SK26094A3 - O-heteroaryl-, o-alkylheteroaryl-, o-alkenylheteroaryl- and o-alkylheteroaryl macrolides compounds, the method of their production and pharmaceutical preparations containing those - Google Patents

O-heteroaryl-, o-alkylheteroaryl-, o-alkenylheteroaryl- and o-alkylheteroaryl macrolides compounds, the method of their production and pharmaceutical preparations containing those Download PDF

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Publication number
SK26094A3
SK26094A3 SK260-94A SK26094A SK26094A3 SK 26094 A3 SK26094 A3 SK 26094A3 SK 26094 A SK26094 A SK 26094A SK 26094 A3 SK26094 A3 SK 26094A3
Authority
SK
Slovakia
Prior art keywords
ethyl
dioxa
tetramethyl
methylvinyl
tetraone
Prior art date
Application number
SK260-94A
Other languages
English (en)
Slovak (sk)
Inventor
Peter J Sinclair
Frederick Wong
Joung Goulet
Mark Goulet
Williams H Parsons
Matthew J Wyvratt
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of SK26094A3 publication Critical patent/SK26094A3/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Transplantation (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Measurement Of Force In General (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
SK260-94A 1991-09-09 1992-09-02 O-heteroaryl-, o-alkylheteroaryl-, o-alkenylheteroaryl- and o-alkylheteroaryl macrolides compounds, the method of their production and pharmaceutical preparations containing those SK26094A3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US75694691A 1991-09-09 1991-09-09
US07/921,851 US5252732A (en) 1991-09-09 1992-08-05 D-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity
PCT/US1992/007508 WO1993005058A1 (en) 1991-09-09 1992-09-02 O-heteroaryl, o-alkylheteroaryl, o-alkenylheteroaryl and o-alkynylheteroarylmacrolides

Publications (1)

Publication Number Publication Date
SK26094A3 true SK26094A3 (en) 1994-08-10

Family

ID=27116312

Family Applications (1)

Application Number Title Priority Date Filing Date
SK260-94A SK26094A3 (en) 1991-09-09 1992-09-02 O-heteroaryl-, o-alkylheteroaryl-, o-alkenylheteroaryl- and o-alkylheteroaryl macrolides compounds, the method of their production and pharmaceutical preparations containing those

Country Status (21)

Country Link
US (2) US5252732A (cs)
EP (1) EP0532088B1 (cs)
JP (1) JPH0813819B2 (cs)
KR (1) KR930006030A (cs)
CN (1) CN1073443A (cs)
AT (1) ATE145915T1 (cs)
AU (1) AU647665B2 (cs)
BG (1) BG98639A (cs)
CA (1) CA2077331A1 (cs)
CZ (1) CZ53194A3 (cs)
DE (1) DE69215615T2 (cs)
FI (1) FI941085A7 (cs)
HU (1) HUT66855A (cs)
IL (1) IL103009A0 (cs)
MX (1) MX9205137A (cs)
NO (1) NO940805L (cs)
NZ (1) NZ244153A (cs)
RO (1) RO114331B1 (cs)
SK (1) SK26094A3 (cs)
WO (1) WO1993005058A1 (cs)
YU (1) YU89792A (cs)

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Also Published As

Publication number Publication date
AU2282992A (en) 1993-03-11
ATE145915T1 (de) 1996-12-15
HU9400686D0 (en) 1994-06-28
US5252732A (en) 1993-10-12
CA2077331A1 (en) 1993-03-10
DE69215615T2 (de) 1997-06-26
JPH06116274A (ja) 1994-04-26
BG98639A (bg) 1995-03-31
JPH0813819B2 (ja) 1996-02-14
NO940805D0 (no) 1994-03-08
KR930006030A (ko) 1993-04-20
WO1993005058A1 (en) 1993-03-18
AU647665B2 (en) 1994-03-24
MX9205137A (es) 1993-04-01
FI941085L (fi) 1994-05-03
CZ53194A3 (en) 1994-08-17
RO114331B1 (ro) 1999-03-30
FI941085A7 (fi) 1994-05-03
US5349061A (en) 1994-09-20
NZ244153A (en) 1995-04-27
HUT66855A (en) 1995-01-30
DE69215615D1 (de) 1997-01-16
FI941085A0 (fi) 1994-03-08
CN1073443A (zh) 1993-06-23
EP0532088A1 (en) 1993-03-17
YU89792A (sh) 1996-01-08
NO940805L (no) 1994-05-06
EP0532088B1 (en) 1996-12-04
IL103009A0 (en) 1993-02-21

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