100650472B1/ko
Priority to TR2001/02728T priority patent/TR200102728T2/xx
Priority to SK1491-2000A priority patent/SK14912000A3/sk
Priority to DE69937077T priority patent/DE69937077T2/de
Priority to IL13929799A priority patent/IL139297A0/xx
Priority to ES99947037T priority patent/ES2249913T3/es
Priority to EP99947038A priority patent/EP1073657B1/en
Priority to DE69928792T priority patent/DE69928792T2/de
Priority to PCT/SE1999/000662 priority patent/WO1999055705A1/en
Priority to DE69927803T priority patent/DE69927803T2/de
Priority to HK01107857.6A priority patent/HK1036984B/xx
Priority to TR2001/02612T priority patent/TR200102612T2/xx
Priority to AT99947038T priority patent/ATE312101T1/de
Priority to CZ20003981A priority patent/CZ293977B6/cs
Priority to KR1020057022787A priority patent/KR100595805B1/ko
Priority to TR2000/03149T priority patent/TR200003149T2/xx
Priority to RU2000127019/04A priority patent/RU2238271C2/ru
Priority to PL343801A priority patent/PL195000B1/pl
Priority to CA002329921A priority patent/CA2329921A1/en
Priority to CNB998078026A priority patent/CN1165535C/zh
Priority to HK01104026.9A priority patent/HK1033457B/en
Priority to EEP200000664A priority patent/EE04916B1/xx
Priority to IDW20002205A priority patent/ID27530A/id
Priority to EP99947037A priority patent/EP1073656B1/en
Priority to AU43007/99A priority patent/AU769190B2/en
Priority to AT04023090T priority patent/ATE372339T1/de
Priority to SI9930850T priority patent/SI1073656T1/sl
Priority to DE69937076T priority patent/DE69937076T2/de
Priority to DK99947038T priority patent/DK1073657T3/da
Priority to CZ20003982A priority patent/CZ292567B6/cs
Priority to BRPI9909996-9A priority patent/BR9909996B1/pt
Priority to KR1020007012027A priority patent/KR100595806B1/ko
Priority to JP2000545864A priority patent/JP3883383B2/ja
Priority to UA2000106033A priority patent/UA67769C2/uk
Priority to PL99343797A priority patent/PL343797A1/xx
Priority to AT99947037T priority patent/ATE307130T1/de
Priority to HU0102425A priority patent/HUP0102425A3/hu
Priority to HK01107808.6A priority patent/HK1036981B/xx
Priority to DK99947037T priority patent/DK1073656T3/da
Priority to PCT/SE1999/000663 priority patent/WO1999055706A1/en
Priority to AT04023091T priority patent/ATE372340T1/de
Priority to CA002329922A priority patent/CA2329922C/en
Priority to US09/319,973 priority patent/US6313137B1/en
Priority to EP04023090A priority patent/EP1491542B1/en
Priority to MYPI99001650A priority patent/MY121379A/en
Priority to MYPI99001649A priority patent/MY121389A/en
Priority to SA99200064A priority patent/SA99200064B1/ar
Priority to SA99200065A priority patent/SA99200065B1/ar
Priority to ZA200005796A priority patent/ZA200005796B/en
Priority to ZA200005797A priority patent/ZA200005797B/en
Priority to IL139200A priority patent/IL139200A/en
Priority to IS5683A priority patent/IS5683A/is
Priority to IS5684A priority patent/IS5684A/is
Priority to IL139297A priority patent/IL139297A/en
Priority to NO20005450A priority patent/NO317262B1/no
Priority to NO20005451A priority patent/NO318203B1/no
Priority to HK05103979.4A priority patent/HK1071140B/en
Priority to HK05103978.5A priority patent/HK1071139B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SE9801526A 1998-04-29 1998-04-29 New compounds SE9801526D0 (sv)

Priority Applications (82)

Application Number Priority Date Filing Date Title
SE9801526A SE9801526D0 (sv) 1998-04-29 1998-04-29 New compounds
TW088106129A TW490466B (en) 1998-04-29 1999-04-16 Imidazo pyridine derivatives which inhibit gastric acid secretion
ARP990101776A AR015768A1 (es) 1998-04-29 1999-04-16 DERIVADOS DE IMIDAZO PIRIDINA QUE INHIBEN LA SECRECIoN DE ÁCIDO GÁSTRICO, COMPOSICIoN FARMACÉUTICA, PROCEDIMIENTOS PARA SU PREPARACIoN, FORMULACIoN FARMACÉUTICA, USO DE DICHOS DERIVADOS PARA PREPARAR MEDICAMENTOS Y COMPUESTOS INTERMEDIARIOS uTILES EN EL PROCEDIMIENTO PARA LA PREPARACIoN DE DICHOS DE
TW088106128A TWI250159B (en) 1998-04-29 1999-04-16 Imidazo pyridine derivatives which inhibit gastric acid secretion
ARP990101777A AR015769A1 (es) 1998-04-29 1999-04-16 Derivados de imidazo piridina que inhiben la secrecion de acido gastrico, procedimiento para la preparacion de dichos derivados, composicion farmaceutica, uso de dichos derivados para la preparacion de medicamentos, y compuestos intermediarios.
ES99947038T ES2252975T3 (es) 1998-04-29 1999-04-23 Derivados de imidazo-piridina que inhiben la secrecion de acido gastrico.
JP2000545865A JP3692034B2 (ja) 1998-04-29 1999-04-23 胃酸分泌を阻害するイミダゾピリジン誘導体
BRPI9909995-0A BR9909995B1 (pt) 1998-04-29 1999-04-23 composto, processo para a preparação de um composto, formulação farmacêutica, e, uso de um composto.
UA2000106034A UA66846C2 (uk) 1998-04-29 1999-04-23 Похідні імідазопіридину, які інгібують секрецію шлункової кислоти
HK01104064.2A HK1033317B (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
IDW20002206A ID26819A (id) 1998-04-29 1999-04-23 Turunan imidazo piridina yang menghambat sekresi asam lambung
HU0102313A HUP0102313A3 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives, process for their preparation pharmaceutical compositions containing the same and intermediates
US09/319,890 US6313136B1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
RU2000127020/04A RU2235725C2 (ru) 1998-04-29 1999-04-23 Производные имидазопиридина, способ их получения и промежуточные соединения, фармацевтический препарат на их основе (варианты), способ ингибирования секреции желудочной кислоты и способ лечения состояний, в которые вовлечено инфицирование h.pylori
IL13920099A IL139200A0 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
EEP200000626A EE04676B1 (et) 1998-04-29 1999-04-23 Imidasopridiini derivaadid, mis inhibeerivad maohappesekretsiooni, protsess nende valmistamiseks ning nende kasutamine
EP04023091A EP1491543B1 (en) 1998-04-29 1999-04-23 Intermediate compounds for the preparation of imidazo-pyridine derivates
NZ507638A NZ507638A (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
SK1492-2000A SK285768B6 (sk) 1998-04-29 1999-04-23 Imidazopyridínové deriváty inhibujúce vylučovaniežalúdočnej kyseliny, spôsob ich prípravy, farmaceutický prostriedok a ich použitie
TR2000/03176T TR200003176T2 (tr) 1998-04-29 1999-04-23 Mide asit salgısını inhibe eden imidazo piridin türevleri
NZ507639A NZ507639A (en) 1998-04-29 1999-04-23 Imidazo pyridine dervatives which inhibit gastric acid secretion
SI9930868T SI1073657T1 (sl) 1998-04-29 1999-04-23 Imidazo piridinski derivati, ki inhibirajo izlocanje zelodcne kisline
CNB998077992A CN1174980C (zh) 1998-04-29 1999-04-23 抑制胃酸分泌的咪唑并吡啶衍生物
AU43006/99A AU769108B2 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
KR1020007012028A KR100650472B1 (ko) 1998-04-29 1999-04-23 위산 분비를 억제하는 이미다조 피리딘 유도체
TR2001/02728T TR200102728T2 (tr) 1998-04-29 1999-04-23 Mide asit salgısını inhibe eden imidazo piridin türevleri
SK1491-2000A SK14912000A3 (sk) 1998-04-29 1999-04-23 Imidazopyridínové deriváty, ktoré inhibujú vylučovanie žalúdočnej kyseliny, spôsob ich prípravy, medziprodukty tohto spôsobu a farmaceutická formulácia
DE69937077T DE69937077T2 (de) 1998-04-29 1999-04-23 Zwischenprodukte für die Herstellung von Imidazo-Pyridin-Derivate
IL13929799A IL139297A0 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
ES99947037T ES2249913T3 (es) 1998-04-29 1999-04-23 Derivados de imidazo-piridina que inhiben la secrecion de acido gastrico.
EP99947038A EP1073657B1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
DE69928792T DE69928792T2 (de) 1998-04-29 1999-04-23 Imidazo-pyridin verbindungen, die die sekretion von magensäure hemmen
PCT/SE1999/000662 WO1999055705A1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
DE69927803T DE69927803T2 (de) 1998-04-29 1999-04-23 Imidazo-pyridin verbindungen, die die sekretion von magensäure hemmen.
HK01107857.6A HK1036984B (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
TR2001/02612T TR200102612T2 (tr) 1998-04-29 1999-04-23 Mide asidi salgılanmasını önleyen imidazo piridin türevleri.
AT99947038T ATE312101T1 (de) 1998-04-29 1999-04-23 Imidazo-pyridin verbindungen, die die sekretion von magensäure hemmen
CZ20003981A CZ293977B6 (cs) 1998-04-29 1999-04-23 Imidazo[1,2-a]pyridinové deriváty inhibující sekreci žaludeční kyseliny, způsob jejich přípravy, farmaceutický prostředek a jejich použití
KR1020057022787A KR100595805B1 (ko) 1998-04-29 1999-04-23 위산 분비를 억제하는 이미다조 피리딘 유도체
TR2000/03149T TR200003149T2 (tr) 1998-04-29 1999-04-23 Mide asidi salgılanmasını önleyen imidazo piridin türevleri.
RU2000127019/04A RU2238271C2 (ru) 1998-04-29 1999-04-23 Производные имидазопиридина, способы их получения и промежуточные соединения, фармацевтический препарат на их основе (варианты), способ ингибирования секреции желудочной кислоты, способ лечения желудочно-кишечных воспалительных заболеваний и способ лечения состояний, в которых вовлечено инфицирование h.pylori
PL343801A PL195000B1 (pl) 1998-04-29 1999-04-23 Pochodne imidazopirydyny, sposób ich wytwarzania, środek farmaceutyczny, zastosowanie tych pochodnych i związki pośrednie
CA002329921A CA2329921A1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
CNB998078026A CN1165535C (zh) 1998-04-29 1999-04-23 抑制胃酸分泌的咪唑并吡啶衍生物
HK01104026.9A HK1033457B (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
EEP200000664A EE04916B1 (et) 1998-04-29 1999-04-23 Imidasopridiini derivaadid, mis inhibeerivad maohappesekretsiooni
IDW20002205A ID27530A (id) 1998-04-29 1999-04-23 Turunan-turunan imidazo piridin yang menghambat keluarnya asam lambung
EP99947037A EP1073656B1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
AU43007/99A AU769190B2 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
AT04023090T ATE372339T1 (de) 1998-04-29 1999-04-23 Zwischenprodukte für die herstellung von imidazo- pyridin-derivate
SI9930850T SI1073656T1 (sl) 1998-04-29 1999-04-23 Imidazo piridinski derivati, ki inhibirajo izlocanje zelodcne kisline
DE69937076T DE69937076T2 (de) 1998-04-29 1999-04-23 Zwischenprodukte für die Herstellung von Imidazo-Pyridin-Derivate
DK99947038T DK1073657T3 (da) 1998-04-29 1999-04-23 Imidazopyridinderivater, der inhiberer mavesyresekretion
CZ20003982A CZ292567B6 (cs) 1998-04-29 1999-04-23 Imidazopyridinové deriváty inhibující sekreci žaludeční kyseliny, způsob jejich přípravy, farmaceutický prostředek a jejich použití
BRPI9909996-9A BR9909996B1 (pt) 1998-04-29 1999-04-23 composto derivado de imidazo piridina, processo para a preparaÇço de um composto, formulaÇço farmacÊutica, e, uso de um composto.
KR1020007012027A KR100595806B1 (ko) 1998-04-29 1999-04-23 위산 분비를 억제하는 이미다조 피리딘 유도체
JP2000545864A JP3883383B2 (ja) 1998-04-29 1999-04-23 胃酸分泌を阻害するイミダゾピリジン誘導体
UA2000106033A UA67769C2 (uk) 1998-04-29 1999-04-23 Похідні імідазопіридину, які інгібують секрецію шлункової кислоти
PL99343797A PL343797A1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
AT99947037T ATE307130T1 (de) 1998-04-29 1999-04-23 Imidazo-pyridin verbindungen, die die sekretion von magensäure hemmen.
HU0102425A HUP0102425A3 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion, process for producing them and pharmaceutical compositions containing them
HK01107808.6A HK1036981B (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
DK99947037T DK1073656T3 (da) 1998-04-29 1999-04-23 Imidazopyridinderivater, der inhiberer mavesyresecernering
PCT/SE1999/000663 WO1999055706A1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
AT04023091T ATE372340T1 (de) 1998-04-29 1999-04-23 Zwischenprodukte für die herstellung von imidazo- pyridin-derivate
CA002329922A CA2329922C (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
US09/319,973 US6313137B1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion
EP04023090A EP1491542B1 (en) 1998-04-29 1999-04-23 Intermediate compounds for the preparation of imidazo-pyridine-derivatives
MYPI99001650A MY121379A (en) 1998-04-29 1999-04-27 Imidazo pyridine derivatives which inhibit gastric acid secretion
MYPI99001649A MY121389A (en) 1998-04-29 1999-04-27 Imidazo pyridine derivatives which inhibit gastric acid secretion
SA99200064A SA99200064B1 (ar) 1998-04-29 1999-05-01 مشتقات إيميدازو بيريدين imidazo pyridine المثبطة لإفراز الحمض المعدي acid secretion
SA99200065A SA99200065B1 (ar) 1998-04-29 1999-05-01 مشتقات الإيمدازو بيريدين Imidazo Pyridine المثبطة لإفراز حمض المعدة
ZA200005796A ZA200005796B (en) 1998-04-29 2000-10-18 Imidazo pyridine derivatives which inhibit gastric acid secretion.
ZA200005797A ZA200005797B (en) 1998-04-29 2000-10-18 Imidazo pyridine derivatives which inhibit gastric acid secretion.
IL139200A IL139200A (en) 1998-04-29 2000-10-23 GASTRIC ACID SECRETION INHIBITING (N - SUBSTITUTED) IMIDAZO [1,2 - a] PYRIDINE - 6 - CARBOXAMIDES CARRYING A BENZYL GROUP IN POSITION 8, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND SOME INTERMEDIATES THEREFOR
IS5683A IS5683A (is) 1998-04-29 2000-10-25 Ímídasópýridínafleiður sem hindra magasýruflæði
IS5684A IS5684A (is) 1998-04-29 2000-10-25 Ímídasópýridínafleiður sem hindra magasýruflæði
IL139297A IL139297A (en) 1998-04-29 2000-10-26 Derivatives of imidazo pyridine that inhibit gastric acid secretion
NO20005450A NO317262B1 (no) 1998-04-29 2000-10-27 Imidazopyridinderivater som inhiberer magesyresekresjon, farmasoytisk formulering som inneholder slike derivater, fremgangsmate for deres fremstilling, anvendelse derav, og mellomprodukter.
NO20005451A NO318203B1 (no) 1998-04-29 2000-10-27 Imidazopyridinderivater som inhiberer magesyresekresjon
HK05103979.4A HK1071140B (en) 1998-04-29 2001-06-12 Intermediate compounds for the preparation of imidazo-pyridine derivates
HK05103978.5A HK1071139B (en) 1998-04-29 2001-06-13 Intermediate compounds for the preparation of imidazo-pyridine-derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9801526A SE9801526D0 (sv) 1998-04-29 1998-04-29 New compounds

Publications (1)

Publication Number Publication Date
SE9801526D0 true SE9801526D0 (sv) 1998-04-29

Family

ID=20411154

Family Applications (1)

Application Number Title Priority Date Filing Date
SE9801526A SE9801526D0 (sv) 1998-04-29 1998-04-29 New compounds

Country Status (33)

Country Link
US (2) US6313137B1 (cs)
EP (4) EP1073656B1 (cs)
JP (2) JP3883383B2 (cs)
KR (3) KR100650472B1 (cs)
CN (2) CN1165535C (cs)
AR (2) AR015769A1 (cs)
AT (4) ATE312101T1 (cs)
AU (2) AU769108B2 (cs)
BR (2) BR9909996B1 (cs)
CA (2) CA2329922C (cs)
CZ (2) CZ293977B6 (cs)
DE (4) DE69937077T2 (cs)
DK (2) DK1073657T3 (cs)
EE (2) EE04676B1 (cs)
ES (2) ES2249913T3 (cs)
HU (2) HUP0102425A3 (cs)
ID (2) ID26819A (cs)
IL (4) IL139200A0 (cs)
IS (2) IS5684A (cs)
MY (2) MY121379A (cs)
NO (2) NO317262B1 (cs)
NZ (2) NZ507638A (cs)
PL (2) PL343797A1 (cs)
RU (2) RU2235725C2 (cs)
SA (2) SA99200064B1 (cs)
SE (1) SE9801526D0 (cs)
SI (1) SI1073656T1 (cs)
SK (2) SK285768B6 (cs)
TR (4) TR200003176T2 (cs)
TW (2) TW490466B (cs)
UA (2) UA67769C2 (cs)
WO (2) WO1999055705A1 (cs)
ZA (2) ZA200005797B (cs)

Families Citing this family (64)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6489346B1 (en) 1996-01-04 2002-12-03 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US5840737A (en) 1996-01-04 1998-11-24 The Curators Of The University Of Missouri Omeprazole solution and method for using same
SE9802794D0 (sv) * 1998-08-21 1998-08-21 Astra Ab New compounds
SE0003186D0 (sv) 2000-09-07 2000-09-07 Astrazeneca Ab New process
US6900324B2 (en) 2000-09-07 2005-05-31 Astrazeneca Ab Process for preparing a substituted imidazopyridine compound
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
SE0100297D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
SE0100295D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
SE0100296D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
CN1491104A (zh) * 2001-02-13 2004-04-21 新型改进释放制剂
JP2004520422A (ja) * 2001-03-08 2004-07-08 アストラゼネカ・アクチエボラーグ 新しい用途
SE0102808D0 (sv) * 2001-08-22 2001-08-22 Astrazeneca Ab New compounds
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
SE0201940D0 (sv) * 2002-06-20 2002-06-20 Astrazeneca Ab New combination II
SE0201939D0 (sv) * 2002-06-20 2002-06-20 Astrazeneca Ab New combination
DE60317529T2 (de) 2002-09-19 2008-09-25 Schering Corp. Imidazopyridine als hemmstoffe cyclin abhängiger kinasen
KR20050086584A (ko) 2002-11-19 2005-08-30 알타나 파마 아게 8-치환 이미다조피리딘
AR043002A1 (es) * 2003-02-18 2005-07-13 Altana Pharma Ag Imidazopirazinas 6-substituidos
RS53118B (sr) * 2003-02-26 2014-06-30 Sugen Inc. Aminoheteroaril jedinjenja kao inhibitori protein kinaze
DK1606261T3 (da) 2003-03-10 2010-01-18 Nycomed Gmbh Hidtil ukendt fremgangsmåde til fremstilling af roflumilast
SE525349C2 (sv) * 2003-06-23 2005-02-08 Volvo Penta Ab Utombordsdrev för båtar
SE0301903D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound III with therapeutic effect
SE0301904D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound II with therapeutic effect
SE0301905D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound I with therapeutic effect
US8993599B2 (en) 2003-07-18 2015-03-31 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
WO2005041961A1 (en) * 2003-11-03 2005-05-12 Astrazeneca Ab Imidazo [1,2-a] pyridine derivatives for the treatment of silent gastro-esophageal reflux
SE0303451D0 (sv) * 2003-12-18 2003-12-18 Astrazeneca Ab New compounds
US20080033006A1 (en) * 2004-01-26 2008-02-07 Altana Pharma Ag 1,2,4-Triazolo[ 1,5-A] Pyridines as Gastric Acid Secretion Inhibitors
US8906940B2 (en) 2004-05-25 2014-12-09 Santarus, Inc. Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
ATE405262T1 (de) * 2004-12-17 2008-09-15 Pfizer Chroman-derivate als säurepumpenantagonisten
AU2006224619B2 (en) 2005-03-16 2012-06-07 Takeda Gmbh Taste masked dosage form containing roflumilast
US7666880B2 (en) 2005-03-21 2010-02-23 S*Bio Pte Ltd. Imidazo[1,2-A]pyridine derivatives: preparation and pharmaceutical applications
MX2007011710A (es) * 2005-03-21 2007-11-20 S Bio Pte Ltd Derivados de imidazo[1,2-a]piridina, preparacion y aplicaciones farmaceuticas.
PE20061110A1 (es) * 2005-03-24 2006-10-20 Glaxo Group Ltd Derivados de imidazopiridina como antagonistas de la bomba de acido (apa)
GB0513423D0 (en) * 2005-06-30 2005-08-03 Glaxo Group Ltd Novel compounds
KR101146852B1 (ko) * 2005-12-05 2012-05-16 화이자 프로덕츠 인크. C?met/hgfr 억제제의 다형체
BRPI0619424B1 (pt) * 2005-12-05 2022-02-08 Pfizer Products Inc Uso de inibidores c-met/hgfrs para a fabricação de medicamentos
BRPI0708808A2 (pt) * 2006-03-17 2011-06-14 Raqualia Pharma Inc Derivados de cromano
WO2008013785A2 (en) 2006-07-24 2008-01-31 Singh-Broemer And Company, Inc. Solid nanoparticle formulation of water insoluble pharmaceutical substances with reduced ostwald ripening
WO2008059373A1 (en) * 2006-11-17 2008-05-22 Raqualia Pharma Inc. Imidazo [1, 2-a] pyrazine derivatives and their use as acid pump antagonists
US8513226B2 (en) * 2008-03-31 2013-08-20 Council Of Scientific And Industrial Research Simultaneous method for the preparation of a mixture of 3-acetoxy-17-acetamido-16-formyl-androst-5,17-diene and 3-acetoxy-2'-chloro-5-androsteno[17,16-b]pyridine
AU2014201644B2 (en) * 2008-12-03 2015-05-21 Cinclus Pharma Holding AB (publ) Imidazopyridine derivatives which inhibit the secretion of gastric acid
FI20086158A0 (fi) * 2008-12-03 2008-12-03 Mikael Dahlstroem Imidatsopyridiinijohdannaiset
RU2403904C1 (ru) * 2009-02-26 2010-11-20 Федеральное государственное учреждение "Научно-исследовательский институт по изучению лепры Федерального агентства по здравоохранению и социальному развитию Росздрава" Способ профилактики острых гастродуоденальных язв у больных колоректальным раком в раннем послеоперационном периоде
US8648080B2 (en) * 2009-07-09 2014-02-11 Raqualia Pharma Inc. Acid pump antagonist for the treatment of diseases involved in abnormal gastrointestinal motility
AR096684A1 (es) * 2013-06-25 2016-01-27 Ptc Therapeutics Inc Compuestos para tratar atrofia muscular espinal
WO2015095128A1 (en) 2013-12-16 2015-06-25 Asana Biosciences, Llc P2x3 and/or p2x2/3 compounds and methods
WO2015148464A1 (en) * 2014-03-24 2015-10-01 Arqule Inc. Process of preparing 3-(3-(4-(1-aminocyclobutyl)phenyl)-5-phenyl-3h-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine
CN106279151A (zh) * 2015-06-26 2017-01-04 江苏太瑞生诺生物医药科技有限公司 5-(2-(8-((2,6-二甲基苄基)氨基)-2,3-二甲基咪唑并[1,2-a]吡啶-6-甲酰胺基)乙氧基)-5-氧代戊酸的固体形式及其制备方法
KR101777971B1 (ko) 2016-07-05 2017-09-12 제일약품주식회사 이미다조[1,2-a]피리딘 유도체, 이의 제조방법 및 이의 용도
KR20190057569A (ko) * 2017-11-20 2019-05-29 제일약품주식회사 7-아미노-1h-인돌-5-카르복사미드 유도체 및 이의 용도
EP3749697A4 (en) 2018-02-05 2021-11-03 Bio-Rad Laboratories, Inc. CHROMATOGRAPHY RESIN WITH LIGAND MIXED MODE ANIONIC / HYDROPHOBIC EXCHANGE
KR102706151B1 (ko) 2018-04-10 2024-09-13 바이엘 악티엔게젤샤프트 2,6-디알킬페닐아세트산을 제조하는 방법
RU2732297C2 (ru) * 2018-11-14 2020-09-15 Общество с ограниченной ответственностью "Гурус БиоФарм" Производные нестероидных противовоспалительных средств
ES2949232T3 (es) 2019-11-04 2023-09-26 Cinclus Pharma Holding Ab Publ Formulación Oral de X842
JP2024542115A (ja) 2021-11-05 2024-11-13 シンクルス・ファーマ・ホールディング・アクチエボラグ リナプラザングルレートのメシラート塩の多形体
JP2024530045A (ja) 2021-11-05 2024-08-14 シンクルス・ファーマ・ホールディング・アクチエボラグ リナプラザングルレート塩酸塩の多形
KR102496869B1 (ko) * 2022-07-29 2023-02-07 제일약품주식회사 이미다조[1,2-a]피리딘 화합물의 신규 염, 이의 결정형 및 제조방법
KR20250132529A (ko) 2023-01-11 2025-09-04 싱클루스 파마 홀딩 에이비 (피유비엘) 리나프라잔 글루레이트의 하이드로브로마이드 염의 다형체
KR20250130654A (ko) 2023-01-11 2025-09-02 싱클루스 파마 홀딩 에이비 (피유비엘) 리나프라잔 글루레이트의 말레산 염의 다형체
CR20250351A (es) * 2023-02-01 2025-10-13 Jeil Pharmaceutical Co Ltd Formulación farmacéutica, método de preparación para la misma y composición de tableta
WO2025215593A1 (en) * 2024-04-12 2025-10-16 Hetero Labs Limited An improved process for preparation of zastaprazan
KR20260002253A (ko) * 2024-06-28 2026-01-06 온코닉테라퓨틱스 주식회사 이미다조[1,2-a]피리딘 화합물의 신규 염 및 이의 제조방법
KR20260002254A (ko) * 2024-06-28 2026-01-06 온코닉테라퓨틱스 주식회사 이미다조[1,2-a]피리딘 화합물의 신규 염의 결정형 및 이의 제조방법

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA81219B (en) * 1980-01-23 1982-01-27 Schering Corp Imidazo (1,2-a) pyridines ,process for their preparation and pharmaceutical compositions containing them
EP0068378B1 (en) * 1981-06-26 1986-03-05 Schering Corporation Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them
US4725601A (en) 1985-06-04 1988-02-16 Fujisawa Pharmaceutical Co., Ltd. Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers
EP0228006A1 (en) * 1985-12-16 1987-07-08 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine compounds and processes for preparation thereof
GB8722488D0 (en) * 1987-09-24 1987-10-28 Fujisawa Pharmaceutical Co Imidazopyridine compound
GB9102997D0 (en) * 1991-02-13 1991-03-27 Pfizer Ltd Therapeutic agents
GB9107513D0 (en) * 1991-04-10 1991-05-29 Fujisawa Pharmaceutical Co Pyrazolopyridine compound and processes for preparation thereof

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