AR219963A1 - Procedimiento para preparar nuevos derivados de (alcoil(c1-c10)-3-isoquinolil-5-imino)-3-tetrahidro-1,5,10,10a-tiazol(3,4-b)- isoquinoleina - Google Patents

Procedimiento para preparar nuevos derivados de (alcoil(c1-c10)-3-isoquinolil-5-imino)-3-tetrahidro-1,5,10,10a-tiazol(3,4-b)- isoquinoleina

Info

Publication number
AR219963A1
AR219963A1 AR275407A AR27540779A AR219963A1 AR 219963 A1 AR219963 A1 AR 219963A1 AR 275407 A AR275407 A AR 275407A AR 27540779 A AR27540779 A AR 27540779A AR 219963 A1 AR219963 A1 AR 219963A1
Authority
AR
Argentina
Prior art keywords
isoquinolil
alcoil
isoquinolein
thiazol
imino
Prior art date
Application number
AR275407A
Other languages
English (en)
Original Assignee
Rhone Poulenc Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7701516A external-priority patent/FR2378030A1/fr
Priority claimed from FR7739028A external-priority patent/FR2412545A1/fr
Application filed by Rhone Poulenc Ind filed Critical Rhone Poulenc Ind
Application granted granted Critical
Publication of AR219963A1 publication Critical patent/AR219963A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/14Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
    • C07D217/16Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
AR275407A 1977-01-20 1979-02-05 Procedimiento para preparar nuevos derivados de (alcoil(c1-c10)-3-isoquinolil-5-imino)-3-tetrahidro-1,5,10,10a-tiazol(3,4-b)- isoquinoleina AR219963A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7701516A FR2378030A1 (fr) 1977-01-20 1977-01-20 Nouveau derive de l'isoquinoleine, sa preparation et les compositions qui le contiennent
FR7739028A FR2412545A1 (fr) 1977-12-23 1977-12-23 Nouveaux derives de l'isoquinoleine, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
AR219963A1 true AR219963A1 (es) 1980-09-30

Family

ID=26219809

Family Applications (2)

Application Number Title Priority Date Filing Date
AR270785A AR217460A1 (es) 1977-01-20 1978-01-20 Procedimiento para preparar derivados de((alquil-3-isoquinolil-5)-imino)-3-tetrahidro-1, 5, 10,10a-tiazol-(3,4-b)-isoquinoleina y sus sales
AR275407A AR219963A1 (es) 1977-01-20 1979-02-05 Procedimiento para preparar nuevos derivados de (alcoil(c1-c10)-3-isoquinolil-5-imino)-3-tetrahidro-1,5,10,10a-tiazol(3,4-b)- isoquinoleina

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR270785A AR217460A1 (es) 1977-01-20 1978-01-20 Procedimiento para preparar derivados de((alquil-3-isoquinolil-5)-imino)-3-tetrahidro-1, 5, 10,10a-tiazol-(3,4-b)-isoquinoleina y sus sales

Country Status (25)

Country Link
US (1) US4153698A (es)
JP (1) JPS5914037B2 (es)
AR (2) AR217460A1 (es)
AT (1) AT361481B (es)
AU (1) AU510044B2 (es)
CA (1) CA1091674A (es)
CH (1) CH633010A5 (es)
CS (2) CS195349B2 (es)
DE (1) DE2802453C3 (es)
DK (1) DK143343C (es)
ES (2) ES466192A1 (es)
FI (1) FI62314C (es)
GB (1) GB1574281A (es)
GR (1) GR61726B (es)
HU (1) HU174219B (es)
IE (1) IE46375B1 (es)
IL (1) IL53841A (es)
LU (1) LU78895A1 (es)
NL (1) NL7800383A (es)
NO (1) NO780202L (es)
NZ (1) NZ186282A (es)
OA (1) OA05859A (es)
PT (1) PT67545B (es)
SE (1) SE7800681L (es)
SU (2) SU730309A3 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU797580A3 (ru) * 1977-11-10 1981-01-15 Рон-Пуленк Эндюстри (Фирма) Способ получени производных изохино-лиНА, иХ СОлЕй, РАцЕМАТОВ или ОпТичЕС-КиХ изОМЕРОВ
FR2456098A2 (fr) * 1977-12-23 1980-12-05 Rhone Poulenc Ind Nouveaux derives de l'isoquinoleine, leur preparation et les compositions pharmaceutiques qui les contiennent
NL7908655A (nl) * 1978-12-07 1980-06-10 Rhone Poulenc Ind Nieuwe thienopyridine-derivaten, de bereiding ervan, alsmede farmaceutische preparaten, die de nieuwe derivaten bevatten.
FR2456111A1 (fr) * 1979-05-09 1980-12-05 Rhone Poulenc Ind Nouveaux derives de l'indole, leur preparation et les medicaments qui les contiennent
GB2048880A (en) * 1979-05-09 1980-12-17 Rhone Poulenc Ind Isoquinoline derivatives
NZ195721A (en) * 1979-12-04 1982-09-14 Rhone Poulenc Ind Thiazolo(3,4-b)isoquinoline derivatives and pharmaceutical compositions
US4269842A (en) * 1979-12-05 1981-05-26 Rhone-Poulenc Industries Method for treating rhinoviral complaints
US6582728B1 (en) * 1992-07-08 2003-06-24 Inhale Therapeutic Systems, Inc. Spray drying of macromolecules to produce inhaleable dry powders

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL169076C (nl) * 1975-08-06 1982-06-01 Rhone Poulenc Ind Werkwijze voor het bereiden of vervaardigen van farmacologische preparaten met een analgetische en antipyretische werking, alsmede werkwijze voor het bereiden van geneeskrachtige verbindingen, welke geschikt zijn voor gebruik in dergelijke preparaten.

Also Published As

Publication number Publication date
CH633010A5 (fr) 1982-11-15
CA1091674A (fr) 1980-12-16
DE2802453B2 (de) 1981-04-02
GB1574281A (en) 1980-09-03
IE46375B1 (en) 1983-05-18
DE2802453C3 (de) 1982-03-25
FI62314B (fi) 1982-08-31
SE7800681L (sv) 1978-07-21
NL7800383A (nl) 1978-07-24
US4153698A (en) 1979-05-08
PT67545B (fr) 1979-06-15
IE780126L (en) 1978-07-20
PT67545A (fr) 1978-02-01
IL53841A0 (en) 1978-04-30
LU78895A1 (fr) 1978-09-18
NZ186282A (en) 1980-02-21
FI62314C (fi) 1982-12-10
AU3261178A (en) 1979-08-02
ES466192A1 (es) 1978-10-16
GR61726B (en) 1978-12-29
DK143343C (da) 1982-01-25
DK27178A (da) 1978-07-21
FI780182A7 (fi) 1978-07-21
AR217460A1 (es) 1980-03-31
ATA39378A (de) 1980-08-15
OA05859A (fr) 1981-05-31
DE2802453A1 (de) 1978-07-27
CS195349B2 (en) 1980-01-31
NO780202L (no) 1978-07-21
AT361481B (de) 1981-03-10
JPS5914037B2 (ja) 1984-04-02
HU174219B (hu) 1979-11-28
CS195350B2 (en) 1980-01-31
SU730309A3 (ru) 1980-04-25
IL53841A (en) 1980-10-26
JPS53116399A (en) 1978-10-11
AU510044B2 (en) 1980-06-05
DK143343B (da) 1981-08-10
SU776560A3 (ru) 1980-10-30
ES468630A1 (es) 1978-12-01

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